Synthesis

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Issue eFirst

Rai, Shweta; Samatha, Polasani; Addipilli, Ramunaidu; Mainkar, Prathama S.; Sripadi, Prabhakar; Adepu, Raju; Chandrasekhar, Srivari: Poly(ethylene glycol) Dimethyl Ethers (PEGDME): Efficient and Recyclable Solvents for Aryne-Involved Reactions
https://www.thieme-connect.de/media/synthesis/202222/i_f0147_ga_10-1055_a-1846-5598.gif
Gillard, Rachel M.; Zhang, Jiajun; Steel, Richard; Wang, Jocelyn; Strull, Jessica L.; Cai, Bin; Chakraborty, Nilanjana; Boger, Dale L.: Aryl Annulation: A Powerful Simplifying Retrosynthetic Disconnection
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0449_ga_10-1055_a-1959-2088.gif
Majhi, Jadab; Zhou, Bohang; Zhuang, Yuxin; Tom, Mai-Jan; Dai, Huifang; Evans, P. Andrew: Palladium-Catalyzed Cross-Coupling of Cyanohydrins with Aryl Bromides: Construction of Biaryl Ketones
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0052_ga_10-1055_a-1850-3687.gif
Khatana, Anil Kumar; Singh, Vikram; Gupta, Manoj Kumar; Tiwari, Bhoopendra: A Highly Efficient NHC-Catalyzed Aerobic Oxidation of Aldehydes to Carboxylic Acids
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0219_ga_10-1055_s-0037-1610069.gif
Liu, Cheng-Yuan; Chen, Ying-Ho; Chen, Chih-Hao; Yu, Ming-Shiuan; Tsai, Fu-Yu; Ong, Tiow-Gan: Selective C(8)–H Activation of Imidazopyridines Mediated by Cooperative Nickel–Aluminum Catalysis
https://www.thieme-connect.de/media/synthesis/201617/i_c0130_ga_10-1055_s-0035-15661438.gif
Kręcijasz, Remigiusz B.; Malinčík, Juraj; Šolomek, Tomáš: Exploring Silyl Protecting Groups for the Synthesis of Carbon Nanohoops
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0520_ga_10-1055_a-2008-9505.gif
Shirke, Rajendra P.; Reddy, Virsinha; Anand, R. Vijaya; Ramasastry, S. S. V.: Furans to Benzofurans: Intramolecular Cross-Benzoin Reactions Catalysed by N-Heterocyclic Carbenes
https://www.thieme-connect.de/media/synthesis/201612/i_c0133_ga_10-1055_s-0035-1560432.gif
Cai, Pin-Wen; You, Zhi-Hao; Xie, Liang-Hui; Tan, Rui; Tong, Zhi-Ping; Liu, Yan-Kai: The Attractive Application of Lactol Chemistry: From Racemic Lactol to Natural Product Skeleton
https://www.thieme-connect.de/media/synthesis/201616/i_c0029_ga_10-1055_s-0035-1561972.gif
Schweighauser, Luca; Bodoky, Ina; Kessler, Simon N.; Häussinger, Daniel; Wegner, Hermann A.: Bidentate Lewis Acid Catalyzed Inverse-Electron-Demand Diels–Alder Reaction for the Selective Functionalization of Aldehydes
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Nori, Valeria; Sinibaldi, Arianna; Pesciaioli, Fabio; Carlone, Armando: Impact of Design of Experiments in the Optimisation of Catalytic Reactions in Academia
https://www.thieme-connect.de/media/synthesis/202219/i_r0735_ga_10-1055_a-1736-6703.gif
Ledovskaya, Maria S.; Voronin, Vladimir V.; Rodygin, Konstantin S.; Ananikov, Valentine P.: Acetylene and Ethylene: Universal C2 Molecular Units in Cycloaddition Reactions
https://www.thieme-connect.de/media/synthesis/202204/i_r0524_ga_10-1055_a-1654-2318.gif
Patra, Subrata; Mosiagin, Ivan; Giri, Rahul; Katayev, Dmitry: Organic Nitrating Reagents
https://www.thieme-connect.de/media/synthesis/202215/i_r0727_ga_10-1055_s-0040-1719905.gif
Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.: IntraMolecular Diels–Alder Reactions of Vinylarenes and Alkynyl Arenes (the IMDAV Reaction)
https://www.thieme-connect.de/media/synthesis/202204/i_z0484_ga_10-1055_s-0040-1705983.gif
Frost, Christopher G.; Edwards, Hannah J.; Penrose, Stephen D.; Gleave, Robert: Exploring Rhodium-Catalysed Conjugate Addition of Chiral Alkenylboronates Using Chiral Olefin Ligands
https://www.thieme-connect.de/media/synthesis/201019/c040_ga.jpg
La Torre, Mathéo; Maton, William; Cleator, Ed; Jouffroy, Matthieu: Pd/C Catalyzed Dehalogenation of (Hetero)aryls Using Triethyl­silane as Hydrogen Donor
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0534_ga_10-1055_s-0042-1753402.gif
Airiau, Etienne; Chemin, Claire; Girard, Nicolas; Lonzi, Giacomo; Mann, André; Petricci, Elena; Salvadori, Jessica; Taddei, Maurizio: Microwave-Assisted Domino Hydroformylation/Cyclization Reactions: Scope and Limitations
https://www.thieme-connect.de/media/synthesis/201017/c034_ga.jpg
Belhomme, Marie-Charlotte; Dru, Delphine; Xiong, Heng-Ying; Cahard, Dominique; Besset, Tatiana; Poisson, Thomas; Pannecoucke, Xavier: Copper-Mediated Direct Functionalization of Unsaturated C–C Bonds with Ethyl Bromo(difluoro)acetate: A Straightforward Access to Highly Valuable Difluoromethylated Alkenes
https://www.thieme-connect.de/media/synthesis/201414/i_c0137_ga_10-1055_s-0033-1338637.gif
Agudelo, Brian Castro; Rigoulet, Florian; Giorgi, Michel; Sayah, Babak; Rodriguez, Jean; Coquerel, Yoann: Synthesis of Axially Chiral Cationic Benzo[c]phenanthridinium Derivatives
https://www.thieme-connect.de/media/synthesis/202222/i_f0170_ga_10-1055_a-1845-3128.gif
Malkina, Anastasiya G.; Stepanov, Anton V.; Sobenina, Lyubov N.; Shemyakina, Olesya A.; Ushakov, Igor A.; Smirnov, Vladimir I.; Trofimov, Boris A.: Organocatalyzed Microwave-Assisted Competing Cyclization of Cyanopropargylic Alcohols with Carboxylic Acids: 4-Cyano-3(2H)-furanones versus 4-Cyano-[(Z)-3-cyanomethylene]-2,3-dihydro­furans
https://www.thieme-connect.de/media/synthesis/201612/i_c0071_ga_10-1055_s-0035-1561591.gif
Dobrydnev, Alexey V.; Popova, Maria V.; Saffon-Merceron, Nathalie; Listunov, Dymytrii; Volovenko, Yulian M.: Synthesis of the First Representatives of Spiro-1λ6-isothiazolidine-1,1,4-triones
https://www.thieme-connect.de/media/synthesis/201517/i_t0209_ga_10-1055_s-0034-1380434.gif
