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10 most-cited SynOpen articles published in 2020/2021
Issue Dedicated to Prof. Issa Yavari
2020/2021 Articles from India
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Kotha, Sambasivarao; Singh, Deepshikha:
Tetraphenylmethane Derivatives Containing Nitrogen Heterocycles
PDF (5628 kb)
Stampolaki, Marianna; Kolocouris, Antonios:
Improved Synthesis of the Antitubercular Agent SQ109
PDF (2715 kb)
Ausgabe 02/2024
Lipson, Victoria V.; Yaremenko, Fedyr G.; Vakula, Volodymyr M.; Kovalenko, Svitlana V.; Kyrychenko, Alexander V.; Desenko, Sergiy M.; Borysko, Petro О.; Zozulya, Sergiy O.:
Discovery of Novel
N
-Acylhydrazone Derivatives as Potent Inhibitors of Sirtuin-1
HTML
PDF (2382 kb)
Ausgabe 01/2024
Subramanyam, Amudala; Sumit, Sumit; Aidhen, Indrapal S.:
Synthesis of
C
-Glucoside Analogues of Naturally Occurring Phenylethanoid
O
-Glucosides
HTML
PDF (719 kb)
Polanco, Jocelyn; Knoell, Theresa; Bakhoda, Abolghasem Gus:
Cobalt–Magnesium and Cobalt–Calcium Heterotrimetallic Dinitrogen Complexes
HTML
PDF (880 kb)
Balázsi, Áron; Bognár, Balázs; Jekő, József; Kálai, Tamás:
Synthesis of 3,4-Disubstituted Pyrroline Nitroxides Containing Diphenylphosphane or Diphenylphosphane Oxide Substituents
HTML
PDF (521 kb)
Pitchai, Manivel; Kaspady, Mahammed; Indasi, Gopikumar; Krishnan, Rajesh; Maheswarappa, Gururaju Sannakki; Vetrichelvan, Muthalagu; Mathur, Arvind; Gupta, Anuradha:
Regioselective C3-Formylation of 2
H
-Indazoles Using Selectfluor under Microwave-Assisted Conditions
HTML
PDF (532 kb)
Ausgabe 04/2023
Li, Li; Dai, Guo-Liang; Zhu, Xue Hua; Yu, Lei; Li, Hai Yan:
Synthesis and Characterization of an Eight-Membered Heterocyclic 1,3,5,7-Tetra(3-pyridyl)-1,3,5,7-tetrazacyclooctane
HTML
PDF (892 kb)
Vetrichelvan, Muthalagu; Lanke, Veeranjaneyulu; Chandu, Bellam; Mathur, Arvind; Gupta, Anuradha:
Cost-Effective and Scalable Synthesis of 4-Bromo-1,2-dimethyl-1
H
-imidazole: A Key Building Block for Bioactive Molecules
HTML
PDF (390 kb)
Yang, Qi-Liang; Lei, Ping-Ping; Hao, Er-Jun; Zhang, Bei-Ning; Zhou, Hong-Hao; Li, Wan-Wan; Guo, Hai-Ming:
Oxidative C–H Sulfonylation of Hydrazones Enabled by Electrochemistry
HTML
PDF (1086 kb)
Mudgal, Deeksha; Singh, Ravi Pratap; Yadav, Nisha; Bharti, Tapeesh; Mishra, Vivek:
Exploring the Catalytic Efficiency of Copper-Doped Magnetic Carbon Aerogel for the Coupling Reaction of Isatin Oxime with Phenylboronic Acid Derivatives
HTML
PDF (4285 kb)
Gavali, Kanchan D.; Chaturbhuj, Ganesh U.:
Truly Catalytic Gewald Synthesis of 2-Aminothiophenes Using Piperidinium Borate (Pip Borate), a Conjugate Acid–Base Pair
HTML
PDF (433 kb)
Prakash, Supriya; Sreedhar, Bojja; Naidu, N. V. S.:
Gum Acacia Stabilized Ag-TiO
2
and Ag-SiO
2
: Sustainable Nanocatalysts for Direct and Convenient Synthesis of 5-Substituted 1
H
-tetrazoles
HTML
PDF (3627 kb)
Lipson, Victoria; Zhikol, Oleg; Shishkina, Svetlana; Semenenko, Alexander; Kulyk, Karina; Mateychenko, Pavel; Musatov, Vladimir; Mazepa, Alexander; Vakula, Vladimir; Borisov, Alexander; Kyrychenko, Alexander:
Low Molecular Weight Supramolecular Allobetuline-, Cyclohexanol-, or Undecanol-Appended 1,2,3-Triazole-Based Gelators: Synthesis and Molecular Dynamics Simulation Study
HTML
PDF (2677 kb)
Ausgabe 03/2023
Prasanthi, A. V. G.; Babu, Bathini Nagendra:
DMSO arbitrated Oxidative Annulation Followed by Homologated N-Alkylation: Microwave-Assisted Efficient and Greener Approach to Access 3-(3-Oxo-3-arylpropyl) Quinazolinones
HTML
PDF (918 kb)
