Synthesis

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Issue eFirst

Rai, Shweta; Samatha, Polasani; Addipilli, Ramunaidu; Mainkar, Prathama S.; Sripadi, Prabhakar; Adepu, Raju; Chandrasekhar, Srivari: Poly(ethylene glycol) Dimethyl Ethers (PEGDME): Efficient and Recyclable Solvents for Aryne-Involved Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0147_ga_10-1055_a-1846-5598.gif
Gillard, Rachel M.; Zhang, Jiajun; Steel, Richard; Wang, Jocelyn; Strull, Jessica L.; Cai, Bin; Chakraborty, Nilanjana; Boger, Dale L.: Aryl Annulation: A Powerful Simplifying Retrosynthetic Disconnection
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0449_ga_10-1055_a-1959-2088.gif
Majhi, Jadab; Zhou, Bohang; Zhuang, Yuxin; Tom, Mai-Jan; Dai, Huifang; Evans, P. Andrew: Palladium-Catalyzed Cross-Coupling of Cyanohydrins with Aryl Bromides: Construction of Biaryl Ketones
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0052_ga_10-1055_a-1850-3687.gif
Khatana, Anil Kumar; Singh, Vikram; Gupta, Manoj Kumar; Tiwari, Bhoopendra: A Highly Efficient NHC-Catalyzed Aerobic Oxidation of Aldehydes to Carboxylic Acids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0219_ga_10-1055_s-0037-1610069.gif
Abuhafez, Naba; Perennes, Antoine; Gramage-Doria, Rafael: Mimicking Enzymes: Taking Advantage of the Substrate-Recognition Properties of Metalloporphyrins in Supramolecular Catalysis
https://www.thieme-connect.de/media/synthesis/202215/i_r0743_ga_10-1055_a-1729-9223.gif
Liu, Cheng-Yuan; Chen, Ying-Ho; Chen, Chih-Hao; Yu, Ming-Shiuan; Tsai, Fu-Yu; Ong, Tiow-Gan: Selective C(8)–H Activation of Imidazopyridines Mediated by Cooperative Nickel–Aluminum Catalysis
https://www.thieme-connect.de/media/synthesis/201617/i_c0130_ga_10-1055_s-0035-15661438.gif
Sarmah, Manashi; Hazarika, Hemanta; Gogoi, Pranjal: Aryne Annulations for the Synthesis of Carbocycles and Heterocycles: An Updated Review
https://www.thieme-connect.de/media/synthesis/202222/i_r0146_ga_10-1055_a-1863-8622.gif
Veth, Lukas; Grab, Hanusch A.; Dydio, Paweł: Recent Trends in Group 9 Catalyzed C–H Borylation Reactions: Different Strategies To Control Site-, Regio-, and Stereoselectivity
https://www.thieme-connect.de/media/synthesis/202215/i_z0615_ga_10-1055_a-1711-5889.gif
Kręcijasz, Remigiusz B.; Malinčík, Juraj; Šolomek, Tomáš: Exploring Silyl Protecting Groups for the Synthesis of Carbon Nanohoops
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0520_ga_10-1055_a-2008-9505.gif
Condon, Sylvie; Nédélec, Jean-Yves: Overview on Nickel-Catalyzed Electrochemical Conjugate Addition of Organic Halides on Electron-Deficient Olefins
https://www.thieme-connect.de/bilder/synthesis/200418/c050_ga
He, Xiao-Yu; Ma, Yu-Hong; Yang, Qing-Qing; Xiao, Wen-Jing: [4+n] Annulation Reactions Using ortho-Chloromethyl Anilines as Aza-ortho-Quinone Methide Precursors
https://www.thieme-connect.de/media/synthesis/202204/i_m0311_ga_10-1055_a-1529-7739.gif
Kimura, Masanari; Kojima, Keisuke; Tamaru, Yoshinao: Nickel-Catalyzed Three-Component Connection Reaction of Dimethylzinc, 1,ω-Ene-Diene, and Acetone: Synthesis of 1,2-Disubstituted Cycloalkanes
https://www.thieme-connect.de/bilder/synthesis/200418/c053_ga
Shirke, Rajendra P.; Reddy, Virsinha; Anand, R. Vijaya; Ramasastry, S. S. V.: Furans to Benzofurans: Intramolecular Cross-Benzoin Reactions Catalysed by N-Heterocyclic Carbenes
https://www.thieme-connect.de/media/synthesis/201612/i_c0133_ga_10-1055_s-0035-1560432.gif
Moragas, Toni; Martin, Ruben: Nickel-Catalyzed Reductive Carboxylation of Cyclopropyl Motifs with Carbon Dioxide
https://www.thieme-connect.de/media/synthesis/201617/i_z0171_ga_10-1055_s-0035-1560439.gif
Shi, Shicheng; Lalancette, Roger; Szostak, Michal: Cyclization of Imides to 2-Azabicycles via Aminoketyl Radicals by Using Samarium(II) Iodide–Water: Reaction Development, Synthetic Scope, and Mechanistic Studies
https://www.thieme-connect.de/media/synthesis/201612/i_c0066_ga_10-1055_s-0035-1560437.gif
Gao, Xing; Han, Jianwei; Wang, Limin: Chiral Iminophosphorane Organocatalyzed Asymmetric Sulfenyl­ation of 3-Substituted Oxindoles: Substrate-Interrelated Enantio­selectivities
https://www.thieme-connect.de/media/synthesis/201616/i_c0026_ga_10-1055_s-0035-1560435.gif
Cai, Pin-Wen; You, Zhi-Hao; Xie, Liang-Hui; Tan, Rui; Tong, Zhi-Ping; Liu, Yan-Kai: The Attractive Application of Lactol Chemistry: From Racemic Lactol to Natural Product Skeleton
https://www.thieme-connect.de/media/synthesis/201616/i_c0029_ga_10-1055_s-0035-1561972.gif
Schweighauser, Luca; Bodoky, Ina; Kessler, Simon N.; Häussinger, Daniel; Wegner, Hermann A.: Bidentate Lewis Acid Catalyzed Inverse-Electron-Demand Diels–Alder Reaction for the Selective Functionalization of Aldehydes
https://www.thieme-connect.de/media/synthesis/201214/c0325_ga.gif
Hayashi, Mikishiro; Michikita, Ryudai; Usuki, Yoshinosuke; Satoh, Tetsuya: Construction of Thienopyrroles through Rhodium-Catalyzed Direct Annulation of (Acetylamino)thiophenes with Alkynes
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0645_ga_10-1055_a-2015-4466.gif
Kumar, Raju Suresh; Almansour, Abdulrahman I.; Arumugam, Natarajan; Menéndez, J. Carlos; Osman, Hasnah; Kumar, Raju Ranjith: Dipolar Cycloaddition-Based Multicomponent Reactions in Ionic Liquids: A Green, Fully Stereoselective Synthesis of Novel Polycyclic Cage Systems with the Generation of Two New Azaheterocyclic Rings
https://www.thieme-connect.de/media/synthesis/201518/i_c0234_ga_10-1055_s-0034-1379931.gif
Nori, Valeria; Sinibaldi, Arianna; Pesciaioli, Fabio; Carlone, Armando: Impact of Design of Experiments in the Optimisation of Catalytic Reactions in Academia
https://www.thieme-connect.de/media/synthesis/202219/i_r0735_ga_10-1055_a-1736-6703.gif
Kabuki, Akira; Yamaguchi, Junichiro: Formal Syntheses of Dictyodendrins B, C, and E by a Multi-Substituted Indole Synthesis
https://www.thieme-connect.de/media/synthesis/202222/i_f0070_ga_10-1055_a-1786-9881.jpg
Berti, Francesco; Favero, Lucilla; Pineschi, Mauro: Asymmetric Synthesis of Methylphenidate and Quinolizidinones by Addition of Aldehydes to Piperidine-Based Conjugated N-Acyl­iminium Ions
https://www.thieme-connect.de/media/synthesis/201616/i_c0250_ga_10-1055_s-0035-1562486.gif
Ledovskaya, Maria S.; Voronin, Vladimir V.; Rodygin, Konstantin S.; Ananikov, Valentine P.: Acetylene and Ethylene: Universal C2 Molecular Units in Cycloaddition Reactions
https://www.thieme-connect.de/media/synthesis/202204/i_r0524_ga_10-1055_a-1654-2318.gif
Brandão, Pedro; Pineiro, Marta; Burke, Anthony J.: Tryptanthrin and Its Derivatives in Drug Discovery: Synthetic Insights
https://www.thieme-connect.de/media/synthesis/202219/i_r0723_ga_10-1055_s-0040-1719901.jpg
Patra, Subrata; Mosiagin, Ivan; Giri, Rahul; Katayev, Dmitry: Organic Nitrating Reagents
https://www.thieme-connect.de/media/synthesis/202215/i_r0727_ga_10-1055_s-0040-1719905.gif
Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)
https://www.thieme-connect.de/media/synthesis/202204/i_z0484_ga_10-1055_s-0040-1705983.gif
Arnold, Jeffrey S.; Nguyen, Hien M.: Rhodium-Catalyzed Asymmetric Amination of Allylic Trichloroacetimidates
https://www.thieme-connect.de/media/synthesis/201315/i_c0145_ga_10-1055_s-0032-1316921.gif
Shimazumi, Ryoma; Kodama, Takuya; Tobisu, Mamoru: Palladium-Catalyzed Unimolecular Fragment Coupling of N-Allylamides Bearing a Tethered Nucleophile with the Translocation of an Amide Group
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0559_ga_10-1055_a-2022-1905.gif
Artigas, Albert; Hagebaum-Reignier, Denis; Carissan, Yannick; Coquerel, Yoann: Multidimensional Isotropic Magnetic Shielding Contour Maps for the Visualization of Aromaticity in ortho-Arynes and Their Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0169_ga_10-1055_a-1867-0674.jpg
Frost, Christopher G.; Edwards, Hannah J.; Penrose, Stephen D.; Gleave, Robert: Exploring Rhodium-Catalysed Conjugate Addition of Chiral Alkenylboronates Using Chiral Olefin Ligands
https://www.thieme-connect.de/media/synthesis/201019/c040_ga.jpg
La Torre, Mathéo; Maton, William; Cleator, Ed; Jouffroy, Matthieu: Pd/C Catalyzed Dehalogenation of (Hetero)aryls Using Triethyl­silane as Hydrogen Donor
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0534_ga_10-1055_s-0042-1753402.gif
Airiau, Etienne; Chemin, Claire; Girard, Nicolas; Lonzi, Giacomo; Mann, André; Petricci, Elena; Salvadori, Jessica; Taddei, Maurizio: Microwave-Assisted Domino Hydroformylation/Cyclization Reactions: Scope and Limitations
https://www.thieme-connect.de/media/synthesis/201017/c034_ga.jpg
Nocera, Giuseppe; Murphy, John A.: Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0401_ga_10-1055_s-0039-1690614.gif
Wang, Li; Wang, Zhi-Qian; Xu, Ming-Hua; Lin, Guo-Qiang: Highly Enantioselective Synthesis of (Diarylmethyl)amines by Rhodium-Catalyzed­ Arylation of N-Nosylimines Using a Chiral Bicyclo[3.3.0]diene Ligand
https://www.thieme-connect.de/media/synthesis/201019/c039_ga.jpg
Parker, Patrick D.; Pierce, Joshua G.: Synthesis of 1,2,4-Oxadiazoles via DDQ-Mediated Oxidative Cyclization of Amidoximes
https://www.thieme-connect.de/media/synthesis/201612/i_c0091_ga_10-1055_s-0035-1561597.gif
Zhang, Qingchen; Wang, Xuan; Qian, Qun; Gong, Hegui: Nickel-Catalyzed Reductive Cross-Coupling of Benzyl Halides with Aryl Halides
https://www.thieme-connect.de/media/synthesis/201617/i_c0285_ga_10-1055_s-0035-1562442.gif
Belhomme, Marie-Charlotte; Dru, Delphine; Xiong, Heng-Ying; Cahard, Dominique; Besset, Tatiana; Poisson, Thomas; Pannecoucke, Xavier: Copper-Mediated Direct Functionalization of Unsaturated C–C Bonds with Ethyl Bromo(difluoro)acetate: A Straightforward Access to Highly Valuable Difluoromethylated Alkenes
https://www.thieme-connect.de/media/synthesis/201414/i_c0137_ga_10-1055_s-0033-1338637.gif
Liu, Jiangguang; Yan, Jiajie; Qin, Dongguang; Cai, Qian: An Unexpected Inversion of Enantioselectivity in a Copper-Catalyzed Intramolecular­ Desymmetric Aryl C–N Coupling Reaction
https://www.thieme-connect.de/media/synthesis/201414/i_c0121_ga_10-1055_s-0033-1338638.gif
Székely, Anna; Sinai, Ádám; Tóth, Edina B.; Novák, Zoltán: Utilization of a Copper on Iron Catalyst for the Synthesis of Biaryl Systems and Benzoxazines via Oxidative Arylation of Anilide Derivatives
https://www.thieme-connect.de/media/synthesis/201414/i_c0145_ga_10-1055_s-0033-1338642.gif
Sperger, Theresa; Schoenebeck, Franziska: α-Arylation of Esters and Ketones Enabled by a Bench-Stable Pd(I) Dimer Catalyst
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0285_ga_10-1055_s-0037-1610087.gif
Agudelo, Brian Castro; Rigoulet, Florian; Giorgi, Michel; Sayah, Babak; Rodriguez, Jean; Coquerel, Yoann: Synthesis of Axially Chiral Cationic Benzo[c]phenanthridinium Derivatives
https://www.thieme-connect.de/media/synthesis/202222/i_f0170_ga_10-1055_a-1845-3128.gif
Liu, Wenting; Hong, Xiaohu; Xu, Bin: Rhodium-Catalyzed Oxidative Coupling of Aryl Hydrazones with Internal Alkynes: Efficient Synthesis of Multisubstituted Isoquinolines
https://www.thieme-connect.de/media/synthesis/201315/i_c0154_ga_10-1055_s-0033-1338417.gif
Sebald, Michael A.; Gebauer, Julian; Koch, Matthias: Concise Syntheses of Alternariol, Alternariol-9-monomethyl Ether and Their D3-Isotopologues
