Synthesis

Issue eFirst

Li, Yanjun; Ye, Ziqi; Cai, Jiaxin; Gong, Lei: Visible-Light-Promoted Asymmetric Catalysis by Chiral Complexes of First-Row Transition Metals

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Neri, Raul; Bossmann, Stefan H.: Isoselenocyanates: Synthesis and Their Use for Preparing Selenium-Based Heterocycles

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Zheng, Songlin; Hu, Yuanyuan; Yuan, Weiming: Recent Advances in C(sp³)–C(sp³) Cross-Coupling via Metalla­photoredox Strategies

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Liu, Jiaming; Chen, Ming: 1,3-Bifunctional Nucleophilic Allylation Reagents: Preparative Methods and Synthetic Applications

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Pellissier, Hélène: The Use of Domino Reactions for the Synthesis of Chiral Rings

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Oh, Eun Hye; Kim, Hyun Jin; Han, Soo Bong: Recent Developments in Visible-Light-Catalyzed Multicomponent Trifluoromethylation of Unsaturated Carbon–Carbon Bonds

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Zhao, Jia-Jia; Zhang, Hong-Hao; Yu, Shouyun: Enantioselective Radical Functionalization of Imines and Iminium Intermediates via Visible-Light Photoredox Catalysis

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Mazumdar, Wrickban; Driver, Tom G.: Recent Advances in the Development of Catalytic Methods that Construct Medium-Ring Lactams, Partially Saturated Benzazepines and Their Derivatives

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Zhao, Baoli; Liu, Yunyun: Step-Economical C–H Activation Reactions Directed by In Situ Amidation

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Rubtsov, Aleksandr E.; Malkov, Andrei V.: Recent Advances in the Synthesis of 2,2′-Bipyridines and Their Derivatives

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Zu, Bing; Guo, Yonghong; Ke, Jie; He, Chuan: Transient- and Native-Directing-Group-Enabled Enantioselective C–H Functionalization

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Inoa, Joan; Dominici, Grecia; Eldabagh, Reem; Foley, Jonathan J.; Xing, Yalan: Synthetic Applications and Computational Perspectives on Eosin Y Induced Direct HAT Process

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Kahlert, Lukas; Schotte, Carsten; Cox, Russell J.: Total Mycosynthesis: Rational Bioconstruction and Bioengineering of Fungal Natural Products

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Li, Qingjiang; Guo, Zhongwu: Enzymatic Synthesis of Glycosphingolipids: A Review

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Singh, Pushpinder; Batra, Aanchal; Singh, Kamal Nain; Mritunjay, Mritunjay: Transition-Metal-Free Strategies for the Synthesis of C-1 Aryl-Substituted Tetrahydroisoquinolines

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Zhou, Wen-Jun; Zhang, Yi-Han; Gui, Yong-Yuan; Sun, Liang; Yu, Da-Gang: Merging Transition-Metal Catalysis with Photoredox Catalysis: An Environmentally Friendly Strategy for C–H Functionalization

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Ashikari, Yosuke; Nagaki, Aiichiro: Homogeneous Catalyzed Aryl–Aryl Cross-Couplings in Flow

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Livingstone, Keith; Little, Gemma; Jamieson, Craig: Recent Advances in the Generation of Nitrilium Betaine 1,3-Dipoles

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Issue Accepted Manuscripts

Pedrood, Keyvan; Nazari Montazer, Mohammad; Larijani, Bagher; Mahdavi, Mohammad: Recent Advances in the Synthesis of Heterocycles by the Aza-Wittig Reaction

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Zhang, Qiaoling; Xi, Jufang; He, Ze; Zeng, Qingle: Syntheses and Transformations of Sulfinamides

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Rehpenn, Andreas; Walter, Alexandra; Storch, Golo: Molecular Editing of Flavins for Catalysis

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Maeda, Kyogo; Motokura, Ken: Recent Advances in Heterogeneous Ir Complex Catalysts for Aromatic C-H Borylation

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Jurunic, Carla Kornowski; Belladona, Andrei Lucca; Schumacher, Ricardo Frederico; Godoi, Benhur: Diorganyl Dichalcogenides, Copper and Iron Salts: Versatile Cyclization System to Achieve Carbo- and Heterocycles from Alkynes

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Roche, Stéphane P.: In the Pursuit of (Ald)Imine Surrogates for the Direct Asymmetric Synthesis of Non-Proteinogenic α-Amino Acids

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Majdecki, Maciej; Niedbała, Patryk; Tyszka-Gumkowska, Agata; Jurczak, Janusz: Assisted by Hydrogen-Bond Donors <i>Cinchona</i> Quaternary Salts as Privileged Chiral Catalysts for Phase-Transfer Reactions

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Zhang, Sheng; Findlater, Michael: Cobalt catalyzed isomerization of alkenes

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Youssef-Saliba, Sparta; Vallée, Yannick: Sulfur amino acids: from prebiotic chemistry to biology and vice versa

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Issue 08/2021

Bartoccini, Francesca; Piersanti, Giovanni: Synthesis and Reactivity of Uhle’s Ketone and Its Derivatives

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Yu, Hsien-Cheng; Mankad, Neal P.: Catalytic Reactions by Heterobimetallic Carbonyl Complexes with Polar Metal–Metal Interactions

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Yu, Jingxun; Luan, Xinjun: Hydroxylamines as One-Atom Nitrogen Sources for Metal-Catalyzed Cycloadditions

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Issue 07/2021

Zhao, Xuchen; Rainier, Jon D.: The Synthesis of Conjugated Bis-Aryl Vinyl Substrates and Their Photoelectrocyclization Reactions towards Phenanthrene Derivatives

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Walther, Melanie; Kipke, Waldemar; Schultzke, Sven; Ghosh, Souvik; Staubitz, Anne: Modification of Azobenzenes by Cross-Coupling Reactions

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Su, Shixia; Wang, Chuan: Catalytic Asymmetric Osmium-Free Dihydroxylation of Alkenes

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Issue 06/2021

Cherepakhin, Valeriy; Williams, Travis J.: Direct Oxidation of Primary Alcohols to Carboxylic Acids

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Jovanovic, Milos D.; Petkovic, Milos R.; Savic, Vladimir M.: Polycyclic Compounds from Allenes via Palladium-Mediated Intramolecular Carbopalladation/Nucleophilic Substitution Cascade Processes

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Nejrotti, Stefano; Prandi, Cristina: Gold Catalysis and Furans: A Powerful Match for Synthetic Connections

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Yang, Chao; Jiang, Chao; Qi, Xiangbing: Alkylzirconocenes in Organic Synthesis: An Overview

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Issue 05/2021

Ura, Yasuyuki: Palladium-Catalyzed Anti-Markovnikov Oxidation of Aromatic and Aliphatic Alkenes to Terminal Acetals and Aldehydes

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Gao, Shuangqiu; Shi, Lili; Chang, Le; Wang, Binglin; Fu, Junkai: Recent Developments in Heck-Type Reaction of Unactivated Alkenes and Alkyl Electrophiles

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Gale-Day, Zachary J.: Recent Advances in Metal-Catalyzed, Electrochemical Coupling Reactions of sp² Halides/Boronic Acids and sp³ Centers

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Wang, Yang; Yang, Bing; Wu, Xin-Xing; Wu, Zheng-Guang: Recent Application of Chiral Aryliodine Based on the 2-Iodo­resorcinol Core in Asymmetric Catalysis

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Issue 04/2021

Chen, Nuan; He, Min; Zhou, Ting; Zhu, Yuqi; Zhang, Hong; Peng, Shiyong: Recent Advances in the Tandem Cyclization/Cycloaddition of Allene Intermediates from Copper-Catalyzed Cross-Coupling of Diazo Compounds with Terminal Alkynes

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Wang, Lili; Ma, Juan; Si, Erbing; Duan, Zheng: Recent Advances in Luminescent Annulated Borepins, Silepins, and Phosphepins

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Xu, Ke; Wang, Ziyuan; Zhu, Tingshun: Recent Progress towards Organocatalyzed Asymmetric (Hetero)Arene Formation

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Gonay, Marie; Batisse, Chloé; Paquin, Jean-François: Recent Advances in the Synthesis of Acyl Fluorides

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Issue 03/2021

Némethová, Ivana; Šebesta, Radovan: Are Organozirconium Reagents Applicable in Current Organic Synthesis?