Phull, Manjinder Singh; Jadav, Surender Singh; Bohara, Chander Singh; Gundla, Rambabu; Mainkar, Prathama S:
Multi-step Flow Synthesis of the Anthelmintic Drug Praziquantel
HTML
PDF (616 kb)
Banwell, Martin G.; Marshall, Sarah; Ward, Jas S.; Schwartz, Brett D.:
Synthesis of the Key Saccharide Fragments of the Glucuronic Acid-Containing Repeat Unit of Pentosan Polysulfate, a Heparin Sulfate Mimetic
HTML
PDF (754 kb)
Nakao, Michiyasu; Nakamura, Akihito; Takesue, Tomoyuki; Kitaike, Syuji; Ito, Hiro-O; Sano, Shigeki:
Synthesis of Novel Phosphorus-Substituted Stable Isoindoles by a Three-Component Coupling Reaction of
ortho
-Phthalaldehyde, 9,10-Dihydro-9-oxa-10-phosphaphenanthrene 10-Oxide, and Primary Amines
HTML
PDF (810 kb)
Katla, Ramesh; Katla, Rakhi:
Pyrrolidinium Acetate (PyrrIL) as a Green and Recyclable Catalyst: Synthesis of 2-Phenyl Benzimidazoles and 2-Phenyl Benzothiazoles under Solvent-Free Conditions at Room Temperature
HTML
PDF (578 kb)
Prachi, Ramteke; Gill, Manjinder Singh:
A Practical and Efficient Method for the Synthesis of Sorafenib and Regorafenib
HTML
PDF (508 kb)
Ausgabe 02/2023
Kumar, Sunil; Yadav, Mangal S.; Singh, Sumit K.; Rajkhowa, Sanchayita; Tiwari, Vinod K.:
Synthesis of Calix[4]arene Appended Lactosylated G
1
and Galactosylated G
2
Generation Glycodendrimers using a ‘CuAAC’ Click Approach
HTML
PDF (815 kb)
Sakhno, Yana; Radchenko, Oleksandr; Saraev, Vyacheslav; Shliapkina, Yuliia; Kaidash, Mariia; Shyshkina, Mariia; Shishkina, Svitlana; Musatov, Vladimir; Desenko, Sergey; Chebanov, Valentyn:
Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction
HTML
PDF (834 kb)
Ausgabe 01/2023
Inyurt, Fevzi Can; Mammadova, Flora; Dengiz, Cagatay:
Click-Type Synthesis of Homoconjugated Push–Pull Chromophores: Computational Investigation of Optical and Nonlinear Optical (NLO) Properties
HTML
PDF (1656 kb)
Miyata, Ryo; Shigeta, Takashi; Kumazawa, Shigenori; Egi, Masahiro:
Selective Syntheses of Coumarin and Benzofuran Derivatives Using Phenols and α-Methoxy-β-ketoesters
HTML
PDF (573 kb)
Goel, Kapil Kumar; Rajput, Satyendra Kumar; Kharb, Rajeev:
Design, Synthesis and Biological Evaluation of Imidazole-Substituted/Fused Aryl Derivatives Targeting Tubulin Polymerization as Anticancer Agents
HTML
PDF (2148 kb)
Mitra, Trisha; Joardar, Soumen; Chakravorty, Santanu; Majumdar, Manoj; Kundu, Mrinalkanti; Roy, Brindaban:
Palladium-Mediated Reductive Heck Cyclization for the Synthesis of Fused Retinoid Derivatives
HTML
PDF (494 kb)
Burke, Adam; Spiccio, Silvia; Di Filippo, Mara; Baumann, Marcus:
Photochemical Synthesis of Pyrazolines from Tetrazoles in Flow
HTML
PDF (701 kb)
Mali, Suraj N.; Pandey, Anima; Thorat, Bapu:
A Chitosan Hydrochloride Mediated, Simple and Efficient Approach for the Synthesis of Hydrazones, their
in vitro
Antimycobacterial Evaluations, and Molecular Modeling Studies (Part III)
HTML
PDF (1759 kb)
Srivastava, Avinash K.; Khandaka, Himanshu; Joshi, Raj Kumar:
CN-Doped Cobalt Oxide Composite: An Economic and Reusable Catalyst with Multitasking Catalytic Capability for Alkyne and Nitrile Hydrations and Nitro Reductions
HTML
PDF (1308 kb)
Mallesham, Poosa; Raghavulu, Karri; Miriyala, Venkatesh; Doddipalla, Raju; Yennam, Satyanarayana; Sanasi, Paul Douglas; Behera, Manoranjan:
Synthesis of Acidiphilamide A–C: Secondary Metabolites from the Genus
Streptacidiphilus
HTML
PDF (693 kb)
Ausgabe 04/2022
Ali, Mohammad Saif; Ramesh, P. I.; Ghosh, Subhash; Babu Tatina, Madhu:
Zinc Acetate Catalyzed Stereoselective 1,2-
trans
-Glycosylation Using Glycosyl Chlorides