https://www.thieme-connect.de/media/synthesis/202219/i_f0536_ga_10-1055_a-1698-8328.gif
Wildermuth, Raphael; Speck, Klaus; Magauer, Thomas: Gold(I)-Catalyzed Enyne Cyclizations: Studies Toward the Total Synthesis of (+)-Aureol
https://www.thieme-connect.de/media/synthesis/201612/i_c0046_ga_10-1055_s-0035-1561589.gif
Liu, Linhao; Doucet, Henri: Scope and Limitations of the Palladium-Catalyzed Direct 1,2-Diheteroarylation of 1,2-Dihalobenzene Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0442_ga_10-1055_a-1981-3213.gif
Endo, Chikako; Inoue, Yurika; Maruyama, Toshifumi; Minoura, Mao; Murai, Toshiaki: Two-Step Transesterification of Phosphates, Phosphorothioates, and Phosphonates with a Binaphthyl Group for the Synthesis of P-Chirogenic Phosphates and Phosphonates
https://www.thieme-connect.de/media/synthesis/202306/i_c0357_ga_10-1055_a-1948-3003.gif
Malkina, Anastasiya G.; Stepanov, Anton V.; Sobenina, Lyubov N.; Shemyakina, Olesya A.; Ushakov, Igor A.; Smirnov, Vladimir I.; Trofimov, Boris A.: Organocatalyzed Microwave-Assisted Competing Cyclization of Cyanopropargylic Alcohols with Carboxylic Acids: 4-Cyano-3(2H)-furanones versus 4-Cyano-[(Z)-3-cyanomethylene]-2,3-dihydro­furans
https://www.thieme-connect.de/media/synthesis/201612/i_c0071_ga_10-1055_s-0035-1561591.gif
Li, Zhilong; Tong, Rongbiao: Asymmetric Total Syntheses of the trans-2-Aryl-6-alkyltetrahydropyrans Diospongin B and Parvistones D and E from a Common Precursor
https://www.thieme-connect.de/media/synthesis/201611/i_c0023_ga_10-1055_s-0035-1561592.gif
Nambu, Hisanori; Ono, Naoki; Yakura, Takayuki: Acid-Catalyzed Ring-Opening Cyclization of Spirocyclopropanes for the Construction of a 2-Arylbenzofuran Skeleton: Total Synthesis of Cuspidan B
https://www.thieme-connect.de/media/synthesis/201612/i_c0077_ga_10-1055_s-0035-1561590.gif
Malik, Chanchal K.; Vaultier, Michel; Ghosh, Subrata: Copper(I)-Catalyzed [2+2] Photocycloaddition of Nonconjugated Alkenes in Room-Temperature Ionic Liquids
https://www.thieme-connect.de/bilder/synthesis/200708/c001_ga
Ma, Yudao; Song, Chun; Chai, Qiang; Ma, Changqin; Andrus, Merritt B.: Palladium-Imidazolium N-Heterocyclic Carbene-Catalyzed Carbonylative Amidation With Boronic Acids, Aryl Diazonium Ions, and Ammonia
https://www.thieme-connect.de/bilder/synthesis/200318/c140_ga
Kabalka, George W.; Yao, Min-Liang: Synthesis of a Potential Boron Neutron Capture Therapy Agent: 1-Aminocyclobutane-1-carboxylic Acid Bearing a Butylboronic Acid Side Chain
https://www.thieme-connect.de/bilder/synthesis/200318/c141_ga
Yamaoka, Yousuke; Taniguchi, Marie; Yamada, Ken-ichi; Takasu, Kiyosei: Asymmetric Total Synthesis of Tylophorine through a Formal [2+2] Cycloaddition Followed by Migrative Ring Opening of a Cyclobutane
https://www.thieme-connect.de/media/synthesis/201518/i_c0267_ga_10-1055_s-0034-1380430.gif
Islam, Kobirul; Das, Deb K.; Akram, Ejaz; Khan, Abu T.: Exploration of C5–C6-Unsubstituted 1,4-Dihydropyridines for the Construction of exo-Hexahydro-1H-chromeno[3,4-h][1,6]naphthyridine-3-carboxylates Using a Stereoselective Povarov Reaction
https://www.thieme-connect.de/media/synthesis/201518/i_c0223_ga_10-1055_s-0034-1380431.gif
Neo, Ana G.; Castellano, Teresa G.; Marcos, Carlos F.: Enol-Ugi Reaction of Hydroxycoumarins: Straightforward Synthesis of Amino Acid Derived Coumarin Enamines
https://www.thieme-connect.de/media/synthesis/201516/i_c0258_ga_10-1055_s-0034-1380436.gif
Dobrydnev, Alexey V.; Popova, Maria V.; Saffon-Merceron, Nathalie; Listunov, Dymytrii; Volovenko, Yulian M.: Synthesis of the First Representatives of Spiro-1λ6-isothiazolidine-1,1,4-triones
https://www.thieme-connect.de/media/synthesis/201517/i_t0209_ga_10-1055_s-0034-1380434.gif
Luo, Guo-Ying; Wu, Hao; Tang, Yu; Li, Hui; Yeom, Hyun-Suk; Yang, Ka; Hsung, Richard P.: A Total Synthesis of (±)-Rhododaurichromanic Acid A via an Oxa-[3+3] Annulation of Resorcinols
https://www.thieme-connect.de/media/synthesis/201518/i_c0219_ga_10-1055_s-0034-1380429.gif
Alouane, Nacira; Vrancken, Emmanuel; Mangeney, Pierre: Preparation of anti-1,2-Disubstituted Homopropargylic Alcohols by Addition of Allenyl(cyano)cuprates to Aldehydes
https://www.thieme-connect.de/bilder/synthesis/200708/c004_ga
Apsunde, Tushar Dattu; Trudell, Mark L.: Microwave-Assisted Iridium-Catalyzed Synthesis of Nicotine and Anabasine Derivatives
https://www.thieme-connect.de/media/synthesis/201315/i_m0987_ga_10-1055_s-0032-1316859.gif
Cole, Charles J. F.; Chi, Hyung Min; DeBacker, Kenneth C.; Snyder, Scott A.: Synthesis of Enhanced, Isolable Disulfanium Salts and their Application to Thiiranium-Promoted Polyene Cyclizations
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0184_ga_10-1055_s-0037-1609754.gif
Wang, Zheng; Ji, Hongtao; He, Wei-Min; Xiong, Yang; Zhang, Guozhu: Chromium-Catalyzed Asymmetric Dearomatization–Addition Reactions of Halomethyloxazoles and Indoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0070_ga_10-1055_s-0037-1609753.gif
Jeganmohan, Masilamani; Cheng, Chien-Hong: Substituted 1-Allyl-2-allenylbenzenes via Palladium-Catalyzed Allylallenylation of Benzyne Derivatives
https://www.thieme-connect.de/bilder/synthesis/200510/c030_ga
Ramírez, Jesus; Fernandez, Elena: Convenient Synthesis of α,α-Difluorinated Carbonyl Compounds from Alkynes through a Fluoro-deboronation Process
https://www.thieme-connect.de/bilder/synthesis/200510/c031_ga
Olson, Christopher A.; Shaner, Courtnay E.; Roche, Sydney C.; Ferrence, Gregory M.; Mitchell, T. Andrew: Hexahydro-1H-Isoindolinone-Like Scaffolds from Electronically Deactivated and Sterically Hindered Dienes: Synthesis in the Context­ of Muironolide A
https://www.thieme-connect.de/media/synthesis/201518/i_c0283_ga_10-1055_s-0034-1380221.gif
Federsel, Hans-Jürgen: Taking the Green Road Towards Pharmaceutical Manufacturing
https://www.thieme-connect.de/media/synthesis/202219/i_r0774_ga_10-1055_a-1752-5471.jpg
Kratzer, Philipp; Gerster, Holger; Maas, Gerhard: Cycloaddition Reactions of Propyne Iminium Salts and Enol Ethers
https://www.thieme-connect.de/media/synthesis/201518/i_c0319_ga_10-1055_s-0034-1380223.gif
Amaya-García, Fabián; Unterlass, Miriam M.: Synthesis of 2,3-Diarylquinoxaline Carboxylic Acids in High-Temperature Water
https://www.thieme-connect.de/media/synthesis/202215/i_t0120_ga_10-1055_s-0040-1719922.gif
Zhang, Li; Shi, Jianxun; Fang, Yewen: An Alternative to the Arbuzov Reaction: Generation and Transformation of α-Dialkyl-Substituted Methylphosphonate Carbanions via an SET Reduction Process
https://www.thieme-connect.de/media/synthesis/202306/i_c0379_ga_10-1055_a-1959-2742.gif
Carreiro, Elisabete P.; Gastalho, Carlos M.; Ernesto, Sofia; Costa, Ana R.; Antunes, Célia M.; Burke, Anthony J.: Synthesis and Antiproliferative Activity of Novel Quercetin-1,2,3-Triazole Hybrids using the 1,3-Dipolar Cycloaddition (Click) Reaction
https://www.thieme-connect.de/media/synthesis/202219/i_t0074_ga_10-1055_s-0040-1719928.gif
Lindner, Marcin; Krasiński, Antoni; Jurczak, Janusz: Facile, Stereocontrolled Synthetic Route towards Bis-functionalised Pyrrolizidines
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0359_ga_10-1055_s-0037-1609582.gif
Ren, Zhi-Hui; Zhao, Mi-Na; Yi, Yukun; Wang, Yao-Yu; Guan, Zheng-Hui: Copper-Catalyzed Aerobic Oxidative Cyclization of Ketoxime Acetates with Pyridines for the Synthesis of Imidazo[1,2-a]pyridines
https://www.thieme-connect.de/media/synthesis/201612/i_c0058_ga_10-1055_s-0035-1561950.gif
Xi, Tuo; Chen, Xu; Zhang, Heyi; Lu, Zhan: Reductive Cyclization of 1,6- and 1,7-Enynes Catalyzed by Iron Complexes
https://www.thieme-connect.de/media/synthesis/201617/i_c0749_ga_10-1055_s-0035-1561957.gif
Chen, Shi; Mondal, Mukulesh; Ibrahim, Ahmad A.; Wheeler, Kraig A.; Kerrigan, Nessan J.: Asymmetric Synthesis of Dipropionate Derivatives through Catalytic Hydrogenation of Enantioenriched E-Ketene Heterodimers
https://www.thieme-connect.de/media/synthesis/201616/i_c0020_ga_10-1055_s-0035-1561958.gif
Dai, Wen; Mi, Yuan; Lv, Ying; Shang, Sensen; Li, Guosong; Chen, Guangwen; Gao, Shuang: Development of a Continuous-Flow Microreactor for Asymmetric Epoxidation of Electron-Deficient Olefins
https://www.thieme-connect.de/media/synthesis/201616/i_c0708_ga_10-1055_s-0035-1561955.gif
Deng, Lu-Jiang; Liu, Jing; Huang, Ji-Qing; Hu, Yanhe; Chen, Mao; Lan, Yu; Chen, Jia-Hua; Lei, Aiwen; Yang, Zhen: Effect of Lithium Chloride on Tuning the Reactivity of Pauson-Khand Reactions­ Catalyzed by Palladium-Tetramethylthiourea
https://www.thieme-connect.de/bilder/synthesis/200716/c037_ga
Yamaoka, Yousuke; Miyabe, Hideto; Yasui, Yoshizumi; Takemoto, Yoshiji: Chiral-Thiourea-Catalyzed Direct Mannich Reaction
https://www.thieme-connect.de/bilder/synthesis/200716/c035_ga
Jiménez Blanco, José L.; Bootello, Purificación; Gutiérrez Gallego, Ricardo; Ortiz Mellet, Carmen; García Fernández, José M.: Synthesis of Thiourea-Linked Glycooligomers that Mimic the Branching Patterns of Natural Oligosaccharides
https://www.thieme-connect.de/bilder/synthesis/200716/c033_ga
Pookkandam Parambil, Shandev; Pulikkal Veettil, Santhini; Dehaen, Wim: The Synthesis of Five-Membered N-Heterocycles by Cycloaddition of Nitroalkenes with (In)Organic Azides and Other 1,3-Dipoles
https://www.thieme-connect.de/media/synthesis/202204/i_t0322_ga_10-1055_a-1547-0196.gif
Wang, Jian; Zu, Liansuo; Li, Hao; Xie, Hexin; Wang, Wei: Cinchona Alkaloid Based Thiourea Promoted Enantioselective Conjugate Addition of N-Heterocycles to Enones
https://www.thieme-connect.de/bilder/synthesis/200716/c036_ga
Miyabe, Hideto: Regiocontrol by Halogen Substituent on Arynes: Generation of 3-Haloarynes and Their Synthetic Reactions
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Pop, Lidia; Golban, Mirabela Ligia; Hădade, Niculina D.; Socaci, Crina; Grosu, Ion: CuAAC Synthesis of Tetragonal Building Blocks Decorated with Nucleobases
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Oberg, Kevin M.; Cochran, Brian M.; Cook, Matthew J.; Rovis, Tomislav: The Catalytic Alkylative Desymmetrization of Anhydrides in a Formal Synthesis of Ionomycin
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Nakayama, Yasuaki; Maeda, Yuichiro; Hama, Naoto; Sato, Takaaki; Chida, Noritaka: Total Synthesis of (–)-Stemoamide by Sequential Overman/Claisen Rearrangement
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Yang, Xiaoyu; Yu, Biao: Synthesis of Landomycin D: Studies on the Saccharide Assembly
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Settambolo, Roberta: Crucial Role of β-Elimination in Determining Regio- and Chemoselectivity of the Rhodium-Catalyzed Hydroformylation of N-Allylpyrroles: A New Approach to 5,6-Dihydroindolizines
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Zhao, Yating; Huang, Binbin; Yang, Chao; Li, Bing; Xia, Wujiong: Metal-Free [3+2] Oxidative Coupling of Phenols with Alkenes: Synthesis of Dihydrobenzofurans
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Vanderghinste, Jaro; Das, Shoubhik: Applications of Photoredox Catalysis for the Radical-Induced Cleavage of C–C Bonds
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Heinz, Benjamin; Djukanovic, Dimitrije; Siemens, Fiona; Idriess, Mohamed; Martin, Benjamin; Knochel, Paul: Regioselective Amination or Alkoxylation of Halogenated Amino-, Thio- or Alkoxypyridines via Pyridyne Intermediates