Luo, Guo-Ying; Wu, Hao; Tang, Yu; Li, Hui; Yeom, Hyun-Suk; Yang, Ka; Hsung, Richard P.: A Total Synthesis of (±)-Rhododaurichromanic Acid A via an Oxa-[3+3] Annulation of Resorcinols
https://www.thieme-connect.de/media/synthesis/201518/i_c0219_ga_10-1055_s-0034-1380429.gif
Kratzer, Philipp; Gerster, Holger; Maas, Gerhard: Cycloaddition Reactions of Propyne Iminium Salts and Enol Ethers
https://www.thieme-connect.de/media/synthesis/201518/i_c0319_ga_10-1055_s-0034-1380223.gif
Carreiro, Elisabete P.; Gastalho, Carlos M.; Ernesto, Sofia; Costa, Ana R.; Antunes, Célia M.; Burke, Anthony J.: Synthesis and Antiproliferative Activity of Novel Quercetin-1,2,3-Triazole Hybrids using the 1,3-Dipolar Cycloaddition (Click) Reaction
https://www.thieme-connect.de/media/synthesis/202219/i_t0074_ga_10-1055_s-0040-1719928.gif
Chen, Shi; Mondal, Mukulesh; Ibrahim, Ahmad A.; Wheeler, Kraig A.; Kerrigan, Nessan J.: Asymmetric Synthesis of Dipropionate Derivatives through Catalytic Hydrogenation of Enantioenriched E-Ketene Heterodimers
https://www.thieme-connect.de/media/synthesis/201616/i_c0020_ga_10-1055_s-0035-1561958.gif
Dai, Wen; Mi, Yuan; Lv, Ying; Shang, Sensen; Li, Guosong; Chen, Guangwen; Gao, Shuang: Development of a Continuous-Flow Microreactor for Asymmetric Epoxidation of Electron-Deficient Olefins
https://www.thieme-connect.de/media/synthesis/201616/i_c0708_ga_10-1055_s-0035-1561955.gif
Deng, Lu-Jiang; Liu, Jing; Huang, Ji-Qing; Hu, Yanhe; Chen, Mao; Lan, Yu; Chen, Jia-Hua; Lei, Aiwen; Yang, Zhen: Effect of Lithium Chloride on Tuning the Reactivity of Pauson-Khand Reactions­ Catalyzed by Palladium-Tetramethylthiourea
https://www.thieme-connect.de/bilder/synthesis/200716/c037_ga
Yamaoka, Yousuke; Miyabe, Hideto; Yasui, Yoshizumi; Takemoto, Yoshiji: Chiral-Thiourea-Catalyzed Direct Mannich Reaction
https://www.thieme-connect.de/bilder/synthesis/200716/c035_ga
Jiménez Blanco, José L.; Bootello, Purificación; Gutiérrez Gallego, Ricardo; Ortiz Mellet, Carmen; García Fernández, José M.: Synthesis of Thiourea-Linked Glycooligomers that Mimic the Branching Patterns of Natural Oligosaccharides
https://www.thieme-connect.de/bilder/synthesis/200716/c033_ga
Pop, Lidia; Golban, Mirabela Ligia; Hădade, Niculina D.; Socaci, Crina; Grosu, Ion: CuAAC Synthesis of Tetragonal Building Blocks Decorated with Nucleobases
https://www.thieme-connect.de/media/synthesis/201518/i_c0288_ga_10-1055_s-0034-1378782.gif
Oberg, Kevin M.; Cochran, Brian M.; Cook, Matthew J.; Rovis, Tomislav: The Catalytic Alkylative Desymmetrization of Anhydrides in a Formal Synthesis of Ionomycin
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0160_ga_10-1055_s-0037-1610108.gif
Nakayama, Yasuaki; Maeda, Yuichiro; Hama, Naoto; Sato, Takaaki; Chida, Noritaka: Total Synthesis of (–)-Stemoamide by Sequential Overman/Claisen Rearrangement
https://www.thieme-connect.de/media/synthesis/201611/i_c0050_ga_10-1055_s-0035-1561948.gif
Heinz, Benjamin; Djukanovic, Dimitrije; Siemens, Fiona; Idriess, Mohamed; Martin, Benjamin; Knochel, Paul: Regioselective Amination or Alkoxylation of Halogenated Amino-, Thio- or Alkoxypyridines via Pyridyne Intermediates
https://www.thieme-connect.de/media/synthesis/202222/i_f0548_ga_10-1055_s-0037-1610786.gif
Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke: Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0368_ga_10-1055_s-0039-1690010.gif
Kousara, Mohammad; Bideau, Franck Le; Ibrahim, Rama; Ferry, Angélique; Venot, Pierre-Etienne; Dejean, Camille; Raingeaud, Joël; Dubois, Joëlle; Retailleau, Pascal; Dumas, Françoise: Suberosanes as Potential Antitumor Agents: First Enantioselective Total Synthesis of (1S)-Suberosanone and Configurational Assignment of Suberosenol A
https://www.thieme-connect.de/media/synthesis/201611/i_c0040_ga_10-1055_s-0035-1561430.jpg
Konda, Saidulu; Khatravath, Mahender; Mallurwar, Naveen Kumar; Rao, Pallavi; Sripelly, Shivashankar; Iqbal, Javed; Arya, Prabhat: Stereoselective Synthesis of the C27–C35 Eribulin Fragment and Its Utilization in Building Structurally Diverse Macrocycles
https://www.thieme-connect.de/media/synthesis/201611/i_c0084_ga_10-1055_s-0035-1561431.gif
Feng, Yangyang; Huang, Ruofeng; Hu, Liangzhen; Xiong, Yan; Coeffard, Vincent: Chiral C2-Symmetric Iodoarene-Catalyzed Asymmetric α-Oxidation of β-Keto Esters
https://www.thieme-connect.de/media/synthesis/201616/i_c0132_ga_10-1055_s-0035-1561442.gif
Zhang, Yongda; Lao, Kendricks S.; Sieber, Joshua D.; Xu, Yibo; Wu, Linglin; Wang, Xiao-Jun; Desrosiers, Jean-Nicolas; Lee, Heewon; Haddad, Nizar; Han, Zhengxu S.; Yee, Nathan K.; Song, Jinhua J.; Howell, Amy R.; Senanayake, Chris H.: Modular Dihydrobenzoazaphosphole Ligands for Suzuki–Miyaura Cross-Coupling
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0181_ga_10-1055_s-0037-1610158.gif
Liddon, John T. R.; Rossi-Ashton, James A.; Clarke, Aimee K.; Lynam, Jason M.; Taylor, Richard J. K.; Unsworth, William P.: Divergent Reactivity of Indole-Tethered Ynones with Silver(I) and Gold(I) Catalysts: A Combined Synthetic and Computational Study
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0211_ga_10-1055_s-0037-1610181.gif
Kumar, Ravindra; Tamai, Eri; Ohnishi, Akira; Nishimura, Akira; Hoshimoto, Yoichi; Ohashi, Masato; Ogoshi, Sensuke: Nickel-Catalyzed Enantioselective Synthesis of Cyclobutenes via [2+2] Cycloaddition of α,β-Unsaturated Carbonyls with 1,3-Enynes
https://www.thieme-connect.de/media/synthesis/201617/i_c0174_ga_10-1055_s-0035-1561669.gif
Marques, Carolina S.; López, Óscar; Leitzbach, Luisa; Fernández-Bolaños, José G.; Stark, Holger; Burke, Anthony J.: Survey of New, Small-Molecule Isatin-Based Oxindole Hybrids as Multi-Targeted Drugs for the Treatment of Alzheimer’s Disease