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Clapham, Margaret L.; Murphy, Emma C.; Douglas, Christopher J.: Synthesis and Crystal Engineering of Rubrene and Its Derivatives

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Jeon, Hongjun; Winkler, Jeffrey D.: Synthesis of Cyclohexane-Angularly-Fused Triquinanes

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Saway, Jason; Salem, Zena M.; Badillo, Joseph J.: Recent Advances in Photoacid Catalysis for Organic Synthesis

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Issue 02/2021

Zhang, Fulin; Xin, Luoting; Yu, Yinghua; Liao, Saihu; Huang, Xueliang: Recent Advances in Palladium-Catalyzed Bridging C–H Activation by Using Alkenes, Alkynes or Diazo Compounds as Bridging Reagents

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Edlová, Tereza; Čubiňák, Marek; Tobrman, Tomáš: Cross-Coupling Reactions of Double or Triple Electrophilic Templates for Alkene Synthesis

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Bandari, Chandrasekhar; Nicholas, Kenneth M.: Deoxygenative Transition-Metal-Promoted Reductive Coupling and Cross-Coupling of Alcohols and Epoxides

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Magyar, Ágnes; Juhász, Kinga; Hell, Zoltán: The Application of 4Å Molecular Sieves in Organic Chemical Syntheses: An Overview

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Issue 01/2021

Muñoz-Molina, José María; Belderrain, Tomás R.; Pérez, Pedro J.: Recent Advances in Copper-Catalyzed Radical C–H Bond Activation Using N–F Reagents

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Shoemaker, Aaron H.; Griffith, Daniel R.: Synthetic Approaches to Non-Tropane, Bridged, Azapolycyclic Ring Systems Containing Seven-Membered Carbocycles

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Carreras, Virginie; Tanbouza, Nour; Ollevier, Thierry: The Power of Iron Catalysis in Diazo Chemistry

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Chen, Tieqiao; Tan, Qihang; Liu, Xue; Liu, Long; Huang, Tianzeng; Han, Li-Biao: Phosphorylation of Carboxylic Acids and Their Derivatives with P(O)–H Compounds Forming P(O)–C Bonds

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Macchia, Antonio; Eitzinger, Andreas; Brière, Jean-François; Waser, Mario; Massa, Antonio: Asymmetric Synthesis of Isoxazol-5-ones and Isoxazolidin-5-ones

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Issue 24/2020

Chen, Jin-Quan; Dong, Zhi-Bing: Recent Progress in Utilization of Functionalized Organometallic Reagents in Cross Coupling Reactions and Nucleophilic Additions

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Al Bujuq, Nader: Methods of Synthesis of Remdesivir, Favipiravir, Hydroxychloroquine, and Chloroquine: Four Small Molecules Repurposed for Clinical Trials during the Covid-19 Pandemic

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Pang, Xiaobo; Peng, Xuejing; Shu, Xing-Zhong: Reductive Cross-Coupling of Vinyl Electrophiles

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Talukdar, Ranadeep: Synthetically Important Ring-Opening Acylations of Alkoxybenzenes

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Yu, Jie; Singh, Anoop S.; Yan, Guobing; Yu, Jian; Tiwari, Vinod K.: Recent Developments on Denitrogenative Functionalization of Benzotriazoles

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Issue 23/2020

Gan, Fuqiang; Luo, Puying; Lin, Junyue; Ding, Qiuping: Recent Advances in the Synthesis and Applications of 2-Arylbenzothiazoles

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Gao, Weiwei; Ding, Shengtao: Progress on Iridium-Catalyzed Hydrosilylation of Alkenes and Alkynes

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Filippov, Ilya P.; Titov, Gleb D.; Rostovskii, Nikolai V.: Recent Advances in Denitrogenative Reactions of Pyridotriazoles

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Khandelwal, Manisha; Ray, Sumit Kumar; Khangarot, Rama Kanwar: Syntheses and Applications of Singh’s Catalyst

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Issue 22/2020

Yorimitsu, Hideki; Yoshimura, Aya; Misaki, Yohji: Catalytic C–H Arylation of Tetrathiafulvalenes for the Synthesis of Functional Materials

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Li, Dan; Chen, Xiaochao; Gao, Wei: Asymmetric Synthesis of C₁-Chiral THIQs with Imines in Isoquinoline Rings

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Issue 21/2020

Mateus-Ruiz, Jeferson B.; Cordero-Vargas, Alejandro: Visible-Light-Mediated Photoredox Reactions in the Total Synthesis of Natural Products

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Moberg, Christina: Silylboranes as Powerful Tools in Organic Synthesis: Stereo- and Regioselective Reactions with 1,n-Enynes

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Issue 20/2020

Calcatelli, Alessio; Cherubini-Celli, Alessio; Carletti, Edoardo; Companyó, Xavier: Unconventional Transformations of Morita–Baylis–Hillman Adducts

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Weißbarth, Hendrik; Mühlhaus, Felix; Gansäuer, Andreas: Titanocene-Catalyzed Regiodivergent Epoxide Opening – From Desymmetrizing meso-Epoxides to Regiodivergent Arylation of Epoxides

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Zhao, Fei; Masci, Domiziana; Tomarelli, Elena; Castagnolo, Daniele: Biocatalytic and Chemo-Enzymatic Approaches for the Synthesis of Heterocycles

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Issue 19/2020

Grygorenko, Oleksandr O.; Moskvina, Viktoriia S.; Hryshchuk, Oleksandr V.; Tymtsunik, Andriy V.: Cycloadditions of Alkenylboronic Derivatives

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Geske, Leander; Sato, Eisuke; Opatz, Till: Anodic Oxidation as an Enabling Tool for the Synthesis of Natural Products

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Arisawa, Mieko: Transition-Metal-Catalyzed Synthesis of Organophosphorus Compounds Involving P–P Bond Cleavage

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Bottcher, Sydney E.; Hutchinson, Lauren E.; Wilger, Dale J.: Nickel-Catalyzed anti-Selective Alkyne Functionalization Reactions

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Issue 18/2020

Large, Benjamin; Prim, Damien: C–H Functionalization Strategies in the Naphthalene Series: Site Selections and Functional Diversity

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Almasalma, Ahmad A.; Mejía, Esteban: Recent Advances on Copper-Catalyzed C–C Bond Formation via C–H Functionalization

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Agrawal, Toolika; Sieber, Joshua D.: Recent Developments in C–C Bond Formation Using Catalytic Reductive Coupling Strategies

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Álvarez-Pérez, Andrea; Saá, Carlos; Varela, Jesús A.: Oxidation of Alkynes via Catalytic Metal-Vinylidenes

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Issue 17/2020

Corti, Vasco; Bertuzzi, Giulio: Organocatalytic Asymmetric Methodologies towards the Synthesis of Atropisomeric N-Heterocycles

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Liang, Dong; Xiao, Wen-Jing; Chen, Jia-Rong: Recent Advances of 1,3,5-Triazinanes in Aminomethylation and Cycloaddition Reactions

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Brechmann, Lea T.; Teichert, Johannes F.: Catch It If You Can: Copper-Catalyzed (Transfer) Hydrogenation Reactions and Coupling Reactions by Intercepting Reactive Intermediates Thereof

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Beltran, Frédéric; Miesch, Laurence: Tertiary Enamides as Versatile and Valuable Substrates to Reach Chemical Diversity

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Issue 16/2020

Yoshimura, Akira; Saito, Akio; Yusubov, Mekhman S.; Zhdankin, Viktor V.: Synthesis of Oxazoline and Oxazole Derivatives by Hypervalent-Iodine-Mediated Oxidative Cycloaddition Reactions

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Liu, Xue; Wu, Xiangmei; Zhang, Ling; Lin, Xiaoyan; Huang, Dayun: Recent Advances in Triarylmethane Synthesis

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Issue 15/2020

Beļaunieks, Rūdolfs; Puriņš, Mikus; Turks, Māris: Manifestation of the β-Silicon Effect in the Reactions of Unsaturated Systems Involving a 1,2-Silyl Shift

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Smolobochkin, Andrey V.; Gazizov, Almir S.; Turmanov, Rakhymzhan A.; Abdullaeva, Dinara S.; Burilov, Alexander R.; Pudovik, Michail A.: N-Phosphorylated Pyrrolidines: An Overview of Synthetic Approaches

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Issue 14/2020

Mittersteiner, Mateus; Bonacorso, Helio G.; Martins, Marcos A. P.; Zanatta, Nilo: Brominated β-Alkoxyvinyl Trihalomethyl Ketones as Promising Synthons in Heterocyclic Synthesis

