DOI: 10.1055/s-00000084

Synthesis

Issue 13 · Volume 45 · July 2013 DOI: 10.1055/s-003-25222

editorial

  • I

    Special Issue Dedicated to Professor Scott E. Denmark - Laudation

    Image for article: Special Issue Dedicated to Professor Scott E. Denmark - Laudation

    • feature article

  • 1719
    Keene, Craig; Kürti, László:

    Regiospecific Synthesis of Novel Cyclic Nitrostyrenes and 3-Substituted 2-Nitronaphthalenes

    Image for article: Regiospecific Synthesis of Novel Cyclic Nitrostyrenes and 3-Substituted 2-Nitronaphthalenes
    Supporting Information (PDF)
  • 1730
    Richers, Matthew T.; Deb, Indubhusan; Platonova, Alena Yu.; Zhang, Chen; Seidel, Daniel:

    Facile Access to Ring-Fused Aminals via Direct α-Amination of Secondary Amines with o-Aminobenzaldehydes: Synthesis of Vasicine, Deoxyvasicine, Deoxyvasicinone, Mackinazolinone, and Ruteacarpine

    Image for article: Facile Access to Ring-Fused Aminals via Direct α-Amination of Secondary Amines with <i>o</i>-Aminobenzaldehydes: Synthesis of Vasicine, Deoxyvasicine, Deoxyvasicinone, Mackinazolinone, and Ruteacarpine
    Supporting Information (PDF)

    • paper

  • 1749
    Qi, Rui; Wang, Xiao-Na; DeKorver, Kyle A.; Tang, Yu; Wang, Chao-Chao; Li, Qian; Li, Hui; Lv, Ming-Can; Yu, Qing; Hsung, Richard P.:

    A Convenient Synthesis of γ-Amino-Ynamides via Additions of Lithiated Ynamides to Aryl Imines; Observation of an Aza-Meyer–Schuster Rearrangement

    Image for article: A Convenient Synthesis of γ-Amino-Ynamides via Additions of Lithiated Ynamides to Aryl Imines; Observation of an Aza-Meyer–Schuster Rearrangement
  • 1759
    Glasspoole, Ben W.; Oderinde, Martins S.; Moore, Brandon D.; Antoft-Finch, Aurora; Crudden, Cathleen M.:

    Highly Chemoselective and Enantiospecific Suzuki–Miyaura Cross-Couplings of Benzylic Organoboronic Esters

    Image for article: Highly Chemoselective and Enantiospecific Suzuki–Miyaura Cross-Couplings of Benzylic Organoboronic Esters
  • 1764
    Baiazitov, Ramil; Du, Wu; Lee, Chang-Sun; Hwang, Seongwoo; Almstead, Neil G.; Moon, Young-Choon:

    Chemoselective Reactions of 4,6-Dichloro-2-(methylsulfonyl)pyrimidine and Related Electrophiles with Amines

    Image for article: Chemoselective Reactions of 4,6-Dichloro-2-(methylsulfonyl)pyrimidine and Related Electrophiles with Amines
    Supporting Information (PDF)
  • 1785
    Calkins, Nathan L.; Harmata, Michael:

    Further Studies of Benzothiazine Metalation

    Image for article: Further Studies of Benzothiazine Metalation
    Supporting Information (PDF)
  • 1791
    Morrill, Christie; Babu, Suresh; Almstead, Neil G.; Moon, Young-Choon:

    Synthesis of 1,4-Disubstituted Pyrazolo[3,4-d]pyrimidines from 4,6-Dichloropyrimidine-5-carboxaldehyde: Insights into Selectivity and Reactivity

    Image for article: Synthesis of 1,4-Disubstituted Pyrazolo[3,4-<i>d</i>]pyrimidines from 4,6-Dichloropyrimidine-5-carboxaldehyde: Insights into Selectivity and Reactivity
    Supporting Information (PDF)
  • 1807
    Xie, Xiaocong; Fox, Joseph M.:

    Diastereoselective Syntheses of Highly Substituted Methylenecyclopropanes via Copper- or Iron-Catalyzed Reactions of 1,2-Disubstituted 3-(Hydroxy­methyl)cyclopropenes with Grignard Reagents

    Image for article: Diastereoselective Syntheses of Highly Substituted Methylenecyclopropanes via Copper- or Iron-Catalyzed Reactions of 1,2-Disubstituted 3-(Hydroxy­methyl)cyclopropenes with Grignard Reagents
    Supporting Information (PDF)
  • 1815
    Wender, Paul A.; Billingsley, Kelvin L.:

    Lead Diversification through a Prins-Driven Macrocyclization Strategy: Application to C13-Diversified Bryostatin Analogues

    Image for article: Lead Diversification through a Prins-Driven Macrocyclization Strategy: Application to C13-Diversified Bryostatin Analogues
  • 1825
    Acharya, Arjun; Eickhoff, John A.; Jeffrey, Christopher S.:

    Intramolecular Aza-[4+3] Cycloaddition Reactions of α-Halohydroxamates

    Image for article: Intramolecular Aza-[4+3] Cycloaddition Reactions of α-Halohydroxamates
    Supporting Information (PDF)
  • 1837
    Liskey, Carl W.; Hartwig, John F.:

    Borylation of Arenes with Bis(hexylene glycolato)diboron

    Image for article: Borylation of Arenes with Bis(hexylene glycolato)diboron
    Supporting Information (PDF)
  • 1843
    Nerurkar, Alok; Chandrasoma, Nalin; Maina, Lincoln; Brassfield, Allen; Luo, Diheng; Brown, Neil; Buszek, Keith R.:

    Further Investigations into the Regioselectivity of 6,7-Indole Aryne Cyclo­additions with 2-Substituted Furans: Remarkable Contrasteric Preference Depends­ on Pyrrole and Benzene Ring Substitution

    Image for article: Further Investigations into the Regioselectivity of 6,7-Indole Aryne Cyclo­additions with 2-Substituted Furans: Remarkable Contrasteric Preference Depends­ on Pyrrole and Benzene Ring Substitution
  • 1853
    Castillo-Ramirez, Jorge; Echevarría, Ileabett; Santiago, Janice; Pérez-Torres, Marianela; Rivera-Claudio, Mirna:

    Synthesis and Characterization of Ferrocene Acetals and Evaluation of Their Antineoplastic Properties by Using Breast Cancer Cell Lines In Vitro

    Image for article: Synthesis and Characterization of Ferrocene Acetals and Evaluation of Their Antineoplastic Properties by Using Breast Cancer Cell Lines In Vitro
    Supporting Information (PDF)
  • 1857
    Hamilton, James Y.; Morandi, Bill; Carreira, Erick M.:

    Homologative Trifluoromethylation of Acetals

    Image for article: Homologative Trifluoromethylation of Acetals
    Supporting Information (PDF)
  • 1863
    Pansare, Sunil V.; Paul, Eldho K.:

    Synthesis of (+)-Febrifugine and a Formal Synthesis of (+)-Halofuginone Employing an Organocatalytic Direct Vinylogous Aldol Reaction

    Image for article: Synthesis of (+)-Febrifugine and a Formal Synthesis of (+)-Halofuginone Employing an Organocatalytic Direct Vinylogous Aldol Reaction
    Supporting Information (PDF)
  • 1870
    Sämann, Christoph; Knochel, Paul:

    A Convenient Synthesis of α-Substituted β,γ-Unsaturated Ketones and Esters via the Direct Addition of Substituted Allylic Zinc Reagents Prepared by Direct Insertion

    Image for article: A Convenient Synthesis of α-Substituted β,γ-Unsaturated Ketones and Esters via the Direct Addition of Substituted Allylic Zinc Reagents Prepared by Direct Insertion
    Supporting Information (PDF)
  • 1877
    Milicevic Sephton, Selena; Mu, Linjing; Dragic, Martina; Krämer, Stefanie D.; Schibli, Roger; Ametamey, Simon M.:

    Synthesis and In Vitro Evaluation of E- and Z-Geometrical Isomers of PSS232 as Potential Metabotropic Glutamate Receptors Subtype 5 (mGlu5) Binders

    Image for article: Synthesis and In Vitro Evaluation of <i>E</i>- and <i>Z</i>-Geometrical Isomers of PSS232 as Potential Metabotropic Glutamate Receptors Subtype 5 (mGlu<SUB>5</SUB>) Binders
    Supporting Information (PDF)
  • 1886
    Brucks, Alexandria P.; Treitler, Daniel S.; Liu, Shu-An; Snyder, Scott A.:

    Explorations into the Potential of Chiral Sulfonium Reagents to Effect Asymmetric Halonium Additions to Isolated Alkenes

    Image for article: Explorations into the Potential of Chiral Sulfonium Reagents to Effect Asymmetric Halonium Additions to Isolated Alkenes
    Supporting Information (PDF)
  • 1899
    Snider, Jason R.; Entrekin, Jordan T.; Snowden, Timothy S.; Dolliver, Debra:

    Synthesis of Potent CERT Inhibitor HPA-12 Featuring a Tandem Corey–Link and Intramolecular Nucleophilic Acyl Substitution Reaction

    Image for article: Synthesis of Potent CERT Inhibitor HPA-12 Featuring a Tandem Corey–Link and Intramolecular Nucleophilic Acyl Substitution Reaction
    Supporting Information (PDF)
  • 1904
    Nguyen, Son T.; Ding, Xiaoyuan; Peet, Norton P.:

    A Remarkable Reductive Dearomatization of Thiophene and Furan Rings

    Image for article: A Remarkable Reductive Dearomatization of Thiophene and Furan Rings
    Supporting Information (PDF)

    • synform

  • A80
    Zanda, Matteo:

    SYNFORM ISSUE 2013/7