A Direct Synthesis of Racemic
1,3,4,5-Tetragalloylapiitol

Please copy the URL and add it into your RSS Feed Reader.

Facebook X Linkedin Weibo

Download PDF

Synthesis 2010(3): 389-391
DOI: 10.1055/s-0029-1217123

SHORTPAPER

George A. Kraus*, Aaron Kempema
Department of Chemistry, Iowa State University, Ames, IA 50011, USA
Fax: +1(515)2940105; e-Mail: gakraus@iastate.edu;

Further Information

Received 7 August 2009
Publication Date:
13 November 2009 (online)

A direct and flexible synthesis of racemic 1,3,4,5-tetragalloylapiitol is described.

apiitol - HIV - osmium tetroxide - deprotection

1 Raskin I. Ribnicky DM. Komarnytsky S. Ilic N. Poulev A. Borisjuk N. Brinker A. Moreno DA. Ripoll C. Yakoby N. O’Neal JM. Cornwell T. Pastor I. Fridlender B. Trends Biotechnol. 2002, 20: 522

Crossref Google Scholar
2 Takada K. Bermingham A. O’Keefe BR. Wamiru A. Beutler JA. Le Grice SFJ. Lloyd J. Gustafson KR. McMahon JB. J. Nat. Prod. 2007, 70: 1647

Crossref PubMed Google Scholar
3 Patel RM. Argade NP. Synthesis 2009, 372

Article in Thieme Connect Google Scholar
4 Sodeoka M. Yamada H. Shibasaki M. J. Am. Chem. Soc. 1990, 112: 4906

Crossref Google Scholar
5 Furegati S. White AJP. Miller AD. Synlett 2005, 2385

Article in Thieme Connect Google Scholar
6 Ren Y. Himmeldirk K. Chen X. J. Med. Chem. 2006, 49: 2829

Crossref PubMed Google Scholar
7 Tully SE. Mabon R. Gama CI. Tsai SM. Liu X. Hiseh-Wilson LC. J. Am. Chem. Soc. 2004, 126: 7736

Crossref PubMed Google Scholar