HTML
PDF (579 kb)
Yasam, Bharath Kumar; Pabbaraja, Srihari:
Total Synthesis of Marine-Derived Azole Resistant Antifungal Agent (–)-Melearoride A and Antibiotic (–)-PF1163B
HTML
PDF (708 kb)
Noble, Jeffrey M.; Chang, Le; Chen, Dan; Wang, Binglin; Dominey, Raymond N.; Cook, Daniel W.; Burns, Justina M.; Stringham, Rodger W.; Cardoso, Flavio S. P.; Snead, David R.:
A Practical and Economical Route to (
S
)-Glycidyl Pivalate
HTML
PDF (746 kb)
Biradar, D. O.; Mane, Y. D.; Sarnikar, Y. P.; Kulkarni, S. G.; Reddy, B. V. Subba; Narsaiah, A. Venkat:
Zn/ZnBr
2
Catalysed Reaction of Aldehydes with Allylbromide: Synthesis of 2,6-Disubstituted 4-Bromotetrahydropyrans
HTML
PDF (496 kb)
Tan, Shen; Lan, Ping; Banwell, Martin G.; White, Lorenzo V.:
Practical, Multigram Preparation of Synthetically Useful, Enantiomerically Pure Building-Blocks from Quinic Acid
HTML
PDF (468 kb)
Biradar, Dhanraj O.; Mane, Yogesh D.; Subba Reddy, Basi V.:
Stereoselective Synthesis of Euscapholide and Tetraketide via Prins Cyclisation and Ring-Closing Metathesis
HTML
PDF (526 kb)
Jesin, C. P. Irfana; Kataria, Ramesh; Nandi, Ganesh Chandra:
Synthesis of α-Sulfoximino Tetrazoles via Azido-Ugi Four-Component Reaction
HTML
PDF (748 kb)
Ausgabe 03/2022
Lin, Zhongren; Tong, Lingfeng; Qiu, Hong; Li, Zheyao; Shen, Lunhua; Chen, Niangen; Yu, Xinhong:
The Synthesis of 5-Hydroxybenzofurans via Tandem
In Situ
Oxidative Coupling and Cyclization
HTML
PDF (445 kb)
Liu, Ying; Zhang, Yiping; Zhou, Yingkai; Zhang, Min; Deng, Hongmei; Song, Liping:
Concise One-Pot Multicomponent Reaction Approach to Monofluorinated Spiro-pyrazole-pyridine Derivatives without Additional Catalyst
HTML
PDF (637 kb)
Devi, Lalita; Mishra, Poornima; Pokhriyal, Ayushi; Rastogi, Namrata:
Organo-photocatalytic Synthesis of Functionalized Pyrroles from 2
H
-Azirines and α-Substituted Nitroalkenes
HTML
PDF (692 kb)
Mkhonazi, Blessing D.; Mabila, Euphrent M.; Moshapo, Paseka T.:
Palladium-Catalysed Reductive Aminocarbonylation of Aryl Bromides and Iodides with Nitroarenes
HTML
PDF (551 kb)
Ausgabe 02/2022
Nie, Hui; Wang, Nian; Huang, Jinwen; Ni, Zhuang; Xue, Kangyan; Song, Lixing; Wang, Mingwei; Wu, Fanhong:
Radiosynthesis and Tumor MicroPET/CT Imaging of
18
F-Fluoroethoxylerianin, an
18
F-Labeled Erianin Analogue
HTML
PDF (695 kb)
Jagadeesha, Gullahalli S.; Mantelingu, Kempegowda; Thimmegowda, Naraganahalli R.; Rangappa, Kanchugarakoppal S.:
Microwave-Assisted, Metal-Free, Chemoselective
N
-Formylation of Amines using 2-Formyl-1,3-dimethyl-1
H
-imidazol-3-ium Iodide and
In Situ
Synthesis of Benzimidazole and Isocyanides
HTML
PDF (620 kb)
Ausgabe 01/2022
Prabhakaran, Srinivasan; Velmathi, Sivan:
Synthesis and Molecular Docking Studies of
N
,
N
-Dimethyl Arylpyranopyrimidinedione Derivatives
HTML
PDF (807 kb)
Tonekaboni, Maryam-Sadat; Tanbakouchian, Zahra; Majedi, Soma; Shiri, Morteza:
Synthesis of [1,4]Oxathiepino[5,6-
b
]quinolines via Base-Mediated Intramolecular Hydroalkoxylation
HTML
PDF (397 kb)
Li, Zhongyuan; Huang, Jinwen; Ni, Zhuang; Sun, Ran; Nie, Hui; Tang, Hui; Song, Lixing; Wu, Fanhong:
Indium-Mediated Reformatsky Reaction of Iododifluoro Ketones with Aldehydes: Preparation of α,α-Difluoro-β-hydroxyketone Derivatives in Water
HTML
PDF (723 kb)
Jagot, Fatema; Minnie, Izak; Rahman, Aliyaah; Ntsimango, Songeziwe; Ngwira, Kennedy J.; de Koning, Charles B.:
Hydrogen-Bonded Xanthones as Potential UV Absorbers: The Synthesis of Xanthones from Bio-Renewable Cardanol Utilizing a Ceric Ammonium Sulfate (CAS)-Mediated Oxidation Reaction
