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Aryne Chemistry in Synthesis
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Cycloadditions – Established and Novel Trends – in Celebration of the 70th Anniversary of the Nobel Prize Awarded to Otto Diels and Kurt Alder
Special Issue dedicated to Prof. Sarah Reisman, recipient of the 2019 Dr. Margaret Faul Women in Chemistry Award
Special Issue Dedicated to Professor Shinji Murai – Part II
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Functional Organic Molecules
Recent Advances in Metal-Catalyzed Ring Construction
Synthesis in Industry
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Halogenation Methods (with a View Towards Radioimaging Applications)
Bürgenstock Special Section 2018
Amination Reactions in Organic Synthesis
Ruthenium in Organic Synthesis
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Issue eFirst
Rai, Shweta; Samatha, Polasani; Addipilli, Ramunaidu; Mainkar, Prathama S.; Sripadi, Prabhakar; Adepu, Raju; Chandrasekhar, Srivari:
Poly(ethylene glycol) Dimethyl Ethers (PEGDME): Efficient and Recyclable Solvents for Aryne-Involved Reactions
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PDF (751 kb)
Gillard, Rachel M.; Zhang, Jiajun; Steel, Richard; Wang, Jocelyn; Strull, Jessica L.; Cai, Bin; Chakraborty, Nilanjana; Boger, Dale L.:
Aryl Annulation: A Powerful Simplifying Retrosynthetic Disconnection
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PDF (536 kb)
Majhi, Jadab; Zhou, Bohang; Zhuang, Yuxin; Tom, Mai-Jan; Dai, Huifang; Evans, P. Andrew:
Palladium-Catalyzed Cross-Coupling of Cyanohydrins with Aryl Bromides: Construction of Biaryl Ketones
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PDF (317 kb)
Khatana, Anil Kumar; Singh, Vikram; Gupta, Manoj Kumar; Tiwari, Bhoopendra:
A Highly Efficient NHC-Catalyzed Aerobic Oxidation of Aldehydes to Carboxylic Acids
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PDF (192 kb)
Abuhafez, Naba; Perennes, Antoine; Gramage-Doria, Rafael:
Mimicking Enzymes: Taking Advantage of the Substrate-Recognition Properties of Metalloporphyrins in Supramolecular Catalysis
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PDF (506 kb)
Liu, Cheng-Yuan; Chen, Ying-Ho; Chen, Chih-Hao; Yu, Ming-Shiuan; Tsai, Fu-Yu; Ong, Tiow-Gan:
Selective C(8)–H Activation of Imidazopyridines Mediated by Cooperative Nickel–Aluminum Catalysis
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PDF (219 kb)
Sarmah, Manashi; Hazarika, Hemanta; Gogoi, Pranjal:
Aryne Annulations for the Synthesis of Carbocycles and Heterocycles: An Updated Review
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PDF (1330 kb)
Veth, Lukas; Grab, Hanusch A.; Dydio, Paweł:
Recent Trends in Group 9 Catalyzed C–H Borylation Reactions: Different Strategies To Control Site-, Regio-, and Stereoselectivity
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Kręcijasz, Remigiusz B.; Malinčík, Juraj; Šolomek, Tomáš:
Exploring Silyl Protecting Groups for the Synthesis of Carbon Nanohoops
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PDF (780 kb)
Condon, Sylvie; Nédélec, Jean-Yves:
Overview on Nickel-Catalyzed Electrochemical Conjugate Addition of Organic Halides on Electron-Deficient Olefins
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He, Xiao-Yu; Ma, Yu-Hong; Yang, Qing-Qing; Xiao, Wen-Jing:
[4+n] Annulation Reactions Using
ortho
-Chloromethyl Anilines as Aza-
ortho
-Quinone Methide Precursors
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PDF (637 kb)
Kimura, Masanari; Kojima, Keisuke; Tamaru, Yoshinao:
Nickel-Catalyzed Three-Component Connection Reaction of Dimethylzinc, 1,ω-Ene-Diene, and Acetone: Synthesis of 1,2-Disubstituted Cycloalkanes
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Shirke, Rajendra P.; Reddy, Virsinha; Anand, R. Vijaya; Ramasastry, S. S. V.:
Furans to Benzofurans: Intramolecular Cross-Benzoin Reactions Catalysed by N-Heterocyclic Carbenes
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Moragas, Toni; Martin, Ruben:
Nickel-Catalyzed Reductive Carboxylation of Cyclopropyl Motifs with Carbon Dioxide
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Shi, Shicheng; Lalancette, Roger; Szostak, Michal:
Cyclization of Imides to 2-Azabicycles via Aminoketyl Radicals by Using Samarium(II) Iodide–Water: Reaction Development, Synthetic Scope, and Mechanistic Studies
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Gao, Xing; Han, Jianwei; Wang, Limin:
Chiral Iminophosphorane Organocatalyzed Asymmetric Sulfenylation of 3-Substituted Oxindoles: Substrate-Interrelated Enantioselectivities
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PDF (216 kb)
Cai, Pin-Wen; You, Zhi-Hao; Xie, Liang-Hui; Tan, Rui; Tong, Zhi-Ping; Liu, Yan-Kai:
The Attractive Application of Lactol Chemistry: From Racemic Lactol to Natural Product Skeleton
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PDF (891 kb)
Schweighauser, Luca; Bodoky, Ina; Kessler, Simon N.; Häussinger, Daniel; Wegner, Hermann A.:
Bidentate Lewis Acid Catalyzed Inverse-Electron-Demand Diels–Alder Reaction for the Selective Functionalization of Aldehydes
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Hayashi, Mikishiro; Michikita, Ryudai; Usuki, Yoshinosuke; Satoh, Tetsuya:
Construction of Thienopyrroles through Rhodium-Catalyzed Direct Annulation of (Acetylamino)thiophenes with Alkynes
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Kumar, Raju Suresh; Almansour, Abdulrahman I.; Arumugam, Natarajan; Menéndez, J. Carlos; Osman, Hasnah; Kumar, Raju Ranjith:
Dipolar Cycloaddition-Based Multicomponent Reactions in Ionic Liquids: A Green, Fully Stereoselective Synthesis of Novel Polycyclic Cage Systems with the Generation of Two New Azaheterocyclic Rings
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Nori, Valeria; Sinibaldi, Arianna; Pesciaioli, Fabio; Carlone, Armando:
Impact of Design of Experiments in the Optimisation of Catalytic Reactions in Academia
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PDF (1900 kb)
Kabuki, Akira; Yamaguchi, Junichiro:
Formal Syntheses of Dictyodendrins B, C, and E by a Multi-Substituted Indole Synthesis
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PDF (1039 kb)
Berti, Francesco; Favero, Lucilla; Pineschi, Mauro:
Asymmetric Synthesis of Methylphenidate and Quinolizidinones by Addition of Aldehydes to Piperidine-Based Conjugated
N
-Acyliminium Ions
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PDF (217 kb)
Ledovskaya, Maria S.; Voronin, Vladimir V.; Rodygin, Konstantin S.; Ananikov, Valentine P.:
Acetylene and Ethylene: Universal C
2
Molecular Units in Cycloaddition Reactions
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PDF (2231 kb)
Brandão, Pedro; Pineiro, Marta; Burke, Anthony J.:
Tryptanthrin and Its Derivatives in Drug Discovery: Synthetic Insights
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Patra, Subrata; Mosiagin, Ivan; Giri, Rahul; Katayev, Dmitry:
Organic Nitrating Reagents
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Krishna, Gaddam; Grudinin, Dmitry G.; Nikitina, Eugeniya V.; Zubkov, Fedor I.:
I
ntra
M
olecular
D
iels–
A
lder Reactions of
V
inylarenes and Alkynyl Arenes (the IMDAV Reaction)
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PDF (8084 kb)
Arnold, Jeffrey S.; Nguyen, Hien M.:
Rhodium-Catalyzed Asymmetric Amination of Allylic Trichloroacetimidates
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Shimazumi, Ryoma; Kodama, Takuya; Tobisu, Mamoru:
Palladium-Catalyzed Unimolecular Fragment Coupling of
N
-Allylamides Bearing a Tethered Nucleophile with the Translocation of an Amide Group
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PDF (279 kb)
Artigas, Albert; Hagebaum-Reignier, Denis; Carissan, Yannick; Coquerel, Yoann:
Multidimensional Isotropic Magnetic Shielding Contour Maps for the Visualization of Aromaticity in
ortho
-Arynes and Their Reactions
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PDF (2569 kb)
Frost, Christopher G.; Edwards, Hannah J.; Penrose, Stephen D.; Gleave, Robert:
Exploring Rhodium-Catalysed Conjugate Addition of Chiral Alkenylboronates Using Chiral Olefin Ligands
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PDF (111 kb)
La Torre, Mathéo; Maton, William; Cleator, Ed; Jouffroy, Matthieu:
Pd/C Catalyzed Dehalogenation of (Hetero)aryls Using Triethylsilane as Hydrogen Donor
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PDF (258 kb)
Airiau, Etienne; Chemin, Claire; Girard, Nicolas; Lonzi, Giacomo; Mann, André; Petricci, Elena; Salvadori, Jessica; Taddei, Maurizio:
Microwave-Assisted Domino Hydroformylation/Cyclization Reactions: Scope and Limitations
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PDF (225 kb)
Nocera, Giuseppe; Murphy, John A.:
Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview
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PDF (247 kb)
Wang, Li; Wang, Zhi-Qian; Xu, Ming-Hua; Lin, Guo-Qiang:
Highly Enantioselective Synthesis of (Diarylmethyl)amines by Rhodium-Catalyzed Arylation of
N
-Nosylimines Using a Chiral Bicyclo[3.3.0]diene Ligand
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PDF (104 kb)
Parker, Patrick D.; Pierce, Joshua G.:
Synthesis of 1,2,4-Oxadiazoles via DDQ-Mediated Oxidative Cyclization of Amidoximes
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PDF (196 kb)
Zhang, Qingchen; Wang, Xuan; Qian, Qun; Gong, Hegui:
Nickel-Catalyzed Reductive Cross-Coupling of Benzyl Halides with Aryl Halides
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PDF (191 kb)
Belhomme, Marie-Charlotte; Dru, Delphine; Xiong, Heng-Ying; Cahard, Dominique; Besset, Tatiana; Poisson, Thomas; Pannecoucke, Xavier:
Copper-Mediated Direct Functionalization of Unsaturated C–C Bonds with Ethyl Bromo(difluoro)acetate: A Straightforward Access to Highly Valuable Difluoromethylated Alkenes
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Liu, Jiangguang; Yan, Jiajie; Qin, Dongguang; Cai, Qian:
An Unexpected Inversion of Enantioselectivity in a Copper-Catalyzed Intramolecular Desymmetric Aryl C–N Coupling Reaction
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Székely, Anna; Sinai, Ádám; Tóth, Edina B.; Novák, Zoltán:
Utilization of a Copper on Iron Catalyst for the Synthesis of Biaryl Systems and Benzoxazines via Oxidative Arylation of Anilide Derivatives
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Sperger, Theresa; Schoenebeck, Franziska:
α-Arylation of Esters and Ketones Enabled by a Bench-Stable Pd(I) Dimer Catalyst
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PDF (209 kb)
Agudelo, Brian Castro; Rigoulet, Florian; Giorgi, Michel; Sayah, Babak; Rodriguez, Jean; Coquerel, Yoann:
Synthesis of Axially Chiral Cationic Benzo[
c
]phenanthridinium Derivatives
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PDF (2477 kb)
Liu, Wenting; Hong, Xiaohu; Xu, Bin:
Rhodium-Catalyzed Oxidative Coupling of Aryl Hydrazones with Internal Alkynes: Efficient Synthesis of Multisubstituted Isoquinolines
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PDF (345 kb)
Sebald, Michael A.; Gebauer, Julian; Koch, Matthias:
Concise Syntheses of Alternariol, Alternariol-9-monomethyl Ether and Their D
3
-Isotopologues
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PDF (823 kb)
Wildermuth, Raphael; Speck, Klaus; Magauer, Thomas:
Gold(I)-Catalyzed Enyne Cyclizations: Studies Toward the Total Synthesis of (+)-Aureol
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PDF (262 kb)
Liu, Linhao; Doucet, Henri:
Scope and Limitations of the Palladium-Catalyzed Direct 1,2-Diheteroarylation of 1,2-Dihalobenzene Derivatives
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PDF (343 kb)
Endo, Chikako; Inoue, Yurika; Maruyama, Toshifumi; Minoura, Mao; Murai, Toshiaki:
Two-Step Transesterification of Phosphates, Phosphorothioates, and Phosphonates with a Binaphthyl Group for the Synthesis of
P
-Chirogenic Phosphates and Phosphonates
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PDF (366 kb)
Malkina, Anastasiya G.; Stepanov, Anton V.; Sobenina, Lyubov N.; Shemyakina, Olesya A.; Ushakov, Igor A.; Smirnov, Vladimir I.; Trofimov, Boris A.:
Organocatalyzed Microwave-Assisted Competing Cyclization of Cyanopropargylic Alcohols with Carboxylic Acids: 4-Cyano-3(2
H
)-furanones versus 4-Cyano-[(
Z
)-3-cyanomethylene]-2,3-dihydrofurans
Full Text
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PDF (913 kb)
Li, Zhilong; Tong, Rongbiao:
Asymmetric Total Syntheses of the
trans
-2-Aryl-6-alkyltetrahydropyrans Diospongin B and Parvistones D and E from a Common Precursor
Full Text
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PDF (1319 kb)
Nambu, Hisanori; Ono, Naoki; Yakura, Takayuki:
Acid-Catalyzed Ring-Opening Cyclization of Spirocyclopropanes for the Construction of a 2-Arylbenzofuran Skeleton: Total Synthesis of Cuspidan B
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PDF (255 kb)
Malik, Chanchal K.; Vaultier, Michel; Ghosh, Subrata:
Copper(I)-Catalyzed [2+2] Photocycloaddition of Nonconjugated Alkenes in Room-Temperature Ionic Liquids
Full Text
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PDF (92 kb)
Ma, Yudao; Song, Chun; Chai, Qiang; Ma, Changqin; Andrus, Merritt B.:
Palladium-Imidazolium
N
-Heterocyclic Carbene-Catalyzed Carbonylative Amidation With Boronic Acids, Aryl Diazonium Ions, and Ammonia
Full Text
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PDF (55 kb)
Kabalka, George W.; Yao, Min-Liang:
Synthesis of a Potential Boron Neutron Capture Therapy Agent: 1-Aminocyclobutane-1-carboxylic Acid Bearing a Butylboronic Acid Side Chain
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PDF (63 kb)
Yamaoka, Yousuke; Taniguchi, Marie; Yamada, Ken-ichi; Takasu, Kiyosei:
Asymmetric Total Synthesis of Tylophorine through a Formal [2+2] Cycloaddition Followed by Migrative Ring Opening of a Cyclobutane
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PDF (209 kb)
Islam, Kobirul; Das, Deb K.; Akram, Ejaz; Khan, Abu T.:
Exploration of C5–C6-Unsubstituted 1,4-Dihydropyridines for the Construction of
exo
-Hexahydro-1
H
-chromeno[3,4-
h
][1,6]naphthyridine-3-carboxylates Using a Stereoselective Povarov Reaction
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PDF (971 kb)
Neo, Ana G.; Castellano, Teresa G.; Marcos, Carlos F.:
Enol-Ugi Reaction of Hydroxycoumarins: Straightforward Synthesis of Amino Acid Derived Coumarin Enamines
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PDF (274 kb)
Dobrydnev, Alexey V.; Popova, Maria V.; Saffon-Merceron, Nathalie; Listunov, Dymytrii; Volovenko, Yulian M.:
Synthesis of the First Representatives of Spiro-1λ
6
-isothiazolidine-1,1,4-triones
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PDF (271 kb)
Luo, Guo-Ying; Wu, Hao; Tang, Yu; Li, Hui; Yeom, Hyun-Suk; Yang, Ka; Hsung, Richard P.:
A Total Synthesis of (±)-Rhododaurichromanic Acid A via an Oxa-[3+3] Annulation of Resorcinols
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PDF (219 kb)
Alouane, Nacira; Vrancken, Emmanuel; Mangeney, Pierre:
Preparation of
anti
-1,2-Disubstituted Homopropargylic Alcohols by Addition of Allenyl(cyano)cuprates to Aldehydes
Full Text
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PDF (89 kb)
Apsunde, Tushar Dattu; Trudell, Mark L.:
Microwave-Assisted Iridium-Catalyzed Synthesis of Nicotine and Anabasine Derivatives
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PDF (184 kb)
Cole, Charles J. F.; Chi, Hyung Min; DeBacker, Kenneth C.; Snyder, Scott A.:
Synthesis of Enhanced, Isolable Disulfanium Salts and their Application to Thiiranium-Promoted Polyene Cyclizations
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PDF (212 kb)
Wang, Zheng; Ji, Hongtao; He, Wei-Min; Xiong, Yang; Zhang, Guozhu:
Chromium-Catalyzed Asymmetric Dearomatization–Addition Reactions of Halomethyloxazoles and Indoles
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PDF (195 kb)
Jeganmohan, Masilamani; Cheng, Chien-Hong:
Substituted 1-Allyl-2-allenylbenzenes via Palladium-Catalyzed Allylallenylation of Benzyne Derivatives
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PDF (266 kb)
Ramírez, Jesus; Fernandez, Elena:
Convenient Synthesis of α,α-Difluorinated Carbonyl Compounds from Alkynes through a Fluoro-deboronation Process
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PDF (161 kb)
Olson, Christopher A.; Shaner, Courtnay E.; Roche, Sydney C.; Ferrence, Gregory M.; Mitchell, T. Andrew:
Hexahydro-1
H
-Isoindolinone-Like Scaffolds from Electronically Deactivated and Sterically Hindered Dienes: Synthesis in the Context of Muironolide A
Full Text
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PDF (1001 kb)
Federsel, Hans-Jürgen:
Taking the Green Road Towards Pharmaceutical Manufacturing
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PDF (1046 kb)
Kratzer, Philipp; Gerster, Holger; Maas, Gerhard:
Cycloaddition Reactions of Propyne Iminium Salts and Enol Ethers
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PDF (397 kb)
Amaya-García, Fabián; Unterlass, Miriam M.:
Synthesis of 2,3-Diarylquinoxaline Carboxylic Acids in High-Temperature Water
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PDF (3473 kb)
Zhang, Li; Shi, Jianxun; Fang, Yewen:
An Alternative to the Arbuzov Reaction: Generation and Transformation of α-Dialkyl-Substituted Methylphosphonate Carbanions via an SET Reduction Process
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PDF (319 kb)
Carreiro, Elisabete P.; Gastalho, Carlos M.; Ernesto, Sofia; Costa, Ana R.; Antunes, Célia M.; Burke, Anthony J.:
Synthesis and Antiproliferative Activity of Novel Quercetin-1,2,3-Triazole Hybrids using the 1,3-Dipolar Cycloaddition (Click) Reaction
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PDF (581 kb)
Lindner, Marcin; Krasiński, Antoni; Jurczak, Janusz:
Facile, Stereocontrolled Synthetic Route towards Bis-functionalised Pyrrolizidines
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PDF (418 kb)
Ren, Zhi-Hui; Zhao, Mi-Na; Yi, Yukun; Wang, Yao-Yu; Guan, Zheng-Hui:
Copper-Catalyzed Aerobic Oxidative Cyclization of Ketoxime Acetates with Pyridines for the Synthesis of Imidazo[1,2-
a
]pyridines
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PDF (204 kb)
Xi, Tuo; Chen, Xu; Zhang, Heyi; Lu, Zhan:
Reductive Cyclization of 1,6- and 1,7-Enynes Catalyzed by Iron Complexes
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PDF (203 kb)
Chen, Shi; Mondal, Mukulesh; Ibrahim, Ahmad A.; Wheeler, Kraig A.; Kerrigan, Nessan J.:
Asymmetric Synthesis of Dipropionate Derivatives through Catalytic Hydrogenation of Enantioenriched
E
-Ketene Heterodimers
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PDF (218 kb)
Dai, Wen; Mi, Yuan; Lv, Ying; Shang, Sensen; Li, Guosong; Chen, Guangwen; Gao, Shuang:
Development of a Continuous-Flow Microreactor for Asymmetric Epoxidation of Electron-Deficient Olefins
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Deng, Lu-Jiang; Liu, Jing; Huang, Ji-Qing; Hu, Yanhe; Chen, Mao; Lan, Yu; Chen, Jia-Hua; Lei, Aiwen; Yang, Zhen:
Effect of Lithium Chloride on Tuning the Reactivity of Pauson-Khand Reactions Catalyzed by Palladium-Tetramethylthiourea
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Yamaoka, Yousuke; Miyabe, Hideto; Yasui, Yoshizumi; Takemoto, Yoshiji:
Chiral-Thiourea-Catalyzed Direct Mannich Reaction
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PDF (117 kb)
Jiménez Blanco, José L.; Bootello, Purificación; Gutiérrez Gallego, Ricardo; Ortiz Mellet, Carmen; García Fernández, José M.:
Synthesis of Thiourea-Linked Glycooligomers that Mimic the Branching Patterns of Natural Oligosaccharides
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PDF (300 kb)
Pookkandam Parambil, Shandev; Pulikkal Veettil, Santhini; Dehaen, Wim:
The Synthesis of Five-Membered N-Heterocycles by Cycloaddition of Nitroalkenes with (In)Organic Azides and Other 1,3-Dipoles
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Wang, Jian; Zu, Liansuo; Li, Hao; Xie, Hexin; Wang, Wei:
Cinchona Alkaloid Based Thiourea Promoted Enantioselective Conjugate Addition of N-Heterocycles to Enones
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PDF (122 kb)
Miyabe, Hideto:
Regiocontrol by Halogen Substituent on Arynes: Generation of 3-Haloarynes and Their Synthetic Reactions
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PDF (459 kb)
Pop, Lidia; Golban, Mirabela Ligia; Hădade, Niculina D.; Socaci, Crina; Grosu, Ion:
CuAAC Synthesis of Tetragonal Building Blocks Decorated with Nucleobases
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Oberg, Kevin M.; Cochran, Brian M.; Cook, Matthew J.; Rovis, Tomislav:
The Catalytic Alkylative Desymmetrization of Anhydrides in a Formal Synthesis of Ionomycin
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Nakayama, Yasuaki; Maeda, Yuichiro; Hama, Naoto; Sato, Takaaki; Chida, Noritaka:
Total Synthesis of (–)-Stemoamide by Sequential Overman/Claisen Rearrangement
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Yang, Xiaoyu; Yu, Biao:
Synthesis of Landomycin D: Studies on the Saccharide Assembly
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Settambolo, Roberta:
Crucial Role of β-Elimination in Determining Regio- and Chemoselectivity of the Rhodium-Catalyzed Hydroformylation of
N