https://www.thieme-connect.de/media/synthesis/202219/i_m0728_ga_10-1055_s-0041-1737343.gif
Carboni, Aude; Dagousset, Guillaume; Magnier, Emmanuel; Masson, Géraldine: Three-Component Photoredox-Mediated Chloro-, Bromo-, or Iodotrifluoromethylation of Alkenes
https://www.thieme-connect.de/media/synthesis/201516/i_c0200_ga_10-1055_s-0034-1378715.gif
Iwata, Takayuki; Hyodo, Mizuki; Fujiwara, Takumi; Kawano, Ryusei; Kuhn, Leah; Alabugin, Igor V.; Shindo, Mitsuru: 3-Trifluoromethylbenzyne: Precise Orientation in Cycloaddition Reaction Enabled Regioselective Synthesis of Trifluoromethylated Triptycenes
https://www.thieme-connect.de/media/synthesis/202222/i_f0130_ga_10-1055_a-1818-0576.gif
Firth, James D.; Zhang, Rong; Morgentin, Rémy; Guilleux, Rachel; Kalliokoski, Tuomo; Warriner, Stuart; Foster, Richard; Marsden, Stephen P.; Nelson, Adam: Exploitation of the Ugi–Joullié Reaction in the Synthesis of Libraries of Drug-Like Bicyclic Hydantoins
https://www.thieme-connect.de/media/synthesis/201516/i_c0208_ga_10-1055_s-0034-1378704.gif
Biswas, Anup; Kundu, Samrat; Pal, Dhananjoy; Pal, Amit; Maji, Modhu Sudan: Organocatalyzed Oxa-Diels–Alder Reactions: Recent Progress
https://www.thieme-connect.de/media/synthesis/202204/i_r0218_ga_10-1055_a-1514-1049.gif
Miller, Daniel K.; Bailey, Christopher A.; Sammelson, Robert E.: Synthesis of Isoxazolines and Isoxazoles Inspired by Fipronil
https://www.thieme-connect.de/media/synthesis/201518/i_c0263_ga_10-1055_s-0034-1378737.gif
Xu, Shibo; Su, Shikuan; Zhang, Huiting; Tian, Lumin; Liang, Pengcheng; Chen, Jiawen; Zhang, Yuan; Li, Chunju; Jia, Xueshun; Li, Jian: Isocyanide-Based Multicomponent Reactions: Rapid Synthesis of a 5,5-Fused Bicyclic Skeleton from α,β-Unsaturated Ketones and Allenoates
https://www.thieme-connect.de/media/synthesis/201516/i_c0250_ga_10-1055_s-0034-1378736.gif
Chuyko, Alexey; Dolgonos, Grygoriy; Shivanyuk, Alexander; Fetyukhin, Volodymyr; Lukin, Oleg: Simple Synthesis of Complex Amines from the Diels–Alder Adducts of (–)-Cytisine
https://www.thieme-connect.de/media/synthesis/202204/i_z0205_ga_10-1055_s-0040-1706282.gif
Ghosh, Prasanjit; Mondal, Swati Lekha; Baidya, Mahiuddin: Ascending of Cycloaddition Strategy for N–O Heterocycles
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Wertjes, William; Ayers, Sloan; Gao, Qi; Simmons, Eric M.; Beutner, Gregory L.: A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0192_ga_10-1055_s-0037-1610140.gif
Hopf, Henning; Sherburn, Michael S.: Allenes in Diels–Alder Cycloadditions
https://www.thieme-connect.de/media/synthesis/202204/i_m0291_ga_10-1055_s-0040-1706052.gif
Yang, Yun; Jones, Christopher R.: The Aryne Ene Reaction
https://www.thieme-connect.de/media/synthesis/202222/i_f0171_ga_10-1055_a-1827-2987.gif
Cormier, Morgan; Chardon, Aurélien; Blanchet, Jérôme; Rouden, Jacques; Maddaluno, Jacques; De Paolis, Michaël: An Organocatalytic Access to Spiro[4.5]decanes and Spiro[4.6]undecanes Containing Aminolactones and 3-Aminopyrrolidines
https://www.thieme-connect.de/media/synthesis/201517/i_c0767_ga_10-1055_s-0034-1380146.gif
Nagai, Akira; Kobayashi, Akihiro; Sakata, Yuki; Minami, Yasunori; Uchida, Keisuke; Hosoya, Takamitsu; Yoshida, Suguru: Synthesis of Multisubstituted Benzenes from Phenols via Multisubstituted Benzynes
https://www.thieme-connect.de/media/synthesis/202222/i_f0139_ga_10-1055_a-1834-2927.gif
Monasson, Olivier; Malinowski, Maciej; Lubin-Germain, Nadège; Ferry, Angélique: Hirao Cross-Coupling Reaction as an Efficient Tool to Build Non-natural C2-Phosphonylated Sugars
https://www.thieme-connect.de/media/synthesis/202215/i_m0624_ga_10-1055_a-1709-3305.gif
Neochoritis, Constantinos G.; Zhang, Ji; Dömling, Alexander: Leuckart–Wallach Approach to Sugar Isocyanides and Its IMCRs
https://www.thieme-connect.de/media/synthesis/201516/i_c0249_ga_10-1055_s-0034-1381046.jpg
Pan, Yuanjia; Lu, Hongjian; Fang, Yewen; Fang, Xinqiang; Chen, Liqun; Qian, Junlu; Wang, Junhua; Li, Chaozhong: Synthesis of Pyrroles via Copper-Catalyzed Coupling of Amines with Bromoenones
https://www.thieme-connect.de/bilder/synthesis/200708/c003_ga
Estéoule, Audrey; Durán, Fernando; Retailleau, Pascal; Dodd, Robert H.; Dauban, Philippe: Enantioselective Intramolecular Copper-Catalyzed Aziridination of Sulfamates
https://www.thieme-connect.de/bilder/synthesis/200708/c002_ga
Seck, Insa; Fall, Alioune; Lago, Carmen; Sène, Massène; Gaye, Mohamed; Seck, Matar; Gómez, Generosa; Fall, Yagamare: Synthesis of a Cholesterol Side-Chain Triazole Analogue via ‘Click’ Chemistry
https://www.thieme-connect.de/media/synthesis/201518/i_c0282_ga_10-1055_s-0034-1381053.gif
Kachkovskyi, Georgii; Cieślak, Marcin; Graczyk, Piotr; Zawadzki, Przemysław; Kalinowska-Tłuścik, Justyna; Werłos, Mateusz: Photocatalytic Approach to α,α-Difluoroalkyl Alcohols
https://www.thieme-connect.de/media/synthesis/202219/i_f0729_ga_10-1055_s-0041-1737546.gif
Fujimoto, Hayato; Yamamura, Shisato; Takenaka, Namiki; Tobisu, Mamoru: Phosphine-Catalyzed Z-Selective Carbofluorination of Alkynoates Bearing an N-Heteroarene Unit
https://www.thieme-connect.de/media/synthesis/202306/i_c0369_ga_10-1055_a-1948-3234.gif
Ugarriza, Iratxe; Reyes, Efraím; Prieto, Liher; Uria, Uxue; Carrillo, Luisa; Vicario, Jose L.: An Approach to the Synthesis of a Hepatitis C Virus Inhibitor through a Proline-Catalyzed 1,3-Dipolar Cycloaddition Using Acrolein
https://www.thieme-connect.de/media/synthesis/202204/i_f0626_ga_10-1055_s-0040-1719858.gif
Sato, Kazuyuki; Tarui, Atsushi; Omote, Masaaki; Ando, Akira; Kumadaki, Itsumaro: Trifluoromethylation of Organic Compounds and Related Reactions