HTML
PDF (757 kb)
Sosunovych, Bohdan; Brown, Alexander J.; Clarke, Paul A.:
Amino Imidate Catalyzed Asymmetric Michael Reactions of Ketones and Nitroalkenes
HTML
PDF (525 kb)
Ausgabe 04/2021
Veverková, Eva; Molnosiová, Pavlína; Šebesta, Radovan:
Asymmetric Sequential Michael Addition and Cyclization Reactions of 2-(2-Nitrovinyl)phenols Catalyzed by Bifunctional Amino-Squaramides
HTML
PDF (529 kb)
Kumar, Nemilikonda Sravan; Ramulu, B. Janaki; Ghosh, Subhash:
Stereoselective Synthesis of the C19–C39 Fragment of Bastimolide A
HTML
PDF (458 kb)
Yadav, Mangal S.; Jaiswal, Manoj K.; Kumar, Sunil; Tiwari, Vinod K.:
Trichloroacetimidate-Triggered Expeditious and Novel Synthesis of
N
-Acylbenzotriazoles
HTML
PDF (753 kb)
Duda, Addison M.; Giurini, Michael T.; Gillmore, Jason G.; Guarr, Thomas F.:
Intramolecular Oxidative Diaryl Coupling of Tetrasubstituted Diphenylamines for the Preparation of Bis(trifluoromethyl) Dimethyl Carbazoles
HTML
PDF (866 kb)
Bardovskyi, Rostyslav; Fabre, Marie; Ronco, Cyril; Benhida, Rachid:
Mild Biamidine-Transfer Conditions for the Synthesis of Aliphatic Biguanides
HTML
PDF (518 kb)
Liang, Zhi-Peng; Yu, Ying-Xin; Sun, Yuan-Yuan; Wang, Yang; Wu, Zheng-Guang:
Oxidative Annulation of Diphenylpropanamides via In Situ Hypervalent Iodine-Promoted Intramolecular C–N/C–O Bond Formation
HTML
PDF (566 kb)
Ausgabe 03/2021
Zullo, Valerio; Petri, Antonella; Iuliano, Anna:
An Efficient and Practical Chemoenzymatic Route to (3
R
,3a
R
,6
R
,6a
R
)-Hexahydrofuro[3,2-
b
]furan-6-amino-3-ol (6-Aminoisomannide) from Renewable Sources
HTML
PDF (711 kb)
Farhid, Hassan; Rostami, Mohammad Mahdi; Shaabani, Ahmad; Notash, Behrouz:
Synthesis of Depsipeptides via Isocyanide-Based Consecutive Bargellini–Passerini Multicomponent Reactions
HTML
PDF (1109 kb)
Ausgabe 02/2021
Saeedi, Marziyeh; Khoshdoun, Maryam; Taheri, Salman; Ziyaei Halimehjani, Azim; Mohammadi, Aliasghar; Halvagar, Mohammad Reza; Amani, Vahid:
Synthesis of Functionalized Bicyclic Pyridones Containing the Dithiocarbamate Group Using Thioazlactones, Diamines, and Nitroketene Dithioacetal
HTML
PDF (689 kb)
Sathish, Kota; Nagaraju, Sakkani; Kashinath, Dhurke:
Synthesis of Spiro Pyrazolone-Oxindole and Bicyclic Pyrazolone Derivatives via Solvent-Dependent Regioselective Aza-1,4/1,6-Michael and Intramolecular Cycloaddition under Catalyst-Free Conditions
HTML
PDF (831 kb)
De Marchi, Elisa; Arnodo, Davide; Maffeis, Elia; Scarpi, Dina; Prandi, Cristina; Occhiato, Ernesto G.:
Enantiodivergent Synthesis of Halofuginone by
Candida antarctica
Lipase B (CAL-B)-Catalyzed Kinetic Resolution in Cyclopentyl Methyl Ether (CPME)
HTML
PDF (552 kb)
Katta, Narenderreddy; Murugan, Arumugavel; Sharma, Sonika; Sharada, Duddu S.:
Visible-Light-Mediated Photocatalytic Oxidative C–C Bond Cleavage of Geminal Diazides: An Approach to Oxamates
HTML
PDF (599 kb)
Ausgabe 01/2021
Kutyashev, Igor B.; Sannikov, Maxim S.; Kochnev, Ivan A.; Barkov, Alexey Y.; Zimnitskiy, Nikolay S.; Korotaev, Vladislav Y.; Sosnovskikh, Vyacheslav Y.:
Diversity-Oriented Synthesis of Novel Trihalomethyl-Containing Spirochromeno[3,4-
a
](thia)pyrrolizidines and Spirochromeno-[3,4-
a
]indolizidines by One-Pot, Three-Component [3+2]-Cycloaddition Reaction
HTML
PDF (1553 kb)
Bracken, Cormac; Batsanov, Andrei S.; Baumann, Marcus:
Development of a Continuous Photochemical Benzyne-Forming Process
HTML
PDF (932 kb)
Ausgabe 04/2020
Guirado, Antonio; Vera, María; Martiz, Bruno; Ródenas, Francisco; Sandoval, José A.; Alarcón, Enrique; Bautista, Delia:
Synthesis and Crystal Structures of 4,5-Dihydroimidazo[1,5-
b
]pyrazol-6-ones
HTML
PDF (1263 kb)
Avula, Satya Kumar; Das, Biswanath; Csuk, Rene; Al-Rawahi, Ahmed; Al-Harrasi, Ahmed:
Total Synthesis of Surinamensinols A and B
HTML
PDF (405 kb)
Nariki, Haruna; Miyamura, Takuya; Matsui, Daiki; Sonoda, Motohiro; Tanimori, Shinji:
Iodine-Mediated Facile One-Pot Access to
N
-Aryl-2-benzoxazolamines
HTML
PDF (518 kb)
Faverio, Chiara; Boselli, Monica Fiorenza; Raimondi, Laura; Benaglia, Maurizio:
Ammonia–Borane-Mediated Reduction of Nitroalkenes
HTML
PDF (498 kb)
Rickertsen, Dillon R. L.; Ma, Longle; Paul, Anirudra; Abboud, Khalil A.; Seidel, Daniel:
Traceless Redox-Annulations of Alicyclic Amines
HTML
PDF (594 kb)
Ausgabe 03/2020
Raghunadh, Akula; Tadiparthi, Krishnaji; Meruva, Suresh Babu; Murthy, V. Narayana; Rao, L. Vaikunta; Kumar, U. K. Syam:
Synthesis of Quinoxalin-2(1
H
)-ones and Hexahydroquinoxalin-2(1
H
)-ones via Oxidative Amidation–Heterocycloannulation
HTML
PDF (510 kb)
Raji Reddy, Chada; Sinare, Sudam N.:
Expedient Approach to the Synthesis of Betrixaban
HTML
PDF (372 kb)
Ausgabe 02/2020
Qin, Ling; Wu, Hui-bin; Weng, Lidong; Shen, Qun; Chen, Huoji:
Aerobic Iron(III)-Catalyzed Direct Thiolation of Imidazo[1,2-
a
]pyridine with Thiols
HTML
PDF (403 kb)
Sharma, Pooja; Singh, Gurdial; Bhongade, Bhoomendra A.; Noolvi, Malleshappa N.; Gadad, Andanappa K.:
Synthesis of 5-Fluoroaminobenzothiazoles
HTML
PDF (565 kb)
Singh, Pargat; Nath, Mahendra:
A Modified Vilsmeier–Haack Strategy to Construct β-Pyridine-Fused 5,10,15,20-Tetraarylporphyrins
HTML
PDF (804 kb)
Ausgabe 04/2019
Jain, Vipin Kumar; Kumar, Mrityunjay:
Synthesis of (–)-Bulgecinine and 5-
epi
-Bulgecinine through Proline-Catalysed Asymmetric α-Hydroxylation of an Aldehyde Derived from
l
-Glutamic Acid
HTML
PDF (445 kb)
Dacho, Vladimír; Nitrayová, Dária; Šoral, Michal; Machyňáková, Andrea; Moncoľ, Ján; Szolcsányi, Peter:
Access to
N
-Alkylpyrazin-2-ones via C–O to C–N Rearrangement of Pyrazinyl Ethers
HTML
PDF (647 kb)
Jain, Vipin Kumar:
Diastereoselective Synthesis of (–)-Bestatin, Epibestatin, Phebestin and (3
S
,4
R
)-4-Amino-3-hydroxy-5-phenylpentanoic Acid from an Aldehyde Derived from
d
-Phenylalanine
HTML
PDF (555 kb)
Sonawane, Rahul B.; Sonawane, Swapnali R.; Rasal, Nishant K.; Jagtap, Sangeeta V.:
Room-Temperature, Base-Mediated Selective Synthesis of 2-(Arylamino)ethanols and 2-Aryloxyethanols
HTML
PDF (753 kb)
Szabó, Tímea; Kormány, Róbert; Dancsó, András; Volk, Balázs; Milen, Mátyás:
Total Synthesis of Bacterial 5-(3-Indolyl)oxazole Alkaloids: Pimprinols A–C
HTML
PDF (529 kb)
Ausgabe 02/2019
Talakokkula, Anil; Baikadi, Karunakar; Narsaiah, A. Venkat:
First Total Synthesis of Artekeiskeanol A, C and Altissimacoumarin D
HTML
PDF (387 kb)
Sharada, Ambati; Kundeti, Lakshmi Srinivasa Rao; Ramakrishna, Kallaganti V. S.; Nagaiah, Kommu:
First Stereoselective Total Synthesis of Ciryneol C
HTML
PDF (466 kb)
Ausgabe 01/2019
Kawtharani, Ranin.; Elmasri, Mirvat; Cherry, Khalil; Jacquemin, Johan; Abarbri, Mohamed:
Highly Regio- and Stereoselective Hydrogermylation of Fluorinated Alkyl Propiolate
HTML
PDF (463 kb)
Debnath, Sudarshan; Mondal, Shovan:
Palladium-Catalysed Intramolecular C–N versus C–C Coupling: The Effect of 1,8-
peri
-Interaction in the Naphthalene System
HTML
PDF (477 kb)
Kitagawa, Saori; Mori, Hiromitsu; Odagiri, Tatsuya; Suzuki, Katsuya; Kikkawa, You; Osugi, Rie; Takizawa, Shinobu; Kimura, Yoshikazu; Kirihara, Masayuki:
A Concise, Catalyst-Free Synthesis of Davis’ Oxaziridines using Sodium Hypochlorite