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Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke: Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite
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Ye, Jian-Liang; Liu, Yang; Zhang, Yu-Feng; Yang, Zhi-Ping; Huang, Pei-Qiang: Studies on the Second-Generation Approach to Loline Alkaloids: Synthesis of N-Bus-norloline through N-tert-Butanesulfinyl Imine Based Asymmetric Vinylogous Mannich Reaction
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Kousara, Mohammad; Bideau, Franck Le; Ibrahim, Rama; Ferry, Angélique; Venot, Pierre-Etienne; Dejean, Camille; Raingeaud, Joël; Dubois, Joëlle; Retailleau, Pascal; Dumas, Françoise: Suberosanes as Potential Antitumor Agents: First Enantioselective Total Synthesis of (1S)-Suberosanone and Configurational Assignment of Suberosenol A
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Konda, Saidulu; Khatravath, Mahender; Mallurwar, Naveen Kumar; Rao, Pallavi; Sripelly, Shivashankar; Iqbal, Javed; Arya, Prabhat: Stereoselective Synthesis of the C27–C35 Eribulin Fragment and Its Utilization in Building Structurally Diverse Macrocycles
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Huang, Jhih-Yi; Delbianco, Martina: Recent Developments in Solid-Phase Glycan Synthesis
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Zhang, Zhou; Yi, Jun-Jie; Aslam, Muhammad; Wan, Jie-Ping; Sun, Meng: Rh(III)-Catalyzed Stereoselective C–H Homoallylation of Indolines with 4-Vinyl-1,3-dioxan-2-ones
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Yu, Mangfei; Zhang, Qian; Wang, Jia; Huang, Peng; Yan, Pengfei; Zhang, Rui; Dong, Dewen: Triflic Anhydride Mediated Ring-Opening/Recyclization Reaction of α-Carbamoyl α-Oximyl Cyclopropanes with DMF: Synthetic Route to 5-Aminoisoxazoles
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Feng, Yangyang; Huang, Ruofeng; Hu, Liangzhen; Xiong, Yan; Coeffard, Vincent: Chiral C2-Symmetric Iodoarene-Catalyzed Asymmetric α-Oxidation of β-Keto Esters
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Zhang, Yongda; Lao, Kendricks S.; Sieber, Joshua D.; Xu, Yibo; Wu, Linglin; Wang, Xiao-Jun; Desrosiers, Jean-Nicolas; Lee, Heewon; Haddad, Nizar; Han, Zhengxu S.; Yee, Nathan K.; Song, Jinhua J.; Howell, Amy R.; Senanayake, Chris H.: Modular Dihydrobenzoazaphosphole Ligands for Suzuki–Miyaura Cross-Coupling
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Komai, Hirotomo; Yoshino, Tatsuhiko; Matsunaga, Shigeki; Kanai, Motomu: Lewis Acid Catalyzed Benzylic C–H Bond Functionalization of Azaarenes; Addition to Imines and Enones
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Mostefaï, Naouël; Sirol, Sabine; Courmarcel, James; Riant, Olivier: Air-Accelerated Enantioselective Hydrosilylation of Ketones Catalyzed by Copper(I) Fluoride-Diphosphine Complexes: Investigations of the Effects of Temperature and Ligand Structure
https://www.thieme-connect.de/bilder/synthesis/200708/c005_ga
Auvil, Tyler J.; Mattson, Anita E.: Internal Lewis Acid Assisted Benzoic Acid Catalysis
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Sugimoto, Kenji; Hoshiba, Yuya; Tsuge, Kiyoshi; Matsuya, Yuji: Synthesis of Substituted Pyrrolo[2,1-a]isoquinolines by Gold-Catalyzed Domino Cyclization of Alkynyl Iminoesters
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Sun, Shutao; Liu, Lei: Catalytic Enantioselective Alkynylation of Tetrahydroisoquinoline-Based N-Acyl Hemiaminals
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Liddon, John T. R.; Rossi-Ashton, James A.; Clarke, Aimee K.; Lynam, Jason M.; Taylor, Richard J. K.; Unsworth, William P.: Divergent Reactivity of Indole-Tethered Ynones with Silver(I) and Gold(I) Catalysts: A Combined Synthetic and Computational Study
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Zhang, Zhiguo; Schreiner, Peter R.: Organocatalytic Biomimetic Reduction of Conjugated Nitroalkenes
https://www.thieme-connect.de/bilder/synthesis/200716/c034_ga
Pan, Jie-Hui; Yang, Min; Gao, Qiang; Zhu, Nian-Yong; Yang, Dan: Bulky Thioureas as New Ligands for Gold(I)-Catalyzed Cyclization of Acetylenic 1,3-Dicarbonyl Compounds
https://www.thieme-connect.de/bilder/synthesis/200716/c032_ga
Kumar, Ravindra; Tamai, Eri; Ohnishi, Akira; Nishimura, Akira; Hoshimoto, Yoichi; Ohashi, Masato; Ogoshi, Sensuke: Nickel-Catalyzed Enantioselective Synthesis of Cyclobutenes via [2+2] Cycloaddition of α,β-Unsaturated Carbonyls with 1,3-Enynes
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Vishwanath, Manjunatha; Prakash, Muthuraj; Vinayagam, Poopathy; Kesavan, Venkitasamy: Construction of Polycyclic Fused Pyrrolidines with Three Contiguous Stereocenters via Michael Addition of Vinylmalononitriles to Nitrostyrenes­ Using l-Proline-Derived Thiourea
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Su, Lin; Xu, Ming-Hua: Asymmetric Reformatsky-Type Reaction of Isatin-Derived N-Sulfinyl Ketimines: Efficient and Practical Synthesis of Enantiopure Chiral 2-Oxoindolinyl-β3,3-Amino Esters
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Marques, Carolina S.; López, Óscar; Leitzbach, Luisa; Fernández-Bolaños, José G.; Stark, Holger; Burke, Anthony J.: Survey of New, Small-Molecule Isatin-Based Oxindole Hybrids as Multi-Targeted Drugs for the Treatment of Alzheimer’s Disease
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Nguyen, Thanh V. Q.; Levoin, Armand; Poli, Lorenzo: Palladium-Catalyzed C7–H (Hetero)arylation of Pyrazolo[1,5-a]pyrazines with Heteroarenes and Aryl Iodides with the Assistance of Silver Salts
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Ribeiro Laia, Fernanda M.; Pinho e Melo, Teresa M. V. D.: Synthesis and Reactivity of Aziridines with Internal Dipolarophiles: An Approach to 1,4-Dihydrochromeno[4,3-b]pyrroles and 3-Methylenechromano[4,3-b]pyrroles
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Peng, Jing; Ran, Guang-Yao; Du, Wei; Chen, Ying-Chun: Tertiary-Amine-Catalyzed Asymmetric [3+2] Annulations of Morita–Baylis–Hillman Carbonates of Isatins with Nitroolefins to Construct Spirooxindoles
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Joshi, Madhur S.; Pigge, F. Christopher: Sequential Pyridine Dearomatization–Mizoroki–Heck Cyclization for the Construction of Fused (Dihydropyrido)isoindolinone Ring Systems
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0093_ga_10-1055_s-0037-1610133.gif
Carboni, Aude; Dagousset, Guillaume; Magnier, Emmanuel; Masson, Géraldine: Three-Component Photoredox-Mediated Chloro-, Bromo-, or Iodotrifluoromethylation of Alkenes
https://www.thieme-connect.de/media/synthesis/201516/i_c0200_ga_10-1055_s-0034-1378715.gif
Iwata, Takayuki; Hyodo, Mizuki; Fujiwara, Takumi; Kawano, Ryusei; Kuhn, Leah; Alabugin, Igor V.; Shindo, Mitsuru: 3-Trifluoromethylbenzyne: Precise Orientation in Cycloaddition Reaction Enabled Regioselective Synthesis of Trifluoromethylated Triptycenes
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Firth, James D.; Zhang, Rong; Morgentin, Rémy; Guilleux, Rachel; Kalliokoski, Tuomo; Warriner, Stuart; Foster, Richard; Marsden, Stephen P.; Nelson, Adam: Exploitation of the Ugi–Joullié Reaction in the Synthesis of Libraries of Drug-Like Bicyclic Hydantoins
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Lanari, Daniela; Piermatti, Oriana; Pizzo, Ferdinando; Vaccaro, Luigi: Copper(II) Triflate–Sodium Dodecyl Sulfate Catalyzed Preparation of 1,2-Diphenyl-2,3-dihydro-4-pyridones in Aqueous Acidic Medium
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Biswas, Anup; Kundu, Samrat; Pal, Dhananjoy; Pal, Amit; Maji, Modhu Sudan: Organocatalyzed Oxa-Diels–Alder Reactions: Recent Progress
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Beckendorf, Stephan; Mancheño, Olga García: 'Click'-BINOLs: A New Class of Tunable Ligands for Asymmetric Catalysis
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Gandeepan, Parthasarathy; Rajamalli, Pachaiyappan; Cheng, Chien-Hong: Palladium-Catalyzed C–H Activation and Cyclization of Anilides with 2-Iodoacetates and 2-Iodobenzoates: An Efficient Method toward Oxindoles and Phenanthridones
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Miller, Daniel K.; Bailey, Christopher A.; Sammelson, Robert E.: Synthesis of Isoxazolines and Isoxazoles Inspired by Fipronil
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Salomó, Ernest; Orgué, Sílvia; Riera, Antoni; Verdaguer, Xavier: Efficient Preparation of (S)- and (R)-tert-Butylmethylphosphine–Borane: A Novel Entry to Important P-Stereogenic Ligands
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Xu, Shibo; Su, Shikuan; Zhang, Huiting; Tian, Lumin; Liang, Pengcheng; Chen, Jiawen; Zhang, Yuan; Li, Chunju; Jia, Xueshun; Li, Jian: Isocyanide-Based Multicomponent Reactions: Rapid Synthesis of a 5,5-Fused Bicyclic Skeleton from α,β-Unsaturated Ketones and Allenoates
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Chuyko, Alexey; Dolgonos, Grygoriy; Shivanyuk, Alexander; Fetyukhin, Volodymyr; Lukin, Oleg: Simple Synthesis of Complex Amines from the Diels–Alder Adducts of (–)-Cytisine
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Ghosh, Prasanjit; Mondal, Swati Lekha; Baidya, Mahiuddin: Ascending of Cycloaddition Strategy for N–O Heterocycles
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Cavitt, Marchello A.; France, Stefan: Aluminum(III)-Catalyzed, Formal Homo-Nazarov-Type Ring-Opening Cyclizations toward the Synthesis of Functionalized Tetrahydroindolizines
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Wertjes, William; Ayers, Sloan; Gao, Qi; Simmons, Eric M.; Beutner, Gregory L.: A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines
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Sugiyama, Yu-ki; Heigozono, Shiori; Tamura, Kazuhiro; Okamoto, Sentaro: Iron-Catalyzed Reductive Metalation–Allylation and Metalative Cyclization of 2,3-Disubstituted Oxetanes and Their Stereoselectivity
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Hopf, Henning; Sherburn, Michael S.: Allenes in Diels–Alder Cycloadditions
https://www.thieme-connect.de/media/synthesis/202204/i_m0291_ga_10-1055_s-0040-1706052.gif
Yang, Yun; Jones, Christopher R.: The Aryne Ene Reaction
https://www.thieme-connect.de/media/synthesis/202222/i_f0171_ga_10-1055_a-1827-2987.gif
Salman, Ghazwan Ali; Ali, Asad; Hussain, Munawar; Khera, Rasheed Ahmad; Langer, Peter: Synthesis of Functionalized Benzofurans by a Double Heck Reaction of 2,3-Dibromofurans and Subsequent 6π-Electrocyclization/Dehydrogenation
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Wu, Zhiqing; Pan, Yinyin; Zhou, Xiangge: Synthesis of 3-Arylimidazo[1,2-a]pyridines by a Catalyst-Free Cascade Process
https://www.thieme-connect.de/media/synthesis/201114/c420_ga.jpg
Cormier, Morgan; Chardon, Aurélien; Blanchet, Jérôme; Rouden, Jacques; Maddaluno, Jacques; De Paolis, Michaël: An Organocatalytic Access to Spiro[4.5]decanes and Spiro[4.6]undecanes Containing Aminolactones and 3-Aminopyrrolidines
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Shaw, Subrata; White, James D.: Asymmetric Catalysis with Iron–Salen Complexes
https://www.thieme-connect.de/media/synthesis/201617/i_c0181_ga_10-1055_s-0035-1562103.gif
Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil: NiIICl(1-Naphthyl)(PCy3)2, An Air-Stable σ-NiII Precatalyst for Quantitative Cross-Coupling of Aryl C–O Electrophiles with Aryl Neopentylglycolboronates
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Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil: An Indefinitely Air-Stable σ-NiII Precatalyst for Quantitative Cross-Coupling of Unreactive Aryl Halides and Mesylates with Aryl Neopentylglycolboronates
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Nagai, Akira; Kobayashi, Akihiro; Sakata, Yuki; Minami, Yasunori; Uchida, Keisuke; Hosoya, Takamitsu; Yoshida, Suguru: Synthesis of Multisubstituted Benzenes from Phenols via Multisubstituted Benzynes
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Urawa, Yoshio; Nishiura, Katsutoshi; Souda, Shigeru; Ogura, Katsuyuki: A Convenient Method for Preparing Aromatic α,β-Unsaturated Ketones from α,β-Unsaturated Acyl Chlorides and Arylboronic Acids via Suzuki-Miyaura Type Coupling Reaction
https://www.thieme-connect.de/bilder/synthesis/200318/c139_ga
Zhang, Ruirui; Peng, Xia; Tan, Jiajing: Recent Advances in Construction of C(sp2)–O Bonds via Aryne Participated Multicomponent Coupling Reactions
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Rosa, Gilber R.; Ebeling, Gunter; Dupont, Jairton; Monteiro, Adriano L.: A Superior Non-Symmetrical NCP Pincer Type Palladacycle Catalyst Precursor for the Coupling of Aryl Boronic Acids with Aryl Chlorides
https://www.thieme-connect.de/bilder/synthesis/200318/c142_ga
Monasson, Olivier; Malinowski, Maciej; Lubin-Germain, Nadège; Ferry, Angélique: Hirao Cross-Coupling Reaction as an Efficient Tool to Build Non-natural C2-Phosphonylated Sugars
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Philipps, Arne R.; Fritze, Lars; Erdmann, Nico; Enders, Dieter: An Asymmetric Organocatalytic Quadruple Domino Reaction Employing a Vinylogous Friedel–Crafts/Michael/Michael/Aldol Condensation Sequence
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Qureshi, Zafar; Schlundt, Waldemar; Lautens, Mark: Introduction of Hindered Electrophiles via C–H Functionalization in a Palladium-Catalyzed Multicomponent Domino Reaction
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Neochoritis, Constantinos G.; Zhang, Ji; Dömling, Alexander: Leuckart–Wallach Approach to Sugar Isocyanides and Its IMCRs
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Högermeier, Jens; Trawny, Daniel; Zimmer, Reinhold; Reissig, Hans-Ulrich: Diels–Alder Reactions of 1,3-Dienes Incorporated into 8-Oxa- and 8-Thiabicyclo[3.2.1]octane Skeletons: A Convenient Access to Complex Tri- and Tetracyclic Compounds
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Kumar, Ketan; Vivekanand, T.; Singh, Bara; Ramasastry, S. S. V.: C(sp3)–H Activation Enabled by (η3-Indolylmethyl)palladium Complexes: Synthesis of Monosubstituted Tetrahydrocarbazoles
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Pan, Yuanjia; Lu, Hongjian; Fang, Yewen; Fang, Xinqiang; Chen, Liqun; Qian, Junlu; Wang, Junhua; Li, Chaozhong: Synthesis of Pyrroles via Copper-Catalyzed Coupling of Amines with Bromoenones
https://www.thieme-connect.de/bilder/synthesis/200708/c003_ga
Estéoule, Audrey; Durán, Fernando; Retailleau, Pascal; Dodd, Robert H.; Dauban, Philippe: Enantioselective Intramolecular Copper-Catalyzed Aziridination of Sulfamates
https://www.thieme-connect.de/bilder/synthesis/200708/c002_ga
Seck, Insa; Fall, Alioune; Lago, Carmen; Sène, Massène; Gaye, Mohamed; Seck, Matar; Gómez, Generosa; Fall, Yagamare: Synthesis of a Cholesterol Side-Chain Triazole Analogue via ‘Click’ Chemistry
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Xiao, Fenfen; Zhang, Qing; Wang, Yunxia; Hu, Xiangdong: Synthetic Studies toward Bi-linderone Lead To Unexpected 6π-Electrocyclization Reactions: A Facile Construction of Highly Congested Spiro Compounds
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Kachkovskyi, Georgii; Cieślak, Marcin; Graczyk, Piotr; Zawadzki, Przemysław; Kalinowska-Tłuścik, Justyna; Werłos, Mateusz: Photocatalytic Approach to α,α-Difluoroalkyl Alcohols
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Lee, Ju Hee; Kim, Dae Young: Organocatalytic Highly Enantioselective Mannich-Type Reactions of Fluoromalonate with N-Boc-Aldimines
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Oonishi, Yoshihiro; Taniuchi, Ai; Sato, Yoshihiro: Rhodium(I)-Catalyzed Hydroacylation/Cycloisomerization Cascade Reaction: Application to the Construction of the Tricyclic Core of Guanacastepenes
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Fujimoto, Hayato; Yamamura, Shisato; Takenaka, Namiki; Tobisu, Mamoru: Phosphine-Catalyzed Z-Selective Carbofluorination of Alkynoates Bearing an N-Heteroarene Unit
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Shibata, Takanori; Fukai, Miku; Sekine, Ryosuke; Hazra, Madhurima; Kanyiva, Kyalo Stephen: Enantioselective Synthesis of Planar-Chiral 1,n-Dioxa[n]paracyclophane-Based Phosphites and Their Application as Chiral Ligands
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Grugel, Holger; Minuth, Tobias; Boysen, Mike M. K.: Novel Olefin-Phosphorus Hybrid and Diene Ligands Derived from Carbohydrates
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Deaton, Kimberly R.; Strouse, Christopher S.; Gin, Mary S.: Selective [2+2+2] Cycloaddition of Nickel-Benzyne and an Asymmetric 1,3-Diyne: An Iterative Route to Substituted [n]Acenes
https://www.thieme-connect.de/bilder/synthesis/200418/c052_ga
Durandetti, Muriel; Périchon, Jacques: Nickel-Catalyzed Electrochemical Coupling of Aryl, Heteroaryl or Vinyl Halides with Activated Alkyl Chlorides: Synthetic and Stereochemical Aspects
https://www.thieme-connect.de/bilder/synthesis/200418/c051_ga
Ambler, Brett R.; Peddi, Santosh; Altman, Ryan A.: Copper-Catalyzed Decarboxylative Trifluoromethylation of Propargyl Bromodifluoroacetates
https://www.thieme-connect.de/media/synthesis/201414/i_c0147_ga_10-1055_s-0033-1339128.gif
Sahoo, Santosh K.; Jena, Himanshu Sekhar; Majji, Ganesh; Patel, Bhisma K.: Formation of Imidazolidine-benzothiazole–Copper(II) Complexes via a Copper-Mediated Room-Temperature C–H Activation of Imidazolidinecarbothioamides
https://www.thieme-connect.de/media/synthesis/201414/i_c0238_ga_10-1055_s-0033-1339127.gif
Barker, Timothy J.; Jarvo, Elizabeth R.: Diene-Ligated Iridium Complexes as Catalysts for Allylation and Methallylation Reactions of Ketones
https://www.thieme-connect.de/media/synthesis/201019/c041_ga.jpg
Luo, Long; Zhang, Jian-Jian; Ling, Wei-Jian; Shao, Yong-Liang; Wang, Ya-Wen; Peng, Yu: Unified Synthesis of (–)-Folicanthine and (–)-Ditryptophenaline Enabled by a Room Temperature Nickel-Mediated Reductive Dimerization
https://www.thieme-connect.de/media/synthesis/201414/i_c0189_ga_10-1055_s-0033-1339126.gif
Ugarriza, Iratxe; Reyes, Efraím; Prieto, Liher; Uria, Uxue; Carrillo, Luisa; Vicario, Jose L.: An Approach to the Synthesis of a Hepatitis C Virus Inhibitor through a Proline-Catalyzed 1,3-Dipolar Cycloaddition Using Acrolein
https://www.thieme-connect.de/media/synthesis/202204/i_f0626_ga_10-1055_s-0040-1719858.gif
Liu, Can; Shen, Ni; Shang, Rui: Photocatalytic Defluoroalkylation of Trifluoroacetates with Alkenes using 4-(Acetamido)thiophenol
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0487_ga_10-1055_a-2019-1532.gif
Zhao, Yanchuan; Zhu, Jieming; Ni, Chuanfa; Hu, Jinbo: Magnesium Metal-Mediated Reductive Trifluoromethylation of Aldehydes with Phenyl Trifluoromethyl Sulfone
https://www.thieme-connect.de/media/synthesis/201011/c008_ga.jpg
Tur, Fernando; Mansilla, Javier; Lillo, Victor J.; Saá, José M.: Constructing Quaternary Centers of Chirality: The Lanthanide Way to Trifluoromethyl-Substituted Tertiary Alcohols
https://www.thieme-connect.de/media/synthesis/201011/c007_ga.jpg
Prakash, G. K. Surya; Do, Clement; Wang, Fang; Mathew, Thomas; Olah, George A.: Cyclodehydration of Fluorinated Diols Using the Mitsunobu Reaction: Highly Efficient Synthesis of Trifluoromethylated Cyclic Ethers
https://www.thieme-connect.de/media/synthesis/201011/c006_ga.jpg
Vasylyev, Maksym; Alper, Howard: Conventional and Tandem Hydroformylation
https://www.thieme-connect.de/media/synthesis/201017/c033_ga.jpg
Sato, Kazuyuki; Tarui, Atsushi; Omote, Masaaki; Ando, Akira; Kumadaki, Itsumaro: Trifluoromethylation of Organic Compounds and Related Reactions
https://www.thieme-connect.de/media/synthesis/201011/c009_ga.jpg
Mahajan, Bhushan; Aand, Dnyaneshwar; Purwa, Mandeep; Mujawar, Taufiqueahmed; Ghosh, Subhash; Pabbaraja, Srihari; Singh, Ajay K.: Elements-Continuous-Flow Platform for Coupling Reactions and Anti-viral Daclatasvir API Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0518_ga_10-1055_a-2022-2063.gif
Guo, Chen; Yue, Xuyi; Qing, Feng-Ling: Palladium-Catalyzed Cross-Coupling of Ethyl α-Bromo-α-fluoroacetate with Arylboronic Acids: Facile Synthesis of α-Aryl-α-fluoroacetates
https://www.thieme-connect.de/media/synthesis/201011/c001_ga.jpg
Peddie, Victoria; Pietsch, Markus; Bromfield, Karen M.; Pike, Robert N.; Duggan, Peter J.; Abell, Andrew D.: Fluorinated β²- and β³-Amino Acids: Synthesis and Inhibition of α-Chymotrypsin
https://www.thieme-connect.de/media/synthesis/201011/c004_ga.jpg
Roger, Julien; Sire, Charline; Tsivery, Anthonia; Cattey, Hélène; Hierso, Jean-Cyrille: Aryl Triflates in Phosphorus-Directed Rhodium(III)-Catalyzed C–H Activation
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0501_ga_10-1055_a-2018-0965.gif
Furuya, Takeru; Klein, Johannes E. M. N.; Ritter, Tobias: Carbon-Fluorine Bond Formation for the Synthesis of Aryl Fluorides
https://www.thieme-connect.de/media/synthesis/201011/c002_ga.jpg
Denizot, Natacha; Guillot, Régis; Kouklovsky, Cyrille; Vincent, Guillaume: N-Iodosuccinimide-Mediated Oxidative Coupling of Indoles and Phenols: A Synthetic Study toward the Benzofuroindoline Moiety of Bipleiophylline
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0092_ga_10-1055_s-0036-1592002.gif
Liu, Zhao; Kumar, Krishna: Trifluoromethyl Derivatization of the Ganglioside, GM1
https://www.thieme-connect.de/media/synthesis/201011/c010_ga.jpg
Yu, Xingxin; Qiu, Guanyinsheng; Liu, Jianping; Wu, Jie: Synthesis of 2,3,4,11b-Tetrahydro-1H-pyridazino[6,1-a]isoquinolines via the Three-Component Reaction of 2-Alkynylbenzaldehydes, a Sulfonohydrazide and Dimethyl Cyclopropane-1,1-dicarboxylate
https://www.thieme-connect.de/media/synthesis/201114/c264_ga.jpg
Vicente-García, Esther; Ramón, Rosario; Lavilla, Rodolfo: New Heterocyclic Inputs for the Povarov Multicomponent Reaction
https://www.thieme-connect.de/media/synthesis/201114/c339_ga.jpg
Tawatari, Tsukasa; Kato, Ritsuki; Takasu, Kiyosei; Takikawa, Hiroshi: Intramolecular Propargylic Ene Reaction of Benzyne En Route to Highly Functionalized Allenes and Allenamides
https://www.thieme-connect.de/media/synthesis/202222/i_f0135_ga_10-1055_a-1826-2545.gif
Bortolato, Tommaso; Dyguda, Mateusz; Vega-Peñaloza, Alberto; Dell’Amico, Luca: Properties and Synthetic Performances of Phenylamino Cyanoarenes under One-Photon Excitation Manifolds
https://www.thieme-connect.de/media/synthesis/202215/i_c0750_ga_10-1055_a-1776-0929.gif
Wang, Weibo; Xu, Bo; Hammond, Gerald B.: Synthesis of Fluorohydrins through Electrophilic Fluorination of Allyl Silanes