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Kramer, Søren: Homogeneous Gold-Catalyzed Aryl–Aryl Coupling Reactions

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Issue 13/2020

Danilkina, Natalia A.; Govdi, Anastasia I.; Balova, Irina A.: 5-Iodo-1H-1,2,3-triazoles as Versatile Building Blocks

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Issue 12/2020

Chai, Zhuo: Catalytic Asymmetric Transformations of Racemic Aziridines

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Issue 11/2020

Khan, Muhammad Kamran; Wang, Dandan; Moloney, Mark G.: Functionalised Nitrogen Heterocycles and the Search for New Antibacterials and Bioactives

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Fischer, Jérôme; Nun, Pierrick; Coeffard, Vincent: Visible-Light-Driven Transformations of Phenols via Energy Transfer Catalysis

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Issue 10/2020

Woltornist, Ryan A.; Ma, Yun; Algera, Russell F.; Zhou, Yuhui; Zhang, Zirong; Collum, David B.: Structure, Reactivity, and Synthetic Applications of Sodium Diisopropylamide

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Issue 09/2020

Tu, Hai-Yong; Zhu, Shengqing; Qing, Feng-Ling; Chu, Lingling: Recent Advances in Nickel-Catalyzed Three-Component Difunctionalization of Unactivated Alkenes

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Zheng, Yue; Shao, Xiaoqing; Ramadoss, Velayudham; Tian, Lifang; Wang, Yahui: Recent Developments in Photochemical and Electrochemical Decarboxylative C(sp³)–N Bond Formation

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Issue 08/2020

Zhu, Yannan; Huang, You: Organocatalyzed [3+3] Annulations for the Construction of Heterocycles

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Issue 07/2020

Salom-Roig, Xavier; Bauder, Claude: Recent Applications in the Use of Sulfoxides as Chiral Auxiliaries for the Asymmetric Synthesis of Natural and Biologically Active Products

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Ping, Yuanyuan; Kong, Wangqing: Ni-Catalyzed Reductive Difunctionalization of Alkenes

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Kuang, Guanghua; Liu, Guangyuan; Zhang, Xingxing; Lu, Naihao; Peng, Yiyuan; Xiao, Qiang; Zhou, Yirong: Directing-Group-Assisted Transition-Metal-Catalyzed Direct C–H Oxidative Annulation of Arenes with Alkynes for Facile Construction of Various Oxygen Heterocycles

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Issue 06/2020

Song, Si-Zhe; Dong, Youren; Ge, Guo-Ping; Li, Qiang; Wei, Wen-Ting: Recent Advances in Radical Nitration Using tert-Butyl Nitrite

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Youn, So Won: Transition-Metal-Catalyzed Annulative Coupling Cascade for the Synthesis of 3-Methyleneisoindolin-1-ones

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Hsieh, Jen-Chieh; Su, Haw-Lih: Synthesis of N-Heterocycles via Transition-Metal-Catalyzed Tandem Addition/Cyclization of a Nitrile

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Issue 05/2020

Akkarasamiyo, Sunisa; Ruchirawat, Somsak; Ploypradith, Poonsaksi; Samec, Joseph S. M.: Transition-Metal-Catalyzed Suzuki–Miyaura-Type Cross-Coupling Reactions of π-Activated Alcohols

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Fatykhov, Ramil F.; Chupakhin, Oleg N.; Inyutina, Anna K.; Khalymbadzha, Igor A.: Synthetic Approaches to Unsymmetrically Substituted 5,7-Dihydroxycoumarins

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Meng, Yan-Ping; Wang, Shi-Meng; Fang, Wan-Yin; Xie, Zhi-Zhong; Leng, Jing; Alsulami, Hamed; Qin, Hua-Li: Ethenesulfonyl Fluoride (ESF) and Its Derivatives in SuFEx Click Chemistry and More

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Issue 04/2020

Uttry, Alexander; van Gemmeren, Manuel: Direct C(sp³)–H Activation of Carboxylic Acids

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Pang, Yue; Moser, Daniel; Cornella, Josep: Pyrylium Salts: Selective Reagents for the Activation of Primary Amino Groups in Organic Synthesis

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Baráth, Eszter: Selective Reduction of Carbonyl Compounds via (Asymmetric) Transfer Hydrogenation on Heterogeneous Catalysts

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Issue 03/2020

Nocera, Giuseppe; Murphy, John A.: Ground State Cross-Coupling of Haloarenes with Arenes Initiated by Organic Electron Donors, Formed in situ: An Overview

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Smyshliaeva, Lidiia A.; Varaksin, Mikhail V.; Charushin, Valery N.; Chupakhin, Oleg N.: Azaheterocyclic Derivatives of ortho-Carborane: Synthetic Strategies and Application Opportunities

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De Luca, Lorena; Mezzetti, Antonio: Catalytic Strategies to Enantiopure Benzoins: Past and Future

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Daley, Ryan A.; Topczewski, Joseph J.: Aryl-Decarboxylation Reactions Catalyzed by Palladium: Scope and Mechanism

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Issue 02/2020

Skotnitzki, Juri; Kremsmair, Alexander; Knochel, Paul: Stereoselective Preparation and Reactions of Chiral Secondary Alkyllithiums

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Xiao, Xuan; Zheng, Zi-Tong; Li, Ting; Zheng, Jing-Lin; Tao, Ting; Chen, Li-Mei; Gu, Jin-Ying; Yao, Xu; Lin, Jin-Hong; Xiao, Ji-Chang: Recent Advances in Difluoromethylthiolation

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Issue 01/2020

Baidilov, Daler: On the Mechanism of the Stevens Rearrangement

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Craig, Alexander J.; Hawkins, Bill C.: The Bonding and Reactivity of α-Carbonyl Cyclopropanes

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Issue 24/2019

Zhang, Tong; Wu, Yue-Hua; Wang, Nai-Xing; Xing, Yalan: Advances in C(sp³)–H Bond Functionalization via Radical Processes

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Levi, Noam; Amir, Dafna; Gershonov, Eytan; Zafrani, Yossi: Recent Progress on the Synthesis of CF₂H-Containing Derivatives

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Issue 23/2019

Rakitin, Oleg A.: Recent Developments in the Synthesis of 1,2,5-Thiadiazoles and 2,1,3-Benzothiadiazoles

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Issue 22/2019

Zeidan, Nicolas; Lautens, Mark: Migratory Insertion Strategies for Dearomatization

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Issue 21/2019

Allouche, Emmanuelle M. D.; Charette, André B.: Cyclopropanation Reactions of Semi-stabilized and Non-stabilized Diazo Compounds

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Issue 20/2019

Li, Yuyang; Kluger, Ronald: Metal-Catalyzed Site-Selective Monoacylation of Diols in Aqueous Media

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Issue 19/2019

Rossignon, Alexandre; Bonifazi, Davide: O-Annulation Leading to Five-, Six-, and Seven-Membered Cyclic Diaryl Ethers Involving C–H Cleavage

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Issue 18/2019

Gazizov, Almir S.; Smolobochkin, Andrey V.; Turmanov, Rahimjan A.; Pudovik, Michail A.; Burilov, Alexander R.; Sinyashin, Oleg G.: Synthesis of Phosphaproline Derivatives: A Short Overview

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Issue 14/2019

Senatore, Raffaele; Ielo, Laura; Monticelli, Serena; Castoldi, Laura; Pace, Vittorio: Weinreb Amides as Privileged Acylating Agents for Accessing α-Substituted Ketones

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Mudarra, Ángel L.; Martínez de Salinas, Sara; Pérez-Temprano, Mónica H.: Nucleophilic Trifluoromethylation Reactions Involving Copper(I) Species: From Organometallic Insights to Scope

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Herraiz, Ana G.; Suero, Marcos G.: New Alkene Cyclopropanation Reactions Enabled by Photoredox Catalysis via Radical Carbenoids

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Kunfi, Attila; London, Gábor: Polydopamine: An Emerging Material in the Catalysis of Organic Transformations

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Issue 13/2019

Steven, Alan: Micelle-Mediated Chemistry in Water for the Synthesis of Drug Candidates

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Issue 12/2019

Sbei, Najoua; Listratova, Anna V.; Titov, Alexander A.; Voskressensky, Leonid G.: Recent Advances in Electrochemistry for the Synthesis of N-Heterocycles