HTML
PDF (361 kb)
Baikadi, Karunakar; Talakokkula, Anil; Narsaiah, A. Venkat:
Stereoselective Total Synthesis of Macrolide Sch-725674 and C-7-
epi
-Sch-725674
HTML
PDF (574 kb)
Sarkar, Sujit; Devi, Namita; Porashar, Bikoshita; Ruidas, Santu; Saikia, Anil K:
Stereoselective Synthesis of 4-
O
-Tosyltetrahydropyrans via Prins Cyclization Reaction of Enol Ethers
HTML
PDF (586 kb)
Ausgabe 04/2018
Kumar, Devarapalli Ravi; Kishore, Dakoju Ravi; Satyanarayana, Gedu:
Palladium-Catalysed Coupling and Acid-Mediated Cyclisation: Synthesis of Fluorenones and Fluorenes
HTML
PDF (738 kb)
Panwar, Rahul; Shally; Shaw, Ranjay; Elagamy, Amr; Shah, Chandan; Pratap, Ramendra:
Substituent-Dependent Chemoselective Synthesis of Highly Functionalized Benzo[
h
]quinolines and 4-Benzylpyrans from 2-Methyl-5-nitro-benzonitrile
HTML
PDF (721 kb)
Bandatmakuru, Sreenivasulareddy; Arava, Veerareddy:
Novel Synthesis of 1,2-Substituted 4-Quinolones
HTML
PDF (491 kb)
Mayooufi, A.; Romdhani-Younes, M.; Thibonnet, J.:
Efficient One-Pot Synthesis of Triazole-Linked Morpholinone Scaffolds by CuAAC in the Presence of 18-Crown-6
HTML
PDF (490 kb)
Delaye, Pierre-Olivier; Pénichon, Mélanie; Boudesocque-Delaye, Leslie; Enguehard-Gueiffier, Cécile; Gueiffier, Alain:
Natural Deep Eutectic Solvents as Sustainable Solvents for Suzuki–Miyaura Cross-Coupling Reactions Applied to Imidazo-Fused Heterocycles
HTML
PDF (514 kb)
Ausgabe 03/2018
Nagalatha, G.; Narala, Siva Ganesh; Narsaiah, A. Venkat:
First Stereoselective Total Synthesis of Tumonoic Acid A and its Derivatives
HTML
PDF (328 kb)
Ausgabe 02/2018
Balalas, T. D.; Stratidis, G.; Papatheodorou, D.; Vlachou, E.-E.; Gabriel, C.; Hadjipavlou-Litina, D. J.; Litinas, K. E.:
One-pot Synthesis of 2-Substituted 4
H
-Chromeno[3,4-
d
]oxazol-4-ones from 4-Hydroxy-3-nitrocoumarin and Acids in the Presence of Triphenylphosphine and Phosphorus Pentoxide under Microwave Irradiation
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PDF (1920 kb)
Ahsan, Mohamed J.; Kumawat, Bhawani S.; Kumawat, Sonu; Sharma, Piush; Bakht, Mohammad A.; Hassan, Mohd Z.; Hussain, Afzal; Saraswat, Pankaj; Khalilullah, Habibullah:
Synthesis and Cytotoxic Evaluation of 3-(4-Fluorophenyl)-4,5-dihydro-5-(3,4,5-trimethoxy/4-nitrophenyl)-
N
-(substituted-phenyl)pyrazole-1-carboxamide Analogues
HTML
PDF (2065 kb)
Kour, M.; Gupta, R.; Saini, R.; Bansal, R. K.:
Diastereoselectivity in the Aza-Michael Reaction of Chiral α-Methylbenzylamines with α,β-Unsaturated Carbonyl Compounds
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PDF (1286 kb)
Mourya, Mohini; Sharma, Himanshu; Joshi, Yogesh C.; Basak, Ashok K.:
[4+3]-Annulation of 3-Cyano-4-aryl-2-iminochromenes with 1,2-Diaminobenzene: An Access to Novel Chromenobenzodiazepines
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PDF (374 kb)
Tiwari, Raju; Nath, Mahendra:
A Divergent Approach to β-Pyrazine-Fused
meso
-Tetraphenyldiporphyrins
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PDF (2209 kb)
Gujjarappa, Raghuram; Vodnala, Nagaraju; Kabi, Arup K.; Kaldhi, Dhananjaya; Kumar, Mohan; Beifuss, Uwe; Malakar, Chandi C.:
Efficient Syntheses of Diverse N-Heterocycles: The Molybdenum(VI)-Catalyzed Reductive Cyclization of Nitroarenes using Pinacol as a Deoxygenating Agent
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PDF (506 kb)
Nagaraju, Kare; Rajesh, Nomula; Krishna, Palakodety Radha:
Synthesis of Phthalimides: A New Entry via TBAI-Catalyzed Intramolecular Cyclization of 2-(Hydroxymethyl)benzamides
