Synthesis

Issue 13 · July 2013

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editorial
I
Special Issue Dedicated to Professor Scott E. Denmark - Laudation
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1719
Keene, Craig; Kürti, László:
Regiospecific Synthesis of Novel Cyclic Nitrostyrenes and 3-Substituted 2-Nitronaphthalenes

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1730
Richers, Matthew T.; Deb, Indubhusan; Platonova, Alena Yu.; Zhang, Chen; Seidel, Daniel:
Facile Access to Ring-Fused Aminals via Direct α-Amination of Secondary Amines with o-Aminobenzaldehydes: Synthesis of Vasicine, Deoxyvasicine, Deoxyvasicinone, Mackinazolinone, and Ruteacarpine

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paper
1749
Qi, Rui; Wang, Xiao-Na; DeKorver, Kyle A.; Tang, Yu; Wang, Chao-Chao; Li, Qian; Li, Hui; Lv, Ming-Can; Yu, Qing; Hsung, Richard P.:
A Convenient Synthesis of γ-Amino-Ynamides via Additions of Lithiated Ynamides to Aryl Imines; Observation of an Aza-Meyer–Schuster Rearrangement

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1759
Glasspoole, Ben W.; Oderinde, Martins S.; Moore, Brandon D.; Antoft-Finch, Aurora; Crudden, Cathleen M.:
Highly Chemoselective and Enantiospecific Suzuki–Miyaura Cross-Couplings of Benzylic Organoboronic Esters

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1764
Baiazitov, Ramil; Du, Wu; Lee, Chang-Sun; Hwang, Seongwoo; Almstead, Neil G.; Moon, Young-Choon:
Chemoselective Reactions of 4,6-Dichloro-2-(methylsulfonyl)pyrimidine and Related Electrophiles with Amines

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1785
Calkins, Nathan L.; Harmata, Michael:
Further Studies of Benzothiazine Metalation

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1791
Morrill, Christie; Babu, Suresh; Almstead, Neil G.; Moon, Young-Choon:
Synthesis of 1,4-Disubstituted Pyrazolo[3,4-d]pyrimidines from 4,6-Dichloropyrimidine-5-carboxaldehyde: Insights into Selectivity and Reactivity

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1807
Xie, Xiaocong; Fox, Joseph M.:
Diastereoselective Syntheses of Highly Substituted Methylenecyclopropanes via Copper- or Iron-Catalyzed Reactions of 1,2-Disubstituted 3-(Hydroxymethyl)cyclopropenes with Grignard Reagents

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1815
Wender, Paul A.; Billingsley, Kelvin L.:
Lead Diversification through a Prins-Driven Macrocyclization Strategy: Application to C13-Diversified Bryostatin Analogues

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1825
Acharya, Arjun; Eickhoff, John A.; Jeffrey, Christopher S.:
Intramolecular Aza-[4+3] Cycloaddition Reactions of α-Halohydroxamates

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1837
Liskey, Carl W.; Hartwig, John F.:
Borylation of Arenes with Bis(hexylene glycolato)diboron

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1843
Nerurkar, Alok; Chandrasoma, Nalin; Maina, Lincoln; Brassfield, Allen; Luo, Diheng; Brown, Neil; Buszek, Keith R.:
Further Investigations into the Regioselectivity of 6,7-Indole Aryne Cycloadditions with 2-Substituted Furans: Remarkable Contrasteric Preference Depends on Pyrrole and Benzene Ring Substitution

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1853
Castillo-Ramirez, Jorge; Echevarría, Ileabett; Santiago, Janice; Pérez-Torres, Marianela; Rivera-Claudio, Mirna:
Synthesis and Characterization of Ferrocene Acetals and Evaluation of Their Antineoplastic Properties by Using Breast Cancer Cell Lines In Vitro

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1857
Hamilton, James Y.; Morandi, Bill; Carreira, Erick M.:
Homologative Trifluoromethylation of Acetals

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1863
Pansare, Sunil V.; Paul, Eldho K.:
Synthesis of (+)-Febrifugine and a Formal Synthesis of (+)-Halofuginone Employing an Organocatalytic Direct Vinylogous Aldol Reaction

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1870
Sämann, Christoph; Knochel, Paul:
A Convenient Synthesis of α-Substituted β,γ-Unsaturated Ketones and Esters via the Direct Addition of Substituted Allylic Zinc Reagents Prepared by Direct Insertion

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1877
Milicevic Sephton, Selena; Mu, Linjing; Dragic, Martina; Krämer, Stefanie D.; Schibli, Roger; Ametamey, Simon M.:
Synthesis and In Vitro Evaluation of E- and Z-Geometrical Isomers of PSS232 as Potential Metabotropic Glutamate Receptors Subtype 5 (mGlu₅) Binders

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1886
Brucks, Alexandria P.; Treitler, Daniel S.; Liu, Shu-An; Snyder, Scott A.:
Explorations into the Potential of Chiral Sulfonium Reagents to Effect Asymmetric Halonium Additions to Isolated Alkenes

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1899
Snider, Jason R.; Entrekin, Jordan T.; Snowden, Timothy S.; Dolliver, Debra:
Synthesis of Potent CERT Inhibitor HPA-12 Featuring a Tandem Corey–Link and Intramolecular Nucleophilic Acyl Substitution Reaction

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1904
Nguyen, Son T.; Ding, Xiaoyuan; Peet, Norton P.:
A Remarkable Reductive Dearomatization of Thiophene and Furan Rings

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synform
A80
Zanda, Matteo:
SYNFORM ISSUE 2013/7
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