https://www.thieme-connect.de/media/synthesis/201011/c009_ga.jpg
Mahajan, Bhushan; Aand, Dnyaneshwar; Purwa, Mandeep; Mujawar, Taufiqueahmed; Ghosh, Subhash; Pabbaraja, Srihari; Singh, Ajay K.: Elements-Continuous-Flow Platform for Coupling Reactions and Anti-viral Daclatasvir API Synthesis
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0518_ga_10-1055_a-2022-2063.gif
Peddie, Victoria; Pietsch, Markus; Bromfield, Karen M.; Pike, Robert N.; Duggan, Peter J.; Abell, Andrew D.: Fluorinated β²- and β³-Amino Acids: Synthesis and Inhibition of α-Chymotrypsin
https://www.thieme-connect.de/media/synthesis/201011/c004_ga.jpg
Roger, Julien; Sire, Charline; Tsivery, Anthonia; Cattey, Hélène; Hierso, Jean-Cyrille: Aryl Triflates in Phosphorus-Directed Rhodium(III)-Catalyzed C–H Activation
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0501_ga_10-1055_a-2018-0965.gif
Furuya, Takeru; Klein, Johannes E. M. N.; Ritter, Tobias: Carbon-Fluorine Bond Formation for the Synthesis of Aryl Fluorides
https://www.thieme-connect.de/media/synthesis/201011/c002_ga.jpg
Vicente-García, Esther; Ramón, Rosario; Lavilla, Rodolfo: New Heterocyclic Inputs for the Povarov Multicomponent Reaction
https://www.thieme-connect.de/media/synthesis/201114/c339_ga.jpg
Bortolato, Tommaso; Dyguda, Mateusz; Vega-Peñaloza, Alberto; Dell’Amico, Luca: Properties and Synthetic Performances of Phenylamino Cyanoarenes under One-Photon Excitation Manifolds
https://www.thieme-connect.de/media/synthesis/202215/i_c0750_ga_10-1055_a-1776-0929.gif
Suzuki, Takeyuki; Ishizaka, Yuka; Ghozati, Kazem; Zhou, Da-Yang; Asano, Kaori; Sasai, Hiroaki: Enantioselective Multicatalytic Synthesis of α-Benzyl-β-hydroxyindan-1-ones
https://www.thieme-connect.de/media/synthesis/201315/i_c0194_ga_10-1055_s-0033-1338479.gif
Duong, Hung A.; Nguyen, Tuan Minh; Rosman, Nurul Zubaidah Binte; Tan, Lionel Jia Liang: Carboxylation of Organoboronic Esters with Potassium Methyl Carbonate under Copper Catalysis
https://www.thieme-connect.de/media/synthesis/201414/i_c0122_ga_10-1055_s-0033-1339119.gif
Zhao, Chenglong; Tan, Zhuozhen; Liang, Zhuye; Deng, Wei; Gong, Hegui: Nickel-Catalyzed Reductive Allylation of Ketones with Allylic Carbonates
https://www.thieme-connect.de/media/synthesis/201414/i_c0174_ga_10-1055_s-0033-1339111.gif
Walkowiak, Justyna; del Campo, Teresa Martinez; Ameduri, Bruno; Gouverneur, Véronique: Syntheses of Mono-, Di-, and Trifluorinated Styrenic Monomers
https://www.thieme-connect.de/media/synthesis/201011/c028_ga.jpg
Murakami, Sho; Brudy, Cosima; Bachmann, Moritz; Takemoto, Yoshiji; Pieber, Bartholomäus: Photocatalytic Cleavage of Trityl Protected Thiols and Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0491_ga_10-1055_a-1979-5933.gif
Hunter, Thomas J.; Wang, Yanping; Zheng, Jiamin; O’Doherty, George A.: Asymmetric Iterative Hydration of Polyene Strategy to Cryptocaryols A and B
https://www.thieme-connect.de/media/synthesis/201611/i_c0125_ga_10-1055_s-0035-1561607.gif
Nishimura, Takahiro; Nagai, Tomotaka; Takechi, Ryosuke; Ebe, Yusuke: Rhodium-Catalyzed Enantioselective Addition of Tricyclopropylboroxin to N-Sulfonylimines
https://www.thieme-connect.de/media/synthesis/201616/i_c0007_ga_10-1055_s-0035-1561605.gif
García-Ruiz, Cristina; Cheng-Sánchez, Iván; Sarabia, Francisco: Synthesis of (–)- and (+)-Gummiferol via Asymmetric Synthesis of Glycidic Amides
https://www.thieme-connect.de/media/synthesis/201611/i_c0102_ga_10-1055_s-0035-1561606.gif
Ferro, Rita; Viduedo, Nuno; Santos, A. Sofia; Silva, Artur M. S.; Royo, Beatriz; Marques, M. Manuel B.: Bimetallic Catalyzed Synthesis of 2-Arylindoles
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0631_ga_10-1055_a-2035-6420.gif
Schäfer, Gabriel; Reber, Stefan; Ahmetovic, Muhamed; Fleischer, Tony; Leuenberger, Daniel; Blumer, Nicole; Udry, Megan; Abele, Stefan: Robust and Scalable Reductive Amination Protocol for Electron-Poor Heterocyclic Amines Using Et3SiH/TFA as Reducing Agent
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0441_ga_10-1055_a-1981-2727.gif
Ziegler, Dorothée S.; Klier, Lydia; Müller, Nicolas; Karaghiosoff, Konstantin; Knochel, Paul: Directed Zincation or Magnesiation of 2- and 4-Pyrones and Their Derivatives
https://www.thieme-connect.de/media/synthesis/EFirst/i_c0411_ga_10-1055_s-0037-1610215.gif
Cserép, Gergely B.; Demeter, Orsolya; Bätzner, Effi; Kállay, Mihály; Wagenknecht, Hans-Achim; Kele, Péter: Synthesis and Evaluation of Nicotinic Acid Derived Tetrazines for Bioorthogonal Labeling
https://www.thieme-connect.de/media/synthesis/201518/i_c0157_ga_10-1055_s-0034-1380721.gif
Zhang, Pengke; Hua, Lin; Takahashi, Tamotsu; Jin, Shengnan; Wang, Qilin: Recent Advances in the Dearomative Skeletal Editing of Mono-azaarenes
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0628_ga_10-1055_a-2013-9885.gif
Khan, Farooq-Ahmad; Yaqoob, Sana; Qasim, Muhammad Wasim; Ali, Shujaat; Wang, Yan; Jiang, Zi-Hua: A Robust, Gram-Scale and High-Yield Synthesis of MDP Congeners for Activation of the NOD2 Receptor and Vaccine Adjuvantation
https://www.thieme-connect.de/media/synthesis/EFirst/i_b0528_ga_10-1055_a-2004-5883.gif
Sara, Alexandru A.; Um-e-Farwa, Um-e-Farwa; Saeed, Aamer; Kalesse, Markus: Recent Applications of the Diels–Alder Reaction in the Synthesis of Natural Products (2017–2020)
https://www.thieme-connect.de/media/synthesis/202204/i_r0249_ga_10-1055_a-1532-4763.gif
Woof, Callum R.; Linford-Wood, Thomas G.; Mahon, Mary F.; Webster, Ruth L.: Catalytic Hydrophosphination of Allenes Using an Iron(II) β-Diketiminate Complex
https://www.thieme-connect.de/media/synthesis/202306/i_c0290_ga_10-1055_a-1902-5592.gif