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Issue 11/2019

Wang, Zhang: The Chemical Syntheses of Nannocystins

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Hollanders, Karlijn; Maes, Bert U. W.; Ballet, Steven: A New Wave of Amide Bond Formations for Peptide Synthesis

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Issue 10/2019

Colomban, Cédric; Châtelet, Bastien; Martinez, Alexandre: Different Strategies for Obtaining Enantiopure Hemicryptophanes

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Li, Jie; Knochel, Paul: Chromium-Catalyzed Cross-Couplings and Related Reactions

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Issue 09/2019

Parisotto, Stefano; Deagostino, Annamaria: π-Allylpalladium Complexes in Synthesis: An Update

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Kotha, Sambasivarao; Meshram, Milind; Panguluri, Nageswara Rao: Advanced Approaches to Post-Assembly Modification of Peptides by Transition-Metal-Catalyzed Reactions

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Rodriguez, Jean; Quintard, Adrien: Acyl Transfer Strategies as Transient Activations for Enantioselective Synthesis

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Issue 08/2019

Eschliman, Kayla; Bossmann, Stefan H.: Synthesis of Isothiocyanates: An Update

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D’Hollander, Agathe C. A.; Peilleron, Laure; Grayfer, Tatyana D.; Cariou, Kevin: Halonium-Induced Polyene Cyclizations

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Issue 07/2019

Vasilenko, Dmitry A.; Sedenkova, Kseniya N.; Kuznetsova, Tamara S.; Averina, Elena B.: Synthetic Approaches to Nitro-Substituted Isoxazoles

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Usman, Muhammad; Zhang, Xiao-Wen; Liu, Wen-Bo: Silicon-Tethered Frameworks as Directing Groups for Carbon–Carbon and Carbon–Heteroatom Bond Formation

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Issue 06/2019

Pellissier, Hélène: Synthesis of Chiral 3-Substituted 3-Amino-2-oxindoles through Enantioselective Catalytic Domino and Tandem Reactions

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Michelotti, Alessia; Roche, Maxime: 40 Years of Hydrogen–Deuterium Exchange Adjacent to Heteroatoms: A Survey

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Issue 05/2019

Zard, Samir Z.: Sulfur Betaines from S-Propargyl Xanthates. Unusual Chemistry from a Simple Functional Group

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Crawford, Jennifer M.; Sigman, Matthew S.: Conformational Dynamics in Asymmetric Catalysis: Is Catalyst Flexibility a Design Element?

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Ferrer, Sofia; Echavarren, Antonio M.: Synthesis of Bullvalenes: Classical Approaches and Recent Developments

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Maraswami, Manikantha; Loh, Teck-Peng: Transition-Metal-Catalyzed Alkenyl sp² C–H Activation: A Short Account

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Sun, Alexandra C.; McAtee, Rory C.; McClain, Edward J.; Stephenson, Corey R. J.: Advancements in Visible-Light-Enabled Radical C(sp)²–H Alkylation of (Hetero)arenes

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Hu, Fan; Ng, Jerome P. L.; Chiu, Pauline: Pyrroles as Dienes in (4+3) Cycloadditions

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Gagosz, Fabien: Gold Vinylidenes as Useful Intermediates in Synthetic Organic Chemistry

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Groso, Emilia J.; Schindler, Corinna S.: Recent Advances in the Application of Ring-Closing Metathesis for the Synthesis of Unsaturated Nitrogen Heterocycles

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Issue 04/2019

Leonardi, Marco; Estévez, Verónica; Villacampa, Mercedes; Menéndez, J. Carlos: The Hantzsch Pyrrole Synthesis: Non-conventional Variations and Applications of a Neglected Classical Reaction

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Palmieri, Alessandro; Petrini, Marino: Recent Advances in the Synthesis of Unsymmetrical Bisindolylmethane Derivatives

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Issue 03/2019

Vaitla, Janakiram; Bayer, Annette: Sulfoxonium Ylide Derived Metal Carbenoids in Organic Synthesis

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Hrdina, Radim: Directed C–H Functionalization of the Adamantane Framework

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Kancherla, Sindhu; Jørgensen, Kåre B.; Fernández-Ibáñez, M. Ángeles: Recent Developments in Palladium-Catalysed Non-Directed C–H Bond Activation in Arenes

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Issue 02/2019

Ghosh, Manoj K.; Rajkiewicz, Adam A.; Kalek, Marcin: Organocatalytic Group Transfer Reactions with Hypervalent Iodine­ Reagents

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Singh, Kuldeep; Kulbir, Kulbir; Gupta, Tarang; Kaur, Rajneesh; Singh, Raman: Applications of Rozen’s Reagent in Oxygen-Transfer and C–H Activation Reactions

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Passador, Kevin; Thorimbert, Serge; Botuha, Candice: ‘Heteroaromatic Rings of the Future’: Exploration of Unconquered Chemical Space

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Issue 01/2019

Murai, Masahito; Takai, Kazuhiko: Unsymmetrical Difunctionalization of Two Different C–H Bonds in One Pot Under Transition-Metal Catalysis

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Karageorgis, George; Waldmann, Herbert: Guided by Evolution: Biology-Oriented Synthesis of Bioactive Compound Classes

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Barrett, Anthony G. M.; Ma, Tsz-Kan; Mies, Thomas: Recent Developments in Polyene Cyclizations and Their Applications in Natural Product Synthesis

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Zhang, Heng; Lei, Aiwen: Electrochemical/Photochemical Aminations Based on Oxidative Cross-Coupling between C–H and N–H

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Piccardi, Riccardo; Turcaud, Serge; Benedetti, Erica; Micouin, Laurent: Synthesis and Reactivity of Mixed Dimethylalkynylaluminum Reagents

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Kiefer, Alexander; Kazmaier, Uli: Syntheses of Cyclomarins – Interesting Marine Natural Products with Distinct Mode of Action towards Malaria and Tuberculosis

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Wu, Xiang; Gong, Liu-Zhu: Palladium(0)-Catalyzed Difunctionalization of 1,3-Dienes: From Racemic to Enantioselective

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Yoshikai, Naohiko: Recent Advances in Enantioselective C–C Bond Formation via Organocobalt Species

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Erb, William; Mongin, Florence: Twofold Ferrocene C–H Lithiations For One-Step Difunctionalizations

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Lübken, Dennis; Saxarra, Marius; Kalesse, Markus: Tris(acetylacetonato) Iron(III): Recent Developments and Synthetic Applications

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Barde, E.; Guérinot, A.; Cossy, J.: α-Arylation of Amides from α-Halo Amides Using Metal-Catalyzed Cross-Coupling Reactions

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Kumagai, Naoya; Shibasaki, Masakatsu: 7-Azaindoline Auxiliary: A Versatile Attachment Facilitating Enantioselective­ C–C Bond-Forming Catalysis

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Issue 24/2018

Soorukram, Darunee; Pohmakotr, Manat; Kuhakarn, Chutima; Reutrakul, Vichai: Stereoselective Synthesis of Tetrahydrofuran Lignans

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Barthelemy, Anne-Laure; Magnier, Emmanuel; Dagousset, Guillaume: Direct Trifluoromethylthiolation Reactions Involving Radical Processes

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Schettini, Rosaria; Sicignano, Marina; De Riccardis, Francesco; Izzo, Irene; Della Sala, Giorgio: Macrocyclic Hosts in Asymmetric Phase-Transfer Catalyzed Reactions

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Issue 23/2018

Martinez de Marigorta, Edorta; de los Santos, Jesús M.; Ochoa de Retana, Ana M.; Vicario, Javier; Palacios, Francisco: Multicomponent Reactions in the Synthesis of γ-Lactams

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Cholewiak, Agnieszka; Stepniak, Pawel; Jurczak, Janusz: Linear Neutral Receptors for Anions: Synthesis, Structure and Applications

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Jin, Tian; Zhao, Lu; Liu, Xiao; Sun, Liang; Lin, Jia-Fu; Zheng, Zhe-Bin: Recent Advances in the Total Synthesis of Clavaminols

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Issue 21/2018

Roulland, Emmanuel: Tiacumicin B: An Antibiotic of Prime Importance and a Natural Product with an Inspiring Complex Structure

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Dimitrov, Ivaylo; Denny, William A.; Jose, Jiney: Syntheses of Ketamine and Related Analogues: A Mini Review

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Yuan, Yu-Chao; Bruneau, Christian; Gramage-Doria, Rafael: Merging Transition-Metal Catalysis with Phthalimides: A New Entry to Useful Building Blocks

