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Issue eFirst
Takahashi, Hiroto; Honjo, Yusaku; Shibata, Yu; Nagashima, Yuki; Tanaka, Ken:
Dienylation of Unfunctionalized Arenes with 1,6-Diynes via Rhodium-Catalyzed Directing-Group-Free C–H Bond Activation
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Gu, Zheng-Yang; Wu, Yang; Jin, Feng; Bao, Xiaoguang; Xia, Ji-Bao:
Intermolecular C–H Amidation of Alkenes with Carbon Monoxide and Azides via Tandem Palladium Catalysis
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PDF (484 kb)
Khatana, Anil Kumar; Singh, Vikram; Gupta, Manoj Kumar; Tiwari, Bhoopendra:
A Highly Efficient NHC-Catalyzed Aerobic Oxidation of Aldehydes to Carboxylic Acids
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PDF (192 kb)
Ryan, Jonathon S.; Schindler, Corinna S.:
Total Synthesis of Mycocyclosin and the Herqulines
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PDF (565 kb)
Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke:
CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones
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PDF (259 kb)
Nocera, Giuseppe; Murphy, John A.:
Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview
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PDF (247 kb)
Sperger, Theresa; Schoenebeck, Franziska:
α-Arylation of Esters and Ketones Enabled by a Bench-Stable Pd(I) Dimer Catalyst
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PDF (209 kb)
Wan, Bin; Zhang, Yanghui:
Synthesis of Unsymmetrically Substituted Tetraphenylenes through Palladium-Catalyzed C(sp
2
)–H Activation
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PDF (312 kb)
Pan, Feng-Feng; Guo, Peng; Huang, Xiaochuang; Shu, Xing-Zhong:
Synthesis of Dibenzyls by Nickel-Catalyzed Homocoupling of Benzyl Alcohols
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PDF (239 kb)
Cole, Charles J. F.; Chi, Hyung Min; DeBacker, Kenneth C.; Snyder, Scott A.:
Synthesis of Enhanced, Isolable Disulfanium Salts and their Application to Thiiranium-Promoted Polyene Cyclizations
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PDF (212 kb)
Wang, Zheng; Ji, Hongtao; He, Wei-Min; Xiong, Yang; Zhang, Guozhu:
Chromium-Catalyzed Asymmetric Dearomatization–Addition Reactions of Halomethyloxazoles and Indoles
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Xu, Wengang; Wu, Mingbo; Yoshikai, Naohiko:
Iron-Catalyzed Remote C–H Alkylation of 8-Amidoquinolines with Cycloalkanes
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PDF (252 kb)
Lindner, Marcin; Krasiński, Antoni; Jurczak, Janusz:
Facile, Stereocontrolled Synthetic Route towards Bis-functionalised Pyrrolizidines
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PDF (418 kb)
Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro:
Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
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Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark:
Recent Advances in Transition-Metal-Free (4+3)-Annulations
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PDF (1989 kb)
Oberg, Kevin M.; Cochran, Brian M.; Cook, Matthew J.; Rovis, Tomislav:
The Catalytic Alkylative Desymmetrization of Anhydrides in a Formal Synthesis of Ionomycin
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PDF (228 kb)
Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke:
Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite
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PDF (180 kb)
Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro:
Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation
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PDF (1169 kb)
Zhang, Yongda; Lao, Kendricks S.; Sieber, Joshua D.; Xu, Yibo; Wu, Linglin; Wang, Xiao-Jun; Desrosiers, Jean-Nicolas; Lee, Heewon; Haddad, Nizar; Han, Zhengxu S.; Yee, Nathan K.; Song, Jinhua J.; Howell, Amy R.; Senanayake, Chris H.:
Modular Dihydrobenzoazaphosphole Ligands for Suzuki–Miyaura Cross-Coupling
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Liddon, John T. R.; Rossi-Ashton, James A.; Clarke, Aimee K.; Lynam, Jason M.; Taylor, Richard J. K.; Unsworth, William P.:
Divergent Reactivity of Indole-Tethered Ynones with Silver(I) and Gold(I) Catalysts: A Combined Synthetic and Computational Study
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Joshi, Madhur S.; Pigge, F. Christopher:
Sequential Pyridine Dearomatization–Mizoroki–Heck Cyclization for the Construction of Fused (Dihydropyrido)isoindolinone Ring Systems
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PDF (269 kb)
Inai, Yasuhito; Usuki, Yoshinosuke; Satoh, Tetsuya:
Synthesis of Benzo-Fused Cyclic Compounds via Rhodium-Catalyzed Decarboxylative Coupling of Aromatic Carboxylic Acids with Alkynes
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PDF (267 kb)
Wertjes, William; Ayers, Sloan; Gao, Qi; Simmons, Eric M.; Beutner, Gregory L.:
A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines
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PDF (531 kb)
Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki:
Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization
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Denizot, Natacha; Guillot, Régis; Kouklovsky, Cyrille; Vincent, Guillaume:
N
-Iodosuccinimide-Mediated Oxidative Coupling of Indoles and Phenols: A Synthetic Study toward the Benzofuroindoline Moiety of Bipleiophylline
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Kawakami, Haruka; Nohira, Itsuki; Chatani, Naoto:
Nickel-Catalyzed C–F/N–H Annulation of 2-(2-Fluoroaryl) N-Heteroaromatic Compounds with Alkynes: Activation of C–F Bonds
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PDF (241 kb)
Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten:
Studies towards the Synthesis of (–)-Pulvomycin: Construction of the C12–C40 Segment by a Stereoselective Aldol Reaction
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Ziegler, Dorothée S.; Klier, Lydia; Müller, Nicolas; Karaghiosoff, Konstantin; Knochel, Paul:
Directed Zincation or Magnesiation of 2- and 4-Pyrones and Their Derivatives
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PDF (273 kb)
Garlets, Zachary J.; Wolfe, John P.:
Asymmetric Synthesis of Six-Membered Cyclic Sulfamides via Palladium-Catalyzed Alkene Carboamination Reactions
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PDF (222 kb)
Fukumoto, Yoshiya; Shiratani, Motohiro; Noguchi, Hikaru; Chatani, Naoto:
Iridium-Catalyzed Direct Amidation of Imidazoles at the C-2 Position with Isocyanates in the Presence of Hydrosilanes Leading to Imidazole-2-Carboxamides
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PDF (267 kb)
Yamamoto, Sonoka; Shibuya, Yushin; Suzuki, Toyoko; Okano, Kentaro; Horie, Masaki; Mori, Atsunori:
One-Shot Deprotonative Metalation/Transmetalation/Polymerization of Halothiophenes Catalyzed by Nickel Complex for Polythiophene Synthesis
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PDF (406 kb)
Issue Accepted Manuscripts
Kiyosu, Yuuki; Tanaka, Shino; Okumura, Sota; Kiyokawa, Kensuke; Minakata, Satoshi:
Synthesis of Fused Diaziridine Derivatives from Cyclic Secondary Amines Utilizing N-Bromosulfonamides as an Aminating Reagent
Full Text
PDF (3702 kb)
You, Jingwen; Chen, Qiang; Nishihara, Yasushi:
Nickel-Catalyzed Decarbonylative Thioetherification of Acyl Fluorides via C-F Bond Activation
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PDF (4410 kb)
Kanyiva, Kyalo Stephen; Nigel Tang, King Hung; Wang, Jiarui; Shibata, Takanori:
Palladium-Catalyzed sp
3
C–H Benzoxylation of Alanine Derivatives Using Aldehydes under Ambient Conditions
Full Text
PDF (1811 kb)
Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto:
C-H bond functionalization using Pd and Au supported catalysts with mechanistic insights of the active species
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PDF (2151 kb)
Dalal, Arup; Arulananda Babu, Srinivasarao:
Pd(II)-catalyzed directing group-aided C-H arylation and alkylation of pyrene core. Synthesis of C1,C2- and C1,C10-disubstituted pyrene motifs
Full Text
PDF (36231 kb)
Oonishi, Yoshihiro; Sakamoto, Shunki; Agata, Shuya; Sato, Yoshihiro:
Rh(I)-Catalyzed Enantioselective Cyclization of Enyne through Site-Selective C(sp3)-H Bond Activation Triggered by Formation of Rhodacycle
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PDF (6626 kb)
De, Pinaki Bhusan; Asako, Sobi; Ilies, Laurean:
Recent Advances in Use of Sodium Dispersion for Organic Synthesis
Full Text
PDF (1739 kb)
Kona, Chandrababu Naidu; Oku, Rikuto; Nishii, Yuji; Miura, Masahiro:
Peri-Selective Direct Acylmethylation and Amidation of Naphthalene Derivatives Using Iridium and Rhodium Catalysts
Full Text
PDF (4746 kb)
Shimazumi, Ryoma; Morita, Kosuke; Yoshida, Tomoki; Yasui, Kousuke; Tobisu, Mamoru:
Late-stage Derivatization of Buflavine by Nickel-catalyzed Direct Substitution of a Methoxy Group via C-O Bond Activation
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PDF (2888 kb)
Ozaki, Tomoya; Kaga, Atsushi; Saito, Hayate; Yorimitsu, Hideki:
Generation of Aryllithium Reagents from N-Arylpyrroles Using Lithium
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PDF (12387 kb)
OHNO, Shohei; MIYOSHI, Makoto; Murai, Kenichi; Arisawa, Mitsuhiro:
Non-directed β- or γ-C(sp3)-H Functionalization of Saturated Nitrogen-containing Heterocycles
Full Text
PDF (1937 kb)
Morimoto, Tsumoru; Wang, Chuang; Tanimoto, Hiroki; Artok, Levent; Kakiuchi, Kiyomi:
Rhodium(I)-Catalyzed CO Gas-Free Arylative Dual-Carbonylation of Alkynes with Arylboronic Acids via the Formyl C-H Activation of Formaldehyde
Full Text
PDF (5489 kb)
Yabe, Ryota; Ebe, Yusuke; Nishimura, Takahiro:
Iridium-Catalyzed Direct C–H Allylation of Ketimines
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PDF (5450 kb)
Vijaykumar, Muniyappa; Punji, Benudhar:
Advances in Transition-Metal-Catalyzed C–H Bond Oxygenation of Amides
Full Text
PDF (3402 kb)