Issue Accepted Manuscripts

Issue 21/2022

Yang, Zhenjie; Cheng, Hong-Gang; Chen, Ruiming; Cao, Liming; Wei, Qiang; Wang, Qingqing; Zhou, Qianghui: Eight-Step Asymmetric Synthesis of (–)-Berkelic Acid
https://www.thieme-connect.de/media/synthesis/202221/i_g0085_ga_10-1055_a-1799-0459.gif
Huang, Long-Tao; Hirata, Yuki; Kato, Yoshimi; Lin, Luqing; Kojima, Masahiro; Yoshino, Tatsuhiko; Matsunaga, Shigeki: Ruthenium(II)/Chiral Carboxylic Acid Catalyzed Enantioselective C–H Functionalization of Sulfoximines
https://www.thieme-connect.de/media/synthesis/202221/i_g0414_ga_10-1055_a-1588-0072.gif
Huang, Xiao-Ling; Li, Chong; Wang, Juan; Yang, Shang-Dong: Direct Copper-Catalyzed C-3 Arylation of Diphenylphosphine Oxide Indoles
https://www.thieme-connect.de/media/synthesis/202221/i_g0472_ga_10-1055_a-1633-8792.gif
Pototskiy, Roman A.; Boym, Mikhail A.; Nelyubina, Yulia V.; Perekalin, Dmitry S.: Synthesis of Ruthenium Catalysts with a Chiral Arene Ligand Derived from Natural Camphor
https://www.thieme-connect.de/media/synthesis/202221/i_g0590_ga_10-1055_a-1668-2075.gif