https://www.thieme-connect.de/media/synthesis/201115/c020_ga.jpg
Roy, Sudipta Raha; Jadhavar, Pradeep S.; Seth, Kapileswar; Sharma, Kulin K.; Chakraborti, Asit K.: Organocatalytic Application of Ionic Liquids: [bmim][MeSO4] as a Recyclable Organocatalyst in the Multicomponent Reaction for the Preparation of Dihydropyrimidinones and -thiones
https://www.thieme-connect.de/media/synthesis/201114/c021_ga.jpg
Suzuki, Takeyuki; Ishizaka, Yuka; Ghozati, Kazem; Zhou, Da-Yang; Asano, Kaori; Sasai, Hiroaki: Enantioselective Multicatalytic Synthesis of α-Benzyl-β-hydroxyindan-1-ones
https://www.thieme-connect.de/media/synthesis/201315/i_c0194_ga_10-1055_s-0033-1338479.gif
Srivastava, Ajay Kumar; Song, Heebum; Park, Seung Bum: Diversity-Oriented Synthesis of Functionalized Polyheterocycles from Garner Aldehyde
https://www.thieme-connect.de/media/synthesis/201114/c014_ga.jpg
Sugiyama, Yu-ki; Okamoto, Sentaro: Regioselective Syntheses of Substituted Pyridines and 2,2′-Bipyridines by Cobalt-Catalyzed [2+2+2] Cycloaddition of α,ω-Diynes with Nitriles
https://www.thieme-connect.de/media/synthesis/201114/c362_ga.jpg
Zhou, Mingxin; Song, Qiuling: Synthesis of α-Ketoamides from Aryl Methyl Ketones and N,N-Dimethylformamide via Copper-Catalyzed Aerobic Oxidative Coupling
https://www.thieme-connect.de/media/synthesis/201414/i_c0127_ga_10-1055_s-0033-1339109.gif
Duong, Hung A.; Nguyen, Tuan Minh; Rosman, Nurul Zubaidah Binte; Tan, Lionel Jia Liang: Carboxylation of Organoboronic Esters with Potassium Methyl Carbonate under Copper Catalysis
https://www.thieme-connect.de/media/synthesis/201414/i_c0122_ga_10-1055_s-0033-1339119.gif
Zhao, Chenglong; Tan, Zhuozhen; Liang, Zhuye; Deng, Wei; Gong, Hegui: Nickel-Catalyzed Reductive Allylation of Ketones with Allylic Carbonates
https://www.thieme-connect.de/media/synthesis/201414/i_c0174_ga_10-1055_s-0033-1339111.gif
Swan, Charlie; Maggi, Lorenzo; Park, Mahri; Taylor, Sophie; Shepherd, William; Ball, Liam T.: Generation of Thiyl Radicals from Air-Stable, Odorless Thiophenol Surrogates: Application to Visible-Light-Promoted C–S Cross-Coupling
https://www.thieme-connect.de/media/synthesis/202215/i_z0611_ga_10-1055_s-0041-1737816.gif
Zajc, Barbara; Kumar, Rakesh: Synthesis of Fluoroolefins via Julia-Kocienski Olefination
https://www.thieme-connect.de/media/synthesis/201011/c005_ga.jpg
Walkowiak, Justyna; del Campo, Teresa Martinez; Ameduri, Bruno; Gouverneur, Véronique: Syntheses of Mono-, Di-, and Trifluorinated Styrenic Monomers
https://www.thieme-connect.de/media/synthesis/201011/c028_ga.jpg
Gurung, Santosh K.; Thapa, Surendra; Shrestha, Bijay; Giri, Ramesh: Copper-Catalyzed Cross-Coupling of Aryl- and Heteroaryltriethoxysilanes with Aryl and Heteroaryl Iodides and Bromides
https://www.thieme-connect.de/media/synthesis/201414/i_c0146_ga_10-1055_s-0033-1339108.gif
Metze, Bryan E.; Bhattacharjee, Avik; McCormick, Theresa M.; Stuart, David R.: Parameterization of Arynophiles: Experimental Investigations towards a Quantitative Understanding of Aryne Trapping Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0166_ga_10-1055_a-1845-3066.gif
Chu, Qiao; Zhou, Yeqin; Ji, Ce; Liu, Ping; Sun, Peipei: Electrochemical Benzylic C(sp3)–H Amidation via Ritter-Type Reaction in the Absence of External Mediator and Oxidant
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0546_ga_10-1055_a-1992-7066.gif
Garbarino, Silvia; Protti, Stefano; Basso, Andrea: Toward a Green Atom Economy: Development of a Sustainable Multicomponent Reaction
https://www.thieme-connect.de/media/synthesis/201516/i_c0183_ga_10-1055_s-0034-1380719.jpg
Murakami, Sho; Brudy, Cosima; Bachmann, Moritz; Takemoto, Yoshiji; Pieber, Bartholomäus: Photocatalytic Cleavage of Trityl Protected Thiols and Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0491_ga_10-1055_a-1979-5933.gif
Wech, Felix; Gellrich, Urs: Hydrogenation of Olefins, Alkynes, Allenes, and Arenes by Borane-Based Frustrated Lewis Pairs
https://www.thieme-connect.de/media/synthesis/202215/i_r0616_ga_10-1055_a-1684-5552.gif
Hunter, Thomas J.; Wang, Yanping; Zheng, Jiamin; O’Doherty, George A.: Asymmetric Iterative Hydration of Polyene Strategy to Cryptocaryols A and B
https://www.thieme-connect.de/media/synthesis/201611/i_c0125_ga_10-1055_s-0035-1561607.gif
Nishimura, Takahiro; Nagai, Tomotaka; Takechi, Ryosuke; Ebe, Yusuke: Rhodium-Catalyzed Enantioselective Addition of Tricyclopropylboroxin to N-Sulfonylimines
https://www.thieme-connect.de/media/synthesis/201616/i_c0007_ga_10-1055_s-0035-1561605.gif
García-Ruiz, Cristina; Cheng-Sánchez, Iván; Sarabia, Francisco: Synthesis of (–)- and (+)-Gummiferol via Asymmetric Synthesis of Glycidic Amides
https://www.thieme-connect.de/media/synthesis/201611/i_c0102_ga_10-1055_s-0035-1561606.gif
Morita, Nobuyoshi; Mashiko, Rie; Hakuta, Dai; Eguchi, Daisuke; Ban, Shintaro; Hashimoto, Yoshimitsu; Okamoto, Iwao; Tamura, Osamu: Gold-Catalyzed Dimeric Cyclization of Isoeugenol and Related 1-Phenylpropenes in Ionic Liquid: Environmentally Friendly and Stereoselective Synthesis of 1,2,3-Trisubstituted 2,3-Dihydro-1H-indenes
https://www.thieme-connect.de/media/synthesis/201612/i_c0078_ga_10-1055_s-0035-1561604.gif
Picthall, Daniel; Surgenor, Brian A.; Kilian, Petr: Convenient and Scalable Synthesis of Aryldichlorophosphines and Primary Arylphosphines via Perthiophosphonic Anhydrides
https://www.thieme-connect.de/media/synthesis/202306/i_c0422_ga_10-1055_a-1994-2301.gif
Ferro, Rita; Viduedo, Nuno; Santos, A. Sofia; Silva, Artur M. S.; Royo, Beatriz; Marques, M. Manuel B.: Bimetallic Catalyzed Synthesis of 2-Arylindoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0631_ga_10-1055_a-2035-6420.gif
Zhu, Mingzhao; Zheng, Nan: Photoinduced Cleavage of N-N Bonds of Aromatic Hydrazines and Hydrazides by Visible Light
https://www.thieme-connect.de/media/synthesis/201114/c016_ga.jpg
Yin, Bin; Inagi, Shinsuke; Fuchigami, Toshio: Selective Electrochemical Fluorodesulfurization of Benzo- and Pyrido-Fused Oxazine Derivatives Using Ex-cell Halogen Mediators
https://www.thieme-connect.de/media/synthesis/201115/c010_ga.jpg
Tovar, John D.: Organic Halogenation Chemistry as a Vital Tool for the Construction of Functional π-Conjugated Materials
https://www.thieme-connect.de/media/synthesis/201115/c215_ga.jpg
Hofmann, Fabian; Gärtner, Cornelius; Kretzschmar, Martin; Schneider, Christoph: Asymmetric Synthesis of Fused Tetrahydroquinolines via Intra­molecular Aza-Diels–Alder Reaction of ortho-Quinone Methide Imines
https://www.thieme-connect.de/media/synthesis/202204/i_t0233_ga_10-1055_a-1517-7515.gif
Schäfer, Gabriel; Reber, Stefan; Ahmetovic, Muhamed; Fleischer, Tony; Leuenberger, Daniel; Blumer, Nicole; Udry, Megan; Abele, Stefan: Robust and Scalable Reductive Amination Protocol for Electron-Poor Heterocyclic Amines Using Et3SiH/TFA as Reducing Agent
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0441_ga_10-1055_a-1981-2727.gif
Chiappe, Cinzia; Sanzone, Angelo: Using the ‘Chemical Tunability’ of Ionic Liquids to Increase Sustainability in the Electrophilic Bromination of Unsaturated Compounds
https://www.thieme-connect.de/media/synthesis/201115/c395_ga.jpg
Kutsumura, Noriki; Kubokawa, Keisuke; Saito, Takao: TBAF-Promoted Elimination of Vicinal Dibromides Having an Adjacent O-Functional Group: Syntheses of 2-Bromoalk-1-enes and Alkynes
https://www.thieme-connect.de/media/synthesis/201115/c359_ga.jpg
Ziegler, Dorothée S.; Klier, Lydia; Müller, Nicolas; Karaghiosoff, Konstantin; Knochel, Paul: Directed Zincation or Magnesiation of 2- and 4-Pyrones and Their Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0411_ga_10-1055_s-0037-1610215.gif
Lopchuk, Justin M.; Song, Mia; Butler, Blythe; Gribble, Gordon W.: Synthesis of Heteroaryl-Substituted Pyrroles via the 1,3-Dipolar Cycloaddition of Unsymmetrical Münchnones and Nitrovinylheterocycles
https://www.thieme-connect.de/media/synthesis/201518/i_c0162_ga_10-1055_s-0034-1380720.gif
Cserép, Gergely B.; Demeter, Orsolya; Bätzner, Effi; Kállay, Mihály; Wagenknecht, Hans-Achim; Kele, Péter: Synthesis and Evaluation of Nicotinic Acid Derived Tetrazines for Bioorthogonal Labeling
https://www.thieme-connect.de/media/synthesis/201518/i_c0157_ga_10-1055_s-0034-1380721.gif
Zhang, Pengke; Hua, Lin; Takahashi, Tamotsu; Jin, Shengnan; Wang, Qilin: Recent Advances in the Dearomative Skeletal Editing of Mono-azaarenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0628_ga_10-1055_a-2013-9885.gif
Zeisel, Lukas; Maier, Martin S.; Thorn-Seshold, Oliver: Efficient and Scalable Syntheses of 1,2-Thiaselenane-4-amine and 1,2-Thiaselenane-5-amine
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0496_ga_10-1055_a-2022-1398.gif
Khan, Farooq-Ahmad; Yaqoob, Sana; Qasim, Muhammad Wasim; Ali, Shujaat; Wang, Yan; Jiang, Zi-Hua: A Robust, Gram-Scale and High-Yield Synthesis of MDP Congeners for Activation of the NOD2 Receptor and Vaccine Adjuvantation
https://www.thieme-connect.de/media/synthesis/EFirst/i_b0528_ga_10-1055_a-2004-5883.gif
Garlets, Zachary J.; Wolfe, John P.: Asymmetric Synthesis of Six-Membered Cyclic Sulfamides via Palladium-Catalyzed Alkene Carboamination Reactions
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0078_ga_10-1055_s-0036-1591574.gif
Sara, Alexandru A.; Um-e-Farwa, Um-e-Farwa; Saeed, Aamer; Kalesse, Markus: Recent Applications of the Diels–Alder Reaction in the Synthesis of Natural Products (2017–2020)
https://www.thieme-connect.de/media/synthesis/202204/i_r0249_ga_10-1055_a-1532-4763.gif
Kageyuki, Ikuo; Yoshida, Hiroto; Takaki, Ken: Three-Component Carboboration of Alkenes under Copper Catalysis
https://www.thieme-connect.de/media/synthesis/201414/i_c0143_ga_10-1055_s-0033-1341267.gif
Orlandi, Simonetta; Colombo, Federica; Benaglia, Maurizio: Chiral Diamine-Copper(I) Complexes as Asymmetric Catalysts in the Enantioselective Addition of Phenylacetylene to Imines
https://www.thieme-connect.de/bilder/synthesis/200510/c034_ga
Fernández, Carlos; Diouf, Ousmane; Momán, Edelmiro; Gómez, Generosa; Fall, Yagamare: OCT Analogues Part 2. Acetylene in the Synthesis of Useful Building Blocks for Analogues of OCT Modified at C-20, C-21, and the D-Ring
https://www.thieme-connect.de/bilder/synthesis/200510/c032_ga
Saejueng, Pranorm; Bates, Craig G.; Venkataraman, D.: Copper(I)-Catalyzed Coupling of Terminal Acetylenes with Aryl or Vinyl Halides
https://www.thieme-connect.de/bilder/synthesis/200510/c033_ga
Ye, Ke-Yin; Zhao, Zhuo-An; Lai, Zeng-Wei; Dai, Li-Xin; You, Shu-Li: Highly Regioselective Allylic Substitution Reactions Catalyzed by an Air-Stable (π-Allyl)iridium Complex Derived from Dinaphthocyclooctatetraene and a Phosphoramidite Ligand
https://www.thieme-connect.de/media/synthesis/201315/i_c0317_ga_10-1055_s-0033-1339187.gif
Woof, Callum R.; Linford-Wood, Thomas G.; Mahon, Mary F.; Webster, Ruth L.: Catalytic Hydrophosphination of Allenes Using an Iron(II) β-Diketiminate Complex
https://www.thieme-connect.de/media/synthesis/202306/i_c0290_ga_10-1055_a-1902-5592.gif
Zhang, Shuang; Hu, Xiu-Qin; Wang, Zhu-Yin; Xu, Peng-Fei: Reactions of Sulfonium Salts with 2,3-Dioxopyrrolidine Derivatives: A Concise Synthesis of Spirocyclopropane
https://www.thieme-connect.de/media/synthesis/201517/i_c0093_ga_10-1055_s-0034-1380522.gif