Wei, Yunlong; Chen, Zhiqi; Wu, Zhen; Xu, Yaohui; Wu, Xinxin; Zhu, Chen:
Radical Carbosulfonylation of Propellane: Synthesis of Sulfonyl β-Keto-Bicyclo[1,1,1]pentanes
Full Text
PDF (4648 kb)
He, Jian; Liu, Qiang:
Highly Efficient Visible-Light-Driven [2+2] cycloaddition of Maleimides to Alkenes/Alkynes for Synthesis of 3‑Azabicyclo[3.2.0]heptane-Fused Scaffolds
Full Text
PDF (13070 kb)
Issue 02/2021
Arjona-Esteban, Alhama; Rausch, Anja; Vysotsky, Myroslav O.; Würthner, Frank:
Merocyanine Dyes with Extended Polymethine Chains by Simple Two-Step Condensation Sequence
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Yoshimura, Aya; Henmi, Keisuke; Kimura, Hitoshi; Sakakibara, Ryo; Ochi, Rika; Shirahata, Takashi; Yorimitsu, Hideki; Misaki, Yohji:
Synthesis of Peripherally Arylated Tetrathiafulvalenes Extended with an Anthraquinoid Spacer via Pd-Catalyzed C–H Arylation and Construction of a Double-Helical Cobalt-Based Metal-Organic Framework
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PDF (2158 kb)
Widner, Florian J.; Kieninger, Christoph; Wurst, Klaus; Deery, Evelyne; Lawrence, Andrew D.; Warren, Martin J.; Kräutler, Bernhard:
Synthesis, Spectral Characterization and Crystal Structure of Chlororhodibalamin: A Synthesis Platform for Rhodium Analogues of Vitamin B
12
and for Rh-Based Antivitamins B
12
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PDF (855 kb)
Yan, Feng-Zhi; Shao, Yuan-Guang; Zhang, Zibin; Shen, Yan-Feng; Huang, Xue-Chun; Zhang, Pei-Ling; Li, Shijun:
Synthesis of Catenanes from a BMP32C10-Based Cryptand Tuned by the Linkage Length of Paraquat Salts
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PDF (842 kb)
Mei, Peifeng; Kurosaki, Ryo; Matsumoto, Akinobu; Yamada, Hiroko; Aratani, Naoki:
One-Pot Synthesis of a Cyclic Pyrene Octamer from Two Bifunctionalized Pyrene Monomers
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Issue 24/2020
Qin, Jing-Hao; Li, Jin-Heng; An, De-Lie:
Recent Advances in Cycloaddition Reactions with Alkynes to Construct Heterocycles
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PDF (1007 kb)
Pellissier, Hélène:
The Use of Domino Reactions for the Synthesis of Chiral Rings
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PDF (632 kb)
Wei, Bin; Li, Ke-Wei; Wu, Yan-Chen; Tong, Shi-Qi; Song, Ren-Jie:
Radical Strategy for the Transition-Metal-Catalyzed Synthesis of γ-Lactones: A Review
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PDF (577 kb)
Huang, Min-Hua; Hao, Wen-Juan; Jiang, Bo:
Iridium(III)-Catalyzed Difluoroalkylation–Bicyclization of 1,7-Enynes toward Benzo[
a
]fluoren-5-ones under Visible-Light Photoredox Conditions
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PDF (261 kb)
Issue 22/2020
Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.:
Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
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Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain:
Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
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PDF (1537 kb)
Wächtler, Andreas; Bremer, Matthias; Maillard, David; Mohr, Thomas:
Controlling the All-
trans
Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds
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PDF (808 kb)
Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis:
Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
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PDF (256 kb)
Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda:
Copper-Catalyzed Asymmetric Hydroamination of Styrenes with
piv
ZPhos as Ligand
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PDF (182 kb)
Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.:
Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
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PDF (253 kb)
Issue 21/2020
Shiri, Morteza; Farajinia-Lehi, Noushin; Salehi, Parvin; Tanbakouchian, Zahra:
Transition Metal and Inner Transition Metal Catalyzed Amide Derivatives Formation through Isocyanide Chemistry
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PDF (1583 kb)
Manne, Srinivasa Rao; de la Torre, Beatriz G.; El-Faham, Ayman; Albericio, Fernando:
OxymaPure Coupling Reagents: Beyond Solid-Phase Peptide Synthesis
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Zhao, Baoli; Liu, Yunyun:
Step-Economical C–H Activation Reactions Directed by In Situ Amidation
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PDF (451 kb)
Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.:
Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis
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PDF (491 kb)
Kolympadi Marković, Maria; Marković, Dean; Laclef, Sylvain:
Amide Synthesis by Transamidation of Primary Carboxamides
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PDF (697 kb)
Shiri, Morteza; Gholami-Koupaei, Zahra; Bandehali-Naeini, Farzaneh; Tonekaboni, Maryam-Sadat; Soheil-Moghaddam, Saeedeh; Ebrahimi, Delaram; Karami, Sima; Notash, Behrouz:
Highly Selective Synthesis of α-Hydroxy, α-Oxy, and α-Oxo Amides by a Post-Passerini Condensation Transformation
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PDF (345 kb)
Movahed, Farzaneh Soleymani; Sawant, Dinesh N.; Bagal, Dattatraya B.; Saito, Susumu:
Tris(
o
-phenylenedioxy)cyclotriphosphazene as a Promoter for the Formation of Amide Bonds Between Aromatic Acids and Amines
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Smolobochkin, Andrey V.; Gazizov, Almir S.; Otegen, Nazerke K.; Voronina, Julia K.; Strelnik, Anna G.; Samigullina, Aida I.; Burilov, Alexander R.; Pudovik, Michail A.:
Nucleophilic Cyclization/Electrophilic Substitution of (2,2-Dialkoxyethyl)ureas: Highly Regioselective Access to Novel 4-(Het)arylimidazolidinones and Benzo[
d
][1,3]diazepinones
Full Text
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PDF (618 kb)
Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.:
Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-
O
-sulfonic Acid in Aqueous Media
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PDF (206 kb)
Kabes, Connor Q.; Gunn, Jack H.; Selbst, Maximilian A.; Lucas, Reagan F.; Gladysz, John A.:
Syntheses of Enantiopure 1,2-Ethylenediamines with Tethered Secondary Amines of the Formula H
2
NCH
2
CH[(CH
2
)
n
NHMe]NH
2
(
n
= 1–4) from α-Amino Acids: New Agents for Asymmetric Catalysis
Full Text
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PDF (516 kb)
Zhang, Rui; Zhang, Jun-Chao; Zhang, Wei-Yi; He, Yu-Qing; Cheng, Hua; Chen, Cheng; Gu, Yu-Cheng:
A Practical Approach for the Transamidation of
N
,
N
-Dimethyl Amides with Primary Amines Promoted by Sodium
tert
-Butoxide under Solvent-Free Conditions
Full Text
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PDF (277 kb)
Issue 08/2020
Connon, Robert; Carroll, Laura; Guiry, Patrick J.:
A Base-Promoted One-Pot Asymmetric Friedel–Crafts Alkylation/Michael Addition of 4-Substituted Indoles
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PDF (927 kb)
Yang, Yuzhong; Zhou, Liwei; Yang, Xiumei; Luo, Xiai; Deng, Guobo; Yang, Yuan; Liang, Yun:
Synthesis of Phenanthrenes via Palladium-Catalyzed Three-Component Domino Reaction of Aryl Iodides, Internal Alkynes, and
o
-Bromobenzoic Acids
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Henkel, Michael; Bach, Thorsten:
Annulation of Indoles with 1,n-Dibromoalkanes by a Pd(II)-Catalyzed and Norbornene-Mediated Reaction Cascade
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PDF (200 kb)
Shen, Zican; Li, Chen; Mercado, Brandon Q.; Ellman, Jonathan A.:
Cobalt(III)-Catalyzed Diastereoselective Three-Component C–H Bond Addition to Butadiene and Activated Ketones
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PDF (267 kb)
Lee, Sumin; Jang, Young Jin; Phipps, Erik J. T.; Lei, Honghui; Rovis, Tomislav:
Rhodium(III)-Catalyzed Three-Component 1,2-Diamination of Unactivated Terminal Alkenes
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PDF (662 kb)
Sun, Manman; Li, Jinshan; Chen, Weida; Wu, Haijian; Yang, Jianguo; Wang, Zhiming:
Palladium-Catalyzed [4+2] Annulation of Aryl and Alkenyl Carboxamides with 1,3-Dienes via C–H Functionalization: Synthesis of 3,4-Dihydroisoquinolones and 5,6-Dihydropyridinones
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Issue 23/2019
Special Topic Cover Page
Full Text
PDF (2080 kb)
Sutherland, Andrew:
Radiohalogenation of Organic Compounds: Practical Considerations and Challenges for Molecular Imaging
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PDF (330 kb)
Milicevic Sephton, Selena; Zhou, Xiaoyun; Thompson, Stephen; Aigbirhio, Franklin I.:
Preparation of the Serotonin Transporter PET Radiotracer 2-({2-[(Dimethylamino)methyl]phenyl}thio)-5-[
18
F]fluoroaniline (4-[
18
F]ADAM): Probing Synthetic and Radiosynthetic Methods
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Kitahara, Kazumasa; Mizutani, Haruna; Iwasa, Seiji; Shibatomi, Kazutaka:
Asymmetric Synthesis of α-Chloro-α-halo Ketones by Decarboxylative Chlorination of α-Halo-β-ketocarboxylic Acids
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PDF (226 kb)
Dubost, Emmanuelle; Babin, Victor; Benoist, Florian; Hébert, Alexandra; Pigrée, Gilbert; Bouillon, Jean-Philippe; Fabis, Frédéric; Cailly, Thomas:
Improvements of C–H Radio-Iodination of
N
-Acylsulfonamides toward Implementation in Clinics
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PDF (684 kb)
Thompson, Stephen; Lee, So Jeong; Jackson, Isaac M.; Ichiishi, Naoko; Brooks, Allen F.; Sanford, Melanie S.; Scott, Peter J. H.:
Synthesis of [
18
F]-γ-Fluoro-α,β-unsaturated Esters and Ketones via Vinylogous
18
F-Fluorination of α-Diazoacetates with [
18
F]AgF
Full Text
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PDF (449 kb)
Sarie, Jérôme C.; Neufeld, Jessica; Daniliuc, Constantin G.; Gilmour, Ryan:
Willgerodt-Type Dichloro(aryl)-λ
3
-Iodanes: A Structural Study
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PDF (3071 kb)