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Issue 20/2018

Gamba-Sánchez, Diego; Prunet, Joëlle: Synthesis of 1,3-Diols by O-Nucleophile Additions to Activated Alkenes

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Nielsen, Christian D.-T.; Abas, Hossay; Spivey, Alan C.: Stereoselective Reactions of ortho-Quinone Methide and ortho-Quinone Methide Imines and Their Utility in Natural Product Synthesis

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Hernández-Ruiz, Raquel; Sanz, Roberto: Dichlorodioxomolybdenum(VI) Complexes: Useful and Readily Available Catalysts in Organic Synthesis

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Issue 19/2018

Ručilová, Veronika; Soural, Miroslav: Recent Advances in the Applications of Triethylsilane in Organic Synthesis

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Rivera-Chao, Eva; Fra, Laura; Fañanás-Mastral, Martín: Synergistic Bimetallic Catalysis for Carboboration of Unsaturated Hydrocarbons

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Dimitrov, Vladimir; Woodward, Simon: Capturing Waste Heat Energy with Charge-Transfer Organic Thermoelectrics

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Chen, Jing-Biao; Whiting, Andrew: Recent Advances in Copper-Catalyzed Asymmetric Hydroboration of Electron-Deficient Alkenes: Methodologies and Mechanism

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Issue 18/2018

Guyon, Hélène; Boussonnière, Anne; Castanet, Anne-Sophie: Transition-Metal-Free Enantioselective Reactions of Organo­magnesium Reagents Mediated by Chiral Ligands

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Oulyadi, Hassan: Recent Advances in NMR: Aggregation, Solvation, and Dynamics of Selected Organolithium Compounds

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Brikci-Nigassa, Nahida Mokhtari; Bentabed-Ababsa, Ghenia; Erb, William; Mongin, Florence: In Situ ‘Trans-Metal Trapping’: An Efficient Way to Extend the Scope of Aromatic Deprotometalation

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Smith, Keith; Alshammari, Mohammed B.; El-Hiti, Gamal A.: Unravelling Factors Affecting Directed Lithiation of Acylamino­aromatics

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Plasseraud, Laurent: Organotin(IV) Complexes Containing Sn–O–Se Moieties: A Structural Inventory

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Dagorne, Samuel: Recent Developments on N-Heterocyclic Carbene Supported Zinc Complexes: Synthesis and Use in Catalysis

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Issue 16/2018

Listunov, Dymytrii; Joly, Etienne; Rullière, Pauline; Gaspard, Hafida; Bernardes-Génisson, Vania; Génisson, Yves; Maraval, Valérie; Chauvin, Remi: From Natural to Artificial Antitumor Lipidic Alkynylcarbinols: Asymmetric Synthesis, Enzymatic Resolution, and Refined SARs

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Issue 15/2018

Segundo, Marcos San; Correa, Arkaitz: Cross-Dehydrogenative Coupling Reactions for the Functionalization of α-Amino Acid Derivatives and Peptides

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Dhara, Ayan; Beuerle, Florian: Synthetic Strategies for the Regioselective Functionalization of Tribenzotriquinacenes

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Issue 14/2018

Gomes, Ana T. P. C.; Forezi, Luana da S. M.; Simões, Mário M. Q.; Gonzaga, Daniel T.; Cardoso, Mariana F. C.; Da Silva, Fernando de C.; Neves, Maria G. P. M. S.; Ferreira, Vítor F.; Cavaleiro, José A. S.: Carbene-Type Species in the Functionalization of Porphyrin Derivatives

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Leitch, Jamie A.; Frost, Christopher G.: Regioselective Transition-Metal-Catalyzed C–H Functionalization of Anilines

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Riley, Darren L.; Neyt, Nicole C.: Approaches for Performing Reductions under Continuous-Flow Conditions

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Issue 13/2018

Dalpozzo, Renato; Mancuso, Raffaella: Enantioselective Vinylogous Reactions of 3-Alkylidene Oxindoles

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da Silva, Amanda F.; Fernandes, Alessandra A. G.; Thurow, Samuel; Stivanin, Mateus L.; Jurberg, Igor D.: Isoxazol-5-ones as Strategic Building Blocks in Organic Synthesis

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Issue 12/2018

Kirupakaran, Sujenth; Korth, Hans-Gert; Hirschhäuser, Christoph: A Complementary Toolbox of Iterative Methods for the Stereo­selective Synthesis of Heteroatom-Rich Motives from C₁-Building Blocks

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Bergman, Jan: Comparison of Two Reagents for Thionations

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Issue 11/2018

Murarka, Sandip; Antonchick, Andrey P.: Metal-Catalyzed Oxidative Coupling of Ketones and Ketone Enolates

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Botubol-Ares, José Manuel; Durán-Peña, María Jesús; Hanson, James R.; Hernández-Galán, Rosario; Collado, Isidro G.: Cp₂Ti(III)Cl and Analogues as Sustainable Templates in Organic Synthesis

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Issue 10/2018

Wu, Wei; Weng, Zhiqiang: Synthesis of Aryl Trifluoromethyl Ketones

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Issue 09/2018

Silva, Eduarda M. P.; Rocha, Djenisa H. A.; Silva, Artur M. S.: Diels–Alder Reactions of 1,2-Dihydropyridines: An Efficient Tool for the Synthesis of Isoquinuclidines

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Fasano, Valerio; Ingleson, Michael J.: Recent Advances in Water-Tolerance in Frustrated Lewis Pair Chemistry

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Issue 08/2018

Mousavizadeh, Farnoush; Meyer, Daniel; Giannis, Athanassios: Synthesis of C-Nor-D-homo-steroidal Alkaloids and Their Derivatives

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Bogdanov, Andrei V.; Mironov, Vladimir F.: Advances in the Synthesis of Isatins: A Survey of the Last Decade

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Issue 07/2018

Boyle, Joshua William; Zhao, Yichao; Chan, Philip Wai Hong: Product Divergence in Coinage-Metal-Catalyzed Reactions of π-Rich Compounds

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Méndez, María V.; Bracca, Andrea B. J.; Kaufman, Teodoro S.: Isolation, Synthesis, and Biological Activity of Quindoline, a Valuable­ Indoloquinoline Natural Product and Useful Key Intermediate­

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Issue 06/2018

Bürglová, Kristýna; Hlaváč, Jan: Application of Trimethylsilanolate Alkali Salts in Organic Synthesis

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Albano, Gianluigi; Aronica, Laura Antonella: Cyclization Reactions for the Synthesis of Phthalans and Isoindolines­

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Meanwell, Michael; Britton, Robert: Synthesis of Heterobenzylic Fluorides

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Issue 05/2018

Wang, Pu-Sheng; Shen, Meng-Lan; Gong, Liu-Zhu: Transition-Metal-Catalyzed Asymmetric Allylation of Carbonyl Compounds with Unsaturated Hydrocarbons

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Balasubramaniam, Sivaraman; Sankaran, Ganapathy Subramanian; Badle, Sneh Sanjay: Perspective on FTY720, an Immunosuppressant

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Chardon, Aurélien; Morisset, Eléonore; Rouden, Jacques; Blanchet, Jérôme: Recent Advances in Amide Reductions

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Issue 04/2018

Ohno, Hiroaki; Inuki, Shinsuke: Recent Progress in Palladium-Catalyzed Cascade Cyclizations for Natural Product Synthesis

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Li, Pengfei; Jia, Xiaodong: tert-Butyl Nitrite (TBN) as a Versatile Reagent in Organic Synthesis

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Len, Christophe; Delbecq, Frederic; Cara Corpas, Cristobal; Ruiz Ramos, Encarnacion: Continuous Flow Conversion of Glycerol into Chemicals: An Overview

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Issue 03/2018

Martín-Heras, Víctor; Parra, Alejandro; Tortosa, Mariola: Cyclopropyl- and Cyclobutylboronates and -silanes: A Stereo­selective Approach

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Kiyokawa, Kensuke; Nagata, Takaya; Minakata, Satoshi: Recent Advances in the Synthesis of β-Ketonitriles

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Richmond, Edward; Moran, Joseph: Recent Advances in Nickel Catalysis Enabled by Stoichiometric Metallic Reducing Agents

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Issue 02/2018

Ramesh, Perla; Suman, Devatha; Reddy, Koti Siva Nagi: Asymmetric Synthetic Strategies of (R)-(–)-Baclofen: An Antispastic Drug