Issue Accepted Manuscripts

Dehnert, Brady W.; Dworkin, Jeremy H.; Kwon, Ohjun: Dealkenylative Functionalization: Conversion of Alkene C(sp3)–C(sp2) Bonds to C(sp3)–X Bonds Using Redox-Based Radical Processes
Sartillo-Piscil, Fernando; Romero-Ibañez, Julio; Sandoval-Lira, Jacinto; Cruz-Gregorio, Silvano; Quintero, Leticia; Hernández-Pérez, Julio: On the Reaction Mechanism of the Selective C(sp3)-H Functionalization of N-Benzyl-Piperidines Mediated by TEMPO Oxoammonium Cation
Delouche, Thomas; Gadiry-Diallo, Abdoul; Besson, Thierry; Ogoshi, Sensuke; Fruit, Corinne: Photocatalyst-Free Visible Light-Mediated C-H Perfluoroalkylation of Quinazolin-4(3H)-ones with perfluoroalkyl iodides
Kaur, Ramandeep; Singh, Harcharan; Arulananda Babu, Srinivasarao: Pd(II)-catalyzed, directing group-aided C-H arylation, alkylation, benzylation and methoxylation of carbazole-3-carboxamides toward C2,C3,C4 functionalized carbazoles
Röckl, Johannes L.; Lundberg, Helena: Samarium and Ytterbium in Organic Electrosynthesis
Naharwal, Sushma; Kharat, Narendra Dinkar; Mahesha, Chikkagundagal K; Bajaj, Kiran; Sakhuja, Rajeev: Palladium-Catalyzed Regioselective C-Arylation and C,N-Diarylation of N-Aryl 2,3-dihydrophthalazine-1,4-diones using Diaryliodonium Salts

Issue 21/2022

Yang, Zhenjie; Cheng, Hong-Gang; Chen, Ruiming; Cao, Liming; Wei, Qiang; Wang, Qingqing; Zhou, Qianghui: Eight-Step Asymmetric Synthesis of (–)-Berkelic Acid
https://www.thieme-connect.de/media/synthesis/202221/i_g0085_ga_10-1055_a-1799-0459.gif
Huang, Long-Tao; Hirata, Yuki; Kato, Yoshimi; Lin, Luqing; Kojima, Masahiro; Yoshino, Tatsuhiko; Matsunaga, Shigeki: Ruthenium(II)/Chiral Carboxylic Acid Catalyzed Enantioselective C–H Functionalization of Sulfoximines
https://www.thieme-connect.de/media/synthesis/202221/i_g0414_ga_10-1055_a-1588-0072.gif
Huang, Xiao-Ling; Li, Chong; Wang, Juan; Yang, Shang-Dong: Direct Copper-Catalyzed C-3 Arylation of Diphenylphosphine Oxide Indoles
https://www.thieme-connect.de/media/synthesis/202221/i_g0472_ga_10-1055_a-1633-8792.gif
Pototskiy, Roman A.; Boym, Mikhail A.; Nelyubina, Yulia V.; Perekalin, Dmitry S.: Synthesis of Ruthenium Catalysts with a Chiral Arene Ligand Derived from Natural Camphor
https://www.thieme-connect.de/media/synthesis/202221/i_g0590_ga_10-1055_a-1668-2075.gif
Wang, Huiying; Wang, Mengmeng; Ma, Biao; Dai, Hui-Xiong: Rhodium-Catalyzed C–H Activation of Indoles for the Construction of Spiroindole Scaffolds
https://www.thieme-connect.de/media/synthesis/202221/i_g0035_ga_10-1055_a-1791-7218.gif
Li, Mingliang; Wang, Jun: Recent Advances on Transition-Metal-Catalyzed Asymmetric C–H Arylation Reactions
https://www.thieme-connect.de/media/synthesis/202221/i_g0577_ga_10-1055_a-1677-5870.gif
Murakami, Kotone; Sakamoto, Kana; Nishimura, Takahiro: Enantioselective C–H Alkylation of N-Arylbenzamides with Vinyl Ethers Catalyzed by an Iridium/Chiral Phosphoramidite–Olefin Complex
https://www.thieme-connect.de/media/synthesis/202221/i_g0582_ga_10-1055_a-1672-6284.gif
Shirai, Tomohiko; Yamamoto, Yasunori: Cationic Iridium/Chiral Bidentate Phosphoramidite Catalyzed Asymmetric Hydroarylation
https://www.thieme-connect.de/media/synthesis/202221/i_g0594_ga_10-1055_a-1683-9455.gif
Xu, Weiwei; Ye, Mengchun: Enantioselective Cobalt-Catalyzed C–H Functionalization
https://www.thieme-connect.de/media/synthesis/202221/i_r0078_ga_10-1055_a-1801-2595.gif
Qian, Pu-Fan; Li, Jun-Yi; Zhou, Tao; Shi, Bing-Feng: Synthesis of P- and S-Stereogenic Compounds via Enantioselective C–H Functionalization
https://www.thieme-connect.de/media/synthesis/202221/i_r0088_ga_10-1055_a-1802-6793.gif
Wang, Pu-Sheng; Gong, Liu-Zhu: Asymmetric C–H Functionalization Enabled by Pd/Chiral Phosphoric Acid Combined Catalysis
https://www.thieme-connect.de/media/synthesis/202221/i_r0530_ga_10-1055_a-1662-7096.gif