Issue 13/2019
Special Topic Cover Page
Full Text
PDF (1732 kb)
Podyacheva, Evgeniya; Afanasyev, Oleg I.; Tsygankov, Alexey A.; Makarova, Maria; Chusov, Denis:
Hitchhiker’s Guide to Reductive Amination
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PDF (1329 kb)
Lai, Wing In; Leung, Man Pan; Choy, Pui Ying; Kwong, Fuk Yee:
Sterically Hindered Amination of Aryl Chlorides Catalyzed by a New Carbazolyl-Derived P,N-Ligand-Composed Palladium Complex
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PDF (686 kb)
Purkait, Anisha; Jana, Chandan K.:
N-Aminations of Benzylamines and Alicyclic Amines with Nitrosoarenes to Hydrazones and Hydrazides
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PDF (339 kb)
Li, Quan-Zhe; Wang, Xun-Hui; Hou, Si-Hua; Ma, Yan-Yan; Zhao, Deng-Gao; Zhang, Shu-Yu; Bai, He-Yuan; Ding, Tong-Mei:
Silver-Catalyzed
para
-Selective C–H Amination of 1-Naphthylamides with Azodicarboxylates at Room Temperature
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PDF (202 kb)
Pratap, Ramendra; Yorimitsu, Hideki:
Palladium-Catalyzed Amination of Aryl Sulfides and Sulfoxides with Azaarylamines of Poor Nucleophilicity
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Zhou, Huan; Zhao, Wenlei; Zhang, Tao; Guo, Haodong; Huang, Haizhou; Chang, Mingxin:
Enantioselective Synthesis of 2-Substituted Pyrrolidines via Intramolecular Reductive Amination
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Issue 12/2019
Special Topic Cover Page
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Zhou, Yongyun; Khan, Ruhima; Fan, Baomin; Xu, Lijin:
Ruthenium-Catalyzed Selective Reduction of Carboxylic Esters and Carboxamides
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Deshmukh, Dewal S.; Bhanage, Bhalchandra M.:
Ruthenium-Catalyzed Annulation of
N
-Cbz Hydrazones via C–H/N–N Bond Activation for the Rapid Synthesis of Isoquinolines
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Das, Riki; Khot, Nandkishor Prakash; Deshpande, Akanksha Santosh; Kapur, Manmohan:
Ruthenium-Catalyzed Directed C(3)–H Olefination of
N
-Acetyl-1,2-dihydroisoquinolines: A Method to Achieve C3-Olefinated Isoquinolines
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Bairy, Gurupada; Nandi, Arijit; Manna, Kartic; Jana, Ranjan:
Ruthenium(II)-Catalyzed Migratory C–H Allylation/Hydroamination Cascade for the Synthesis of Rutaecarpine Analogues
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Tran, Christine; Haddad, Mansour; Ratovelomanana-Vidal, Virginie:
Ruthenium-Catalyzed [2+2+2] Cycloaddition of α,ω-Diynes and Selenocyanates: An Entry to Selenopyridine Derivatives
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Kawano, Teruhiro; Watari, Ryo; Kayaki, Yoshihito; Ikariya, Takao:
Catalytic Hydrogenation of Carboxamides with a Bifunctional Cp*Ru Catalyst Bearing an Imidazol-2-ylidene with a Protic Aminoethyl Side Chain
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Issue 17/2018
Special Topic Cover Page
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Oh, Eun Hye; Kim, Hyun Jin; Han, Soo Bong:
Recent Developments in Visible-Light-Catalyzed Multicomponent Trifluoromethylation of Unsaturated Carbon–Carbon Bonds
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Zhou, Wen-Jun; Zhang, Yi-Han; Gui, Yong-Yuan; Sun, Liang; Yu, Da-Gang:
Merging Transition-Metal Catalysis with Photoredox Catalysis: An Environmentally Friendly Strategy for C–H Functionalization
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Du, Yuliu; Wei, Zheng; Wang, Ting:
Visible-Light-Mediated Synthesis of Oxidized Amides via Organic Photoredox Catalysis
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An, Xiao-De; Yu, Shouyun:
Photoredox-Catalyzed Radical Relay Reaction Toward Functionalized Vicinal Diamines
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Voutyritsa, Errika; Nikitas, Nikolaos F.; Apostolopoulou, Mary K.; Gerogiannopoulou, Anna Dimitra D.; Kokotos, Christoforos G.:
Photoorganocatalytic Atom Transfer Radical Addition of Bromoacetonitrile to Aliphatic Olefins
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Otomura, Nobutaka; Okugawa, Yuto; Hirano, Koji; Miura, Masahiro:
Bromine Cation Initiated
vic
-Diphosphination of Styrenes with Diphosphines under Photoredox Catalysis
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Issue 16/2018
Special Topic Cover Page
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Baumann, Andreas N.; Eisold, Michael; Music, Arif; Didier, Dorian:
One-Pot Preparation of Stable Organoboronate Reagents for the Functionalization of Unsaturated Four- and Five-Membered Carbo- and Heterocycles
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Yamaguchi, Eiji; Kamito, Yuji; Matsuo, Kazuki; Ishihara, Jun; Itoh, Akichika:
Photooxidative Keto-Trifluoromethylation of Styrenes by Means of an Anthraquinone-Based Organocatalyst
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Chen, Yizhou; Wang, Shanlu; Zhao, Li; Rong, Chenyan; Liu, Tong; Sun, Han; Wang, Yuping; Zhang, Jian; Zhong, Guofu:
A Metal-Free Synthesis of 3-Phenoxyimidazo Heterocycles by Catalytic Oxidative Cyclization of 2-Amino-azaarenes with Lignin Models
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Suen, Linda M.; Wang, Cheng; Hunter, David N.; Mitchell, Helen J.; Converso, Antonella; ElMarrouni, Abdellatif:
Synthesis of HIV NNRTI Doravirine Analogues via Visible-Light Photoredox Decarboxylative Cross-Coupling
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Liu, Yang; Daka, Mario; Bandini, Marco:
Regio- and Stereoselective Nickel-Catalyzed Coupling of Boronic Acids with Allenoates
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Park, Jaerim; Song, Kwang Ho; Lee, Sunwoo:
Palladium-Catalyzed Decarboxylative Coupling Reactions of Propiolic Acid Derivatives and Arylsulfonyl Hydrazide
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Torregrosa, Robert R. P.; Mendis, Shehani N.; Davies, Alex; Tunge, Jon A.:
Palladium-Catalyzed Decarboxylative Benzylation of Acetylides and Enolates
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Li, Jing; Wang, Zhong-Xia:
Nickel-Catalyzed Transformation of Aryl 2-Pyridyl Ethers via Cleavage of the Carbon–Oxygen Bond: Synthesis of Mono-α-arylated Ketones
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De, Pinaki Bhusan; Pradhan, Sourav; Shah, Tariq A.; Punniyamurthy, Tharmalingam:
Iodine-Mediated Intramolecular C–H Amination of Benzimidazoles: A Metal-Free Route to Dihydroimidazobenzimidazoles
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Guan, Weiye; Liao, Jennie; Watson, Mary P.:
Vinylation of Benzylic Amines via C–N Bond Functionalization of Benzylic Pyridinium Salts
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Yin, Zhiping; Power, Dennis J.; Wang, Zechao; Stewart, Scott G.; Wu, Xiao-Feng:
Synthesis of 1,3,4-Oxadiazoles via Annulation of Hydrazides and Benzene-1,3,5-triyl Triformate under Metal-Free Conditions
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Issue 15/2018
Special Topic Cover Page
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Zhang, Qi; Raveendra Babu, Kaki; Huang, Zhouliang; Song, Jinna; Bi, Xihe:
Visible-Light-Induced Radical Polynitration of Arylboronic Acids: Synthesis of Polynitrophenols
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Wu, Kui; Fang, Cheng; Kaur, Sarbjeet; Liu, Peng; Wang, Ting:
Methylene Blue-Catalyzed Oxidative Cleavage of N-Carbonylated Indoles
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Wang, Guang-Zu; Shang, Rui; Fu, Yao:
Irradiation-Induced Palladium-Catalyzed Direct C–H Alkylation of Heteroarenes with Tertiary and Secondary Alkyl Bromides
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Hamsath, Akil; Galloway, Jordan D.; Baxter, Ryan D.:
Quinone C–H Alkylations via Oxidative Radical Processes
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Li, Longji; Yang, Qi; Jia, Zongbin; Luo, Sanzhong:
Organocatalytic Electrochemical C–H Lactonization of Aromatic Carboxylic Acids
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Levin, Vitalij V.; Agababyan, Daniil P.; Struchkova, Marina I.; Dilman, Alexander D.:
Dimerization of Benzyl and Allyl Halides via Photoredox-Mediated Disproportionation of Organozinc Reagents
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Manick, Anne-Doriane; Tanaka, Hirotaka; Oisaki, Kounosuke; Kanai, Motomu:
Organophotoredox/Copper Hybrid Catalysis for Regioselective Allylic Aminodecarboxylation of β,γ-Unsaturated Carboxylic Acids
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Egami, Hiromichi; Ito, Yuta; Ide, Takafumi; Masuda, Shuya; Hamashima, Yoshitaka:
Simple Photo-Induced Trifluoromethylation of Aromatic Rings
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Gharpure, Santosh J.; Niranjana, P.; Porwal, Suheel K.:
Cascade Radical Cyclization to Vinylogous Carbonates/Carbamates for the Synthesis of Oxa- and Aza-Angular Triquinanes: Diastereoselectivity Depends on the Ring Size of Radical Precursor
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Li, Cheng-Kun; Zhang, Dong-Liang; Olamiji, Ogundipe Olukayode; Zhang, Pei-Zhi; Shoberu, Adedamola; Zou, Jian-Ping; Zhang, Wei:
Mn(OAc)
3
-Mediated Regioselective Radical Alkoxycarbonylation of Indoles, Pyrimidinones, and Pyridinones
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Deng, Weili; Li, Yajun; Li, You-Gui; Bao, Hongli:
Iron-Catalyzed Carboiodination of Alkynes
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Zhao, Xinxin; Chen, Ming; Huang, Binbin; Yang, Chao; Gao, Yuan; Xia, Wujiong:
Photoinduced Cross-Coupling of Amines with 1,2-Diiodobenzene and Its Application in the Synthesis of Carbazoles
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Luo, Kai; Zhang, Ling; Wei, Kai; Yang, Wen-Chao; Wu, Lei:
Latent Radical Cleavage of α-Allenylic C–O Bonds: Potassium Persulfate Mediated Thiolation of Allenylphosphine Oxides
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Mei, Chong; Hu, Yixin; Lu, Wenjun:
Visible-Light-Driven Oxidation of
N
-Alkylamides to Imides Using Oxone/H
2
O and Catalytic KBr
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Das, Dipendu; Khan, Hina P. A.; Chakraborty, Tushar Kanti:
Ti(III)-Mediated Radical-Induced Approach to a Bicyclic δ-Lactone with a Bridgehead β-Hydroxy Group
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Fukuyama, Takahide; Bando, Takanobu; Ryu, Ilhyong:
Electron-Transfer-Induced Intramolecular Heck Carbonylation Reactions Leading to Benzolactones and Benzolactams
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Baguia, Hajar; Deldaele, Christopher; Romero, Eugénie; Michelet, Bastien; Evano, Gwilherm:
Copper-Catalyzed Photoinduced Radical Domino Cyclization of Ynamides and Cyanamides: A Unified Entry to Rosettacin, Luotonin A, and Deoxyvasicinone
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Issue 21/2017
Special Topic Cover Page
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Takenouchi, Yuta; Ito, Hajime:
Copper(I)-Catalyzed Boryl Substitution of Allyl Aminals: Selective Synthesis of Linear γ-Aminoallylboronates
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Miura, Wataru; Hirano, Koji; Miura, Masahiro:
Iridium-Catalyzed Site-Selective C–H Borylation of 2-Pyridones
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Jang, Won Jun; Han, Jung Tae; Yun, Jaesook:
NHC-Copper-Catalyzed Tandem Hydrocupration and Allylation of Alkenyl Boronates
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Pinet, Sandra; Liautard, Virginie; Debiais, Mégane; Pucheault, Mathieu:
Radical Metal-Free Borylation of Aryl Iodides
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Saito, Hayate; Nogi, Keisuke; Yorimitsu, Hideki:
Palladium-Catalyzed Double Borylation of Diaryl Sulfoxides with Diboron
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Farre, Albert; Briggs, Rachel; Pubill-Ulldemolins, Cristina; Bonet, Amadeu:
Developing a Bench-Scale Green Diboration Reaction toward Industrial Application
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Issue 20/2017
Special Topic Cover Page
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Couly, Florence; Dubouilh-Benard, Carole; Besson, Thierry; Fruit, Corinne:
Late-Stage C–H Arylation of Thiazolo[5,4-
f
]quinazolin-9(8
H
)-one Backbone: Synthesis of an Array of Potential Kinase Inhibitors
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Sabat, Nazarii; Smoleń, Sabina; Nauš, Petr; Perlíková, Pavla; Cebová, Magdaléna; Poštová Slavětínská, Lenka; Hocek, Michal:
Synthesis of 2,6-Substituted 7-(Het)aryl-7-deazapurine Nucleobases (2,4-Disubstituted 5-(Het)aryl-pyrrolo[2,3-
d
]pyrimidines)
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Skonieczny, Kamil; Jaźwiński, Jarosław; Gryko, Daniel T.:
The Synthesis of Imidazo[1,2-
f
]phenanthridines, Phenanthro-[9,10-
d
]imidazoles, and Phenanthro[9′,10′:4,5]imidazo[1,2-
f
]-phenanthridines via Intramolecular Oxidative Aromatic Coupling
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Yu, Zhao; Bo, Tang; Aiying, Guan; Weiwei, Wang; Zhenhua, Zhang; Mingan, Wang:
Synthesis and Fungicidal Activity of (
E
)-5-[1-(4-Phenyl-2-oxo-1-oxaspiro[4.5]dec-3-en-3-yl)ethylidene]-2-aminoimidazolin-4-one Derivatives
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Tokumaru, Kazuyuki; Bera, Kalisankar; Johnston, Jeffrey N.:
1,3,4-Oxadiazole and Heteroaromatic-Fused 1,2,4-Triazole Synthesis Using Diverted Umpolung Amide Synthesis
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Lessi, Marco; Panzetta, Gianmarco; Marianetti, Giulia; Bellina, Fabio:
Improved Synthesis of Symmetrical 2,5-Diarylimidazoles by One-Pot Palladium-Catalyzed Direct Arylation Tailored on the Electronic Features of the Aryl Halide
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Zhang, Xiaojuan; Han, Xiuling; Hu, Zhiyong; Lu, Xiyan:
Synthesis of Substituted Piperidines via Cationic Palladium(II)-Catalyzed Reductive Coupling of
N
-Tosyl-Tethered Alkynones
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Shang, Xiao-Jie; Liu, Zhong-Quan:
A Catalyzed Aerobic Intramolecular C–O Bond Formation: Facile Access to Ring-Fused Dihydrobenzoxazine Derivatives
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Issue 18/2017
Special Topic Cover Page
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Abe, Takumi; Haruyama, Tomohiro; Yamada, Koji:
C4 Pictet–Spengler Reactions for the Synthesis of Core Structures in Hyrtiazepine Alkaloids
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Pertschi, Romain; Miaskiewicz, Solène; Weibel, Jean-Marc; Pale, Patrick; Blanc, Aurélien:
Gold(I)-Catalyzed Cascade: Synthesis of 2,5-Disubstituted Pyrroles from
N
-Sulfonyl-2-(1-ethoxypropargyl)azetidines through Cyclization/Nucleophilic Substitution/Elimination
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Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna:
2-(Aminomethyl)-3-arylindoles from 3-(
o
-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach
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Zheng, Min; Chen, Kai; Zhu, Shifa:
One-Pot Synthesis of Indole Derivatives from the Reaction of Nitroalkynes and Alkynes via a Mercury-Carbene Intermediate
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Shimizu, Maki; Hayama, Noboru; Kimachi, Tetsutaro; Inamoto, Kiyofumi:
Copper-Catalyzed Intramolecular C–H Amination: A New Entry to Substituted Xanthine Derivatives
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Opsomer, Tomas; Thomas, Joice; Dehaen, Wim:
Chemoselectivity in the Synthesis of 1,2,3-Triazoles from Enolizable Ketones, Primary Alkylamines, and 4-Nitrophenyl Azide
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Fujita, Shoji; Shibuya, Masatoshi; Yamamoto, Yoshihiko:
Intramolecular Hydroalkoxylation/Reduction and Hydroamination/Reduction of Unactivated Alkynes Using a Silane–Iodine Catalytic System
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Paul, Kartick; Jalal, Swapnadeep; Kundal, Sandip; Chakraborty, Baitan; Jana, Umasish:
Iron-Catalyzed Intramolecular Alkyne–Carbonyl Metathesis: A New Cyclization Strategy for the Synthesis of Benzocarbazole and Azepino[1,2-
a
]indole Derivatives
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Li, Xue-Fei; Lin, Jin-Shun; Liu, Xin-Yuan:
Catalytic Radical Intramolecular Aminoperfluoroalkylation and Aminodifluoromethylation of Unactivated Alkenes with Fluoroalkylsulfonyl Chlorides
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Mullapudi, Venkannababu; Bhogade, Ravindra B.; Deshpande, Mukund V.; Ramana, Chepuri V.:
Phenol Oxidative Dearomatization of Modified Nucleoside Templates: A Simple Access to the C7-Spiroannulated Octosyl Acid Framework
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Ghosh, Arun K.; Tomaine, Anthony J.; Cantwell, Kelsey E.:
Lewis Acid Mediated Cyclizations: Diastereoselective Synthesis of Six- to Eight-Membered Substituted Cyclic Ethers
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Lee, Sang Eun; Lee, Seong Jong; Cheon, Cheol-Hong:
Concise Total Syntheses of Paullone and Kenpaullone via Cyanide-Catalyzed Intramolecular Imino-Stetter Reaction
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Triandafillidi, Ierasia; Sideri, Ioanna K.; Tzaras, Dimitrios Ioannis; Spiliopoulou, Nikoleta; Kokotos, Christoforos G.:
Green Organocatalytic Synthesis of Dihydrobenzofurans by Oxidation–Cyclization of Allylphenols
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Nayak, Sanatan; Prabagar, B.; Ghosh, Nayan; Mallick, Rajendra K.; Sahoo, Akhila K.:
Ag(I)-Catalyzed Cycloisomerization and Cyclization of Ketene Aminals: Construction of Azepine and 1,2-Dihydropyridine Derivatives
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Nagamoto, Midori; Nishimura, Takahiro; Yorimitsu, Hideki:
Iridium-Catalyzed Intramolecular Oxidative Cyclization of Alkenyl Amides and Alkenoic Acids
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Li, Dianjun; Li, Ying; Yu, Wei:
tert
-Butyl Hypochlorite Induced Cyclization of Ethyl 2-(
N
-Arylcarbamoyl)-2-iminoacetates
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Li, Jie; Xiao, Jun-An; Zhao, Shu-Juan; Xiang, Hao-Yue; Yang, Hua:
Facile Construction of Pyrrolo[1,2-
a
]indolenine Scaffold via Diastereoselective [3+2] Annulation of Donor–Acceptor Cyclopropane with Indolenine
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Issue 17/2017
Special Topic Cover Page
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Hammann, Jeffrey M.; Hofmayer, Maximilian S.; Lutter, Ferdinand H.; Thomas, Lucie; Knochel, Paul:
Recent Advances in Cobalt-Catalyzed Csp
2
and Csp
3
Cross-Couplings
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Ferrand, Laura; Lyu, Ye; Rivera-Hernández, Alejandro; Fallon, Brendan J.; Amatore, Muriel; Aubert, Corinne; Petit, Marc:
Hydroboration and Diboration of Internal Alkynes Catalyzed by a Well-Defined Low-Valent Cobalt Catalyst
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Joshi, Hemant; Ghosh, Subrata K.; Gladysz, John A.:
Enantioselective Additions of Stabilized Carbanions to Imines Generated from α-Amido Sulfones By Using Lipophilic Salts of Chiral Tris(1,2-diphenylethylenediamine) Cobalt(III) Trications as Hydrogen Bond Donor Catalysts
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Suo, Jian-Feng; Zhao, Xue-Mei; Zhang, Kai-Xin; Zhou, Sheng-Li; Niu, Jun-Long; Song, Mao-Ping:
Cobalt-Catalyzed Perfluoroalkylation of Quinoline Amides at the C5 Position
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Hofmayer, Maximilian S.; Hammann, Jeffrey M.; Lutter, Ferdinand H.; Knochel, Paul:
Large-Scale Cobalt-Catalyzed Cross-Couplings of Functionalized Bench-Stable Arylzinc Pivalates with (Hetero)Aryl and Alkenyl Halides
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Xu, Kun; Tan, Zhoumei; Zhang, Haonan; Zhang, Sheng:
Cobalt-Catalyzed Monoselective
ortho
-C–H Ethylation of Carboxamides with Triethylaluminum