Issue 17/2022

Remete, Attila M.; Nonn, Melinda; Volk, Balázs; Kiss, Loránd: Developments in the Alkynyltrifluoromethylations of Alkenes and Alkynes
https://www.thieme-connect.de/media/synthesis/202217/i_r0123_ga_10-1055_a-1811-8679.gif
Fichez, Jeanne; Dupommier, Dorian; Besset, Tatiana: Direct Synthesis of Disubstituted Trifluoromethylthiolated Alkenes
https://www.thieme-connect.de/media/synthesis/202217/i_r0707_ga_10-1055_s-0040-1719891.gif
Gonda, Zsombor; Földesi, Tamás; Nagy, Bálint; Novák, Zoltán: Modular Synthesis of Carbazole-Substituted Phthalimides as Potential Photocatalysts
https://www.thieme-connect.de/media/synthesis/202217/i_z0437_ga_10-1055_a-1647-7292.jpg
Salamon-Krokosz, Katarzyna; Gołdyn, Mateusz; Siodła, Tomasz; Bartoszak-Adamska, Elżbieta; Koroniak, Henryk; Koroniak-Szejn, Katarzyna: Fluorinated Olefinic Lactams: The Case of Amino Acids – Preparation and Mechanistic Studies
https://www.thieme-connect.de/media/synthesis/202217/i_c0658_ga_10-1055_s-0041-1737346.jpg
El Haimer, Mohamed; Faragó, Tünde; Schelz, Zsuzsanna; Zupkó, István; Palkó, Márta: Synthesis of Alicyclic 2-Methylenethiazolo[2,3-b]quinazolinone Derivatives via Base-Promoted Cascade Reactions
https://www.thieme-connect.de/media/synthesis/202217/i_t0623_ga_10-1055_s-0040-1720028.gif
Garnes-Portolés, Francisco; Miguélez, Rubén; Grayson, Matthew N.; Barrio, Pablo: Heteroatom-Tethered ω-Alkenylallylboronates: Stereoselective Synthesis of Heterocyclic Derived Alcohols
https://www.thieme-connect.de/media/synthesis/202217/i_t0690_ga_10-1055_s-0040-1719890.gif
Dargó, Gyula; Nagy, Sándor; Kis, Dávid; Bagi, Péter; Mátravölgyi, Béla; Tóth, Blanka; Huszthy, Péter; Drahos, László; Kupai, József: Application of Proline-Derived (Thio)squaramide Organocatalysts in Asymmetric Diels–Alder and Conjugate Addition Reactions
https://www.thieme-connect.de/media/synthesis/202217/i_z0619_ga_10-1055_s-0040-1719886.gif
Raji, Mounir; Le, Tam Minh; Csámpai, Antal; Nagy, Viktória; Zupkó, István; Szakonyi, Zsolt: Stereoselective Synthesis and Applications of Pinane-Based Chiral 1,4-Amino Alcohol Derivatives
https://www.thieme-connect.de/media/synthesis/202217/i_z0668_ga_10-1055_s-0040-1719887.gif
Cserép, Gergely B.; Németh, Krisztina; Szatmári, Ágnes; Horváth, Flóra; Imre, Tímea; Németh, Krisztina; Kele, Péter: Beyond the Bioorthogonal Inverse-Electron-Demand Diels–Alder Reactions of Tetrazines: 2-Pyrone-Functionalized Fluorogenic Probes
https://www.thieme-connect.de/media/synthesis/202217/i_t0622_ga_10-1055_a-1761-4672.jpg
Szabó, Tímea; Görür, Funda Lidya; Horváth, Simon; Volk, Balázs; Milen, Mátyás: Synthesis of Racemic and Enantiopure Forms of β-Carboline Alkaloid Brevicolline
https://www.thieme-connect.de/media/synthesis/202217/i_t0720_ga_10-1055_s-0041-1737830.gif
Berecz, Gábor; Dancsó, András; Németh, Dóra R.; Kiss, Loránd; Simig, Gyula; Volk, Balázs: Towards Tianeptine Analogues: Synthesis of New Ring Systems Containing a Dibenzo[c,f][1,2]thiazepine S,S-Dioxide Core
https://www.thieme-connect.de/media/synthesis/202217/i_t0733_ga_10-1055_s-0040-1719885.gif
Takao, Go; Hakozaki, Tomohiro; Miura, Keisuke; Urushibara, Yusuke; Fuchibe, Kohei; Ichikawa, Junji: Construction of Substituted [4]Acene Frameworks Based on Double Cationic Cyclizations of Fluoroalkenes
https://www.thieme-connect.de/media/synthesis/202217/i_f0693_ga_10-1055_s-0037-1610791.gif
Harsági, Nikoletta; Kiss, Nóra Zsuzsa; Drahos, László; Keglevich, György: Synthesis of Cyclic Phosphinates by Microwave-Assisted Ionic-Liquid-Promoted Alcoholysis
https://www.thieme-connect.de/media/synthesis/202217/i_t0208_ga_10-1055_a-1504-8924.gif