-Allylpyrroles: A New Approach to 5,6-Dihydroindolizines
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Zhao, Yating; Huang, Binbin; Yang, Chao; Li, Bing; Xia, Wujiong:
Metal-Free [3+2] Oxidative Coupling of Phenols with Alkenes: Synthesis of Dihydrobenzofurans
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PDF (208 kb)
Vanderghinste, Jaro; Das, Shoubhik:
Applications of Photoredox Catalysis for the Radical-Induced Cleavage of C–C Bonds
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Heinz, Benjamin; Djukanovic, Dimitrije; Siemens, Fiona; Idriess, Mohamed; Martin, Benjamin; Knochel, Paul:
Regioselective Amination or Alkoxylation of Halogenated Amino-, Thio- or Alkoxypyridines via Pyridyne Intermediates
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PDF (269 kb)
Pang, Jia Hao; Ong, Derek Yiren; Watanabe, Kohei; Takita, Ryo; Chiba, Shunsuke:
Leaving Group Ability in Nucleophilic Aromatic Amination by Sodium Hydride–Lithium Iodide Composite
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Ye, Jian-Liang; Liu, Yang; Zhang, Yu-Feng; Yang, Zhi-Ping; Huang, Pei-Qiang:
Studies on the Second-Generation Approach to Loline Alkaloids: Synthesis of
N
-Bus-norloline through
N
-
tert
-Butanesulfinyl Imine Based Asymmetric Vinylogous Mannich Reaction
Full Text
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PDF (632 kb)
Kousara, Mohammad; Bideau, Franck Le; Ibrahim, Rama; Ferry, Angélique; Venot, Pierre-Etienne; Dejean, Camille; Raingeaud, Joël; Dubois, Joëlle; Retailleau, Pascal; Dumas, Françoise:
Suberosanes as Potential Antitumor Agents: First Enantioselective Total Synthesis of (1
S
)-Suberosanone and Configurational Assignment of Suberosenol A
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Konda, Saidulu; Khatravath, Mahender; Mallurwar, Naveen Kumar; Rao, Pallavi; Sripelly, Shivashankar; Iqbal, Javed; Arya, Prabhat:
Stereoselective Synthesis of the C27–C35 Eribulin Fragment and Its Utilization in Building Structurally Diverse Macrocycles
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Huang, Jhih-Yi; Delbianco, Martina:
Recent Developments in Solid-Phase Glycan Synthesis
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Zhang, Zhou; Yi, Jun-Jie; Aslam, Muhammad; Wan, Jie-Ping; Sun, Meng:
Rh(III)-Catalyzed Stereoselective C–H Homoallylation of Indolines with 4-Vinyl-1,3-dioxan-2-ones
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Yu, Mangfei; Zhang, Qian; Wang, Jia; Huang, Peng; Yan, Pengfei; Zhang, Rui; Dong, Dewen:
Triflic Anhydride Mediated Ring-Opening/Recyclization Reaction of α-Carbamoyl α-Oximyl Cyclopropanes with DMF: Synthetic Route to 5-Aminoisoxazoles
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Feng, Yangyang; Huang, Ruofeng; Hu, Liangzhen; Xiong, Yan; Coeffard, Vincent:
Chiral
C
2
-Symmetric Iodoarene-Catalyzed Asymmetric α-Oxidation of β-Keto Esters
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Zhang, Yongda; Lao, Kendricks S.; Sieber, Joshua D.; Xu, Yibo; Wu, Linglin; Wang, Xiao-Jun; Desrosiers, Jean-Nicolas; Lee, Heewon; Haddad, Nizar; Han, Zhengxu S.; Yee, Nathan K.; Song, Jinhua J.; Howell, Amy R.; Senanayake, Chris H.:
Modular Dihydrobenzoazaphosphole Ligands for Suzuki–Miyaura Cross-Coupling
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Komai, Hirotomo; Yoshino, Tatsuhiko; Matsunaga, Shigeki; Kanai, Motomu:
Lewis Acid Catalyzed Benzylic C–H Bond Functionalization of Azaarenes; Addition to Imines and Enones
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Mostefaï, Naouël; Sirol, Sabine; Courmarcel, James; Riant, Olivier:
Air-Accelerated Enantioselective Hydrosilylation of Ketones Catalyzed by Copper(I) Fluoride-Diphosphine Complexes: Investigations of the Effects of Temperature and Ligand Structure
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Auvil, Tyler J.; Mattson, Anita E.:
Internal Lewis Acid Assisted Benzoic Acid Catalysis
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Sugimoto, Kenji; Hoshiba, Yuya; Tsuge, Kiyoshi; Matsuya, Yuji:
Synthesis of Substituted Pyrrolo[2,1-
a
]isoquinolines by Gold-Catalyzed Domino Cyclization of Alkynyl Iminoesters
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Sun, Shutao; Liu, Lei:
Catalytic Enantioselective Alkynylation of Tetrahydroisoquinoline-Based
N
-Acyl Hemiaminals
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Liddon, John T. R.; Rossi-Ashton, James A.; Clarke, Aimee K.; Lynam, Jason M.; Taylor, Richard J. K.; Unsworth, William P.:
Divergent Reactivity of Indole-Tethered Ynones with Silver(I) and Gold(I) Catalysts: A Combined Synthetic and Computational Study
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Zhang, Zhiguo; Schreiner, Peter R.:
Organocatalytic Biomimetic Reduction of Conjugated Nitroalkenes
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Pan, Jie-Hui; Yang, Min; Gao, Qiang; Zhu, Nian-Yong; Yang, Dan:
Bulky Thioureas as New Ligands for Gold(I)-Catalyzed Cyclization of Acetylenic 1,3-Dicarbonyl Compounds
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Kumar, Ravindra; Tamai, Eri; Ohnishi, Akira; Nishimura, Akira; Hoshimoto, Yoichi; Ohashi, Masato; Ogoshi, Sensuke:
Nickel-Catalyzed Enantioselective Synthesis of Cyclobutenes via [2+2] Cycloaddition of α,β-Unsaturated Carbonyls with 1,3-Enynes
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Vishwanath, Manjunatha; Prakash, Muthuraj; Vinayagam, Poopathy; Kesavan, Venkitasamy:
Construction of Polycyclic Fused Pyrrolidines with Three Contiguous Stereocenters via Michael Addition of Vinylmalononitriles to Nitrostyrenes Using
l
-Proline-Derived Thiourea
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Su, Lin; Xu, Ming-Hua:
Asymmetric Reformatsky-Type Reaction of Isatin-Derived
N
-Sulfinyl Ketimines: Efficient and Practical Synthesis of Enantiopure Chiral 2-Oxoindolinyl-β
3,3
-Amino Esters
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Marques, Carolina S.; López, Óscar; Leitzbach, Luisa; Fernández-Bolaños, José G.; Stark, Holger; Burke, Anthony J.:
Survey of New, Small-Molecule Isatin-Based Oxindole Hybrids as Multi-Targeted Drugs for the Treatment of Alzheimer’s Disease
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Nguyen, Thanh V. Q.; Levoin, Armand; Poli, Lorenzo:
Palladium-Catalyzed C7–H (Hetero)arylation of Pyrazolo[1,5-
a
]pyrazines with Heteroarenes and Aryl Iodides with the Assistance of Silver Salts
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Ribeiro Laia, Fernanda M.; Pinho e Melo, Teresa M. V. D.:
Synthesis and Reactivity of Aziridines with Internal Dipolarophiles: An Approach to 1,4-Dihydrochromeno[4,3-
b
]pyrroles and 3-Methylenechromano[4,3-
b
]pyrroles
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Peng, Jing; Ran, Guang-Yao; Du, Wei; Chen, Ying-Chun:
Tertiary-Amine-Catalyzed Asymmetric [3+2] Annulations of Morita–Baylis–Hillman Carbonates of Isatins with Nitroolefins to Construct Spirooxindoles
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Joshi, Madhur S.; Pigge, F. Christopher:
Sequential Pyridine Dearomatization–Mizoroki–Heck Cyclization for the Construction of Fused (Dihydropyrido)isoindolinone Ring Systems
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Carboni, Aude; Dagousset, Guillaume; Magnier, Emmanuel; Masson, Géraldine:
Three-Component Photoredox-Mediated Chloro-, Bromo-, or Iodotrifluoromethylation of Alkenes
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Iwata, Takayuki; Hyodo, Mizuki; Fujiwara, Takumi; Kawano, Ryusei; Kuhn, Leah; Alabugin, Igor V.; Shindo, Mitsuru:
3-Trifluoromethylbenzyne: Precise Orientation in Cycloaddition Reaction Enabled Regioselective Synthesis of Trifluoromethylated Triptycenes
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Firth, James D.; Zhang, Rong; Morgentin, Rémy; Guilleux, Rachel; Kalliokoski, Tuomo; Warriner, Stuart; Foster, Richard; Marsden, Stephen P.; Nelson, Adam:
Exploitation of the Ugi–Joullié Reaction in the Synthesis of Libraries of Drug-Like Bicyclic Hydantoins
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Lanari, Daniela; Piermatti, Oriana; Pizzo, Ferdinando; Vaccaro, Luigi:
Copper(II) Triflate–Sodium Dodecyl Sulfate Catalyzed Preparation of 1,2-Diphenyl-2,3-dihydro-4-pyridones in Aqueous Acidic Medium
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Biswas, Anup; Kundu, Samrat; Pal, Dhananjoy; Pal, Amit; Maji, Modhu Sudan:
Organocatalyzed Oxa-Diels–Alder Reactions: Recent Progress
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Beckendorf, Stephan; Mancheño, Olga García:
'Click'-BINOLs: A New Class of Tunable Ligands for Asymmetric Catalysis
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Gandeepan, Parthasarathy; Rajamalli, Pachaiyappan; Cheng, Chien-Hong:
Palladium-Catalyzed C–H Activation and Cyclization of Anilides with 2-Iodoacetates and 2-Iodobenzoates: An Efficient Method toward Oxindoles and Phenanthridones
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Miller, Daniel K.; Bailey, Christopher A.; Sammelson, Robert E.:
Synthesis of Isoxazolines and Isoxazoles Inspired by Fipronil
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Salomó, Ernest; Orgué, Sílvia; Riera, Antoni; Verdaguer, Xavier:
Efficient Preparation of (
S
)- and (
R
)-
tert
-Butylmethylphosphine–Borane: A Novel Entry to Important P-Stereogenic Ligands
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Xu, Shibo; Su, Shikuan; Zhang, Huiting; Tian, Lumin; Liang, Pengcheng; Chen, Jiawen; Zhang, Yuan; Li, Chunju; Jia, Xueshun; Li, Jian:
Isocyanide-Based Multicomponent Reactions: Rapid Synthesis of a 5,5-Fused Bicyclic Skeleton from α,β-Unsaturated Ketones and Allenoates
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Chuyko, Alexey; Dolgonos, Grygoriy; Shivanyuk, Alexander; Fetyukhin, Volodymyr; Lukin, Oleg:
Simple Synthesis of Complex Amines from the Diels–Alder Adducts of (–)-Cytisine
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Ghosh, Prasanjit; Mondal, Swati Lekha; Baidya, Mahiuddin:
Ascending of Cycloaddition Strategy for N–O Heterocycles
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Cavitt, Marchello A.; France, Stefan:
Aluminum(III)-Catalyzed, Formal Homo-Nazarov-Type Ring-Opening Cyclizations toward the Synthesis of Functionalized Tetrahydroindolizines
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Wertjes, William; Ayers, Sloan; Gao, Qi; Simmons, Eric M.; Beutner, Gregory L.:
A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines
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Sugiyama, Yu-ki; Heigozono, Shiori; Tamura, Kazuhiro; Okamoto, Sentaro:
Iron-Catalyzed Reductive Metalation–Allylation and Metalative Cyclization of 2,3-Disubstituted Oxetanes and Their Stereoselectivity