Issue 17/2022

Remete, Attila M.; Nonn, Melinda; Volk, Balázs; Kiss, Loránd: Developments in the Alkynyltrifluoromethylations of Alkenes and Alkynes
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Fichez, Jeanne; Dupommier, Dorian; Besset, Tatiana: Direct Synthesis of Disubstituted Trifluoromethylthiolated Alkenes
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Gonda, Zsombor; Földesi, Tamás; Nagy, Bálint; Novák, Zoltán: Modular Synthesis of Carbazole-Substituted Phthalimides as Potential Photocatalysts
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Salamon-Krokosz, Katarzyna; Gołdyn, Mateusz; Siodła, Tomasz; Bartoszak-Adamska, Elżbieta; Koroniak, Henryk; Koroniak-Szejn, Katarzyna: Fluorinated Olefinic Lactams: The Case of Amino Acids – Preparation and Mechanistic Studies
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Uchikura, Tatsuhiro; Yokohama, Sosuke; Murakami, Mona; Akiyama, Takahiko: Chiral Calcium Phosphate Catalyzed Enantioselective Synthesis of All-Carbon Quaternary Center by Friedel–Crafts Alkylation Reaction of Pyrroles and Trifluoromethylated Nitrostyrenes
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Cruz-Hernández, Carlos; Juaristi, Eusebio: On the Synthesis of a Novel Chiral Phosphorodiamidic Acid Containing­ the α-Phenylethyl Moiety: Insights on its Conformation and Reactivity
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El Haimer, Mohamed; Faragó, Tünde; Schelz, Zsuzsanna; Zupkó, István; Palkó, Márta: Synthesis of Alicyclic 2-Methylenethiazolo[2,3-b]quinazolinone Derivatives via Base-Promoted Cascade Reactions
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Garnes-Portolés, Francisco; Miguélez, Rubén; Grayson, Matthew N.; Barrio, Pablo: Heteroatom-Tethered ω-Alkenylallylboronates: Stereoselective Synthesis of Heterocyclic Derived Alcohols
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Dargó, Gyula; Nagy, Sándor; Kis, Dávid; Bagi, Péter; Mátravölgyi, Béla; Tóth, Blanka; Huszthy, Péter; Drahos, László; Kupai, József: Application of Proline-Derived (Thio)squaramide Organocatalysts in Asymmetric Diels–Alder and Conjugate Addition Reactions
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Raji, Mounir; Le, Tam Minh; Csámpai, Antal; Nagy, Viktória; Zupkó, István; Szakonyi, Zsolt: Stereoselective Synthesis and Applications of Pinane-Based Chiral 1,4-Amino Alcohol Derivatives
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Molnár, István G.; Mucsi, Zoltán; Kovács, Ervin; Nyerges, Miklós: Electrocyclization and Unexpected Reactions of Non-Stabilized α,β:γ,δ-Unsaturated Azomethine Ylides: Experimental and Theoretical Studies
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Cserép, Gergely B.; Németh, Krisztina; Szatmári, Ágnes; Horváth, Flóra; Imre, Tímea; Németh, Krisztina; Kele, Péter: Beyond the Bioorthogonal Inverse-Electron-Demand Diels–Alder Reactions of Tetrazines: 2-Pyrone-Functionalized Fluorogenic Probes
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Szabó, Tímea; Görür, Funda Lidya; Horváth, Simon; Volk, Balázs; Milen, Mátyás: Synthesis of Racemic and Enantiopure Forms of β-Carboline Alkaloid Brevicolline
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Berecz, Gábor; Dancsó, András; Németh, Dóra R.; Kiss, Loránd; Simig, Gyula; Volk, Balázs: Towards Tianeptine Analogues: Synthesis of New Ring Systems Containing a Dibenzo[c,f][1,2]thiazepine S,S-Dioxide Core
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Takao, Go; Hakozaki, Tomohiro; Miura, Keisuke; Urushibara, Yusuke; Fuchibe, Kohei; Ichikawa, Junji: Construction of Substituted [4]Acene Frameworks Based on Double Cationic Cyclizations of Fluoroalkenes
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Harsági, Nikoletta; Kiss, Nóra Zsuzsa; Drahos, László; Keglevich, György: Synthesis of Cyclic Phosphinates by Microwave-Assisted Ionic-Liquid-Promoted Alcoholysis
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Issue 04/2022

He, Jian; Liu, Qiang: Highly Efficient Visible-Light-Driven [2+2] Cycloaddition of Maleimides to Alkenes and Alkynes for the Synthesis of 3-Aza­bicyclo[3.2.0]heptane-Fused Scaffolds
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Qureshi, Asif Ali; Sanjeeva Kumar, Arpula; Chauhan, Sachin; Kumara Swamy, K. C.: Stereo- and Regioselective [3+2] Cycloaddition of Acetoxy Allenoates with Azides: Metal-Free Synthesis of Multisubstituted Triazoles
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Barday, Manuel; Nicolas, Eva; Higginson, Bradley; Delmotte, François; Appelmans, Martin; Aïssa, Christophe: Tandem Nickel-Catalyzed Dimerization/(4+2) Cycloaddition of Terminal Alkynes with Four-Membered Ring Ketones
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Issue 22/2021

Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations
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Ryan, Jonathon S.; Schindler, Corinna S.: Total Synthesis of Mycocyclosin and the Herqulines
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Sokol, Kevin Rafael; Magauer, Thomas: Total Synthesis of Oxepin and Dihydrooxepin Containing Natural Products
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Martín-Heras, Víctor; Daniliuc, Constantin G.; Gilmour, Ryan: An I(I)/I(III) Catalysis Route to the Heptafluoroisopropyl Group: A Privileged Module in Contemporary Agrochemistry
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Wood, Devin P.; Guan, Weiyang; Lin, Song: Titanium and Cobalt Bimetallic Radical Redox Relay for the Isomerization of N-Bz Aziridines to Allylic Amides
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Garry, Olivia L.; Mansfield, Steven J.; Anderson, Edward A.: Regio- and Stereoselective Addition of Brønsted Acids to Yndiamides: Synthesis of N,O,N- and N,S,N-Trisubstituted Ketene Acetals
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Tien, Chieh-Hung; Trofimova, Alina; Shao, Wenjie; Yudin, Andrei K.: Synthesis of Borylated Hydrazino Acid Derivatives
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Kasim, Johanes K.; Kavianinia, Iman; Bull, Matthew; Harris, Paul W. R.; Smaill, Jeff B.; Patterson, Adam V.; Brimble, Margaret A.: Fourth-Generation Analogues of the Anticancer Peptaibol Culicinin D: Probing the Effects of Hydrophobicity and Halogenation on Cytotoxicity
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Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten: Studies towards the Synthesis of (–)-Pulvomycin: Construction of the C12–C40 Segment by a Stereoselective Aldol Reaction
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El Khoury, Anton; Seidler, Paul M.; Eisenberg, David S.; Harran, Patrick G.: Catalytic Synthesis of PEGylated EGCG Conjugates that Disaggregate Alzheimer’s Tau
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Caldora, Henry P.; Govaerts, Sebastian; Dighe, Shashikant U.; Turner, Oliver J.; Leonori, Daniele: A de novo Synthesis of Oxindoles from Cyclohexanone-Derived γ-Keto-Ester Acceptors Using a Desaturative Amination–Cyclization Approach
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Wong, Jonathan J.; Chen, Xiangyang; Houk, Kendall N.; Vollhardt, K. Peter C.: The Trajectory of the (η5-Cyclopentadienyl)cobalt-Mediated Cycloisomerization of Ene-Yne-Ene-Type Allyl Propargylic Ethers to Furans: A DFT Appraisal
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Davis, Christopher W.; Bingham, Tanner W.; Okumura, Mikiko; Sarlah, David: Dearomative syn-1,2-Diamination of Benzene and Naphthalene
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Jaye, Joseph A.; Sletten, Ellen M.: Simple Synthesis of Fluorinated Ene-Ynes via In Situ Generation of Allenes
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Wang, Lin; Ni, Shengyang; Cornella, Josep: Validation of Arylphosphorothiolates as Convergent Substrates for Ar-SF4Cl and Ar-SF5 Synthesis
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Issue 18/2021

Basak, Sumon; Biswas, Jyoti Prasad; Maiti, Debabrata: Transition-Metal-Catalyzed C–H Arylation Using Organoboron Reagents
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De, Pinaki Bhusan; Asako, Sobi; Ilies, Laurean: Recent Advances in the Use of Sodium Dispersion for Organic Synthesis
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Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki: Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization
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Misal Castro, Luis C.; Sultan, Ibrahim; Tsurugi, Hayato; Mashima, Kazushi: Pyridine-Mediated B–B Bond Activation of (RO)2B–B(OR)2 for Generating Borylpyridine Anions and Pyridine-Stabilized Boryl Radicals as Useful Boryl Reagents in Organic Synthesis
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Maeda, Kyogo; Motokura, Ken: Recent Advances in Heterogeneous Ir Complex Catalysts for Aromatic C–H Borylation
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Doiuchi, Daiki; Uchida, Tatsuya: Recent Strategies in Non-Heme-Type Metal Complex-Catalyzed Site-, Chemo-, and Enantioselective C–H Oxygenations
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Sihag, Pinki; Jeganmohan, Masilamani: Recent Advances in Transition-Metal-Catalyzed C–H Functionalization Reactions Involving Aza/Oxabicyclic Alkenes
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Jung, Jieun; Saito, Susumu: Recent Advances in Light-Driven Carbon–Carbon Bond Formation via Carbon Dioxide Activation
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Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto: C–H Bond Functionalization Using Pd- and Au-Supported Catalysts with Mechanistic Insights of the Active Species
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Zhang, Zhuo-Zhuo; Zhou, Gang; Huang, Fan-Rui; Shi, Bing-Feng: Cobalt-Catalyzed Oxidative [4+2] Annulation of Benzamides with Dihydrofuran: A Facile Route to Tetrahydrofuro[2,3-c]isoquinolinones
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Wan, Bin; Zhang, Yanghui: Synthesis of Unsymmetrically Substituted Tetraphenylenes through Palladium-Catalyzed C(sp2)–H Activation
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Dalal, Arup; Babu, Srinivasarao Arulananda: Pd(II)-Catalyzed Directing-Group-Aided C–H Arylation and Alkylation of Pyrene Core: Synthesis of C1,C2- and C1,C10-Disubstituted Pyrene Motifs
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Wei, Yunlong; Chen, Zhiqi; Wu, Zhen; Xu, Yaohui; Wu, Xinxin; Zhu, Chen: Radical Carbosulfonylation of Propellane: Synthesis of Sulfonyl β-Keto-bicyclo[1,1,1]pentanes
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Hassan, Mirja Md Mahamudul; Hoque, Md Emdadul; Dey, Sayan; Guria, Saikat; Roy, Brindaban; Chattopadhyay, Buddhadeb: Iridium-Catalyzed Site-Selective Borylation of 8-Arylquinolines
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Yuan, Shuqing; Ling, Liang; Tang, Jinghua; Luo, Meiming; Zeng, Xiaoming: Chromium-Catalyzed Reductive Cleavage of Unactivated Aromatic and Benzylic C–O Bonds
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Minami, Yasunori; Matsuyama, Nao; Matsuo, Yasuaki; Tamura, Masanori; Sato, Kazuhiko; Nakajima, Yumiko: Catalytic Reductive Cleavage of Poly(phenylene sulfide) Using a Hydrosilane
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Xu, Wei; Kohei, Miki; Shibasaki, Masakatsu; Kumagai, Naoya: Strategic Synthesis of Asymmetrically Substituted C4N4 Fluorophores
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Gu, Zheng-Yang; Wu, Yang; Jin, Feng; Bao, Xiaoguang; Xia, Ji-Bao: Intermolecular C–H Amidation of Alkenes with Carbon Monoxide and Azides via Tandem Palladium Catalysis
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Morimoto, Tsumoru; Wang, Chuang; Tanimoto, Hiroki; Artok, Levent; Kakiuchi, Kiyomi: Rhodium(I)-Catalyzed CO-Gas-Free Arylative Dual-Carbonylation of Alkynes with Arylboronic Acids via the Formyl C–H Activation of Formaldehyde
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Kimura, Naoki; Katta, Shiori; Kitazawa, Yoichi; Kochi, Takuya; Kakiuchi, Fumitoshi: Deuterium-Labeling Studies on the C–H/Olefin Coupling of Aromatic Ketones Catalyzed by Fe(PMe3)4
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Jinnai, Seihou; Oi, Ayumi; Seo, Takuji; Moriyama, Taichi; Minami, Ryunosuke; Higashida, Suguru; Ie, Yutaka: Electron-Accepting π-Conjugated Compound Containing Cyano-Substituted Naphthobisthiadiazole as Nonfullerene Acceptor in Organic Solar Cells
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Rawat, Vishal Kumar; Higashida, Kosuke; Sawamura, Masaya: Nickel-Catalyzed Homocoupling of Aryl Ethers with Magnesium Anthracene Reductant
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Fukuyama, Takahide; Hamada, Yuki; Ryu, Ilhyong: A New Protocol for Catalytic Reduction of Alkyl Chlorides Using an Iridium/Bis(benzimidazol-2′-yl)pyridine Catalyst and Triethylsilane
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Issue 17/2021