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Kalsi, Deepti; Barsu, Nagaraju; Dahiya, Pardeep; Sundararaju, Basker:
C–H and N–H Bond Annulation of Benzamides with Isonitriles Catalyzed by Cobalt(III)
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Cabré, Albert; Verdaguer, Xavier; Riera, Antoni:
Ethylene Glycol Assisted Intermolecular Pauson–Khand Reaction
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Jamieson, Megan L.; Brant, Nicola Z.; Brimble, Margaret A.; Furkert, Daniel P.:
Remarkable Influence of Cobalt Catalysis on Epoxide Ring-Opening with Sulfoxonium Ylides
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Midya, Siba P.; Mondal, Akash; Begum, Ayesha; Balaraman, Ekambaram:
A Simple Cobalt(II) Chloride Catalyzed
N
-Alkylation of Amines with Alcohols
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Issue 16/2017
Special Topic Cover Page
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Watabe, Yota; Kanazawa, Kohei; Fujita, Takeshi; Ichikawa, Junji:
Nickel-Catalyzed Hydroalkenylation of Alkynes through C–F Bond Activation: Synthesis of 2-Fluoro-1,3-dienes
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Xiao, Jian; Wang, Ya-Wen; Peng, Yu:
Nickel-Promoted Reductive Cyclization Cascade: A Short Synthesis of a New Aromatic Strigolactone Analogue
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PDF (740 kb)
Barday, Manuel; Janot, Christopher; Clare, Daniel; Carr-Knox, Caitlin; Higginson, Bradley; Ho, Kelvin Y. T.; Aïssa, Christophe:
On the Regioselectivity of the Nickel-Catalyzed Insertion of Alkynes into the Carbon–Carbon Bond of Oxetan-3-one
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Sumida, Yuto; Sumida, Tomoe; Hosoya, Takamitsu:
Nickel-Catalyzed Reductive Cross-Coupling of Aryl Triflates and Nonaflates with Alkyl Iodides
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Shi, Shicheng; Szostak, Michal:
Nickel-Catalyzed Negishi Cross-Coupling of
N
-Acylsuccinimides: Stable, Amide-Based, Twist-Controlled Acyl-Transfer Reagents via N–C Activation
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Issue 13/2017
Special Topic Cover Page
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Parmeggiani, Camilla; Matassini, Camilla; Cardona, Francesca; Goti, Andrea:
On the Oxidation of Hydroxylamines with
o
-Iodoxybenzoic Acid (IBX)
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Muñiz, Kilian; Fra, Laura:
Enantioselective 4-Hydroxylation of Phenols under Chiral Organoiodine(I/III) Catalysis
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Kiyokawa, Kensuke; Takemoto, Kenta; Yahata, Shunsuke; Kojima, Takumi; Minakata, Satoshi:
Oxidative Cyclization of β,γ-Unsaturated Carboxylic Acids Using Hypervalent Iodine Reagents: An Efficient Synthesis of 4-Substituted Furan-2-ones
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Fujita, Morifumi; Lee, Hee Jin; Ichihara, Chisaki; Sugimura, Takashi:
E
/
Z
-Selectivity Controlled by Participation of Internal Oxy Group During Electrophilic Substitution of Alk-1-enylboronate with Bis(2,4,6-trimethylpyridine)iodonium Salt
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Li, Guangchen; Zhang-Negrerie, Daisy; Du, Yunfei:
Synthesis of N-Substituted 2-Amino-3,4-diiodofurans from Allenes via NIS-Mediated Intramolecular Electrophilic Iodocyclization
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Dagenais, Robin; Lauriers, Antoine Jobin-Des; Legault, Claude Y.:
Iodine(III)-Mediated Oxidative Hydrolysis of Haloalkenes: Investigation of the Effect of Iodine(III) Reagents
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Issue 17/2016
Shaw, Subrata; White, James D.:
Asymmetric Catalysis with Iron–Salen Complexes
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Liu, Cheng-Yuan; Chen, Ying-Ho; Chen, Chih-Hao; Yu, Ming-Shiuan; Tsai, Fu-Yu; Ong, Tiow-Gan:
Selective C(8)–H Activation of Imidazopyridines Mediated by Cooperative Nickel–Aluminum Catalysis
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Kumar, Ravindra; Tamai, Eri; Ohnishi, Akira; Nishimura, Akira; Hoshimoto, Yoichi; Ohashi, Masato; Ogoshi, Sensuke:
Nickel-Catalyzed Enantioselective Synthesis of Cyclobutenes via [2+2] Cycloaddition of α,β-Unsaturated Carbonyls with 1,3-Enynes
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Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil:
An Indefinitely Air-Stable σ-Ni
II
Precatalyst for Quantitative Cross-Coupling of Unreactive Aryl Halides and Mesylates with Aryl Neopentylglycolboronates
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Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil:
Ni
II
Cl(1-Naphthyl)(PCy
3
)
2
, An Air-Stable σ-Ni
II
Precatalyst for Quantitative Cross-Coupling of Aryl C–O Electrophiles with Aryl Neopentylglycolboronates
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Moragas, Toni; Martin, Ruben:
Nickel-Catalyzed Reductive Carboxylation of Cyclopropyl Motifs with Carbon Dioxide
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Sugiyama, Yu-ki; Heigozono, Shiori; Tamura, Kazuhiro; Okamoto, Sentaro:
Iron-Catalyzed Reductive Metalation–Allylation and Metalative Cyclization of 2,3-Disubstituted Oxetanes and Their Stereoselectivity
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Zhang, Qingchen; Wang, Xuan; Qian, Qun; Gong, Hegui:
Nickel-Catalyzed Reductive Cross-Coupling of Benzyl Halides with Aryl Halides
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Xi, Tuo; Chen, Xu; Zhang, Heyi; Lu, Zhan:
Reductive Cyclization of 1,6- and 1,7-Enynes Catalyzed by Iron Complexes
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Issue 16/2016
Cai, Pin-Wen; You, Zhi-Hao; Xie, Liang-Hui; Tan, Rui; Tong, Zhi-Ping; Liu, Yan-Kai:
The Attractive Application of Lactol Chemistry: From Racemic Lactol to Natural Product Skeleton
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PDF (891 kb)
Su, Lin; Xu, Ming-Hua:
Asymmetric Reformatsky-Type Reaction of Isatin-Derived
N
-Sulfinyl Ketimines: Efficient and Practical Synthesis of Enantiopure Chiral 2-Oxoindolinyl-β
3,3
-Amino Esters
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PDF (906 kb)
Gao, Xing; Han, Jianwei; Wang, Limin:
Chiral Iminophosphorane Organocatalyzed Asymmetric Sulfenylation of 3-Substituted Oxindoles: Substrate-Interrelated Enantioselectivities
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Nishimura, Takahiro; Nagai, Tomotaka; Takechi, Ryosuke; Ebe, Yusuke:
Rhodium-Catalyzed Enantioselective Addition of Tricyclopropylboroxin to
N
-Sulfonylimines
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Chen, Shi; Mondal, Mukulesh; Ibrahim, Ahmad A.; Wheeler, Kraig A.; Kerrigan, Nessan J.:
Asymmetric Synthesis of Dipropionate Derivatives through Catalytic Hydrogenation of Enantioenriched
E
-Ketene Heterodimers
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Sun, Shutao; Liu, Lei:
Catalytic Enantioselective Alkynylation of Tetrahydroisoquinoline-Based
N
-Acyl Hemiaminals
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Feng, Yangyang; Huang, Ruofeng; Hu, Liangzhen; Xiong, Yan; Coeffard, Vincent:
Chiral
C
2
-Symmetric Iodoarene-Catalyzed Asymmetric α-Oxidation of β-Keto Esters
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Berti, Francesco; Favero, Lucilla; Pineschi, Mauro:
Asymmetric Synthesis of Methylphenidate and Quinolizidinones by Addition of Aldehydes to Piperidine-Based Conjugated
N
-Acyliminium Ions
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Dai, Wen; Mi, Yuan; Lv, Ying; Shang, Sensen; Li, Guosong; Chen, Guangwen; Gao, Shuang:
Development of a Continuous-Flow Microreactor for Asymmetric Epoxidation of Electron-Deficient Olefins
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Salomó, Ernest; Orgué, Sílvia; Riera, Antoni; Verdaguer, Xavier:
Efficient Preparation of (
S
)- and (
R
)-
tert
-Butylmethylphosphine–Borane: A Novel Entry to Important P-Stereogenic Ligands
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Shibata, Takanori; Fukai, Miku; Sekine, Ryosuke; Hazra, Madhurima; Kanyiva, Kyalo Stephen:
Enantioselective Synthesis of Planar-Chiral 1,
n
-Dioxa[
n
]paracyclophane-Based Phosphites and Their Application as Chiral Ligands
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Vishwanath, Manjunatha; Prakash, Muthuraj; Vinayagam, Poopathy; Kesavan, Venkitasamy:
Construction of Polycyclic Fused Pyrrolidines with Three Contiguous Stereocenters via Michael Addition of Vinylmalononitriles to Nitrostyrenes Using
l
-Proline-Derived Thiourea
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Issue 12/2016
Wildermuth, Raphael; Speck, Klaus; Magauer, Thomas:
Gold(I)-Catalyzed Enyne Cyclizations: Studies Toward the Total Synthesis of (+)-Aureol
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Shi, Shicheng; Lalancette, Roger; Szostak, Michal:
Cyclization of Imides to 2-Azabicycles via Aminoketyl Radicals by Using Samarium(II) Iodide–Water: Reaction Development, Synthetic Scope, and Mechanistic Studies
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Sugimoto, Kenji; Hoshiba, Yuya; Tsuge, Kiyoshi; Matsuya, Yuji:
Synthesis of Substituted Pyrrolo[2,1-
a
]isoquinolines by Gold-Catalyzed Domino Cyclization of Alkynyl Iminoesters
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Shirke, Rajendra P.; Reddy, Virsinha; Anand, R. Vijaya; Ramasastry, S. S. V.:
Furans to Benzofurans: Intramolecular Cross-Benzoin Reactions Catalysed by N-Heterocyclic Carbenes
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Gandeepan, Parthasarathy; Rajamalli, Pachaiyappan; Cheng, Chien-Hong:
Palladium-Catalyzed C–H Activation and Cyclization of Anilides with 2-Iodoacetates and 2-Iodobenzoates: An Efficient Method toward Oxindoles and Phenanthridones
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Malkina, Anastasiya G.; Stepanov, Anton V.; Sobenina, Lyubov N.; Shemyakina, Olesya A.; Ushakov, Igor A.; Smirnov, Vladimir I.; Trofimov, Boris A.:
Organocatalyzed Microwave-Assisted Competing Cyclization of Cyanopropargylic Alcohols with Carboxylic Acids: 4-Cyano-3(2