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Hopf, Henning; Sherburn, Michael S.:
Allenes in Diels–Alder Cycloadditions
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Yang, Yun; Jones, Christopher R.:
The Aryne Ene Reaction
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Salman, Ghazwan Ali; Ali, Asad; Hussain, Munawar; Khera, Rasheed Ahmad; Langer, Peter:
Synthesis of Functionalized Benzofurans by a Double Heck Reaction of 2,3-Dibromofurans and Subsequent 6π-Electrocyclization/Dehydrogenation
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Wu, Zhiqing; Pan, Yinyin; Zhou, Xiangge:
Synthesis of 3-Arylimidazo[1,2-
a
]pyridines by a Catalyst-Free Cascade Process
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Cormier, Morgan; Chardon, Aurélien; Blanchet, Jérôme; Rouden, Jacques; Maddaluno, Jacques; De Paolis, Michaël:
An Organocatalytic Access to Spiro[4.5]decanes and Spiro[4.6]undecanes Containing Aminolactones and 3-Aminopyrrolidines
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Shaw, Subrata; White, James D.:
Asymmetric Catalysis with Iron–Salen Complexes
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Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil:
Ni
II
Cl(1-Naphthyl)(PCy
3
)
2
, An Air-Stable σ-Ni
II
Precatalyst for Quantitative Cross-Coupling of Aryl C–O Electrophiles with Aryl Neopentylglycolboronates
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Malineni, Jagadeesh; Jezorek, Ryan L.; Zhang, Na; Percec, Virgil:
An Indefinitely Air-Stable σ-Ni
II
Precatalyst for Quantitative Cross-Coupling of Unreactive Aryl Halides and Mesylates with Aryl Neopentylglycolboronates
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Nagai, Akira; Kobayashi, Akihiro; Sakata, Yuki; Minami, Yasunori; Uchida, Keisuke; Hosoya, Takamitsu; Yoshida, Suguru:
Synthesis of Multisubstituted Benzenes from Phenols via Multisubstituted Benzynes
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Urawa, Yoshio; Nishiura, Katsutoshi; Souda, Shigeru; Ogura, Katsuyuki:
A Convenient Method for Preparing Aromatic α,β-Unsaturated Ketones from α,β-Unsaturated Acyl Chlorides and Arylboronic Acids via Suzuki-Miyaura Type Coupling Reaction
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Zhang, Ruirui; Peng, Xia; Tan, Jiajing:
Recent Advances in Construction of C(sp
2
)–O Bonds via Aryne Participated Multicomponent Coupling Reactions
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Rosa, Gilber R.; Ebeling, Gunter; Dupont, Jairton; Monteiro, Adriano L.:
A Superior Non-Symmetrical NCP Pincer Type Palladacycle Catalyst Precursor for the Coupling of Aryl Boronic Acids with Aryl Chlorides
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Monasson, Olivier; Malinowski, Maciej; Lubin-Germain, Nadège; Ferry, Angélique:
Hirao Cross-Coupling Reaction as an Efficient Tool to Build Non-natural C2-Phosphonylated Sugars
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Philipps, Arne R.; Fritze, Lars; Erdmann, Nico; Enders, Dieter:
An Asymmetric Organocatalytic Quadruple Domino Reaction Employing a Vinylogous Friedel–Crafts/Michael/Michael/Aldol Condensation Sequence
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Qureshi, Zafar; Schlundt, Waldemar; Lautens, Mark:
Introduction of Hindered Electrophiles via C–H Functionalization in a Palladium-Catalyzed Multicomponent Domino Reaction
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Neochoritis, Constantinos G.; Zhang, Ji; Dömling, Alexander:
Leuckart–Wallach Approach to Sugar Isocyanides and Its IMCRs
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Högermeier, Jens; Trawny, Daniel; Zimmer, Reinhold; Reissig, Hans-Ulrich:
Diels–Alder Reactions of 1,3-Dienes Incorporated into 8-Oxa- and 8-Thiabicyclo[3.2.1]octane Skeletons: A Convenient Access to Complex Tri- and Tetracyclic Compounds
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Kumar, Ketan; Vivekanand, T.; Singh, Bara; Ramasastry, S. S. V.:
C(sp
3
)–H Activation Enabled by (η
3
-Indolylmethyl)palladium Complexes: Synthesis of Monosubstituted Tetrahydrocarbazoles
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Pan, Yuanjia; Lu, Hongjian; Fang, Yewen; Fang, Xinqiang; Chen, Liqun; Qian, Junlu; Wang, Junhua; Li, Chaozhong:
Synthesis of Pyrroles via Copper-Catalyzed Coupling of Amines with Bromoenones
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Estéoule, Audrey; Durán, Fernando; Retailleau, Pascal; Dodd, Robert H.; Dauban, Philippe:
Enantioselective Intramolecular Copper-Catalyzed Aziridination of Sulfamates
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Seck, Insa; Fall, Alioune; Lago, Carmen; Sène, Massène; Gaye, Mohamed; Seck, Matar; Gómez, Generosa; Fall, Yagamare:
Synthesis of a Cholesterol Side-Chain Triazole Analogue via ‘Click’ Chemistry
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Xiao, Fenfen; Zhang, Qing; Wang, Yunxia; Hu, Xiangdong:
Synthetic Studies toward Bi-linderone Lead To Unexpected 6π-Electrocyclization Reactions: A Facile Construction of Highly Congested Spiro Compounds
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Kachkovskyi, Georgii; Cieślak, Marcin; Graczyk, Piotr; Zawadzki, Przemysław; Kalinowska-Tłuścik, Justyna; Werłos, Mateusz:
Photocatalytic Approach to α,α-Difluoroalkyl Alcohols
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Lee, Ju Hee; Kim, Dae Young:
Organocatalytic Highly Enantioselective Mannich-Type Reactions of Fluoromalonate with
N
-Boc-Aldimines
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Oonishi, Yoshihiro; Taniuchi, Ai; Sato, Yoshihiro:
Rhodium(I)-Catalyzed Hydroacylation/Cycloisomerization Cascade Reaction: Application to the Construction of the Tricyclic Core of Guanacastepenes
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Fujimoto, Hayato; Yamamura, Shisato; Takenaka, Namiki; Tobisu, Mamoru:
Phosphine-Catalyzed
Z
-Selective Carbofluorination of Alkynoates Bearing an N-Heteroarene Unit
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Shibata, Takanori; Fukai, Miku; Sekine, Ryosuke; Hazra, Madhurima; Kanyiva, Kyalo Stephen:
Enantioselective Synthesis of Planar-Chiral 1,
n
-Dioxa[
n
]paracyclophane-Based Phosphites and Their Application as Chiral Ligands
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Grugel, Holger; Minuth, Tobias; Boysen, Mike M. K.:
Novel Olefin-Phosphorus Hybrid and Diene Ligands Derived from Carbohydrates
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Deaton, Kimberly R.; Strouse, Christopher S.; Gin, Mary S.:
Selective [2+2+2] Cycloaddition of Nickel-Benzyne and an Asymmetric 1,3-Diyne: An Iterative Route to Substituted [
n
]Acenes
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Durandetti, Muriel; Périchon, Jacques:
Nickel-Catalyzed Electrochemical Coupling of Aryl, Heteroaryl or Vinyl Halides with Activated Alkyl Chlorides: Synthetic and Stereochemical Aspects
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Ambler, Brett R.; Peddi, Santosh; Altman, Ryan A.:
Copper-Catalyzed Decarboxylative Trifluoromethylation of Propargyl Bromodifluoroacetates
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Sahoo, Santosh K.; Jena, Himanshu Sekhar; Majji, Ganesh; Patel, Bhisma K.:
Formation of Imidazolidine-benzothiazole–Copper(II) Complexes via a Copper-Mediated Room-Temperature C–H Activation of Imidazolidinecarbothioamides
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Barker, Timothy J.; Jarvo, Elizabeth R.:
Diene-Ligated Iridium Complexes as Catalysts for Allylation and Methallylation Reactions of Ketones
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Luo, Long; Zhang, Jian-Jian; Ling, Wei-Jian; Shao, Yong-Liang; Wang, Ya-Wen; Peng, Yu:
Unified Synthesis of (–)-Folicanthine and (–)-Ditryptophenaline Enabled by a Room Temperature Nickel-Mediated Reductive Dimerization
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Ugarriza, Iratxe; Reyes, Efraím; Prieto, Liher; Uria, Uxue; Carrillo, Luisa; Vicario, Jose L.:
An Approach to the Synthesis of a Hepatitis C Virus Inhibitor through a Proline-Catalyzed 1,3-Dipolar Cycloaddition Using Acrolein
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Liu, Can; Shen, Ni; Shang, Rui:
Photocatalytic Defluoroalkylation of Trifluoroacetates with Alkenes using 4-(Acetamido)thiophenol
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Zhao, Yanchuan; Zhu, Jieming; Ni, Chuanfa; Hu, Jinbo:
Magnesium Metal-Mediated Reductive Trifluoromethylation of Aldehydes with Phenyl Trifluoromethyl Sulfone
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Tur, Fernando; Mansilla, Javier; Lillo, Victor J.; Saá, José M.:
Constructing Quaternary Centers of Chirality: The Lanthanide Way to Trifluoromethyl-Substituted Tertiary Alcohols
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Prakash, G. K. Surya; Do, Clement; Wang, Fang; Mathew, Thomas; Olah, George A.:
Cyclodehydration of Fluorinated Diols Using the Mitsunobu Reaction: Highly Efficient Synthesis of Trifluoromethylated Cyclic Ethers
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Vasylyev, Maksym; Alper, Howard:
Conventional and Tandem Hydroformylation
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Sato, Kazuyuki; Tarui, Atsushi; Omote, Masaaki; Ando, Akira; Kumadaki, Itsumaro:
Trifluoromethylation of Organic Compounds and Related Reactions
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Mahajan, Bhushan; Aand, Dnyaneshwar; Purwa, Mandeep; Mujawar, Taufiqueahmed; Ghosh, Subhash; Pabbaraja, Srihari; Singh, Ajay K.:
Elements-Continuous-Flow Platform for Coupling Reactions and Anti-viral Daclatasvir API Synthesis
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Guo, Chen; Yue, Xuyi; Qing, Feng-Ling:
Palladium-Catalyzed Cross-Coupling of Ethyl α-Bromo-α-fluoroacetate with Arylboronic Acids: Facile Synthesis of α-Aryl-α-fluoroacetates
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Peddie, Victoria; Pietsch, Markus; Bromfield, Karen M.; Pike, Robert N.; Duggan, Peter J.; Abell, Andrew D.:
Fluorinated β
²
- and β
³
-Amino Acids: Synthesis and Inhibition of α-Chymotrypsin
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Roger, Julien; Sire, Charline; Tsivery, Anthonia; Cattey, Hélène; Hierso, Jean-Cyrille:
Aryl Triflates in Phosphorus-Directed Rhodium(III)-Catalyzed C–H Activation
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Furuya, Takeru; Klein, Johannes E. M. N.; Ritter, Tobias:
Carbon-Fluorine Bond Formation for the Synthesis of Aryl Fluorides
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Denizot, Natacha; Guillot, Régis; Kouklovsky, Cyrille; Vincent, Guillaume:
N
-Iodosuccinimide-Mediated Oxidative Coupling of Indoles and Phenols: A Synthetic Study toward the Benzofuroindoline Moiety of Bipleiophylline
