DOI: 10.1055/s-00000083

Synlett

Issue 03 · Volume 24 · February 2013 DOI: 10.1055/s-003-24466

synform

  • A15
    Zanda, Matteo:

    SYNFORM ISSUE 2013/2

    • synpacts

  • 269
    Lalic, Gojko; Rucker, Richard P.:

    Copper-Catalyzed Electrophilic Amination of Organoboron Compounds

    Image for article: Copper-Catalyzed Electrophilic Amination of Organoboron Compounds
  • 276
    Streuff, Jan:

    An Update on Catalytic Strategies for the Synthesis of α-Hydroxyketones

    Image for article: An Update on Catalytic Strategies for the Synthesis of α-Hydroxyketones

    • account

  • 281
    Gualandi, Andrea; Cozzi, Pier Giorgio:

    Stereoselective Organocatalytic Alkylations with Carbenium Ions

    Image for article: Stereoselective Organocatalytic Alkylations with Carbenium Ions

    • cluster

  • 297

    Cluster Cover Page

  • 298
    Yasuda, Nobuyoshi:

    Cluster Preface: Process Chemistry

    Image for article: Cluster Preface: Process Chemistry
  • 301
    Chen, Ying; Crockett, Richard D.; Wang, Xin; Larsen, Robert D.; Cui, Sheng; Faul, Margaret M.:

    Development of a Scalable Synthesis of a VEGFR Inhibitor

    Image for article: Development of a Scalable Synthesis of a VEGFR Inhibitor
    Supporting Information (PDF)
  • 305
    Mudryk, Boguslaw; Joshi, Amit; Ortiz, Adrian; Young, Ian S.; Sawyer, James R.; Zheng, Bin; Sugiyama, Masano; Shi, Zhongping; Müslehiddinoğlu, Jale; Corbett, R. Michael; Kronenthal, David R.; Conlon, David A.:

    Evolution of the Process for the Preparation of a Selective ErbB VEGF Receptor Inhibitor

    Image for article: Evolution of the Process for the Preparation of a Selective ErbB VEGF Receptor Inhibitor
    Supporting Information (PDF)
  • 313
    Houpis, Ioannis N.; Lemaire, Sebastien; Farina, Vittorio; Xiao, Tingting; Liu, Renmao; Nettekoven, Ulrike; Wang, Youchu:

    New Synthesis of 2′,4′-Functionalized Nucleotides via Stereospecific Hydrogenation and Azidation Reactions

    Image for article: New Synthesis of 2′,4′-Functionalized Nucleotides via Stereospecific Hydrogenation and Azidation Reactions
  • 317
    Lu, Bruce Z.; Li, Guisheng; Rodriguez, Sonia; Liu, Jianxu; Eriksson, Magnus C.; Tan, Zhulin; Song, Jinhua J.; Yee, Nathan K.; Farina, Vittorio; Senanayake, Chris H.:

    Development of a Practical Synthesis of 4-[6-(Morpholinomethyl)-pyridin-3-yl]naphthalen-1-amine, a Key Intermediate for the Synthesis of BIRB 1017, a Potent p38 MAP Kinase Inhibitor

    Image for article: Development of a Practical Synthesis of 4-[6-(Morpholinomethyl)-pyridin-3-yl]naphthalen-1-amine, a Key Intermediate for the Synthesis of BIRB 1017, a Potent p38 MAP Kinase Inhibitor
  • 323
    Chase, Charles E.; Fang, Francis G.; Lewis, Bryan M.; Wilkie, Gordon D.; Schnaderbeck, Matthew J.; Zhu, Xiaojie:

    Process Development of Halaven®: Synthesis of the C1–C13 Fragment from d-(–)-Gulono-1,4-lactone

    Image for article: Process Development of Halaven<SUP>®</SUP>: Synthesis of the C1–C13 Fragment from <sc> d</sc>-(–)-Gulono-1,4-lactone
  • 327
    Austad, Brian C.; Benayoud, Farid; Calkins, Trevor L.; Campagna, Silvio; Chase, Charles E.; Choi, Hyeong-wook; Christ, William; Costanzo, Robert; Cutter, James; Endo, Atsushi; Fang, Francis G.; Hu, Yongbo; Lewis, Bryan M.; Lewis, Michael D.; McKenna, Shawn; Noland, Thomas A.; Orr, John D.; Pesant, Marc; Schnaderbeck, Matthew J.; Wilkie, Gordon D.; Abe, Taichi; Asai, Naoki; Asai, Yumi; Kayano, Akio; Kimoto, Yuichi; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Mizuno, Masanori; Nakamura, Taiju; Omae, Takao; Ozeki, Naoki; Suzuki, Taeko; Takigawa, Teiji; Watanabe, Tomohiro; Yoshizawa, Kazuhiro:

    Process Development of Halaven®: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization

    Image for article: Process Development of Halaven<SUP>®</SUP>: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization
    Primary Data (ZIP)
  • 333
    Austad, Brian C.; Calkins, Trevor L.; Chase, Charles E.; Fang, Francis G.; Horstmann, Thomas E.; Hu, Yongbo; Lewis, Bryan M.; Niu, Xiang; Noland, Thomas A.; Orr, John D.; Schnaderbeck, Matthew J.; Zhang, Huiming; Asakawa, Naoki; Asai, Naoki; Chiba, Hiroyuki; Hasebe, Takashi; Hoshino, Yorihisa; Ishizuka, Hiroyuki; Kajima, Takashi; Kayano, Akio; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Miyazawa, Mamoru; Tagami, Katsuya; Watanabe, Tomohiro:

    Commercial Manufacture of Halaven®: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones

    Image for article: Commercial Manufacture of Halaven<SUP>®</SUP>: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones
    Supporting Information (PDF) Primary Data (ZIP)

    • letter

  • 338
    Mayer, Marilyn Graziano; Nador, Fabiana; Volpe, María Alicia; Radivoy, Gabriel:

    High Surface Area CeO2 Promoted Suzuki–Miyaura Cross-Coupling of Arylboronic Acids and Aryl Iodides

    Image for article: High Surface Area CeO<SUB>2</SUB> Promoted Suzuki–Miyaura Cross-Coupling of Arylboronic Acids and Aryl Iodides
  • 343
    Spork, Anatol P.; Ducho, Christian:

    Stereocontrolled Synthesis of 5′- and 6′-Epimeric Analogues of Muraymycin Nucleoside Antibiotics

    Image for article: Stereocontrolled Synthesis of 5′- and 6′-Epimeric Analogues of Muraymycin Nucleoside Antibiotics
    Supporting Information (PDF)
  • 347
    Dighe, Mahesh G.; Lonkar, Sachin L.; Degani, Mariam S.:

    Mechanistic Insights into Palladium Leaching in Novel Pd/C-Catalyzed Boron-Heck Reaction of Arylboronic Acid

    Image for article: Mechanistic Insights into Palladium Leaching in Novel Pd/C-Catalyzed Boron-Heck Reaction of Arylboronic Acid
    Supporting Information (PDF)
  • 351
    Pereshivko, Olga P.; Peshkov, Vsevolod A.; Ermolat’ev, Denis S.; Van der Eycken, Erik V.:

    Fast Assembly of 1H-Imidazo[1,2-a]imidazol-5-amines via Groebke–Blackburn–Bienaymé Reaction with 2-Aminoimidazoles

    Image for article: Fast Assembly of 1<i>H</i>-Imidazo[1,2-<i>a</i>]imidazol-5-amines via Groebke–Blackburn–Bienaymé Reaction with 2-Aminoimidazoles
    Supporting Information (PDF)
  • 355
    Titanyuk, Igor D.; Beletskaya, Irina P.:

    Palladium-Catalyzed Hydroarylation of Diazoacetic Ester

    Image for article: Palladium-Catalyzed Hydroarylation of Diazoacetic Ester
    Supporting Information (PDF)
  • 359
    Ehlers, Peter; Petrosyan, Andranik; Ghochikyan, Tariel V.; Saghyan, Ashot S.; Neubauer, Antje; Lochbrunner, Stefan; Langer, Peter:

    Suzuki–Miyaura Reactions of 2,7-Dichloro-1,8-naphthyridine

    Image for article: Suzuki–Miyaura Reactions of 2,7-Dichloro-1,8-naphthyridine
    Supporting Information (PDF)
  • 363
    Craven, Philip G. E.; Taylor, Richard J. K.:

    Stereocontrolled Routes to 4-Methoxypentadienoates for Use in Natural Product Synthesis

    Image for article: Stereocontrolled Routes to 4-Methoxypentadienoates for Use in Natural Product Synthesis
  • 369
    Varghese, Vimal; Hudlicky, Tomas:

    Total Synthesis of Dihydrocodeine and Hydrocodone via a Double Claisen Rearrangement and C-10/C-11 Closure Strategy

    Image for article: Total Synthesis of Dihydrocodeine and Hydrocodone via a Double Claisen Rearrangement and C-10/C-11 Closure Strategy
  • 375
    Narayama, Akira; Shibatomi, Kazutaka; Soga, Yoshinori; Muto, Tsubasa; Iwasa, Seiji:

    Copper(II)-Catalyzed Enantioselective Fluorination of β-Keto Esters Using Chiral Spiro Oxazoline Ligands

    Image for article: Copper(II)-Catalyzed Enantioselective Fluorination of β-Keto Esters Using Chiral Spiro Oxazoline Ligands
    Supporting Information (PDF)
  • 379
    Choi, Juhee; Kim, Hyunseok; Park, Sangyun; Tae, Jinsung:

    Asymmetric Total Synthesis of (–)-Galanthamine via Intramolecular Heck Reaction of Conjugated Diene

    Image for article: Asymmetric Total Synthesis of (–)-Galanthamine via Intramolecular Heck Reaction of Conjugated Diene
    Supporting Information (PDF)
  • 383
    Xu, Xiangsheng; Li, Tao; Li, Xiaoqing; Shao, Jiangbin:

    Synthesis of Substituted Fluorenes by Cascade Allenylation, Electrocyclization and Intramolecular Friedel–Crafts Reaction of 1,3-Diene-Substituted Propargylic Alcohols

    Image for article: Synthesis of Substituted Fluorenes by Cascade Allenylation, Electrocyclization and Intramolecular Friedel–Crafts Reaction of 1,3-Diene-Substituted Propargylic Alcohols
    Supporting Information (PDF)
  • 389
    Gao, Detian; Back, Thomas G.:

    Synthesis of the Reverse Transcriptase Inhibitor L-737,126 and the CB2 Cannabinoid Receptor Agonist Pravadoline by a Copper-Catalyzed Intramolecular Cross-Coupling

    Image for article: Synthesis of the Reverse Transcriptase Inhibitor L-737,126 and the CB<SUB>2</SUB> Cannabinoid Receptor Agonist Pravadoline by a Copper-Catalyzed Intramolecular Cross-Coupling
  • 394
    Voltrova, Svatava; Srogl, Jiri:

    Expedient Method for Samarium(II) Iodide Preparation Utilizing a Flow Approach

    Image for article: Expedient Method for Samarium(II) Iodide Preparation Utilizing a Flow Approach

    • spotlight

  • 397
    Fintelman Dias, Flaviana Rodrigues:

    Ethyl 2-Diazoacetoacetate

  • 399
    Gigant, Nicolas:

    Triflic Acid

    • erratum

  • e1
    Chase, Charles E.; Fang, Francis G.; Lewis, Bryan M.; Wilkie, Gordon D.; Schnaderbeck, Matthew J.; Zhu, Xiaojie:

    Process Development of Halaven®: Synthesis of the C1–C13 Fragment from d-(–)-Gulono-1,4-lactone

  • e2
    Austad, Brian C.; Benayoud, Farid; Calkins, Trevor L.; Campagna, Silvio; Chase, Charles E.; Choi, Hyeong-wook; Christ, William; Costanzo, Robert; Cutter, James; Endo, Atsushi; Fang, Francis G.; Hu, Yongbo; Lewis, Bryan M.; Lewis, Michael D.; McKenna, Shawn; Noland, Thomas A.; Orr, John D.; Pesant, Marc; Schnaderbeck, Matthew J.; Wilkie, Gordon D.; Abe, Taichi; Asai, Naoki; Asai, Yumi; Kayano, Akio; Kimoto, Yuichi; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Mizuno, Masanori; Nakamura, Taiju; Omae, Takao; Ozeki, Naoki; Suzuki, Taeko; Takigawa, Teiji; Watanabe, Tomohiro; Yoshizawa, Kazuhiro:

    Process Development of Halaven®: Synthesis of the C14–C35 Fragment via Iterative Nozaki–Hiyama–Kishi Reaction–Williamson Ether Cyclization

  • e3
    Austad, Brian C.; Calkins, Trevor L.; Chase, Charles E.; Fang, Francis G.; Horstmann, Thomas E.; Hu, Yongbo; Lewis, Bryan M.; Niu, Xiang; Noland, Thomas A.; Orr, John D.; Schnaderbeck, Matthew J.; Zhang, Huiming; Asakawa, Naoki; Asai, Naoki; Chiba, Hiroyuki; Hasebe, Takashi; Hoshino, Yorihisa; Ishizuka, Hiroyuki; Kajima, Takashi; Kayano, Akio; Komatsu, Yuki; Kubota, Manabu; Kuroda, Hirofumi; Miyazawa, Mamoru; Tagami, Katsuya; Watanabe, Tomohiro:

    Commercial Manufacture of Halaven®: Chemoselective Transformations En Route to Structurally Complex Macrocyclic Ketones