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PDF (348 kb)
Pathan, Mosim Amin; Khan, Faiz Ahmed:
Synthesis of Substituted Pyrido-oxazine through Tandem S
N
2 and S
N
Ar Reaction
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PDF (2148 kb)
Matziari, Magdalini; Xie, Yixin:
One-Pot Synthesis of α-Substituted Acrylates
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PDF (457 kb)
Shields, Samuel W. J.; Buist, Peter H.; Manthorpe, Jeffrey M.:
Asymmetric and Regiospecific Synthesis of Isotopically Labelled Cyclopropane Fatty Acid (9
R
,10
S
)-Dihydrosterculic Acid: Overcoming Spontaneous Protonation During Lithium-Sulfoxide Exchange
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PDF (528 kb)
Rana, Anil; Kumar, Varun; Tiwari, Lata; Thakur, Anamika; Meena, Chhuttan Lal; Mahajan, Dinesh:
Triflic Anhydride Promoted Synthesis of Primary Amides and their Conversion into Nitriles
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PDF (676 kb)
Grollmisch, A.; Kragl, U.; Großeheilmann, J.:
Enzyme Immobilization in Polymerized Ionic Liquids-based Hydrogels for Active and Reusable Biocatalysts
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PDF (1049 kb)
Rahman, Masood ur; Ayoob, Iram; Rehman, Shakeel u; Bhat, Khursheed A.; Ara, Tabassum:
Microwave-Assisted Synthesis of Andrographolide Analogues as Potent β-Glycosidase Inhibitors
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PDF (702 kb)
Choudhary, Rakhee; Bai, Rekha; Singh, Pratibha; Sharma, Mahesh C.; Badsara, Satpal Singh:
Room Temperature, Open-Flask C–P Bond-Formation on Water under Catalyst-Free Conditions
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PDF (541 kb)
Ausgabe 01/2018
Songsichan, T.; Katrun, P.; Khaikate, O.; Soorukram, D.; Pohmakotr, M.; Reutrakul, V.; Kuhakarn, C.:
Thiocyanation of Pyrazoles Using KSCN/K
2
S
2
O
8
Combination
HTML
PDF (649 kb)
Kummari, Bhaskar; Ramesh, Perla; Polkam, Naveen; Malthum, Shankaraiah; Vishnuvardhan, M. V. P. S.; Anireddy, Jaya Shree:
Design, Synthesis, and Cytotoxic Evaluation of Etodolac-1,3,4-oxadiazole-1,2,3-triazole Molecules
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PDF (569 kb)
Uma, Pathki; Rajanna, Kamatala Chinna; Sriram, Yelike Hemanth; Premalatha, Akarapu; Saipraksh, Pondichery Kuppuswamy:
Synthesis of 3-(4-(Benzo[
d
]thiazol-2-yl)phenyl)-5-aryl-1,3,5-oxadiazinane-4-thiones and 1-(4-(Benzo[
d
]thiazol-2-yl)phenyl)-5-methyl-3-aryl-1,3,5-triazinane-2-thiones
HTML
PDF (379 kb)
Caillé, Julien; Setzer, Paul; Boeda, Fabien; Pearson-Long, Morwenna S. M.; Bertus, Philippe:
Asymmetric Titanium-Catalyzed Cyclopropanation of Nitriles with Grignard Reagents
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Nakao, Michiyasu; Nishikiori, Nanako; Nakamura, Akihito; Miyagi, Murasaki; Shibata, Nao; Kitaike, Syuji; Fukui, Makoto; Ito, Hiro-O; Sano, Shigeki:
Synthesis of Sterically Protected Isoindoles from
ortho
-Phthalaldehyde
HTML
PDF (2131 kb)
Reddy, A. Maheswara; Sabitha, Gowravaram:
First Total Synthesis of Cryptopyranmoscatone A3 and Cryptopyranmoscatone B4
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PDF (802 kb)
Menczinger, B.; Nemes, A.; Csámpai, A.; Rábai, J.:
Synthesis of 3-(Arylthio)propionic Acids from Nonactivated Aryl Iodides and their Use as Odorless Aryl Mercaptan Surrogates
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PDF (2519 kb)
Ausgabe 01/2017
Zeng, Meng-Tian; Xu, Wan; Liu, Min; Liu, Xing; Chang, Cai-Zhu; Zhu, Hui; Dong, Zhi-Bing:
Iodobenzene-Promoted Pd-Catalysed