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Liu, Zhao; Kumar, Krishna:
Trifluoromethyl Derivatization of the Ganglioside, G
M1
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Yu, Xingxin; Qiu, Guanyinsheng; Liu, Jianping; Wu, Jie:
Synthesis of 2,3,4,11b-Tetrahydro-1
H
-pyridazino[6,1-
a
]isoquinolines via the Three-Component Reaction of 2-Alkynylbenzaldehydes, a Sulfonohydrazide and Dimethyl Cyclopropane-1,1-dicarboxylate
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Vicente-García, Esther; Ramón, Rosario; Lavilla, Rodolfo:
New Heterocyclic Inputs for the Povarov Multicomponent Reaction
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Tawatari, Tsukasa; Kato, Ritsuki; Takasu, Kiyosei; Takikawa, Hiroshi:
Intramolecular Propargylic Ene Reaction of Benzyne En Route to Highly Functionalized Allenes and Allenamides
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Bortolato, Tommaso; Dyguda, Mateusz; Vega-Peñaloza, Alberto; Dell’Amico, Luca:
Properties and Synthetic Performances of Phenylamino Cyanoarenes under One-Photon Excitation Manifolds
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Wang, Weibo; Xu, Bo; Hammond, Gerald B.:
Synthesis of Fluorohydrins through Electrophilic Fluorination of Allyl Silanes
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Roy, Sudipta Raha; Jadhavar, Pradeep S.; Seth, Kapileswar; Sharma, Kulin K.; Chakraborti, Asit K.:
Organocatalytic Application of Ionic Liquids: [bmim][MeSO
4
] as a Recyclable Organocatalyst in the Multicomponent Reaction for the Preparation of Dihydropyrimidinones and -thiones
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Suzuki, Takeyuki; Ishizaka, Yuka; Ghozati, Kazem; Zhou, Da-Yang; Asano, Kaori; Sasai, Hiroaki:
Enantioselective Multicatalytic Synthesis of α-Benzyl-β-hydroxyindan-1-ones
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Srivastava, Ajay Kumar; Song, Heebum; Park, Seung Bum:
Diversity-Oriented Synthesis of Functionalized Polyheterocycles from Garner Aldehyde
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Sugiyama, Yu-ki; Okamoto, Sentaro:
Regioselective Syntheses of Substituted Pyridines and 2,2′-Bipyridines by Cobalt-Catalyzed [2+2+2] Cycloaddition of α,ω-Diynes with Nitriles
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Zhou, Mingxin; Song, Qiuling:
Synthesis of α-Ketoamides from Aryl Methyl Ketones and
N
,
N
-Dimethylformamide via Copper-Catalyzed Aerobic Oxidative Coupling
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Duong, Hung A.; Nguyen, Tuan Minh; Rosman, Nurul Zubaidah Binte; Tan, Lionel Jia Liang:
Carboxylation of Organoboronic Esters with Potassium Methyl Carbonate under Copper Catalysis
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Zhao, Chenglong; Tan, Zhuozhen; Liang, Zhuye; Deng, Wei; Gong, Hegui:
Nickel-Catalyzed Reductive Allylation of Ketones with Allylic Carbonates
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Swan, Charlie; Maggi, Lorenzo; Park, Mahri; Taylor, Sophie; Shepherd, William; Ball, Liam T.:
Generation of Thiyl Radicals from Air-Stable, Odorless Thiophenol Surrogates: Application to Visible-Light-Promoted C–S Cross-Coupling
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Zajc, Barbara; Kumar, Rakesh:
Synthesis of Fluoroolefins via Julia-Kocienski Olefination
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Walkowiak, Justyna; del Campo, Teresa Martinez; Ameduri, Bruno; Gouverneur, Véronique:
Syntheses of Mono-, Di-, and Trifluorinated Styrenic Monomers
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Gurung, Santosh K.; Thapa, Surendra; Shrestha, Bijay; Giri, Ramesh:
Copper-Catalyzed Cross-Coupling of Aryl- and Heteroaryltriethoxysilanes with Aryl and Heteroaryl Iodides and Bromides
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Metze, Bryan E.; Bhattacharjee, Avik; McCormick, Theresa M.; Stuart, David R.:
Parameterization of Arynophiles: Experimental Investigations towards a Quantitative Understanding of Aryne Trapping Reactions
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Chu, Qiao; Zhou, Yeqin; Ji, Ce; Liu, Ping; Sun, Peipei:
Electrochemical Benzylic C(sp
3
)–H Amidation via Ritter-Type Reaction in the Absence of External Mediator and Oxidant
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Garbarino, Silvia; Protti, Stefano; Basso, Andrea:
Toward a Green Atom Economy: Development of a Sustainable Multicomponent Reaction
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Murakami, Sho; Brudy, Cosima; Bachmann, Moritz; Takemoto, Yoshiji; Pieber, Bartholomäus:
Photocatalytic Cleavage of Trityl Protected Thiols and Alcohols
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Wech, Felix; Gellrich, Urs:
Hydrogenation of Olefins, Alkynes, Allenes, and Arenes by Borane-Based Frustrated Lewis Pairs
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Hunter, Thomas J.; Wang, Yanping; Zheng, Jiamin; O’Doherty, George A.:
Asymmetric Iterative Hydration of Polyene Strategy to Cryptocaryols A and B
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Nishimura, Takahiro; Nagai, Tomotaka; Takechi, Ryosuke; Ebe, Yusuke:
Rhodium-Catalyzed Enantioselective Addition of Tricyclopropylboroxin to
N
-Sulfonylimines
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García-Ruiz, Cristina; Cheng-Sánchez, Iván; Sarabia, Francisco:
Synthesis of (–)- and (+)-Gummiferol via Asymmetric Synthesis of Glycidic Amides
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Morita, Nobuyoshi; Mashiko, Rie; Hakuta, Dai; Eguchi, Daisuke; Ban, Shintaro; Hashimoto, Yoshimitsu; Okamoto, Iwao; Tamura, Osamu:
Gold-Catalyzed Dimeric Cyclization of Isoeugenol and Related 1-Phenylpropenes in Ionic Liquid: Environmentally Friendly and Stereoselective Synthesis of 1,2,3-Trisubstituted 2,3-Dihydro-1
H
-indenes
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Picthall, Daniel; Surgenor, Brian A.; Kilian, Petr:
Convenient and Scalable Synthesis of Aryldichlorophosphines and Primary Arylphosphines via Perthiophosphonic Anhydrides
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Ferro, Rita; Viduedo, Nuno; Santos, A. Sofia; Silva, Artur M. S.; Royo, Beatriz; Marques, M. Manuel B.:
Bimetallic Catalyzed Synthesis of 2-Arylindoles
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Zhu, Mingzhao; Zheng, Nan:
Photoinduced Cleavage of N-N Bonds of Aromatic Hydrazines and Hydrazides by Visible Light
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Yin, Bin; Inagi, Shinsuke; Fuchigami, Toshio:
Selective Electrochemical Fluorodesulfurization of Benzo- and Pyrido-Fused Oxazine Derivatives Using Ex-cell Halogen Mediators
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Tovar, John D.:
Organic Halogenation Chemistry as a Vital Tool for the Construction of Functional π-Conjugated Materials
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Hofmann, Fabian; Gärtner, Cornelius; Kretzschmar, Martin; Schneider, Christoph:
Asymmetric Synthesis of Fused Tetrahydroquinolines via Intramolecular Aza-Diels–Alder Reaction of
ortho
-Quinone Methide Imines
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Schäfer, Gabriel; Reber, Stefan; Ahmetovic, Muhamed; Fleischer, Tony; Leuenberger, Daniel; Blumer, Nicole; Udry, Megan; Abele, Stefan:
Robust and Scalable Reductive Amination Protocol for Electron-Poor Heterocyclic Amines Using Et
3
SiH/TFA as Reducing Agent
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Chiappe, Cinzia; Sanzone, Angelo:
Using the ‘Chemical Tunability’ of Ionic Liquids to Increase Sustainability in the Electrophilic Bromination of Unsaturated Compounds
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Kutsumura, Noriki; Kubokawa, Keisuke; Saito, Takao:
TBAF-Promoted Elimination of Vicinal Dibromides Having an Adjacent O-Functional Group: Syntheses of 2-Bromoalk-1-enes and Alkynes
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Ziegler, Dorothée S.; Klier, Lydia; Müller, Nicolas; Karaghiosoff, Konstantin; Knochel, Paul:
Directed Zincation or Magnesiation of 2- and 4-Pyrones and Their Derivatives
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Lopchuk, Justin M.; Song, Mia; Butler, Blythe; Gribble, Gordon W.:
Synthesis of Heteroaryl-Substituted Pyrroles via the 1,3-Dipolar Cycloaddition of Unsymmetrical Münchnones and Nitrovinylheterocycles
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Cserép, Gergely B.; Demeter, Orsolya; Bätzner, Effi; Kállay, Mihály; Wagenknecht, Hans-Achim; Kele, Péter:
Synthesis and Evaluation of Nicotinic Acid Derived Tetrazines for Bioorthogonal Labeling
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Zhang, Pengke; Hua, Lin; Takahashi, Tamotsu; Jin, Shengnan; Wang, Qilin:
Recent Advances in the Dearomative Skeletal Editing of Mono-azaarenes
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Zeisel, Lukas; Maier, Martin S.; Thorn-Seshold, Oliver:
Efficient and Scalable Syntheses of 1,2-Thiaselenane-4-amine and 1,2-Thiaselenane-5-amine
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Khan, Farooq-Ahmad; Yaqoob, Sana; Qasim, Muhammad Wasim; Ali, Shujaat; Wang, Yan; Jiang, Zi-Hua:
A Robust, Gram-Scale and High-Yield Synthesis of MDP Congeners for Activation of the NOD2 Receptor and Vaccine Adjuvantation
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Garlets, Zachary J.; Wolfe, John P.:
Asymmetric Synthesis of Six-Membered Cyclic Sulfamides via Palladium-Catalyzed Alkene Carboamination Reactions
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Sara, Alexandru A.; Um-e-Farwa, Um-e-Farwa; Saeed, Aamer; Kalesse, Markus:
Recent Applications of the Diels–Alder Reaction in the Synthesis of Natural Products (2017–2020)
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Kageyuki, Ikuo; Yoshida, Hiroto; Takaki, Ken:
Three-Component Carboboration of Alkenes under Copper Catalysis
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Orlandi, Simonetta; Colombo, Federica; Benaglia, Maurizio:
Chiral Diamine-Copper(I) Complexes as Asymmetric Catalysts in the Enantioselective Addition of Phenylacetylene to Imines
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Fernández, Carlos; Diouf, Ousmane; Momán, Edelmiro; Gómez, Generosa; Fall, Yagamare:
OCT Analogues Part 2. Acetylene in the Synthesis of Useful Building Blocks for Analogues of OCT Modified at C-20, C-21, and the D-Ring
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Saejueng, Pranorm; Bates, Craig G.; Venkataraman, D.:
Copper(I)-Catalyzed Coupling of Terminal Acetylenes with Aryl or Vinyl Halides
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Ye, Ke-Yin; Zhao, Zhuo-An; Lai, Zeng-Wei; Dai, Li-Xin; You, Shu-Li:
Highly Regioselective Allylic Substitution Reactions Catalyzed by an Air-Stable (π-Allyl)iridium Complex Derived from Dinaphthocyclooctatetraene and a Phosphoramidite Ligand
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Woof, Callum R.; Linford-Wood, Thomas G.; Mahon, Mary F.; Webster, Ruth L.:
Catalytic Hydrophosphination of Allenes Using an Iron(II) β-Diketiminate Complex
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Zhang, Shuang; Hu, Xiu-Qin; Wang, Zhu-Yin; Xu, Peng-Fei:
Reactions of Sulfonium Salts with 2,3-Dioxopyrrolidine Derivatives: A Concise Synthesis of Spirocyclopropane
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Issue Accepted Manuscripts
Dehnert, Brady W.; Dworkin, Jeremy H.; Kwon, Ohjun:
Dealkenylative Functionalization: Conversion of Alkene C(sp3)–C(sp2) Bonds to C(sp3)–X Bonds Using Redox-Based Radical Processes
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Sartillo-Piscil, Fernando; Romero-Ibañez, Julio; Sandoval-Lira, Jacinto; Cruz-Gregorio, Silvano; Quintero, Leticia; Hernández-Pérez, Julio:
On the Reaction Mechanism of the Selective C(sp3)-H Functionalization of N-Benzyl-Piperidines Mediated by TEMPO Oxoammonium Cation
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Delouche, Thomas; Gadiry-Diallo, Abdoul; Besson, Thierry; Ogoshi, Sensuke; Fruit, Corinne:
Photocatalyst-Free Visible Light-Mediated C-H Perfluoroalkylation of Quinazolin-4(3H)-ones with perfluoroalkyl iodides
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Kaur, Ramandeep; Singh, Harcharan; Arulananda Babu, Srinivasarao:
Pd(II)-catalyzed, directing group-aided C-H arylation, alkylation, benzylation and methoxylation of carbazole-3-carboxamides toward C2,C3,C4 functionalized carbazoles
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Röckl, Johannes L.; Lundberg, Helena:
Samarium and Ytterbium in Organic Electrosynthesis
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Naharwal, Sushma; Kharat, Narendra Dinkar; Mahesha, Chikkagundagal K; Bajaj, Kiran; Sakhuja, Rajeev:
Palladium-Catalyzed Regioselective C-Arylation and C,N-Diarylation of N-Aryl 2,3-dihydrophthalazine-1,4-diones using Diaryliodonium Salts
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Issue 21/2022
Yang, Zhenjie; Cheng, Hong-Gang; Chen, Ruiming; Cao, Liming; Wei, Qiang; Wang, Qingqing; Zhou, Qianghui:
Eight-Step Asymmetric Synthesis of (–)-Berkelic Acid
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Huang, Long-Tao; Hirata, Yuki; Kato, Yoshimi; Lin, Luqing; Kojima, Masahiro; Yoshino, Tatsuhiko; Matsunaga, Shigeki:
Ruthenium(II)/Chiral Carboxylic Acid Catalyzed Enantioselective C–H Functionalization of Sulfoximines
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Huang, Xiao-Ling; Li, Chong; Wang, Juan; Yang, Shang-Dong:
Direct Copper-Catalyzed C-3 Arylation of Diphenylphosphine Oxide Indoles
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Pototskiy, Roman A.; Boym, Mikhail A.; Nelyubina, Yulia V.; Perekalin, Dmitry S.:
Synthesis of Ruthenium Catalysts with a Chiral Arene Ligand Derived from Natural Camphor
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Wang, Huiying; Wang, Mengmeng; Ma, Biao; Dai, Hui-Xiong:
Rhodium-Catalyzed C–H Activation of Indoles for the Construction of Spiroindole Scaffolds
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Li, Mingliang; Wang, Jun:
Recent Advances on Transition-Metal-Catalyzed Asymmetric C–H Arylation Reactions
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Murakami, Kotone; Sakamoto, Kana; Nishimura, Takahiro:
Enantioselective C–H Alkylation of
N
-Arylbenzamides with Vinyl Ethers Catalyzed by an Iridium/Chiral Phosphoramidite–Olefin Complex
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Shirai, Tomohiko; Yamamoto, Yasunori:
Cationic Iridium/Chiral Bidentate Phosphoramidite Catalyzed Asymmetric Hydroarylation
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Xu, Weiwei; Ye, Mengchun:
Enantioselective Cobalt-Catalyzed C–H Functionalization
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Qian, Pu-Fan; Li, Jun-Yi; Zhou, Tao; Shi, Bing-Feng:
Synthesis of
P
- and
S
-Stereogenic Compounds via Enantioselective C–H Functionalization
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Wang, Pu-Sheng; Gong, Liu-Zhu:
Asymmetric C–H Functionalization Enabled by Pd/Chiral Phosphoric Acid Combined Catalysis
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Issue 17/2022
Remete, Attila M.; Nonn, Melinda; Volk, Balázs; Kiss, Loránd:
Developments in the Alkynyltrifluoromethylations of Alkenes and Alkynes
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Fichez, Jeanne; Dupommier, Dorian; Besset, Tatiana:
Direct Synthesis of Disubstituted Trifluoromethylthiolated Alkenes
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Gonda, Zsombor; Földesi, Tamás; Nagy, Bálint; Novák, Zoltán:
Modular Synthesis of Carbazole-Substituted Phthalimides as Potential Photocatalysts
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Salamon-Krokosz, Katarzyna; Gołdyn, Mateusz; Siodła, Tomasz; Bartoszak-Adamska, Elżbieta; Koroniak, Henryk; Koroniak-Szejn, Katarzyna:
Fluorinated Olefinic Lactams: The Case of Amino Acids – Preparation and Mechanistic Studies
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Uchikura, Tatsuhiro; Yokohama, Sosuke; Murakami, Mona; Akiyama, Takahiko:
Chiral Calcium Phosphate Catalyzed Enantioselective Synthesis of All-Carbon Quaternary Center by Friedel–Crafts Alkylation Reaction of Pyrroles and Trifluoromethylated Nitrostyrenes
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Cruz-Hernández, Carlos; Juaristi, Eusebio:
On the Synthesis of a Novel Chiral Phosphorodiamidic Acid Containing the α-Phenylethyl Moiety: Insights on its Conformation and Reactivity
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El Haimer, Mohamed; Faragó, Tünde; Schelz, Zsuzsanna; Zupkó, István; Palkó, Márta:
Synthesis of Alicyclic 2-Methylenethiazolo[2,3-
b
]quinazolinone Derivatives via Base-Promoted Cascade Reactions
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Garnes-Portolés, Francisco; Miguélez, Rubén; Grayson, Matthew N.; Barrio, Pablo:
Heteroatom-Tethered ω-Alkenylallylboronates: Stereoselective Synthesis of Heterocyclic Derived Alcohols
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Dargó, Gyula; Nagy, Sándor; Kis, Dávid; Bagi, Péter; Mátravölgyi, Béla; Tóth, Blanka; Huszthy, Péter; Drahos, László; Kupai, József:
Application of Proline-Derived (Thio)squaramide Organocatalysts in Asymmetric Diels–Alder and Conjugate Addition Reactions
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Raji, Mounir; Le, Tam Minh; Csámpai, Antal; Nagy, Viktória; Zupkó, István; Szakonyi, Zsolt:
Stereoselective Synthesis and Applications of Pinane-Based Chiral 1,4-Amino Alcohol Derivatives
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Molnár, István G.; Mucsi, Zoltán; Kovács, Ervin; Nyerges, Miklós:
Electrocyclization and Unexpected Reactions of Non-Stabilized α,β:γ,δ-Unsaturated Azomethine Ylides: Experimental and Theoretical Studies
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Cserép, Gergely B.; Németh, Krisztina; Szatmári, Ágnes; Horváth, Flóra; Imre, Tímea; Németh, Krisztina; Kele, Péter:
Beyond the Bioorthogonal Inverse-Electron-Demand Diels–Alder Reactions of Tetrazines: 2-Pyrone-Functionalized Fluorogenic Probes
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Szabó, Tímea; Görür, Funda Lidya; Horváth, Simon; Volk, Balázs; Milen, Mátyás:
Synthesis of Racemic and Enantiopure Forms of β-Carboline Alkaloid Brevicolline
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Berecz, Gábor; Dancsó, András; Németh, Dóra R.; Kiss, Loránd; Simig, Gyula; Volk, Balázs:
Towards Tianeptine Analogues: Synthesis of New Ring Systems Containing a Dibenzo[
c
,
f
][1,2]thiazepine
S
,
S
-Dioxide Core
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Takao, Go; Hakozaki, Tomohiro; Miura, Keisuke; Urushibara, Yusuke; Fuchibe, Kohei; Ichikawa, Junji:
Construction of Substituted [4]Acene Frameworks Based on Double Cationic Cyclizations of Fluoroalkenes
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Harsági, Nikoletta; Kiss, Nóra Zsuzsa; Drahos, László; Keglevich, György:
Synthesis of Cyclic Phosphinates by Microwave-Assisted Ionic-Liquid-Promoted Alcoholysis
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Issue 04/2022
He, Jian; Liu, Qiang:
Highly Efficient Visible-Light-Driven [2+2] Cycloaddition of Maleimides to Alkenes and Alkynes for the Synthesis of 3-Azabicyclo[3.2.0]heptane-Fused Scaffolds
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Qureshi, Asif Ali; Sanjeeva Kumar, Arpula; Chauhan, Sachin; Kumara Swamy, K. C.:
Stereo- and Regioselective [3+2] Cycloaddition of Acetoxy Allenoates with Azides: Metal-Free Synthesis of Multisubstituted Triazoles
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Barday, Manuel; Nicolas, Eva; Higginson, Bradley; Delmotte, François; Appelmans, Martin; Aïssa, Christophe:
Tandem Nickel-Catalyzed Dimerization/(4+2) Cycloaddition of Terminal Alkynes with Four-Membered Ring Ketones
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Issue 22/2021
Lam, Heather; Abel-Snape, Xavier; Köllen, Martin F.; Lautens, Mark:
Recent Advances in Transition-Metal-Free (4+3)-Annulations
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Ryan, Jonathon S.; Schindler, Corinna S.:
Total Synthesis of Mycocyclosin and the Herqulines
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Sokol, Kevin Rafael; Magauer, Thomas:
Total Synthesis of Oxepin and Dihydrooxepin Containing Natural Products
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Martín-Heras, Víctor; Daniliuc, Constantin G.; Gilmour, Ryan:
An I(I)/I(III) Catalysis Route to the Heptafluoroisopropyl Group: A Privileged Module in Contemporary Agrochemistry
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Wood, Devin P.; Guan, Weiyang; Lin, Song:
Titanium and Cobalt Bimetallic Radical Redox Relay for the Isomerization of
N
-Bz Aziridines to Allylic Amides
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Garry, Olivia L.; Mansfield, Steven J.; Anderson, Edward A.:
Regio- and Stereoselective Addition of Brønsted Acids to Yndiamides: Synthesis of
N
,
O
,
N
- and
N
,
S
,
N
-Trisubstituted Ketene Acetals
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Tien, Chieh-Hung; Trofimova, Alina; Shao, Wenjie; Yudin, Andrei K.:
Synthesis of Borylated Hydrazino Acid Derivatives
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Kasim, Johanes K.; Kavianinia, Iman; Bull, Matthew; Harris, Paul W. R.; Smaill, Jeff B.; Patterson, Adam V.; Brimble, Margaret A.:
Fourth-Generation Analogues of the Anticancer Peptaibol Culicinin D: Probing the Effects of Hydrophobicity and Halogenation on Cytotoxicity
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Wienhold, Sebastian; Fritz, Lukas; Judt, Tatjana; Hackl, Sabrina; Neubauer, Thomas; Sauerer, Bastian; Bach, Thorsten:
Studies towards the Synthesis of (–)-Pulvomycin: Construction of the C12–C40 Segment by a Stereoselective Aldol Reaction
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El Khoury, Anton; Seidler, Paul M.; Eisenberg, David S.; Harran, Patrick G.:
Catalytic Synthesis of PEGylated EGCG Conjugates that Disaggregate Alzheimer’s Tau
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Caldora, Henry P.; Govaerts, Sebastian; Dighe, Shashikant U.; Turner, Oliver J.; Leonori, Daniele:
A
de novo
Synthesis of Oxindoles from Cyclohexanone-Derived γ-Keto-Ester Acceptors Using a Desaturative Amination–Cyclization Approach
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Wong, Jonathan J.; Chen, Xiangyang; Houk, Kendall N.; Vollhardt, K. Peter C.:
The Trajectory of the (
η
5
-Cyclopentadienyl)cobalt-Mediated Cycloisomerization of Ene-Yne-Ene-Type Allyl Propargylic Ethers to Furans: A DFT Appraisal
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Davis, Christopher W.; Bingham, Tanner W.; Okumura, Mikiko; Sarlah, David:
Dearomative
syn
-1,2-Diamination of Benzene and Naphthalene
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Jaye, Joseph A.; Sletten, Ellen M.:
Simple Synthesis of Fluorinated Ene-Ynes via In Situ Generation of Allenes
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Wang, Lin; Ni, Shengyang; Cornella, Josep:
Validation of Arylphosphorothiolates as Convergent Substrates for Ar-SF
4
Cl and Ar-SF
5
Synthesis
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Issue 18/2021
Basak, Sumon; Biswas, Jyoti Prasad; Maiti, Debabrata:
Transition-Metal-Catalyzed C–H Arylation Using Organoboron Reagents
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De, Pinaki Bhusan; Asako, Sobi; Ilies, Laurean:
Recent Advances in the Use of Sodium Dispersion for Organic Synthesis
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Tang, Zhi; Tong, Zhou; Qiu, Renhua; Yin, Shuang-Feng; Kambe, Nobuaki:
Recent Advances on Benzofuranones: Synthesis and Transformation via C–H Functionalization
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Misal Castro, Luis C.; Sultan, Ibrahim; Tsurugi, Hayato; Mashima, Kazushi:
Pyridine-Mediated B–B Bond Activation of (RO)
2
B–B(OR)
2
for Generating Borylpyridine Anions and Pyridine-Stabilized Boryl Radicals as Useful Boryl Reagents in Organic Synthesis
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Maeda, Kyogo; Motokura, Ken:
Recent Advances in Heterogeneous Ir Complex Catalysts for Aromatic C–H Borylation
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Doiuchi, Daiki; Uchida, Tatsuya:
Recent Strategies in Non-Heme-Type Metal Complex-Catalyzed Site-, Chemo-, and Enantioselective C–H Oxygenations
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Sihag, Pinki; Jeganmohan, Masilamani:
Recent Advances in Transition-Metal-Catalyzed C–H Functionalization Reactions Involving Aza/Oxabicyclic Alkenes
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Jung, Jieun; Saito, Susumu:
Recent Advances in Light-Driven Carbon–Carbon Bond Formation via Carbon Dioxide Activation
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Ishida, Tamao; Zhang, Zhenzhong; Murayama, Haruno; Yamamoto, Eiji; Tokunaga, Makoto:
C–H Bond Functionalization Using Pd- and Au-Supported Catalysts with Mechanistic Insights of the Active Species
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Zhang, Zhuo-Zhuo; Zhou, Gang; Huang, Fan-Rui; Shi, Bing-Feng:
Cobalt-Catalyzed Oxidative [4+2] Annulation of Benzamides with Dihydrofuran: A Facile Route to Tetrahydrofuro[2,3-
c
]isoquinolinones
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Wan, Bin; Zhang, Yanghui:
Synthesis of Unsymmetrically Substituted Tetraphenylenes through Palladium-Catalyzed C(sp
2
)–H Activation
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Dalal, Arup; Babu, Srinivasarao Arulananda:
Pd(II)-Catalyzed Directing-Group-Aided C–H Arylation and Alkylation of Pyrene Core: Synthesis of C1,C2- and C1,C10-Disubstituted Pyrene Motifs
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Wei, Yunlong; Chen, Zhiqi; Wu, Zhen; Xu, Yaohui; Wu, Xinxin; Zhu, Chen:
Radical Carbosulfonylation of Propellane: Synthesis of Sulfonyl β-Keto-bicyclo[1,1,1]pentanes
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Hassan, Mirja Md Mahamudul; Hoque, Md Emdadul; Dey, Sayan; Guria, Saikat; Roy, Brindaban; Chattopadhyay, Buddhadeb:
Iridium-Catalyzed Site-Selective Borylation of 8-Arylquinolines
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Yuan, Shuqing; Ling, Liang; Tang, Jinghua; Luo, Meiming; Zeng, Xiaoming:
Chromium-Catalyzed Reductive Cleavage of Unactivated Aromatic and Benzylic C–O Bonds
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Minami, Yasunori; Matsuyama, Nao; Matsuo, Yasuaki; Tamura, Masanori; Sato, Kazuhiko; Nakajima, Yumiko:
Catalytic Reductive Cleavage of Poly(phenylene sulfide) Using a Hydrosilane
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Xu, Wei; Kohei, Miki; Shibasaki, Masakatsu; Kumagai, Naoya:
Strategic Synthesis of Asymmetrically Substituted C4N4 Fluorophores
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Gu, Zheng-Yang; Wu, Yang; Jin, Feng; Bao, Xiaoguang; Xia, Ji-Bao:
Intermolecular C–H Amidation of Alkenes with Carbon Monoxide and Azides via Tandem Palladium Catalysis
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Morimoto, Tsumoru; Wang, Chuang; Tanimoto, Hiroki; Artok, Levent; Kakiuchi, Kiyomi:
Rhodium(I)-Catalyzed CO-Gas-Free Arylative Dual-Carbonylation of Alkynes with Arylboronic Acids via the Formyl C–H Activation of Formaldehyde
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Kimura, Naoki; Katta, Shiori; Kitazawa, Yoichi; Kochi, Takuya; Kakiuchi, Fumitoshi:
Deuterium-Labeling Studies on the C–H/Olefin Coupling of Aromatic Ketones Catalyzed by Fe(PMe
3
)
4
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Jinnai, Seihou; Oi, Ayumi; Seo, Takuji; Moriyama, Taichi; Minami, Ryunosuke; Higashida, Suguru; Ie, Yutaka:
Electron-Accepting π-Conjugated Compound Containing Cyano-Substituted Naphthobisthiadiazole as Nonfullerene Acceptor in Organic Solar Cells
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Rawat, Vishal Kumar; Higashida, Kosuke; Sawamura, Masaya:
Nickel-Catalyzed Homocoupling of Aryl Ethers with Magnesium Anthracene Reductant
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Fukuyama, Takahide; Hamada, Yuki; Ryu, Ilhyong:
A New Protocol for Catalytic Reduction of Alkyl Chlorides Using an Iridium/Bis(benzimidazol-2′-yl)pyridine Catalyst and Triethylsilane
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Issue 17/2021
Korvorapun, Korkit; Samanta, Ramesh C.; Rogge, Torben; Ackermann, Lutz:
Remote C–H Functionalizations by Ruthenium Catalysis
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Vijaykumar, Muniyappa; Punji, Benudhar:
Advances in Transition-Metal-Catalyzed C–H Bond Oxygenation of Amides
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Ohno, Shohei; Miyoshi, Makoto; Murai, Kenichi; Arisawa, Mitsuhiro:
Non-Directed β- or γ-C(sp
3
)–H Functionalization of Saturated Nitrogen-Containing Heterocycles
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Aldhous, Timothy P.; Chung, Raymond W. M.; Dalling, Andrew G.; Bower, John F.:
Enantioselective Intermolecular Murai-Type Alkene Hydroarylation Reactions
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Oonishi, Yoshihiro; Sakamoto, Shunki; Agata, Shuya; Sato, Yoshihiro:
Rhodium(I)-Catalyzed Enantioselective Cyclization of Enynes through Site-Selective C(sp
3
)–H Bond Activation Triggered by Formation of Rhodacycle
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Watanabe, Hikaru; Nakajima, Kazuki; Ekuni, Kento; Edagawa, Ryota; Akagi, Yuta; Okuda, Yasuhiro; Wakamatsu, Kan; Orita, Akihiro:
Custom-Made Pyrene Photocatalyst-Promoted Desulfonylation of Arylethenyl Sulfones Using Green-Light-Emitting Diodes
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Akahori, Shuhei; Fujihara, Tetsuaki; Tsuji, Yasushi; Shinokubo, Hiroshi; Miyake, Yoshihiro:
Synthesis of Tetrasilatetrathia[8]circulenes through C–I and C–H Silylation
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Seo, Jia; Chen, Che-Wei; Lee, Woohyeong; Jeon, Ju Eun; Chen, Pei-Ling; Chuang, Shih-Ching; Joo, Jung Min:
Palladium-Catalyzed C–H Benzannulation of Functionalized Furans and Pyrroles with Alkynes
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Fukumoto, Yoshiya; Shiratani, Motohiro; Noguchi, Hikaru; Chatani, Naoto:
Iridium-Catalyzed Direct Amidation of Imidazoles at the C-2 Position with Isocyanates in the Presence of Hydrosilanes Leading to Imidazole-2-Carboxamides
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Ozaki, Tomoya; Kaga, Atsushi; Saito, Hayate; Yorimitsu, Hideki:
Generation of Aryllithium Reagents from
N
-Arylpyrroles Using Lithium
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Inai, Yasuhito; Usuki, Yoshinosuke; Satoh, Tetsuya:
Synthesis of Benzo-Fused Cyclic Compounds via Rhodium-Catalyzed Decarboxylative Coupling of Aromatic Carboxylic Acids with Alkynes
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Shimazumi, Ryoma; Morita, Kosuke; Yoshida, Tomoki; Yasui, Kosuke; Tobisu, Mamoru:
Late-Stage Derivatization of Buflavine by Nickel-Catalyzed Direct Substitution of a Methoxy Group via C–O Bond Activation
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You, Jingwen; Chen, Qiang; Nishihara, Yasushi:
Nickel-Catalyzed Decarbonylative Thioetherification of Acyl Fluorides via C–F Bond Activation
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Yabe, Ryota; Ebe, Yusuke; Nishimura, Takahiro:
Iridium-Catalyzed Direct C–H Allylation of Ketimines
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Ohmura, Toshimichi; Yagi, Kaito; Torigoe, Takeru; Suginome, Michinori:
Intramolecular Addition of a Dimethylamino C(sp
3
)–H Bond across C–C Triple Bonds Using IrCl(DTBM-SEGPHOS)(ethylene) Catalyst: Synthesis of Indoles from 2-Alkynyl-
N
-methylanilines
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Takahashi, Hiroto; Honjo, Yusaku; Shibata, Yu; Nagashima, Yuki; Tanaka, Ken:
Dienylation of Unfunctionalized Arenes with 1,6-Diynes via Rhodium-Catalyzed Directing-Group-Free C–H Bond Activation
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Kawakami, Haruka; Nohira, Itsuki; Chatani, Naoto:
Nickel-Catalyzed C–F/N–H Annulation of 2-(2-Fluoroaryl) N-Heteroaromatic Compounds with Alkynes: Activation of C–F Bonds
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Yamamoto, Sonoka; Shibuya, Yushin; Suzuki, Toyoko; Okano, Kentaro; Horie, Masaki; Mori, Atsunori:
One-Shot Deprotonative Metalation/Transmetalation/Polymerization of Halothiophenes Catalyzed by Nickel Complex for Polythiophene Synthesis
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Kanyiva, Kyalo Stephen; Tang, King Hung Nigel; Wang, Jiarui; Shibata, Takanori:
Palladium-Catalyzed sp
3
C–H Benzoxylation of Alanine Derivatives Using Aldehydes under Ambient Conditions
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Pan, Feng-Feng; Guo, Peng; Huang, Xiaochuang; Shu, Xing-Zhong:
Synthesis of Dibenzyls by Nickel-Catalyzed Homocoupling of Benzyl Alcohols
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Kiyosu, Yuuki; Tanaka, Shino; Okumura, Sota; Kiyokawa, Kensuke; Minakata, Satoshi:
Synthesis of Fused Diaziridine Derivatives from Cyclic Secondary Amines by Utilizing
N
-Bromosulfonamides as an Aminating Reagent
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Ninokata, Ryo; Korogi, Riho; Nakao, Junya; Fukuda, Tsutomu; Onodera, Gen; Kimura, Masanari:
Reconstruction of Carbon Bond Frameworks via Oxapalladacycles Promoted by the Synergistic Effect of Palladium Catalyst and Triethylborane
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Tanaka, Shinji; Iwase, Shoutaro; Kanda, Sena; Kato, Marie; Kiriyama, Yutaro; Kitamura, Masato:
Ruthenium-Catalyzed Asymmetric Dehydrative Allylic Cyclization of Five-Membered Chalcogen Heteroaromatics
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Kona, Chandrababu Naidu; Oku, Rikuto; Nishii, Yuji; Miura, Masahiro:
Peri
-Selective Direct Acylmethylation and Amidation of Naphthalene Derivatives Using Iridium and Rhodium Catalysts
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Ishida, Naoyoshi; Iwamoto, Hiroaki; Sunagawa, Denise Eimi; Ohashi, Masato; Ogoshi, Sensuke:
CsF-Catalyzed Fluoroacylation of Tetrafluoroethylene Using Acyl Fluorides for the Synthesis of Pentafluoroethyl Ketones
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Xu, Wengang; Wu, Mingbo; Yoshikai, Naohiko:
Iron-Catalyzed Remote C–H Alkylation of 8-Amidoquinolines with Cycloalkanes
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Issue 02/2021
Arjona-Esteban, Alhama; Rausch, Anja; Vysotsky, Myroslav O.; Würthner, Frank:
Merocyanine Dyes with Extended Polymethine Chains by Simple Two-Step Condensation Sequence
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Yoshimura, Aya; Henmi, Keisuke; Kimura, Hitoshi; Sakakibara, Ryo; Ochi, Rika; Shirahata, Takashi; Yorimitsu, Hideki; Misaki, Yohji:
Synthesis of Peripherally Arylated Tetrathiafulvalenes Extended with an Anthraquinoid Spacer via Pd-Catalyzed C–H Arylation and Construction of a Double-Helical Cobalt-Based Metal-Organic Framework
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Widner, Florian J.; Kieninger, Christoph; Wurst, Klaus; Deery, Evelyne; Lawrence, Andrew D.; Warren, Martin J.; Kräutler, Bernhard:
Synthesis, Spectral Characterization and Crystal Structure of Chlororhodibalamin: A Synthesis Platform for Rhodium Analogues of Vitamin B
12
and for Rh-Based Antivitamins B
12
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Yan, Feng-Zhi; Shao, Yuan-Guang; Zhang, Zibin; Shen, Yan-Feng; Huang, Xue-Chun; Zhang, Pei-Ling; Li, Shijun:
Synthesis of Catenanes from a BMP32C10-Based Cryptand Tuned by the Linkage Length of Paraquat Salts
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Mei, Peifeng; Kurosaki, Ryo; Matsumoto, Akinobu; Yamada, Hiroko; Aratani, Naoki:
One-Pot Synthesis of a Cyclic Pyrene Octamer from Two Bifunctionalized Pyrene Monomers
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Issue 24/2020
Qin, Jing-Hao; Li, Jin-Heng; An, De-Lie:
Recent Advances in Cycloaddition Reactions with Alkynes to Construct Heterocycles
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Pellissier, Hélène:
The Use of Domino Reactions for the Synthesis of Chiral Rings
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Wei, Bin; Li, Ke-Wei; Wu, Yan-Chen; Tong, Shi-Qi; Song, Ren-Jie:
Radical Strategy for the Transition-Metal-Catalyzed Synthesis of γ-Lactones: A Review
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Huang, Min-Hua; Hao, Wen-Juan; Jiang, Bo:
Iridium(III)-Catalyzed Difluoroalkylation–Bicyclization of 1,7-Enynes toward Benzo[
a
]fluoren-5-ones under Visible-Light Photoredox Conditions
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Issue 22/2020
Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.:
Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
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Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain:
Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
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Wächtler, Andreas; Bremer, Matthias; Maillard, David; Mohr, Thomas:
Controlling the All-
trans
Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds
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Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis:
Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
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Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda:
Copper-Catalyzed Asymmetric Hydroamination of Styrenes with
piv
ZPhos as Ligand
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Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.:
Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
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Issue 21/2020
Shiri, Morteza; Farajinia-Lehi, Noushin; Salehi, Parvin; Tanbakouchian, Zahra:
Transition Metal and Inner Transition Metal Catalyzed Amide Derivatives Formation through Isocyanide Chemistry
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Manne, Srinivasa Rao; de la Torre, Beatriz G.; El-Faham, Ayman; Albericio, Fernando:
OxymaPure Coupling Reagents: Beyond Solid-Phase Peptide Synthesis
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Zhao, Baoli; Liu, Yunyun:
Step-Economical C–H Activation Reactions Directed by In Situ Amidation
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Spiliopoulou, Nikoleta; Constantinou, Constantinos T.; Triandafillidi, Ierasia; Kokotos, Christoforos G.:
Synthetic Approaches to Acyl Hydrazides and Their Use as Synthons in Organic Synthesis
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Kolympadi Marković, Maria; Marković, Dean; Laclef, Sylvain:
Amide Synthesis by Transamidation of Primary Carboxamides
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Shiri, Morteza; Gholami-Koupaei, Zahra; Bandehali-Naeini, Farzaneh; Tonekaboni, Maryam-Sadat; Soheil-Moghaddam, Saeedeh; Ebrahimi, Delaram; Karami, Sima; Notash, Behrouz:
Highly Selective Synthesis of α-Hydroxy, α-Oxy, and α-Oxo Amides by a Post-Passerini Condensation Transformation
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Movahed, Farzaneh Soleymani; Sawant, Dinesh N.; Bagal, Dattatraya B.; Saito, Susumu:
Tris(
o
-phenylenedioxy)cyclotriphosphazene as a Promoter for the Formation of Amide Bonds Between Aromatic Acids and Amines
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Smolobochkin, Andrey V.; Gazizov, Almir S.; Otegen, Nazerke K.; Voronina, Julia K.; Strelnik, Anna G.; Samigullina, Aida I.; Burilov, Alexander R.; Pudovik, Michail A.:
Nucleophilic Cyclization/Electrophilic Substitution of (2,2-Dialkoxyethyl)ureas: Highly Regioselective Access to Novel 4-(Het)arylimidazolidinones and Benzo[
d
][1,3]diazepinones
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Verma, Saumya; Kumar, Puneet; Khatana, Anil K.; Chandra, Dinesh; Yadav, Ajay K.; Tiwari, Bhoopendra; Jat, Jawahar L.:
Zinc(II)-Catalyzed Synthesis of Secondary Amides from Ketones via Beckmann Rearrangement Using Hydroxylamine-
O
-sulfonic Acid in Aqueous Media
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Kabes, Connor Q.; Gunn, Jack H.; Selbst, Maximilian A.; Lucas, Reagan F.; Gladysz, John A.:
Syntheses of Enantiopure 1,2-Ethylenediamines with Tethered Secondary Amines of the Formula H
2
NCH
2
CH[(CH
2
)
n
NHMe]NH
2
(
n
= 1–4) from α-Amino Acids: New Agents for Asymmetric Catalysis
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Zhang, Rui; Zhang, Jun-Chao; Zhang, Wei-Yi; He, Yu-Qing; Cheng, Hua; Chen, Cheng; Gu, Yu-Cheng:
A Practical Approach for the Transamidation of
N
,
N
-Dimethyl Amides with Primary Amines Promoted by Sodium
tert
-Butoxide under Solvent-Free Conditions
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Issue 08/2020
Connon, Robert; Carroll, Laura; Guiry, Patrick J.:
A Base-Promoted One-Pot Asymmetric Friedel–Crafts Alkylation/Michael Addition of 4-Substituted Indoles
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Yang, Yuzhong; Zhou, Liwei; Yang, Xiumei; Luo, Xiai; Deng, Guobo; Yang, Yuan; Liang, Yun:
Synthesis of Phenanthrenes via Palladium-Catalyzed Three-Component Domino Reaction of Aryl Iodides, Internal Alkynes, and
o
-Bromobenzoic Acids
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Henkel, Michael; Bach, Thorsten:
Annulation of Indoles with 1,n-Dibromoalkanes by a Pd(II)-Catalyzed and Norbornene-Mediated Reaction Cascade
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Shen, Zican; Li, Chen; Mercado, Brandon Q.; Ellman, Jonathan A.:
Cobalt(III)-Catalyzed Diastereoselective Three-Component C–H Bond Addition to Butadiene and Activated Ketones
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Lee, Sumin; Jang, Young Jin; Phipps, Erik J. T.; Lei, Honghui; Rovis, Tomislav:
Rhodium(III)-Catalyzed Three-Component 1,2-Diamination of Unactivated Terminal Alkenes
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Sun, Manman; Li, Jinshan; Chen, Weida; Wu, Haijian; Yang, Jianguo; Wang, Zhiming:
Palladium-Catalyzed [4+2] Annulation of Aryl and Alkenyl Carboxamides with 1,3-Dienes via C–H Functionalization: Synthesis of 3,4-Dihydroisoquinolones and 5,6-Dihydropyridinones
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Issue 23/2019
Special Topic Cover Page
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Sutherland, Andrew:
Radiohalogenation of Organic Compounds: Practical Considerations and Challenges for Molecular Imaging
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Milicevic Sephton, Selena; Zhou, Xiaoyun; Thompson, Stephen; Aigbirhio, Franklin I.:
Preparation of the Serotonin Transporter PET Radiotracer 2-({2-[(Dimethylamino)methyl]phenyl}thio)-5-[
18
F]fluoroaniline (4-[
18
F]ADAM): Probing Synthetic and Radiosynthetic Methods
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