Korvorapun, Korkit; Samanta, Ramesh C.; Rogge, Torben; Ackermann, Lutz: Remote C–H Functionalizations by Ruthenium Catalysis
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Vijaykumar, Muniyappa; Punji, Benudhar: Advances in Transition-Metal-Catalyzed C–H Bond Oxygenation of Amides
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Ohno, Shohei; Miyoshi, Makoto; Murai, Kenichi; Arisawa, Mitsuhiro: Non-Directed β- or γ-C(sp3)–H Functionalization of Saturated Nitrogen-Containing Heterocycles
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Aldhous, Timothy P.; Chung, Raymond W. M.; Dalling, Andrew G.; Bower, John F.: Enantioselective Intermolecular Murai-Type Alkene Hydroarylation Reactions
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Oonishi, Yoshihiro; Sakamoto, Shunki; Agata, Shuya; Sato, Yoshihiro: Rhodium(I)-Catalyzed Enantioselective Cyclization of Enynes through Site-Selective C(sp3)–H Bond Activation Triggered by Formation of Rhodacycle
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Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
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Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro: Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation
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Seo, Jia; Chen, Che-Wei; Lee, Woohyeong; Jeon, Ju Eun; Chen, Pei-Ling; Chuang, Shih-Ching; Joo, Jung Min: Palladium-Catalyzed C–H Benzannulation of Functionalized Furans and Pyrroles with Alkynes
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Fukumoto, Yoshiya; Shiratani, Motohiro; Noguchi, Hikaru; Chatani, Naoto: Iridium-Catalyzed Direct Amidation of Imidazoles at the C-2 Position with Isocyanates in the Presence of Hydrosilanes Leading to Imidazole-2-Carboxamides
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Ozaki, Tomoya; Kaga, Atsushi; Saito, Hayate; Yorimitsu, Hideki: Generation of Aryllithium Reagents from N-Arylpyrroles Using Lithium
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Inai, Yasuhito; Usuki, Yoshinosuke; Satoh, Tetsuya: Synthesis of Benzo-Fused Cyclic Compounds via Rhodium-Catalyzed Decarboxylative Coupling of Aromatic Carboxylic Acids with Alkynes
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Shimazumi, Ryoma; Morita, Kosuke; Yoshida, Tomoki; Yasui, Kosuke; Tobisu, Mamoru: Late-Stage Derivatization of Buflavine by Nickel-Catalyzed Direct Substitution of a Methoxy Group via C–O Bond Activation
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You, Jingwen; Chen, Qiang; Nishihara, Yasushi: Nickel-Catalyzed Decarbonylative Thioetherification of Acyl Fluorides via C–F Bond Activation
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Yabe, Ryota; Ebe, Yusuke; Nishimura, Takahiro: Iridium-Catalyzed Direct C–H Allylation of Ketimines
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Ohmura, Toshimichi; Yagi, Kaito; Torigoe, Takeru; Suginome, Michinori: Intramolecular Addition of a Dimethylamino C(sp3)–H Bond across C–C Triple Bonds Using IrCl(DTBM-SEGPHOS)(ethylene) Catalyst: Synthesis of Indoles from 2-Alkynyl-N-methylanilines
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Takahashi, Hiroto; Honjo, Yusaku; Shibata, Yu; Nagashima, Yuki; Tanaka, Ken: Dienylation of Unfunctionalized Arenes with 1,6-Diynes via Rhodium-Catalyzed Directing-Group-Free C–H Bond Activation
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Kawakami, Haruka; Nohira, Itsuki; Chatani, Naoto: Nickel-Catalyzed C–F/N–H Annulation of 2-(2-Fluoroaryl) N-Heteroaromatic Compounds with Alkynes: Activation of C–F Bonds
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Yamamoto, Sonoka; Shibuya, Yushin; Suzuki, Toyoko; Okano, Kentaro; Horie, Masaki; Mori, Atsunori: One-Shot Deprotonative Metalation/Transmetalation/Polymerization of Halothiophenes Catalyzed by Nickel Complex for Polythiophene Synthesis
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Kanyiva, Kyalo Stephen; Tang, King Hung Nigel; Wang, Jiarui; Shibata, Takanori: Palladium-Catalyzed sp3 C–H Benzoxylation of Alanine Derivatives Using Aldehydes under Ambient Conditions
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Pan, Feng-Feng; Guo, Peng; Huang, Xiaochuang; Shu, Xing-Zhong: Synthesis of Dibenzyls by Nickel-Catalyzed Homocoupling of Benzyl Alcohols
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Kiyosu, Yuuki; Tanaka, Shino; Okumura, Sota; Kiyokawa, Kensuke; Minakata, Satoshi: Synthesis of Fused Diaziridine Derivatives from Cyclic Secondary Amines by Utilizing N-Bromosulfonamides as an Aminating Reagent
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Ninokata, Ryo; Korogi, Riho; Nakao, Junya; Fukuda, Tsutomu; Onodera, Gen; Kimura, Masanari: Reconstruction of Carbon Bond Frameworks via Oxapalladacycles Promoted by the Synergistic Effect of Palladium Catalyst and Triethylborane
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Tanaka, Shinji; Iwase, Shoutaro; Kanda, Sena; Kato, Marie; Kiriyama, Yutaro; Kitamura, Masato: Ruthenium-Catalyzed Asymmetric Dehydrative Allylic Cyclization of Five-Membered Chalcogen Heteroaromatics
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Kona, Chandrababu Naidu; Oku, Rikuto; Nishii, Yuji; Miura, Masahiro: Peri-Selective Direct Acylmethylation and Amidation of Naphthalene Derivatives Using Iridium and Rhodium Catalysts
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Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke: CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones
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Xu, Wengang; Wu, Mingbo; Yoshikai, Naohiko: Iron-Catalyzed Remote C–H Alkylation of 8-Amidoquinolines with Cycloalkanes
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Issue 02/2021

Arjona-Esteban, Alhama; Rausch, Anja; Vysotsky, Myroslav O.; Würthner, Frank: Merocyanine Dyes with Extended Polymethine Chains by Simple Two-Step Condensation Sequence
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Yoshimura, Aya; Henmi, Keisuke; Kimura, Hitoshi; Sakakibara, Ryo; Ochi, Rika; Shirahata, Takashi; Yorimitsu, Hideki; Misaki, Yohji: Synthesis of Peripherally Arylated Tetrathiafulvalenes Extended with an Anthraquinoid Spacer via Pd-Catalyzed C–H Arylation and Construction of a Double-Helical Cobalt-Based Metal-Organic Framework
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Widner, Florian J.; Kieninger, Christoph; Wurst, Klaus; Deery, Evelyne; Lawrence, Andrew D.; Warren, Martin J.; Kräutler, Bernhard: Synthesis, Spectral Characterization and Crystal Structure of Chlororhodibalamin: A Synthesis Platform for Rhodium Analogues of Vitamin B12 and for Rh-Based Antivitamins B12
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Yan, Feng-Zhi; Shao, Yuan-Guang; Zhang, Zibin; Shen, Yan-Feng; Huang, Xue-Chun; Zhang, Pei-Ling; Li, Shijun: Synthesis of Catenanes from a BMP32C10-Based Cryptand Tuned by the Linkage Length of Paraquat Salts
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Mei, Peifeng; Kurosaki, Ryo; Matsumoto, Akinobu; Yamada, Hiroko; Aratani, Naoki: One-Pot Synthesis of a Cyclic Pyrene Octamer from Two Bifunctionalized Pyrene Monomers
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Issue 24/2020

Qin, Jing-Hao; Li, Jin-Heng; An, De-Lie: Recent Advances in Cycloaddition Reactions with Alkynes to Construct Heterocycles
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Pellissier, Hélène: The Use of Domino Reactions for the Synthesis of Chiral Rings
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Wei, Bin; Li, Ke-Wei; Wu, Yan-Chen; Tong, Shi-Qi; Song, Ren-Jie: Radical Strategy for the Transition-Metal-Catalyzed Synthesis of γ-Lactones: A Review
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Huang, Min-Hua; Hao, Wen-Juan; Jiang, Bo: Iridium(III)-Catalyzed Difluoroalkylation–Bicyclization of 1,7-Enynes toward Benzo[a]fluoren-5-ones under Visible-Light Photoredox Conditions
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Issue 22/2020

Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
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Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain: Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
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Wächtler, Andreas; Bremer, Matthias; Maillard, David; Mohr, Thomas: Controlling the All-trans Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds
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Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis: Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
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Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda: Copper-Catalyzed Asymmetric Hydroamination of Styrenes with pivZPhos as Ligand
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Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.: Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
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Issue 21/2020

Shiri, Morteza; Farajinia-Lehi, Noushin; Salehi, Parvin; Tanbakouchian, Zahra: Transition Metal and Inner Transition Metal Catalyzed Amide Derivatives Formation through Isocyanide Chemistry
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Manne, Srinivasa Rao; de la Torre, Beatriz G.; El-Faham, Ayman; Albericio, Fernando: OxymaPure Coupling Reagents: Beyond Solid-Phase Peptide Synthesis
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Zhao, Baoli; Liu, Yunyun: Step-Economical C–H Activation Reactions Directed by In Situ Amidation
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Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.: Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis
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Kolympadi Marković, Maria; Marković, Dean; Laclef, Sylvain: Amide Synthesis by Transamidation of Primary Carboxamides
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Shiri, Morteza; Gholami-Koupaei, Zahra; Bandehali-Naeini, Farzaneh; Tonekaboni, Maryam-Sadat; Soheil-Moghaddam, Saeedeh; Ebrahimi, Delaram; Karami, Sima; Notash, Behrouz: Highly Selective Synthesis of α-Hydroxy, α-Oxy, and α-Oxo Amides by a Post-Passerini Condensation Transformation
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Movahed, Farzaneh Soleymani; Sawant, Dinesh N.; Bagal, Dattatraya B.; Saito, Susumu: Tris(o-phenylenedioxy)cyclotriphosphazene as a Promoter for the Formation of Amide Bonds Between Aromatic Acids and Amines
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Smolobochkin, Andrey V.; Gazizov, Almir S.; Otegen, Nazerke K.; Voronina, Julia K.; Strelnik, Anna G.; Samigullina, Aida I.; Burilov, Alexander R.; Pudovik, Michail A.: Nucleophilic Cyclization/Electrophilic Substitution of (2,2-Dialkoxyethyl)ureas: Highly Regioselective Access to Novel 4-(Het)arylimidazolidinones and Benzo[d][1,3]diazepinones
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Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.: Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-O-sulfonic Acid in Aqueous Media
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Kabes, Connor Q.; Gunn, Jack H.; Selbst, Maximilian A.; Lucas, Reagan F.; Gladysz, John A.: Syntheses of Enantiopure 1,2-Ethylenediamines with Tethered Secondary Amines of the Formula H2NCH2CH[(CH2)nNHMe]NH2 (n = 1–4) from α-Amino Acids: New Agents for Asymmetric Catalysis
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Zhang, Rui; Zhang, Jun-Chao; Zhang, Wei-Yi; He, Yu-Qing; Cheng, Hua; Chen, Cheng; Gu, Yu-Cheng: A Practical Approach for the Transamidation of N,N-Dimethyl Amides with Primary Amines Promoted by Sodium tert-Butoxide under Solvent-Free Conditions
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Issue 08/2020

Connon, Robert; Carroll, Laura; Guiry, Patrick J.: A Base-Promoted One-Pot Asymmetric Friedel–Crafts Alkylation/Michael Addition of 4-Substituted Indoles
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Yang, Yuzhong; Zhou, Liwei; Yang, Xiumei; Luo, Xiai; Deng, Guobo; Yang, Yuan; Liang, Yun: Synthesis of Phenanthrenes via Palladium-Catalyzed Three-Component Domino Reaction of Aryl Iodides, Internal Alkynes, and o-Bromobenzoic Acids
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Henkel, Michael; Bach, Thorsten: Annulation of Indoles with 1,n-Dibromoalkanes by a Pd(II)-Catalyzed and Norbornene-Mediated Reaction Cascade
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Shen, Zican; Li, Chen; Mercado, Brandon Q.; Ellman, Jonathan A.: Cobalt(III)-Catalyzed Diastereoselective Three-Component C–H Bond Addition to Butadiene and Activated Ketones
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Lee, Sumin; Jang, Young Jin; Phipps, Erik J. T.; Lei, Honghui; Rovis, Tomislav: Rhodium(III)-Catalyzed Three-Component 1,2-Diamination of Unactivated Terminal Alkenes
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Sun, Manman; Li, Jinshan; Chen, Weida; Wu, Haijian; Yang, Jianguo; Wang, Zhiming: Palladium-Catalyzed [4+2] Annulation of Aryl and Alkenyl Carboxamides with 1,3-Dienes via C–H Functionalization: Synthesis of 3,4-Dihydroisoquinolones and 5,6-Dihydropyridinones
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Issue 23/2019

Special Topic Cover Page
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Sutherland, Andrew: Radiohalogenation of Organic Compounds: Practical Considerations and Challenges for Molecular Imaging
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Milicevic Sephton, Selena; Zhou, Xiaoyun; Thompson, Stephen; Aigbirhio, Franklin I.: Preparation of the Serotonin Transporter PET Radiotracer 2-({2-[(Dimethylamino)methyl]phenyl}thio)-5-[18F]fluoroaniline (4-[18F]ADAM): Probing Synthetic and Radiosynthetic Methods
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