H
)-furanones versus 4-Cyano-[(
Z
)-3-cyanomethylene]-2,3-dihydrofurans
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Nambu, Hisanori; Ono, Naoki; Yakura, Takayuki:
Acid-Catalyzed Ring-Opening Cyclization of Spirocyclopropanes for the Construction of a 2-Arylbenzofuran Skeleton: Total Synthesis of Cuspidan B
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Parker, Patrick D.; Pierce, Joshua G.:
Synthesis of 1,2,4-Oxadiazoles via DDQ-Mediated Oxidative Cyclization of Amidoximes
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Cavitt, Marchello A.; France, Stefan:
Aluminum(III)-Catalyzed, Formal Homo-Nazarov-Type Ring-Opening Cyclizations toward the Synthesis of Functionalized Tetrahydroindolizines
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Ren, Zhi-Hui; Zhao, Mi-Na; Yi, Yukun; Wang, Yao-Yu; Guan, Zheng-Hui:
Copper-Catalyzed Aerobic Oxidative Cyclization of Ketoxime Acetates with Pyridines for the Synthesis of Imidazo[1,2-
a
]pyridines
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Morita, Nobuyoshi; Mashiko, Rie; Hakuta, Dai; Eguchi, Daisuke; Ban, Shintaro; Hashimoto, Yoshimitsu; Okamoto, Iwao; Tamura, Osamu:
Gold-Catalyzed Dimeric Cyclization of Isoeugenol and Related 1-Phenylpropenes in Ionic Liquid: Environmentally Friendly and Stereoselective Synthesis of 1,2,3-Trisubstituted 2,3-Dihydro-1
H
-indenes
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Yu, Mangfei; Zhang, Qian; Wang, Jia; Huang, Peng; Yan, Pengfei; Zhang, Rui; Dong, Dewen:
Triflic Anhydride Mediated Ring-Opening/Recyclization Reaction of α-Carbamoyl α-Oximyl Cyclopropanes with DMF: Synthetic Route to 5-Aminoisoxazoles
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Issue 11/2016
Li, Zhilong; Tong, Rongbiao:
Asymmetric Total Syntheses of the
trans
-2-Aryl-6-alkyltetrahydropyrans Diospongin B and Parvistones D and E from a Common Precursor
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Kousara, Mohammad; Bideau, Franck Le; Ibrahim, Rama; Ferry, Angélique; Venot, Pierre-Etienne; Dejean, Camille; Raingeaud, Joël; Dubois, Joëlle; Retailleau, Pascal; Dumas, Françoise:
Suberosanes as Potential Antitumor Agents: First Enantioselective Total Synthesis of (1
S
)-Suberosanone and Configurational Assignment of Suberosenol A
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Nakayama, Yasuaki; Maeda, Yuichiro; Hama, Naoto; Sato, Takaaki; Chida, Noritaka:
Total Synthesis of (–)-Stemoamide by Sequential Overman/Claisen Rearrangement
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García-Ruiz, Cristina; Cheng-Sánchez, Iván; Sarabia, Francisco:
Synthesis of (–)- and (+)-Gummiferol via Asymmetric Synthesis of Glycidic Amides
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Konda, Saidulu; Khatravath, Mahender; Mallurwar, Naveen Kumar; Rao, Pallavi; Sripelly, Shivashankar; Iqbal, Javed; Arya, Prabhat:
Stereoselective Synthesis of the C27–C35 Eribulin Fragment and Its Utilization in Building Structurally Diverse Macrocycles
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Ye, Jian-Liang; Liu, Yang; Zhang, Yu-Feng; Yang, Zhi-Ping; Huang, Pei-Qiang:
Studies on the Second-Generation Approach to Loline Alkaloids: Synthesis of
N
-Bus-norloline through
N
-
tert
-Butanesulfinyl Imine Based Asymmetric Vinylogous Mannich Reaction
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Yang, Xiaoyu; Yu, Biao:
Synthesis of Landomycin D: Studies on the Saccharide Assembly
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Hunter, Thomas J.; Wang, Yanping; Zheng, Jiamin; O’Doherty, George A.:
Asymmetric Iterative Hydration of Polyene Strategy to Cryptocaryols A and B
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Issue 19/2015
Liu, Le; Zhang-Negrerie, Daisy; Du, Yunfei; Zhao, Kang:
Hypervalent Iodine Mediated C–C Double Bond Activation: A Cascade Access to α-Keto Diacetates from Readily Available Cinnamic Acids
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Sun, Gui-Jun; Wang, Yong; Kang, Qiang:
Palladium-Catalyzed Allylic Amination of Homoallylic Alcohols with Amines via Carbon–Carbon Bond Cleavage
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Okuma, Kentaro; Horigami, Kenta; Nagahora, Noriyoshi; Shioji, Kosei:
Enantioselective Synthesis of 4,4′-Biaryl-BINOLs from Arynes and β-Diketones
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Aoyama, Tadashi; Hayakawa, Mamiko; Kubota, Sho; Ogawa, Sumire; Nakajima, Erika; Mitsuyama, Emi; Iwabuchi, Taku; Kaneko, Haruki; Obara, Rina; Takido, Toshio; Kodomari, Mitsuo; Ouchi, Akihiko:
Simple Method for sp
2
–sp
3
and sp
3
–sp
3
Carbon–Carbon Bond Activation in 2-Substituted 1,3-Diketones
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Choi, Jeongae; Jung, Hyunuk; Yeo, Jeong-Eun; Koo, Sangho:
Synthesis of Tribenzotropone by Ring Expansion of Phenanthrene-9,10-dione
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Shadrin, Ivan A.; Rzhevskii, Sergey A.; Rybakov, Victor B.; Babaev, Eugene V.:
Sonogashira Reaction of the Indolizine Ring
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Parida, Amarchand; Sharique, Mohd.; Kakde, Badrinath N.; Ghosh, Santanu; Bisai, Alakesh:
Efficient Synthesis of 3-Alkynyl-2-(hydroxymethyl)cyclohex-2-en-1-ones by a Stork–Danheiser Sequence from Vinylogous Esters and Terminal Alkynes
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Ou, Yang; Qin, Chong; Song, Song; Jiao, Ning:
An Iron-Catalyzed Direct Approach to Amides from Benzyl Azides via C–C Bond Cleavage
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Issue 18/2015
Luo, Guo-Ying; Wu, Hao; Tang, Yu; Li, Hui; Yeom, Hyun-Suk; Yang, Ka; Hsung, Richard P.:
A Total Synthesis of (±)-Rhododaurichromanic Acid A via an Oxa-[3+3] Annulation of Resorcinols
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Kumar, Raju Suresh; Almansour, Abdulrahman I.; Arumugam, Natarajan; Menéndez, J. Carlos; Osman, Hasnah; Kumar, Raju Ranjith:
Dipolar Cycloaddition-Based Multicomponent Reactions in Ionic Liquids: A Green, Fully Stereoselective Synthesis of Novel Polycyclic Cage Systems with the Generation of Two New Azaheterocyclic Rings
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Zhao, Yating; Huang, Binbin; Yang, Chao; Li, Bing; Xia, Wujiong:
Metal-Free [3+2] Oxidative Coupling of Phenols with Alkenes: Synthesis of Dihydrobenzofurans
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Cserép, Gergely B.; Demeter, Orsolya; Bätzner, Effi; Kállay, Mihály; Wagenknecht, Hans-Achim; Kele, Péter:
Synthesis and Evaluation of Nicotinic Acid Derived Tetrazines for Bioorthogonal Labeling
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Islam, Kobirul; Das, Deb K.; Akram, Ejaz; Khan, Abu T.:
Exploration of C5–C6-Unsubstituted 1,4-Dihydropyridines for the Construction of
exo
-Hexahydro-1
H
-chromeno[3,4-
h
][1,6]naphthyridine-3-carboxylates Using a Stereoselective Povarov Reaction
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Olson, Christopher A.; Shaner, Courtnay E.; Roche, Sydney C.; Ferrence, Gregory M.; Mitchell, T. Andrew:
Hexahydro-1
H
-Isoindolinone-Like Scaffolds from Electronically Deactivated and Sterically Hindered Dienes: Synthesis in the Context of Muironolide A
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Högermeier, Jens; Trawny, Daniel; Zimmer, Reinhold; Reissig, Hans-Ulrich:
Diels–Alder Reactions of 1,3-Dienes Incorporated into 8-Oxa- and 8-Thiabicyclo[3.2.1]octane Skeletons: A Convenient Access to Complex Tri- and Tetracyclic Compounds
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Lopchuk, Justin M.; Song, Mia; Butler, Blythe; Gribble, Gordon W.:
Synthesis of Heteroaryl-Substituted Pyrroles via the 1,3-Dipolar Cycloaddition of Unsymmetrical Münchnones and Nitrovinylheterocycles
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Ribeiro Laia, Fernanda M.; Pinho e Melo, Teresa M. V. D.:
Synthesis and Reactivity of Aziridines with Internal Dipolarophiles: An Approach to 1,4-Dihydrochromeno[4,3-
b
]pyrroles and 3-Methylenechromano[4,3-
b
]pyrroles
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Miller, Daniel K.; Bailey, Christopher A.; Sammelson, Robert E.:
Synthesis of Isoxazolines and Isoxazoles Inspired by Fipronil
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Pop, Lidia; Golban, Mirabela Ligia; Hădade, Niculina D.; Socaci, Crina; Grosu, Ion:
CuAAC Synthesis of Tetragonal Building Blocks Decorated with Nucleobases
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Kratzer, Philipp; Gerster, Holger; Maas, Gerhard:
Cycloaddition Reactions of Propyne Iminium Salts and Enol Ethers
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Yamaoka, Yousuke; Taniguchi, Marie; Yamada, Ken-ichi; Takasu, Kiyosei:
Asymmetric Total Synthesis of Tylophorine through a Formal [2+2] Cycloaddition Followed by Migrative Ring Opening of a Cyclobutane
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Seck, Insa; Fall, Alioune; Lago, Carmen; Sène, Massène; Gaye, Mohamed; Seck, Matar; Gómez, Generosa; Fall, Yagamare:
Synthesis of a Cholesterol Side-Chain Triazole Analogue via ‘Click’ Chemistry
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Issue 17/2015
Dobrydnev, Alexey V.; Popova, Maria V.; Saffon-Merceron, Nathalie; Listunov, Dymytrii; Volovenko, Yulian M.:
Synthesis of the First Representatives of Spiro-1λ
6
-isothiazolidine-1,1,4-triones
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Zhang, Shuang; Hu, Xiu-Qin; Wang, Zhu-Yin; Xu, Peng-Fei:
Reactions of Sulfonium Salts with 2,3-Dioxopyrrolidine Derivatives: A Concise Synthesis of Spirocyclopropane
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Peng, Jing; Ran, Guang-Yao; Du, Wei; Chen, Ying-Chun:
Tertiary-Amine-Catalyzed Asymmetric [3+2] Annulations of Morita–Baylis–Hillman Carbonates of Isatins with Nitroolefins to Construct Spirooxindoles
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Xiao, Fenfen; Zhang, Qing; Wang, Yunxia; Hu, Xiangdong:
Synthetic Studies toward Bi-linderone Lead To Unexpected 6π-Electrocyclization Reactions: A Facile Construction of Highly Congested Spiro Compounds
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Cormier, Morgan; Chardon, Aurélien; Blanchet, Jérôme; Rouden, Jacques; Maddaluno, Jacques; De Paolis, Michaël:
An Organocatalytic Access to Spiro[4.5]decanes and Spiro[4.6]undecanes Containing Aminolactones and 3-Aminopyrrolidines
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Issue 16/2015
Philipps, Arne R.; Fritze, Lars; Erdmann, Nico; Enders, Dieter:
An Asymmetric Organocatalytic Quadruple Domino Reaction Employing a Vinylogous Friedel–Crafts/Michael/Michael/Aldol Condensation Sequence
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PDF (257 kb)
Garbarino, Silvia; Protti, Stefano; Basso, Andrea:
Toward a Green Atom Economy: Development of a Sustainable Multicomponent Reaction
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Firth, James D.; Zhang, Rong; Morgentin, Rémy; Guilleux, Rachel; Kalliokoski, Tuomo; Warriner, Stuart; Foster, Richard; Marsden, Stephen P.; Nelson, Adam:
Exploitation of the Ugi–Joullié Reaction in the Synthesis of Libraries of Drug-Like Bicyclic Hydantoins
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Neochoritis, Constantinos G.; Zhang, Ji; Dömling, Alexander:
Leuckart–Wallach Approach to Sugar Isocyanides and Its IMCRs
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Xu, Shibo; Su, Shikuan; Zhang, Huiting; Tian, Lumin; Liang, Pengcheng; Chen, Jiawen; Zhang, Yuan; Li, Chunju; Jia, Xueshun; Li, Jian:
Isocyanide-Based Multicomponent Reactions: Rapid Synthesis of a 5,5-Fused Bicyclic Skeleton from α,β-Unsaturated Ketones and Allenoates
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Neo, Ana G.; Castellano, Teresa G.; Marcos, Carlos F.:
Enol-Ugi Reaction of Hydroxycoumarins: Straightforward Synthesis of Amino Acid Derived Coumarin Enamines
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Carboni, Aude; Dagousset, Guillaume; Magnier, Emmanuel; Masson, Géraldine:
Three-Component Photoredox-Mediated Chloro-, Bromo-, or Iodotrifluoromethylation of Alkenes
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Qureshi, Zafar; Schlundt, Waldemar; Lautens, Mark:
Introduction of Hindered Electrophiles via C–H Functionalization in a Palladium-Catalyzed Multicomponent Domino Reaction
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Issue 15/2015
Du, Haiying; Rodriguez, Jean; Bugaut, Xavier; Constantieux, Thierry:
Michael Addition Initiated Substrate- or Catalyst-Controlled Chemodivergent Three-Component Construction of Fused and Bridged Polycyclic Heterocycles
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Vízcaíno-Milla, Pascuala; Sansano, José M.; Nájera, Carmen; Fiser, Béla; Gómez-Bengoa, Enrique:
Primary Amine–2-Aminopyrimidine Chiral Organocatalysts for the Enantioselective Conjugate Addition of Branched Aldehydes to Maleimides
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Fu, Niankai; Guo, Yinliang; Zhang, Long; Luo, Sanzhong:
Chiral Primary Amine Catalyzed Asymmetric Tandem Reduction–Michael Addition–Protonation Reaction between Alkylidene Meldrum’s Acid and α-Substituted Vinyl Ketones
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Rideau, Emeline; Mäsing, Florian; Fletcher, Stephen P.:
Asymmetric Conjugate Addition of Alkylzirconocenes to Cyclopent-4-ene-1,3-dione Monoacetals
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Tai, Hung-Che; Chavan, Arjun S.; Chuang, Shih-Ching:
Nucleophilic Conjugate 1,5-Addition of Gilman Reagents to (
E
)-Hex-2-en-4-ynedioates: An Access to β(γ′)-Substituted Muconates
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Roscales, Silvia; Sancho, Ainhoa; Csákÿ, Aurelio G.:
Metal-Free Conjugate Addition of Alkenylboronic Acids to Enedicarbonyl Compounds towards the Synthesis of Pyridazine Derivatives
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Peck, Cheryl L.; Calderone, Joseph A.; Santos, Webster L.:
Copper(II)-Catalyzed β-Borylation of Acetylenic Esters in Water
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Witte, Swjatoslaw N. R.; Voigt, Benjamin; Mahrwald, Rainer:
Amine-Catalyzed Cascade Reactions of Unprotected and Unactivated Carbohydrates: Direct Access to C-Glycosides
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Nishimura, Katsumi; Fukuyama, Naoshi; Yamashita, Mitsuaki; Sumiyoshi, Takaaki; Yamamoto, Yasutomo; Yamada, Ken-ichi; Tomioka, Kiyoshi:
Cyclic Model for the Asymmetric Conjugate Addition of Organolithiums with Enoates
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Sugiura, Masaharu; Ishikawa, Wakoto; Kuboyama, Yukinobu; Nakajima, Makoto:
Conjugate Addition of Diboron Catalyzed by
O
-Monoacyltartaric Acids
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Issue 17/2014
Mori, Yasuyuki; Mori, Takamichi; Onodera, Gen; Kimura, Masanari:
Nickel-Catalyzed Multicomponent Coupling of Alkyne, Buta-1,3-diene, and Dimethylzinc under Carbon Dioxide
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Strack, Martin; Metzler-Nolte, Nils; Albada, H. Bauke:
Copper-Free Cleavage-Sonogashira Conjugation of Silylacetylene Immobilized Peptides
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Ma, Wenbo; Ackermann, Lutz:
Silver-Mediated Alkyne Annulations by C–H/P–H Functionalizations: Step-Economical Access to Benzophospholes
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PDF (237 kb)
Park, Youngchul; Kang, Dongjin; Jeon, Woo Hyung; Ryu, Taekyu; Lee, Phil Ho:
Synthesis of Ethyl Arylpropiolates through Palladium-Catalyzed Cross-Coupling Reactions of Aryl Iodides with In Situ Generated Lithium Tetrakis(ethoxycarbonylethynyl)indates
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Issue 16/2014
Guo, Wei; Xia, Yuanzhi:
THF Solvent as a Proton Shuttle in the AuCl
3
-Catalyzed Cycloisomerization of a Bromoallenyl Ketone: A Mechanistic DFT Study
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Lee, Ji Hyung; Jeong, Wook; Rhee, Young Ho:
Unique Divergent Reactivity of Boc-Protected Homopropargylic Alkoxyalkylamines in the Gold(I)-Catalyzed Domino Catalytic Reactions: Application to the Formal Synthesis of (–)-Pseudodistomin B
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Liu, Meng-Qi; Zhou, Ai-Hua; Jiang, Shuang; Wang, Jia-Qi; Ye, Long-Wu:
Highly Diastereoselective Synthesis of Cyclopentenones via a One-Pot Gold Catalysis, Nazarov Cyclization and Alkylation Cascade
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Wei, Fang; Wang, Xianghua; Peng, Shasha; Jia, Qiuhui; Jiang, Chao; Liu, Shili; Xu, Zhenghu:
Direct Gold-Catalyzed Regioselective Tetrafunctionalization of Nonactivated Alkynes
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Issue 14/2014
Zhou, Mingxin; Song, Qiuling:
Synthesis of α-Ketoamides from Aryl Methyl Ketones and
N
,
N
-Dimethylformamide via Copper-Catalyzed Aerobic Oxidative Coupling
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PDF (193 kb)
Belhomme, Marie-Charlotte; Dru, Delphine; Xiong, Heng-Ying; Cahard, Dominique; Besset, Tatiana; Poisson, Thomas; Pannecoucke, Xavier:
Copper-Mediated Direct Functionalization of Unsaturated C–C Bonds with Ethyl Bromo(difluoro)acetate: A Straightforward Access to Highly Valuable Difluoromethylated Alkenes
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Székely, Anna; Sinai, Ádám; Tóth, Edina B.; Novák, Zoltán:
Utilization of a Copper on Iron Catalyst for the Synthesis of Biaryl Systems and Benzoxazines via Oxidative Arylation of Anilide Derivatives
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Duong, Hung A.; Nguyen, Tuan Minh; Rosman, Nurul Zubaidah Binte; Tan, Lionel Jia Liang:
Carboxylation of Organoboronic Esters with Potassium Methyl Carbonate under Copper Catalysis
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Sahoo, Santosh K.; Jena, Himanshu Sekhar; Majji, Ganesh; Patel, Bhisma K.:
Formation of Imidazolidine-benzothiazole–Copper(II) Complexes via a Copper-Mediated Room-Temperature C–H Activation of Imidazolidinecarbothioamides
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Zhao, Chenglong; Tan, Zhuozhen; Liang, Zhuye; Deng, Wei; Gong, Hegui:
Nickel-Catalyzed Reductive Allylation of Ketones with Allylic Carbonates
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Luo, Long; Zhang, Jian-Jian; Ling, Wei-Jian; Shao, Yong-Liang; Wang, Ya-Wen; Peng, Yu:
Unified Synthesis of (–)-Folicanthine and (–)-Ditryptophenaline Enabled by a Room Temperature Nickel-Mediated Reductive Dimerization
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Liu, Jiangguang; Yan, Jiajie; Qin, Dongguang; Cai, Qian:
An Unexpected Inversion of Enantioselectivity in a Copper-Catalyzed Intramolecular Desymmetric Aryl C–N Coupling Reaction
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Kageyuki, Ikuo; Yoshida, Hiroto; Takaki, Ken:
Three-Component Carboboration of Alkenes under Copper Catalysis
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Gurung, Santosh K.; Thapa, Surendra; Shrestha, Bijay; Giri, Ramesh:
Copper-Catalyzed Cross-Coupling of Aryl- and Heteroaryltriethoxysilanes with Aryl and Heteroaryl Iodides and Bromides
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Ambler, Brett R.; Peddi, Santosh; Altman, Ryan A.:
Copper-Catalyzed Decarboxylative Trifluoromethylation of Propargyl Bromodifluoroacetates
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Issue 10/2014
Tang, Weijun; Xiao, Jianliang:
Asymmetric Hydrogenation of Imines via Metal–Organo Cooperative Catalysis
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Deiana, Luca; Ghisu, Lorenza; Córdova, Oscar; Afewerki, Samson; Zhang, Renyun; Córdova, Armando:
Efficient and Highly Enantioselective Aerobic Oxidation–Michael–Carbocyclization Cascade Transformations by Integrated Pd(0)-CPG Nanoparticle/Chiral Amine Relay Catalysis
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Diezel, Sonja; Breit, Bernhard:
Tandem Regioselective Rhodium-Catalyzed Hydroformylation–Enantioselective Aminocatalytic