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Vorobyeva, Daria V.; Osipov, Sergey N.: Selective Synthesis of 2- and 7-Substituted Indole Derivatives via Chelation-Assisted Metallocarbenoid C–H Bond Functionalization

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Largeron, Martine; Nguyen, Khac Minh Huy: Recent Advances in the Synthesis of Benzimidazole Derivatives from the Oxidative Coupling of Primary Amines

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Issue 01/2018

Ajay, Sama; Shaw, Arun K.: Studies Towards the Synthesis of (+)- and (–)-Anisomycin and Their Analogues

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Chen, Yue-Gang; Xu, Xue-Tao; Zhang, Kun; Li, Yi-Qian; Zhang, Li-Pu; Fang, Ping; Mei, Tian-Sheng: Transition-Metal-Catalyzed Carboxylation of Organic Halides and Their Surrogates with Carbon Dioxide

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Eivgi, Or; Lemcoff, N. Gabriel: Turning the Light On: Recent Developments in Photoinduced Olefin Metathesis

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Issue 24/2017

Castro-Alvarez, Alejandro; Carneros, Héctor; Costa, Anna M; Vilarrasa, Jaume: Computer-Aided Insight into the Relative Stability of Enamines

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Wang, Chuan: Electrophilic Ring Opening of Small Heterocycles

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Issue 23/2017

Pankova, Alena S.; Kuznetsov, Mikhail A.: Recent Advances in the Chemistry of 2-Acylaziridines

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Kimura, Tsutomu: Recent Advances in Magnesium Carbenoid Chemistry

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Issue 22/2017

Hu, Wen-Li; Hu, Xiang-Guo; Hunter, Luke: Recent Developments in the Deoxyfluorination of Alcohols and Phenols: New Reagents, Mechanistic Insights, and Applications

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Pathipati, Stalin R.; van der Werf, Angela; Selander, Nicklas: Indium(III)-Catalyzed Transformations of Alkynes: Recent Advances in Carbo- and Heterocyclization Reactions

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Issue 21/2017

Gusarova, Nina K.; Chernysheva, Nataliya A.; Trofimov, Boris A.: Catalyst- and Solvent-Free Addition of the P–H Species to Alkenes and Alkynes: A Green Methodology for C–P Bond Formation

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Zhao, Qun; Poisson, Thomas; Pannecoucke, Xavier; Besset, Tatiana: The Transient Directing Group Strategy: A New Trend in Transition-Metal-Catalyzed C–H Bond Functionalization

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Issue 20/2017

Aziz, Jessy; Piguel, Sandrine: An Update on Direct C–H Bond Functionalization of Nitrogen-Containing Fused Heterocycles

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Henry, Martyn C.; Mostafa, Mohamed A. B.; Sutherland, Andrew: Recent Advances in Transition-Metal-Catalyzed, Directed Aryl C–H/N–H Cross-Coupling Reactions

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Issue 19/2017

Feng, Minghao; Jiang, Xuefeng: Reactions of Arynes Involving Transition-Metal Catalysis

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Barroso, Raquel; Cabal, María P.; Valdés, Carlos: Pd-catalyzed Auto-Tandem Cascades Based on N-Sulfonylhydrazones: Hetero- and Carbocyclization Processes

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Issue 18/2017

Míguez-Lago, Sandra; Cid, María Magdalena: Axially Chiral Shape-Persistent Encapsulating Agents

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Issue 17/2017

Guo, Qihang; Lu, Zhan: Recent Advances in Nitrogen–Nitrogen Bond Formation

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Pfund, Emmanuel; Lequeux, Thierry: Synthesis of Fluoropyrrolidines and (Fluoroalkyl)pyrrolidines

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Issue 16/2017

Arava, Shlomy; Diesendruck, Charles E.: Strategies for the Synthesis of N-Arylammonium Salts

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Issue 15/2017

Chen, Yi-Hung; Ellwart, Mario; Malakhov, Vladimir; Knochel, Paul: Solid Organozinc Pivalates: A New Class of Zinc Organometallics with Greatly Enhanced Air- and Moisture-Stability

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Breugst, Martin; von der Heiden, Daniel; Schmauck, Julie: Novel Noncovalent Interactions in Catalysis: A Focus on Halogen, Chalcogen, and Anion-π Bonding

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Bartolo, Nicole D.; Read, Jacquelyne A.; Valentín, Elizabeth M.; Woerpel, K. A.: Reactions of Allylmagnesium Halides with Carbonyl Compounds: Reactivity, Structure, and Mechanism

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Mąkosza, Mieczysław: How Does Nucleophilic Aromatic Substitution in Nitroarenes Really Proceed: General Mechanism

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Tabolin, Andrey A.; Sukhorukov, Alexey Yu.; Ioffe, Sema L.; Dilman, Alexander D.: Recent Advances in the Synthesis and Chemistry of Nitronates

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Parchomyk, Tobias; Koszinowski, Konrad: Iron-Catalyzed Cross-Coupling: Mechanistic Insight for Rational Applications in Synthesis

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Dana, Suman; Ramakrishna, Isai; Baidya, Mahiuddin: Ambident Reactivity of Nitroso Compounds for Direct Amination and Hydroxylation of Carbonyls

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Reissig, Hans-Ulrich; Zimmer, Reinhold: Cyclizations of Alkoxyallenes: Mechanisms, Intermediates, ­Products – A Personal Account on Solved and Unsolved Problems with Unique Allene Building Blocks

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Hartley, Will C.; O’Riordan, Timothy J. C.; Smith, Andrew D.: Aryloxide-Promoted Catalyst Turnover in Lewis Base Organo­catalysis

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Fantin, Marco; Lorandi, Francesca; Gennaro, Armando; Isse, Abdirisak A.; Matyjaszewski, Krzysztof: Electron Transfer Reactions in Atom Transfer Radical Polymerization

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Armstrong, Roly J.; Aggarwal, Varinder K.: 50 Years of Zweifel Olefination: A Transition-Metal-Free Coupling

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Abe, Manabu; Chitose, Youhei; Jakkampudi, Satish; Thuy, Pham Thi Thu; Lin, Qianghua; Van, Bui Thi; Yamada, Ayato; Oyama, Ryoko; Sasaki, Miyu; Katan, Claudine: Design and Synthesis of Two-Photon Responsive Chromophores for Near-Infrared Light-Induced Uncaging Reactions

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Micheletti, Gabriele; Boga, Carla: Nucleophile/Electrophile Combinations in Aromatic Substitution: From Wheland to Wheland–Meisenheimer Intermediates Using Strongly Activated Arenes

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Zhao, Rong; Chang, Denghu; Shi, Lei: Recent Advances in Cyclic Diacyl Peroxides: Reactivity and Selectivity Enhancement Brought by the Cyclic Structure

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Asahara, Haruyasu: Recent Advances in the Carbon–Carbon Bond-Forming Reactions of N-Acylketimines

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Maji, Biplab; Barman, Milan K.: Recent Developments of Manganese Complexes for Catalytic Hydrogenation and Dehydrogenation Reactions

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Krishnamoorthy, Sankarganesh; Prakash, G. K. Surya: Silicon-Based Reagents for Difluoromethylation and Difluoromethylenation Reactions

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Gao, Pin; Gu, Yu-Rui; Duan, Xin-Hua: Direct C–H Functionalization of Heteroarenes via Redox-Neutral Radical Process: A Facile Route to C–C Bonds Formation

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Denegri, Bernard; Matić, Mirela; Kronja, Olga: Impact of Electronic Effects on the Nucleofugality of Leaving Groups

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Gualandi, Andrea; Mengozzi, Luca; Cozzi, Pier Giorgio: Stereoselective S_N1-Type Reaction of Enols and Enolates

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Quint, Valentin; Noël-Duchesneau, Ludovik; Lagadic, Elodie; Morlet-Savary, Fabrice; Lalevée, Jacques; Gaumont, Annie- Claude; Lakhdar, Sami: Metal-Free Generation of Phosphorus-Centered Radicals for the Synthesis of Phosphorus-Based Heterocycles: A Personal Account

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Issue 14/2017

Budynina, Ekaterina M.; Ivanov, Konstantin L.; Sorokin, Ivan D.; Melnikov, Mikhail Ya.: Ring Opening of Donor–Acceptor Cyclopropanes with N-Nucleo­philes

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Keglevich, György; Kiss, Nóra Zsuzsa; Grün, Alajos; Bálint, Erika; Kovács, Tamara: Advantages of the Microwave Tool in Organophosphorus Syntheses