Issue 04/2022

Issue 22/2021

Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark: Recent Advances in Transition-Metal-Free (4+3)-Annulations
https://www.thieme-connect.de/media/synthesis/202122/i_z0520_ga_10-1055_s-0040-1706023.gif
Ryan, Jonathon S.; Schindler, Corinna S.: Total Synthesis of Mycocyclosin and the Herqulines
https://www.thieme-connect.de/media/synthesis/202122/i_m0034_ga_10-1055_a-1403-4312.gif
Tien, Chieh-Hung; Trofimova, Alina; Shao, Wenjie; Yudin, Andrei K.: Synthesis of Borylated Hydrazino Acid Derivatives
https://www.thieme-connect.de/media/synthesis/202122/i_t0192_ga_10-1055_s-0040-1706046.gif
Kasim, Johanes K.; Kavianinia, Iman; Bull, Matthew; Harris, Paul W. R.; Smaill, Jeff B.; Patterson, Adam V.; Brimble, Margaret A.: Fourth-Generation Analogues of the Anticancer Peptaibol Culicinin D: Probing the Effects of Hydrophobicity and Halogenation on Cytotoxicity
https://www.thieme-connect.de/media/synthesis/202122/i_m0124_ga_10-1055_s-0040-1706264.gif
Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten: Studies towards the Synthesis of (–)-Pulvomycin: Construction of the C12–C40 Segment by a Stereoselective Aldol Reaction
https://www.thieme-connect.de/media/synthesis/202122/i_m0156_ga_10-1055_a-1464-2576.gif
El Khoury, Anton; Seidler, Paul M.; Eisenberg, David S.; Harran, Patrick G.: Catalytic Synthesis of PEGylated EGCG Conjugates that Disaggregate Alzheimer’s Tau
https://www.thieme-connect.de/media/synthesis/202122/i_m0212_ga_10-1055_a-1509-5904.gif
Caldora, Henry P.; Govaerts, Sebastian; Dighe, Shashikant U.; Turner, Oliver J.; Leonori, Daniele: A de novo Synthesis of Oxindoles from Cyclohexanone-Derived γ-Keto-Ester Acceptors Using a Desaturative Amination–Cyclization Approach
https://www.thieme-connect.de/media/synthesis/202122/i_m0336_ga_10-1055_a-1538-8429.gif
Davis, Christopher W.; Bingham, Tanner W.; Okumura, Mikiko; Sarlah, David: Dearomative syn-1,2-Diamination of Benzene and Naphthalene
https://www.thieme-connect.de/media/synthesis/202122/i_m0523_ga_10-1055_s-0040-1719842.gif

Issue 18/2021

Basak, Sumon; Biswas, Jyoti Prasad; Maiti, Debabrata: Transition-Metal-Catalyzed C–H Arylation Using Organoboron Reagents
https://www.thieme-connect.de/media/synthesis/202118/i_f0145_ga_10-1055_a-1485-4666.gif
Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki: Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization
https://www.thieme-connect.de/media/synthesis/202118/i_f0039_ga_10-1055_a-1405-5761.gif
Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto: C–H Bond Functionalization Using Pd- and Au-Supported Catalysts with Mechanistic Insights of the Active Species
https://www.thieme-connect.de/media/synthesis/202118/i_f0140_ga_10-1055_a-1468-1455.jpg
Wei, Yunlong; Chen, Zhiqi; Wu, Zhen; Xu, Yaohui; Wu, Xinxin; Zhu, Chen: Radical Carbosulfonylation of Propellane: Synthesis of Sulfonyl β-Keto-bicyclo[1,1,1]pentanes
https://www.thieme-connect.de/media/synthesis/202118/i_f0143_ga_10-1055_a-1484-1028.gif
Hassan, Mirja Md Mahamudul; Hoque, Md Emdadul; Dey, Sayan; Guria, Saikat; Roy, Brindaban; Chattopadhyay, Buddhadeb: Iridium-Catalyzed Site-Selective Borylation of 8-Arylquinolines
https://www.thieme-connect.de/media/synthesis/202118/i_f0179_ga_10-1055_a-1506-3884.gif
Yuan, Shuqing; Ling, Liang; Tang, Jinghua; Luo, Meiming; Zeng, Xiaoming: Chromium-Catalyzed Reductive Cleavage of Unactivated Aromatic and Benzylic C–O Bonds
https://www.thieme-connect.de/media/synthesis/202118/i_f0232_ga_10-1055_a-1507-6419.gif
Minami, Yasunori; Matsuyama, Nao; Matsuo, Yasuaki; Tamura, Masanori; Sato, Kazuhiko; Nakajima, Yumiko: Catalytic Reductive Cleavage of Poly(phenylene sulfide) Using a Hydrosilane
https://www.thieme-connect.de/media/synthesis/202118/i_f0259_ga_10-1055_a-1518-9010.gif
Xu, Wei; Kohei, Miki; Shibasaki, Masakatsu; Kumagai, Naoya: Strategic Synthesis of Asymmetrically Substituted C4N4 Fluorophores
https://www.thieme-connect.de/media/synthesis/202118/i_f0270_ga_10-1055_a-1516-9399.jpg
Kimura, Naoki; Katta, Shiori; Kitazawa, Yoichi; Kochi, Takuya; Kakiuchi, Fumitoshi: Deuterium-Labeling Studies on the C–H/Olefin Coupling of Aromatic Ketones Catalyzed by Fe(PMe3)4
https://www.thieme-connect.de/media/synthesis/202118/i_f0186_ga_10-1055_s-0040-1706040.gif
Jinnai, Seihou; Oi, Ayumi; Seo, Takuji; Moriyama, Taichi; Minami, Ryunosuke; Higashida, Suguru; Ie, Yutaka: Electron-Accepting π-Conjugated Compound Containing Cyano-Substituted Naphthobisthiadiazole as Nonfullerene Acceptor in Organic Solar Cells
https://www.thieme-connect.de/media/synthesis/202118/i_f0214_ga_10-1055_a-1528-1632.gif