anti
-Mannich Reaction
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Gualandi, Andrea; Mengozzi, Luca; Wilson, Claire Margaret; Cozzi, Pier Giorgio:
Synergistic Stereoselective Organocatalysis with Indium(III) Salts
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Lee, Hwa-Jung; Shyam, Pranab Kumar; Yoon, Woojin; Yun, Hoseop; Jang, Hye-Young:
Diastereo- and Enantioselective Synthesis of Hexasubstituted Cyclohexanes via a Metal–Organocatalytic Quadruple Cascade Sequence
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Praveen, Chandrasekaran; Levêque, Sabine; Vitale, Maxime R.; Michelet, Véronique; Ratovelomanana-Vidal, Virginie:
Synergistic Iron-and-Amine Catalysis in Carbocyclizations
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Liu, Lu; Daka, Philias; Sarkisian, Ryan; Deng, Yongming; Wheeler, Kraig; Wang, Hong:
Oxa-Diels–Alder Reaction of Isatins and Acyclic α,β-Unsaturated Methyl Ketones through Cooperative Dienamine and Metal Lewis Acid Catalysis
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Jing, Changcheng; Xing, Dong; Qian, Yu; Hu, Wenhao:
Rh
2
(OAc)
4
and Chiral Phosphoric Acid Cocatalyzed Highly Diastereo- and Enantioselective Four-Component Reactions: Facile Synthesis of Chiral α,β-Diamino Acid Derivatives
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Li, Nan; Chen, Dian-Feng; Wang, Pu-Sheng; Han, Zhi-Yong; Gong, Liu-Zhu:
Relay Catalytic Cascade Hydrosiloxylation and Asymmetric Hetero-Diels–Alder Reaction
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Yang, Jinming; Yu, Xingxin; Wu, Jie:
A Facile Route to
H
-Pyrazolo[5,1-
a
]isoquinolines through a Multicomponent Reaction of 2-Alkynylbenzaldehyde, Sulfonylhydrazine, and Benzyne
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Yoshida, Masanori; Masaki, Erika; Terumine, Tatsuaki; Hara, Shoji:
Asymmetric α-Allylation of α-Branched Aldehydes with Allyl Alcohols by Synergistic Catalysis Using an Achiral Palladium Complex and a Chiral Primary Amino Acid
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Issue 19/2013
Reboredo, Silvia; Vicario, Jose L.; Carrillo, Luisa; Reyes, Efraím; Uria, Uxue:
A Simple Synthesis of Polysubstituted Pyrrolidines by an Organocatalytic Three-Component Approach Featuring a One-Pot Condensation and [3+2]-Cycloaddition Reaction in Aqueous Medium
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Reitel, Kärt; Lippur, Kristin; Järving, Ivar; Kudrjašova, Marina; Lopp, Margus; Kanger, Tõnis:
Asymmetric Aminocatalytic Michael Addition of Cyclopropane-Containing Aldehydes to Nitroalkenes
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Shimada, Yoshiko; Hattori, Kasumi; Tada, Norihiro; Miura, Tsuyoshi; Itoh, Akichika:
Facile Aerobic Photooxidation of Alcohols Using 2-Chloroanthraquinone under Visible Light Irradiation
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Paria, Suva; Pirtsch, Michael; Kais, Viktor; Reiser, Oliver:
Visible-Light-Induced Intermolecular Atom-Transfer Radical Addition of Benzyl Halides to Olefins: Facile Synthesis of Tetrahydroquinolines
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Cismesia, Megan A.; Ischay, Michael A.; Yoon, Tehshik P.:
Reductive Cyclizations of Nitroarenes to Hydroxamic Acids by Visible Light Photoredox Catalysis
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Issue 15/2013
Mochizuki, Katsufumi; Sakai, Kazunori; Kochi, Takuya; Kakiuchi, Fumitoshi:
Rhodium-Catalyzed Dimerization of Arylacetylenes and Addition of Malonates to 1,3-Enynes
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Yamada, Yoichi M. A.; Ohta, Hidetoshi; Yuyama, Yoshinari; Uozumi, Yasuhiro:
Polymeric Bimetallic Catalyst-Promoted In-Water Dehydrative Alkylation of Ammonia and Amines with Alcohols
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Arnold, Jeffrey S.; Nguyen, Hien M.:
Rhodium-Catalyzed Asymmetric Amination of Allylic Trichloroacetimidates
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Ye, Ke-Yin; Zhao, Zhuo-An; Lai, Zeng-Wei; Dai, Li-Xin; You, Shu-Li:
Highly Regioselective Allylic Substitution Reactions Catalyzed by an Air-Stable (π-Allyl)iridium Complex Derived from Dinaphthocyclooctatetraene and a Phosphoramidite Ligand
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Obora, Yasushi; Sawaguchi, Takuya; Tsubakimoto, Keiko; Yoshida, Hiroshi; Ogawa, Shinji; Hatanaka, Shintaro:
Iridium-Catalyzed Synthesis of ω-Hydroxy Homoallylic Alcohols
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Apsunde, Tushar Dattu; Trudell, Mark L.:
Microwave-Assisted Iridium-Catalyzed Synthesis of Nicotine and Anabasine Derivatives
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Wang, Hui; Xu, Ming-Hua:
Rhodium-Catalyzed Highly Enantioselective Addition of Arylboronic Acids to Cyclic Aldimines: Practical Asymmetric Synthesis of Cyclic Sulfamidates
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Suzuki, Takeyuki; Ishizaka, Yuka; Ghozati, Kazem; Zhou, Da-Yang; Asano, Kaori; Sasai, Hiroaki:
Enantioselective Multicatalytic Synthesis of α-Benzyl-β-hydroxyindan-1-ones
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Liu, Wenting; Hong, Xiaohu; Xu, Bin:
Rhodium-Catalyzed Oxidative Coupling of Aryl Hydrazones with Internal Alkynes: Efficient Synthesis of Multisubstituted Isoquinolines
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Issue 12/2013
Fukata, Yukihiro; Miyaji, Ryota; Okamura, Takaaki; Asano, Keisuke; Matsubara, Seijiro:
Asymmetric Cycloetherifications by Bifunctional Aminothiourea Catalysts: The Importance of Hydrogen Bonding
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Jakab, Gergely; Hosseini, Abolfazl; Hausmann, Heike; Schreiner, Peter R.:
Mild and Selective Organocatalytic Iodination of Activated Aromatic Compounds
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Kumar, Vikas; Ray, Bidisha; Rathi, Preeti; Mukherjee, Santanu:
Catalytic Asymmetric Direct Vinylogous Michael Addition of γ-Aryl-Substituted Deconjugated Butenolides to Nitroolefins and
N
-Phenylmaleimide
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Duan, Shu-Wen; Liu, Yi-Yin; Ding, Wei; Li, Tian-Ren; Shi, De-Qing; Chen, Jia-Rong; Xiao, Wen-Jing:
Chiral Squaramide Catalyzed Asymmetric Conjugate Additions of 3-Substituted Oxindoles to Vinylphosphonates
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Chen, Guo-Ying; Lu, Yixin:
Highly Enantioselective Michael Addition of α-Substituted Nitrophosphonates to a Vinyl Sulfone
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Raimondi, Wilfried; Sanchez Duque, Maria del Mar; Goudedranche, Sébastien; Quintard, Adrien; Constantieux, Thierry; Bugaut, Xavier; Bonne, Damien; Rodriguez, Jean:
Activation of 1,2- and 1,3-Ketoamides with Thiourea Organocatalyst for the Enantioselective Domino Synthesis of Functionalized Cyclohexanes
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Issue 18/2012
Hassink, Matthew D.; Fox, Joseph M.:
Functionalized Cyclopropenes and Methylenecyclopropenes from Dianions of 3-Hydroxymethylcyclopropenes
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Rotstein, Benjamin H.; Yudin, Andrei K.:
Aziridine-2-carboxaldehyde Dimers Undergo Homo-Ugi 4-Component-5-center Reactions
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Walker, Daniel P.; Eklov, Brian M.; Bedore, Matthew W.:
Practical Synthesis of 3-Oxa-6-azabicyclo[3.1.1]heptane Hydrotosylate; A Novel Morpholine-Based Building Block
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Di Bussolo, Valeria; Frau, Ileana; Pineschi, Mauro; Crotti, Paolo:
d
-Allal- and
d
-Galactal-Derived Vinyl
N
-Mesylaziridines: Regio- and Stereoselectivity in Addition Reactions of O-, C-, N-, and S-Nucleophiles
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Florio, Saverio:
Unraveling the Synthetic Utility of the Regio- and Stereoselective Lithiation of Aziridines
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Issue 16/2012
Lei, Ming; Tian, Wan; Hu, Ruijun; Li, Wei; Zhang, Hong:
An Efficient Synthesis of 2-(Trifluoromethyl)-2
H
-[1,3]oxazino[2,3-
a
]isoquinolines via a Three-Component Cascade Approach Using a Continuous-Flow Microreactor
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Rodriguez, Antonio M.; Juan, Alberto; Gómez, M. Victoria; Moreno, Andres; de la Hoz, Antonio:
Continuous-Flow Microliter Microwave Irradiation in the Synthesis of Isoxazole Derivatives: An Optimization Procedure
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Slocum, D. W.; Reinscheld, Thomas K.; Austin, Nick D.; Kusmic, Damir; Whitley, Paul E.:
Near-Ambient Temperature Halogen–Lithium Exchange of
p
-Bromoanisole and Related Substrates: Flow/Batch Studies
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Pagano, Nicholas; Heil, Marintha L.; Cosford, Nicholas D. P.:
Automated Multistep Continuous Flow Synthesis of 2-(1
H
-Indol-3-yl)thiazole Derivatives
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Ullah, Farman; Zang, Qin; Javed, Salim; Porubsky, Patrick; Neuenswander, Benjamin; Lushington, Gerald H.; Hanson, Paul R.; Organ, Michael G.:
Synthesis of an Isoindoline-Annulated, Tricyclic Sultam Library via Microwave-Assisted, Continuous-Flow Organic Synthesis (MACOS)
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Fukuyama, Takahide; Kajihara, Yoshito; Ryu, Ilhyong; Studer, Armido:
Nitroxide-Mediated Polymerization of Styrene, Butyl Acrylate, or Methyl Methacrylate by Microflow Reactor Technology
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Issue 14/2012
Wu, Xingxing; Zhang, Junliang:
Y(OTf)
3
-Catalyzed Diastereoselective [3+2] Cycloaddition of
N
-Tosylaziridines and Imines; Efficient Synthesis of Multisubstituted Imidazolidines
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Yamazaki, Shoko; Fukushima, Yugo; Ukai, Tetsuma; Tatsumi, Kohei; Ogawa, Akiya:
Lewis Acid Promoted Reactions of 1,1-Diarylallenes and Ketone Derivatives: Synthesis of Indenes by an Addition/Cyclization Reaction
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