ortho
-Directed C–H Activation: The Synthesis of Benzothiazoles via Intramolecular Coupling
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PDF (447 kb)
Ghosal, Nirnita Chakraborty; Mahato, Sachinta; Chatterjee, Rana; Santra, Sougata; Zyryanov, Grigory V.; Majee, Adinath:
A Mild and Efficient Method for the Syntheses and Regioselective Ring-Opening of Aziridines
HTML
PDF (848 kb)
Diez-Martinez, Alba; Krishnamurthy, Ramanarayanan:
Investigations towards the Synthesis of 5-Amino-
l
-lyxofuranosides and 4-Amino-lyxopyranosides and NMR Analysis
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PDF (1536 kb)
Panda, Siva S.; Asiri, Abdullah M.; Elagawany, Mohamed; Buchanan, Devan D.; Torkian, Behrad; Bathala, Keerthana; Thomas, Sean J.; Capito, Jason E.; Arshad, Muhammad N.; Al-Romaizan, Abeer N.:
Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates
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PDF (846 kb)
Ge, Haihong; Liu, Shuang; Cai, Yan; Gao, Zenghui; Du, Siyi; Miao, Zhiwei; Xie, Guixian:
Diastereoselective [Cu(MeCN)
4
BF
4
/BF
3
·Et
2
O]-Catalyzed Cyclopropenation of Alkynes: Asymmetric Synthesis of β-Amino-α-cyclopropenyl Phosphonates
HTML
PDF (510 kb)
Li, Jihui; Yu, Weiguang; Hou, Yifeng; Fu, Wenxing; Xu, Shuying; Zhang, Yucang:
An Efficient Protocol for the Synthesis of
O
-Fluoroalkylisoureas through Copper-Catalysed, Three-Component Reaction of Cyanamides, Fluoroalcohols and Diaryliodonium Triflates
HTML
PDF (509 kb)
Nosik, Pavel S.; Artamonov, Oleksiy S.; Ryabukhin, Sergey V.; Grygorenko, Oleksandr O.:
An Approach to 1,1-Disubstituted Pyrazolylcyclopropane Building Blocks
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PDF (443 kb)
Cívicos, José F.; Costa, Paulo R. R.; Domingos, Jorge L. O.:
Palladium-Catalyzed α-Arylation of Dimethyl Malonate and Ethyl Cyanoacetate with
o
-Alkoxybromobenzenes for the Synthesis of Phenylacetic Acid, Esters and Phenylacetonitriles
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PDF (438 kb)
Don Lawson, Chioma; Maza-Iglesias, Max; Sirhan, Muthana M.; Al Dulayymi, Jumaa R.; Baird, Mark S.:
The Synthesis of Single Enantiomers of α-Mycolic Acids of
Mycobacterium tuberculosis
and Related Organisms, with Alternative Cyclopropane Stereochemistries
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PDF (787 kb)
Majeed, Anju; Nagabhushanam, Kalyanam; Majeed, Muhammed; Thomas, Samuel Manoharan; Thajuddin, Nooruddin:
An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues
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PDF (773 kb)
Zhao, Lingyu; Shen, Guodong; Zhang, Tongxin; Wang, Zhen; Liang, Yuhua:
Pd/C-Catalyzed Intramolecular C–H Arylation for the Synthesis of Phenanthridinones and Dibenzo-α-pyrones
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PDF (568 kb)
Yang, Yi-Qiu; Ke, Long-Zhi; Wang, Gui-Fei; Song, Shu-Yong; Qiu, Ming-Ning; Liu, Jian-Jun; Huang, Yun-Sheng:
Synthesis of
N
-Pyridin-2-ylmethyl and
N
-Quinolin-2-ylmethyl Substituted Ethane-1,2-diamines
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PDF (670 kb)
Barcia, Jose C.; Cruces, Jacobo; Salas, Cristian O.; Estévez, Juan C.; Cuellar, Mauricio A.; Tapia, Ricardo A.; Estévez, Ramón J.:
A New Approach to the Synthesis of Benzo[
b
]naphtho[2,3-
b
]furan-6,11-diones and 2-Benzyl-3-hydroxynaphthalene-1,4-diones
HTML
PDF (592 kb)
Maheshwar Reddy, A.; Sabitha, Gowravaram:
Synthesis of the C1–C9, C11–C19 Pyran Core and C19–C24 Fragments of Macrolactin 3
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PDF (506 kb)