Issue 17/2021

Korvorapun, Korkit; Samanta, Ramesh C.; Rogge, Torben; Ackermann, Lutz: Remote C–H Functionalizations by Ruthenium Catalysis
https://www.thieme-connect.de/media/synthesis/202117/i_f0171_ga_10-1055_a-1485-5156.gif
Aldhous, Timothy P.; Chung, Raymond W. M.; Dalling, Andrew G.; Bower, John F.: Enantioselective Intermolecular Murai-Type Alkene Hydroarylation Reactions
https://www.thieme-connect.de/media/synthesis/202117/i_f0144_ga_10-1055_s-0040-1720406.gif
Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro: Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
https://www.thieme-connect.de/media/synthesis/202117/i_f0005_ga_10-1055_s-0040-1706025.gif
Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro: Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation
https://www.thieme-connect.de/media/synthesis/202117/i_f0107_ga_10-1055_a-1437-9917.gif
Seo, Jia; Chen, Che-Wei; Lee, Woohyeong; Jeon, Ju Eun; Chen, Pei-Ling; Chuang, Shih-Ching; Joo, Jung Min: Palladium-Catalyzed C–H Benzannulation of Functionalized Furans and Pyrroles with Alkynes
https://www.thieme-connect.de/media/synthesis/202117/i_f0134_ga_10-1055_a-1502-3641.gif
Ozaki, Tomoya; Kaga, Atsushi; Saito, Hayate; Yorimitsu, Hideki: Generation of Aryllithium Reagents from N-Arylpyrroles Using Lithium
https://www.thieme-connect.de/media/synthesis/202117/i_z0120_ga_10-1055_a-1482-2567.gif
Yabe, Ryota; Ebe, Yusuke; Nishimura, Takahiro: Iridium-Catalyzed Direct C–H Allylation of Ketimines
https://www.thieme-connect.de/media/synthesis/202117/i_f0137_ga_10-1055_a-1477-7059.gif
Kanyiva, Kyalo Stephen; Tang, King Hung Nigel; Wang, Jiarui; Shibata, Takanori: Palladium-Catalyzed sp3 C–H Benzoxylation of Alanine Derivatives Using Aldehydes under Ambient Conditions
https://www.thieme-connect.de/media/synthesis/202117/i_f0024_ga_10-1055_a-1422-9632.gif
Pan, Feng-Feng; Guo, Peng; Huang, Xiaochuang; Shu, Xing-Zhong: Synthesis of Dibenzyls by Nickel-Catalyzed Homocoupling of Benzyl Alcohols
https://www.thieme-connect.de/media/synthesis/202117/i_f0108_ga_10-1055_a-1467-2432.gif
Tanaka, Shinji; Iwase, Shoutaro; Kanda, Sena; Kato, Marie; Kiriyama, Yutaro; Kitamura, Masato: Ruthenium-Catalyzed Asymmetric Dehydrative Allylic Cyclization of Five-Membered Chalcogen Heteroaromatics
https://www.thieme-connect.de/media/synthesis/202117/i_f0141_ga_10-1055_a-1523-6826.gif
Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke: CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones
https://www.thieme-connect.de/media/synthesis/202117/i_f0481_ga_10-1055_s-0040-1705962.gif

Issue 02/2021

Arjona-Esteban, Alhama; Rausch, Anja; Vysotsky, Myroslav O.; Würthner, Frank: Merocyanine Dyes with Extended Polymethine Chains by Simple Two-Step Condensation Sequence
https://www.thieme-connect.de/media/synthesis/202102/i_c0240_ga_10-1055_s-0040-1707896.gif
Widner, Florian J.; Kieninger, Christoph; Wurst, Klaus; Deery, Evelyne; Lawrence, Andrew D.; Warren, Martin J.; Kräutler, Bernhard: Synthesis, Spectral Characterization and Crystal Structure of Chlororhodibalamin: A Synthesis Platform for Rhodium Analogues of Vitamin B12 and for Rh-Based Antivitamins B12
https://www.thieme-connect.de/media/synthesis/202102/i_c0397_ga_10-1055_s-0040-1707288.gif
Yan, Feng-Zhi; Shao, Yuan-Guang; Zhang, Zibin; Shen, Yan-Feng; Huang, Xue-Chun; Zhang, Pei-Ling; Li, Shijun: Synthesis of Catenanes from a BMP32C10-Based Cryptand Tuned by the Linkage Length of Paraquat Salts
https://www.thieme-connect.de/media/synthesis/202102/i_c0428_ga_10-1055_s-0040-1707290.gif
Mei, Peifeng; Kurosaki, Ryo; Matsumoto, Akinobu; Yamada, Hiroko; Aratani, Naoki: One-Pot Synthesis of a Cyclic Pyrene Octamer from Two Bifunctionalized Pyrene Monomers
https://www.thieme-connect.de/media/synthesis/202102/i_c0439_ga_10-1055_s-0040-1705950.gif

Issue 24/2020

Issue 22/2020

Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
https://www.thieme-connect.de/media/synthesis/202022/i_c0045_ga_10-1055_s-0040-1707994.gif
Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain: Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
https://www.thieme-connect.de/media/synthesis/202022/i_c0232_ga_10-1055_s-0040-1707339.jpg
Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis: Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
https://www.thieme-connect.de/media/synthesis/202022/i_c0207_ga_10-1055_s-0040-1707859.gif
Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda: Copper-Catalyzed Asymmetric Hydroamination of Styrenes with pivZPhos as Ligand
https://www.thieme-connect.de/media/synthesis/202022/i_c0264_ga_10-1055_s-0040-1707346.gif
Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.: Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
https://www.thieme-connect.de/media/synthesis/202022/i_c0401_ga_10-1055_s-0040-1707279.gif

Issue 21/2020

Manne, Srinivasa Rao; de la Torre, Beatriz G.; El-Faham, Ayman; Albericio, Fernando: OxymaPure Coupling Reagents: Beyond Solid-Phase Peptide Synthesis
https://www.thieme-connect.de/media/synthesis/202021/i_c0384_ga_10-1055_s-0040-1706296.jpg
Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.: Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis
https://www.thieme-connect.de/media/synthesis/202021/i_c0186_ga_10-1055_s-0040-1707394.gif
Kolympadi Marković, Maria; Marković, Dean; Laclef, Sylvain: Amide Synthesis by Transamidation of Primary Carboxamides
https://www.thieme-connect.de/media/synthesis/202021/i_c0202_ga_10-1055_s-0040-1707133.gif
Shiri, Morteza; Gholami-Koupaei, Zahra; Bandehali-Naeini, Farzaneh; Tonekaboni, Maryam-Sadat; Soheil-Moghaddam, Saeedeh; Ebrahimi, Delaram; Karami, Sima; Notash, Behrouz: Highly Selective Synthesis of α-Hydroxy, α-Oxy, and α-Oxo Amides by a Post-Passerini Condensation Transformation
https://www.thieme-connect.de/media/synthesis/202021/i_c0210_ga_10-1055_s-0040-1707132.gif
Smolobochkin, Andrey V.; Gazizov, Almir S.; Otegen, Nazerke K.; Voronina, Julia K.; Strelnik, Anna G.; Samigullina, Aida I.; Burilov, Alexander R.; Pudovik, Michail A.: Nucleophilic Cyclization/Electrophilic Substitution of (2,2-Dialkoxyethyl)ureas: Highly Regioselective Access to Novel 4-(Het)arylimidazolidinones and Benzo[d][1,3]diazepinones
https://www.thieme-connect.de/media/synthesis/202021/i_c0158_ga_10-1055_s-0040-1707864.gif
Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.: Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-O-sulfonic Acid in Aqueous Media
https://www.thieme-connect.de/media/synthesis/202021/i_c0225_ga_10-1055_s-0040-1707809.gif

Issue 08/2020

Issue 23/2019