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Issue 13/2017

Broggini, Gianluigi; Borelli, Tea; Giofré, Sabrina; Mazza, Alberto: Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C–H Functionalization of Unactivated Olefins

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Döndas, H. Ali; de Gracia Retamosa, María; Sansano, José M.: Current Trends towards the Synthesis of Bioactive Heterocycles and Natural Products Using 1,3-Dipolar Cycloadditions (1,3-DC) with Azomethine Ylides

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Issue 12/2017

Glinsky-Olivier, Nicolas; Guinchard, Xavier: Enantioselective Catalytic Methods for the Elaboration of Chiral Tetrahydro-β-carbolines and Related Scaffolds

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Naidoo, Shivani; Jeena, Vineet: Synthesis of 2,4-Disubstituted Quinoline Derivatives via A³-Coupling: An EcoScale Evaluation

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Issue 11/2017

Pires, Marina J. D.; Purificação, Sara I.; Santos, A. Sofia; Marques, M. Manuel B.: The Role of PEG on Pd- and Cu-Catalyzed Cross-Coupling Reactions

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Fuse, Shinichiro; Morita, Taiki; Nakamura, Hiroyuki: Step-by-Step Multifunctionalization of Isoxazoles Based On S_EAr Reactions and C–H Direct Arylations

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Mostinski, Yelena; Lankri, David; Tsvelikhovsky, Dmitry: Transition-Metal-Catalyzed Synthesis of Spirolactones

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Issue 10/2017

Annibaletto, Julien; Oudeyer, Sylvain; Levacher, Vincent; Brière, Jean-François: Catalytic Enantioselective Syntheses of Isoxazolidin-5-ones

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Issue 09/2017

Carraro, Massimo; Pisano, Luisa; Azzena, Ugo: Silica Gel Stabilized Na and Na/K Alloys: Highly Effective, Versatile and Environmentally Friendly Reducing Agents

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Merad, Jérémy; Candy, Mathieu; Pons, Jean-Marc; Bressy, Cyril: Catalytic Enantioselective Desymmetrization of Meso Compounds in Total Synthesis of Natural Products: Towards an Economy of Chiral Reagents

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Issue 08/2017

Schröder, Birte; Gaich, Tanja: Methoxatin as a Target in Total Synthesis

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Polák, Peter; Dvořák, Dalimil; Tobrman, Tomáš: Cyanogen: A Versatile Reagent for Diversity-Oriented Synthesis

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Blouin, Sarah; Blond, Gaelle; Donnard, Morgan; Gulea, Mihaela; Suffert, Jean: Cyclocarbopalladation as a Key Step in Cascade Reactions: Recent Developments

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Jackman, Mary M.; Cai, Yu; Castle, Steven L.: Recent Advances in Iminyl Radical Cyclizations

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Issue 07/2017

Fraile, José M.; García, José I.; Herrerías, Clara I.; Pires, Elisabet: Synthetic Transformations for the Valorization of Fatty Acid Derivatives

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Thaima, Thanaphat; Zamani, Farzad; Hyland, Christopher J. T.; Pyne, Stephen G.: Allenylation and Propargylation Reactions of Ketones, Aldehydes, Imines, and Iminium Ions Using Organoboronates and Related Derivatives

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Coussanes, Guilhem; Vila, Xavier; Diaba, Faïza; Bonjoch, Josep: Radical Cyclization of Trichloroacetamides: Synthesis of Lactams

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Lebœuf, David; Gandon, Vincent: Carbon–Carbon and Carbon–Heteroatom Bond-Forming Transformations Catalyzed by Calcium(II) Triflimide

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Issue 06/2017

Zhang, Min; Zhu, Chunyin; Ye, Long-Wu: Recent Advances in Dual Visible Light Photoredox and Gold-Catalyzed­ Reactions

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Lepori, Clément; Hannedouche, Jérôme: First-Row Late Transition Metals for Catalytic (Formal) Hydro­amination of Unactivated Alkenes

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Comas-Barceló, Júlia; Harrity, Joseph P. A.: Metal Acetylides in Cycloaddition Reactions

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Grimaud, Laurence; Jutand, Anny: Role of Fluoride Ions in Palladium-Catalyzed Cross-Coupling Reactions­

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Issue 05/2017

Liu, Jie; Wang, Lei: Recent Advances in Asymmetric Reactions Catalyzed by Proline and Its Derivatives

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Lanari, Daniela; Piermatti, Oriana; Morozzi, Chiara; Santoro, Stefano; Vaccaro, Luigi: Recent Applications of Solid-Supported Ammonium Fluorides in Organic Synthesis

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Mizar, Pushpak; Wirth, Thomas: Iodoaminations of Alkenes

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Ordóñez, Mario; Viveros-Ceballos, José Luis; Sayago, Francisco J.; Cativiela, Carlos: Stereoselective Synthesis of α-Amino-H-phosphinic Acids and Derivatives

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Issue 04/2017

Legnani, Luca; Bhawal, Benjamin N.; Morandi, Bill: Recent Developments in the Direct Synthesis of Unprotected Primary­ Amines

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Adeleke, A. Francis; Brown, Alexander P. N.; Cheng, Li-Jie; Mosleh, Kari A. M.; Cordier, Christopher J.: Recent Advances in Catalytic Transformations Involving Copper Acetylides

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Otero-Fraga, Jorge; Montesinos-Magraner, Marc; Mendoza, Abraham: Perspectives on Intermolecular Azomethine Ylide [3+2] Cycloadditions with Non-Electrophilic Olefins

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Chen, Wenyi; Bakewell, Clare; Crimmin, Mark R.: Functionalisation of Carbon–Fluorine Bonds with Main Group Reagents

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Eisink, Niek N. H. M.; Minnaard, Adriaan J.; Witte, Martin D.: Chemo- and Regioselective Oxidation of Secondary Alcohols in Vicinal Diols

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Mayer, Susanne; Lang, Kathrin: Tetrazines in Inverse-Electron-Demand Diels–Alder Cycloadditions and Their Use in Biology

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Issue 03/2017

Barré, Anaïs; Ţînţaş, Mihaela-Liliana; Levacher, Vincent; Papamicaël, Cyril; Gembus, Vincent: An Overview of the Synthesis of Highly Versatile N-Hydroxysuccinimide Esters

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Aullón, Gabriel; Romea, Pedro; Urpí, Fèlix: Substrate-Controlled Aldol Reactions from Chiral α-Hydroxy Ketones

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Yuan, Ling-Zhi; Hamze, Abdallah; Alami, Mouad; Provot, Olivier: Synthesis of Substituted Benzils from Diarylalkyne Oxidation

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Mangeney, Pierre; Gérard, Hélène; Vrancken, Emmanuel: Li⁺-Controlled Diastereoselectivity of the Addition of Allenyl Cuprate Reagents to Aldehydes

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Issue 02/2017

Moegling, Julian; Hoffmann, Alexander; Herres-Pawlis, Sonja: Insights into Copper-Poly(pyrazolyl)methane-Catalyzed Reactions for Organic Transformations

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Schmid, Fabian; Baro, Angelika; Laschat, Sabine: Strategies for the Synthesis of Deoxypropionates

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Issue 01/2017

Qureshi, Zafar; Toker, Christina; Lautens, Mark: Secondary Alkyl Groups in Palladium-Catalyzed Cross-Coupling Reactions

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Selter, Lars; Zygalski, Lukas; Kerste, Eric; Koert, Ulrich: Vicinal Tricarbonyl Compounds: Versatile Building Blocks for Natural Product Synthesis

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Jalani, Hitesh B.; Karagöz, Aysun Çapcı; Tsogoeva, Svetlana B.: Synthesis of Substituted 1,2,3-Triazoles via Metal-Free Click Cycloaddition Reactions and Alternative Cyclization Methods

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Issue 24/2016

Ganesh, Venkataraman; Chandrasekaran, Srinivasan: Recent Advances in the Synthesis and Reactivity of Vinylcyclopropanes

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Shang, Ming; Sun, Shang-Zheng; Wang, Hong-Li; Wang, Ming-Ming; Dai, Hui-Xiong: Recent Progress on Copper-Mediated Directing-Group-Assisted C(sp²)–H Activation

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Indukuri, Kiran; Cornelissen, Loïc; Riant, Olivier: Recent Developments in the Chemistry of Vinylsiloxanes

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Issue 23/2016

Tian, Qingshan; Zhang, Guozhu: Recent Advances in the Asymmetric Nozaki–Hiyama–Kishi Reaction

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Moni, Lisa; Banfi, Luca; Riva, Renata; Basso, Andrea: External-Oxidant-Based Multicomponent Reactions

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Pons, Amandine; Poisson, Thomas; Pannecoucke, Xavier; Charette, André B.; Jubault, Philippe: Synthesis and Applications of Fluorocyclopropanes

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Issue 22/2016

Rintjema, Jeroen; Kleij, Arjan W.: Substrate-Assisted Carbon Dioxide Activation as a Versatile Approach for Heterocyclic Synthesis

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Besson, Thierry; Fruit, Corinne: Recent Developments in Microwave-Assisted Metal-Catalyzed C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications

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Vargas-Caporali, Jorge; Juaristi, Eusebio: The Diamino Analogues of Privileged Corey–Bakshi–Shibata and Jørgensen–Hayashi Catalysts: A Comparison of Their Performance

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Issue 21/2016

Zani, Lorenzo; Mordini, Alessandro; Calamante, Massimo; Reginato, Gianna: Preparation of Reduced Pyrazino[2,1-a]isoquinoline Derivatives: Important Heterocycles in the Field of Bioactive Compounds

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Renaud, Jean-Luc; Gaillard, Sylvain: Recent Advances in Iron- and Cobalt-Complex-Catalyzed Tandem/Consecutive Processes Involving Hydrogenation

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Fülöpová, Veronika; Soural, Miroslav: Solid-Phase Synthesis of Heterocycles with α-Haloketones as the Key Building Blocks

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Issue 20/2016

Ajitha, Manjaly J.; Huang, Kuo-Wei: Non-Classical C–H···X Hydrogen Bonding and Its Role in Asymmetric Organocatalysis

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Serrano-Molina, David; Martín-Castro, Ana M.: Tandem Sequences Involving Michael Additions and Sigmatropic Rearrangements

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Varela, Jesús A.; Saá, Carlos: Metal-Catalyzed Cyclizations to Pyran and Oxazine Derivatives

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Issue 18/2016

Sloan, Nikki L.; Sutherland, Andrew: Recent Advances in Transition-Metal-Catalyzed Iodination of Arenes

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Wencel-Delord, Joanna; Colobert, Françoise: Stereoselective Metal-Catalyzed C–C Bond Coupling Reactions by Stereoconvergence, Dynamic Kinetic Asymmetric Transformation, or Dynamic Kinetic Resolution

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Alezra, Valérie; Kawabata, Takeo: Recent Progress in Memory Of Chirality (MOC): An Advanced Chiral Pool

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Issue 17/2016

Amat, Mercedes; Llor, Núria; Guignard, Guillaume; Bosch, Joan: Synthesis of Fluvirucins and Their Aglycons, the Fluvirucinins

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Giustiniano, Mariateresa; Novellino, Ettore; Tron, Gian Cesare: Nitrile N-Oxides and Nitrile Imines as New Fuels for the Discovery of Novel Isocyanide-Based Multicomponent Reactions

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Nielsen, Mogens Brøndsted: Sonogashira-Like Coupling Reactions with Phosphine–Gold(I) Alkynyl Complexes

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Issue 16/2016

Echeverria, Pierre-Georges; Ayad, Tahar; Phansavath, Phannarath; Ratovelomanana-Vidal, Virginie: Recent Developments in Asymmetric Hydrogenation and Transfer Hydrogenation of Ketones and Imines through Dynamic Kinetic Resolution

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Yoshida, Hiroto: Stannylation Reactions under Base Metal Catalysis: Some Recent Advances

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Roselló, María Sánchez; del Pozo, Carlos; Fustero, Santos: A Decade of Advance in the Asymmetric Vinylogous Mannich Reaction

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Issue 15/2016

García-Cabeza, Ana Leticia; Moreno-Dorado, F. Javier; Ortega, María J.; Guerra, Francisco M.: Copper-Catalyzed Oxidation of Alkenes and Heterocycles

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Vicente, Rubén: Recent Progresses towards the Strengthening of Cyclopropene Chemistry

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Banert, Klaus: The Chemistry of Unusually Functionalized Azides

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Issue 14/2016

Zeng, Yuwen; Hu, Jinbo: Bridging Fluorine and Aryne Chemistry: Vicinal Difunctionalization of Arynes Involving Nucleophilic Fluorination, Trifluoromethylation, or Trifluoromethylthiolation

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Montesinos-Magraner, Marc; Vila, Carlos; Blay, Gonzalo; Pedro, José R.: Catalytic Enantioselective Friedel–Crafts Reactions of Naphthols and Electron-Rich Phenols

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Sánchez-Sancho, Francisco; Csákÿ, Aurelio G.: C–H Bond Formation with Boronic Acids and Derivatives by Transition-Metal-Free Conjugate Addition Reactions

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Issue 13/2016

Sasaki, I.: Recent Uses of Kröhnke Methodology: A Short Survey

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Florio, Saverio; Salomone, Antonio: Heterocycle-Mediated ortho-Functionalization of Aromatic Compounds: The DoM Methodology and Synthetic Utility

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Tanoury, Gerald J.: Photochemical Synthesis of Azaheterocycles

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Issue 12/2016

Chen, Zhang-Pei; Zhou, Yong-Gui: Asymmetric Hydrogenation of Heteroarenes with Multiple Heteroatoms

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Hoffmann, Norbert: Photochemical Electron and Hydrogen Transfer in Organic Synthesis: The Control of Selectivity

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Issue 11/2016

Kindt, Stephanie; Heinrich, Markus R.: Recent Advances in Meerwein Arylation Chemistry

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Heinrich, Clément F.; Peter, Clovis; Miesch, Laurence; Geoffroy, Philippe; Miesch, Michel: Diastereo- and Enantioselective Synthesis of Polyfunctionalized Diquinanes, Hydrindanes, and Decalins Bearing a Hydroxyl Group at the Ring Junction

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Issue 10/2016

Erhardt, Hellmuth; Kirsch, Stefan F.: Geminal Bis- and Tristriazoles: Long-known but still Uncommon Heterocyclic Entities

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Collins, Súil; Bartlett, Sean; Nie, Feilin; Sore, Hannah F.; Spring, David R.: Diversity-Oriented Synthesis of Macrocycle Libraries for Drug Discovery and Chemical Biology

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Issue 09/2016

Das, Sudarshan; Santra, Sougata; Mondal, Pallab; Majee, Adinath; Hajra, Alakananda: Zwitterionic Imidazolium Salt: Recent Advances in Organocatalysis

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Nishiwaki, Nagatoshi: Development of a Pseudo-Intramolecular Process

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Issue 08/2016

Benischke, Andreas D.; Ellwart, Mario; Becker, Matthias R.; Knochel, Paul: Polyfunctional Zinc and Magnesium Organometallics for Organic Synthesis: Some Perspectives

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Issue 07/2016

Meazza, Marta; Rios, Ramon: Merging Transition-Metal Activation and Aminocatalysis

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Issue 06/2016

Bag, Sukdev; Maiti, Debabrata: Palladium-Catalyzed Olefination of Aryl C–H Bonds by Using Directing­ Scaffolds

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Issue 05/2016

Lundberg, Helena; Adolfsson, Hans: Catalytic α-Alkylation/Reduction of Ketones with Primary Alcohols To Furnish Secondary Alcohols

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Merino, Pedro; Tejero, Tomás; Delso, Ignacio; Matute, Rosa: Recent Advances on Asymmetric Nitroso Aldol Reaction

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Issue 04/2016

Pullarkat, Sumod A.: Recent Progress in Palladium-Catalyzed Asymmetric Hydrophos­phination

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Issue 03/2016

Dai, Qiang; Jiang, Yan; Yu, Jin-Tao; Cheng, Jiang: Peroxide: A Novel Methylating Reagent

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Issue 02/2016

Tilly, David; Chevallier, Floris; Mongin, Florence: Synthesis of Heterobiaryls Featuring 1,4 N···S Inter-Ring Interactions

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Issue 01/2016

Jia, Xiaodong: Radical Cation Salts: From Single-Electron Oxidation to C–H Activation­

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Issue 23/2015

Xu, Zheng; Huang, Wei-Sheng; Zhang, Jin; Xu, Li-Wen: Recent Advances in Transition-Metal-Catalyzed Silylations of Arenes with Hydrosilanes: C–X Bond Cleavage or C–H Bond Activation­ Synchronized with Si–H Bond Activation