DOI: 10.1055/s-00000083

Synlett

Issue 01 · Volume 26 · January 2015 DOI: 10.1055/s-004-28259

editorial

  • I

    Editorial

    • synform

  • A1
    Zanda, Matteo:

    SYNFORM ISSUE 2015/01

    • synpacts

  • 1
    Glas, Adrian; Grossmann, Tom N.:

    Constraining Peptide Conformations with the Help of Ring-Closing Metathesis

    Image for article: Constraining Peptide Conformations with the Help of Ring-Closing Metathesis

    • account

  • 6
    Ma, Ying-Xian; Meng, Zheng; Chen, Chuan-Feng:

    Synthesis of Substituted Iptycenes

    Image for article: Synthesis of Substituted Iptycenes

    • cluster

  • 31

    Cluster Cover Page

    Image for article: Cluster Cover Page
  • 33
    Browne, Duncan L.:

    Cluster Preface: Progress in Organo-Fluorine Chemistry

    Image for article: Cluster Preface: Progress in Organo-Fluorine Chemistry
  • 36
    Xu, Peng; Guo, Shuo; Wang, Liyan; Tang, Pingping:

    Recent Advances in the Synthesis of Difluoromethylated Arenes

    Image for article: Recent Advances in the Synthesis of Difluoromethylated Arenes
  • 40
    Dai, Xiaoyang; Cahard, Dominique:

    Regio- and Stereocontrolled Nucleophilic Trifluoromethylthiolation of Morita–Baylis–Hillman Carbonates

    Image for article: Regio- and Stereocontrolled Nucleophilic Trifluoromethylthiolation of Morita–Baylis–Hillman Carbonates
    Supporting Information (PDF)
  • 45
    Lishchynskyi, Anton; Mazloomi, Zahra; Grushin, Vladimir V.:

    Trifluoromethylation and Pentafluoroethylation of Vinylic Halides with Low-Cost RfH-Derived CuRf (Rf = CF3, C2F5)

    Image for article: Trifluoromethylation and Pentafluoroethylation of Vinylic Halides with Low-Cost R<sub>f</sub>H-Derived CuR<sub>f</sub> (R<sub>f</sub> = CF<sub>3</sub>, C<sub>2</sub>F<sub>5</sub>)
    Supporting Information (PDF)
  • 51
    Breen, Jessica R.; Sandford, Graham; Patel, Bhairavi; Fray, Jonathan:

    Synthesis of 4,4-Difluoro-1H-pyrazole Derivatives

    Image for article: Synthesis of 4,4-Difluoro-1<i>H</i>-pyrazole Derivatives
    Supporting Information (PDF)
  • 55
    Tarui, Atsushi; Miyata, Erina; Tanaka, Ayumi; Sato, Kazuyuki; Omote, Masaaki; Ando, Akira:

    Stereoselective Suzuki Coupling Reaction of an α-Bromo-α-fluoro-β-lactam

    Image for article: Stereoselective Suzuki Coupling Reaction of an α-Bromo-α-fluoro-β-lactam
    Supporting Information (PDF)
  • 59
    Zhang, Zhikun; Feng, Jiajie; Xu, Yan; Zhang, Songnan; Ye, Yuxuan; Li, Tianjiao; Wang, Xi; Chen, Jun; Zhang, Yan; Wang, Jianbo:

    Synthesis of Trifluoromethylated Cycloheptatrienes from N-Tosylhydrazones: Transition-Metal-Free Büchner Ring Expansion

    Image for article: Synthesis of Trifluoromethylated Cycloheptatrienes from <i>N</i>-Tosylhydrazones: Transition-Metal-Free Büchner Ring Expansion
    Supporting Information (PDF)
  • 63
    Kageshima, Yoshiya; Suzuki, Chiharu; Oshiro, Kojun; Amii, Hideki:

    Highly Controlled Ring-Opening of Siloxydifluorocyclopropanes: A Versatile Route to Cyclic Fluoroketones

    Image for article: Highly Controlled Ring-Opening of Siloxydifluorocyclopropanes: A Versatile Route to Cyclic Fluoroketones
    Supporting Information (PDF)
  • 67
    Liu, Yingle; Yang, Yi; Huang, Yangen; Xu, Xiu-Hua; Qing, Feng-Ling:

    Regio- and Diastereoselective Vinylogous Mannich Addition of 3-Alkenyl-2-oxindoles to α-Fluoroalkyl Aldimines

    Image for article: Regio- and Diastereoselective Vinylogous Mannich Addition of 3-Alkenyl-2-oxindoles to α-Fluoroalkyl Aldimines
    Supporting Information (PDF)
  • 73
    Hendriks, Christine M. M.; Reball, Jens; Bolm, Carsten:

    Methyl 4-Pentafluorosulfanylphenyl Sulfoximines

    Image for article: Methyl 4-Pentafluorosulfanylphenyl Sulfoximines
    Supporting Information (PDF)
  • 76
    Alazet, Sébastien; Billard, Thierry:

    Electrophilic Aromatic Trifluoromethylthiolation with the Second Generation of Trifluoromethanesulfenamide

    Image for article: Electrophilic Aromatic Trifluoromethylthiolation with the Second Generation of Trifluoromethanesulfenamide
    Supporting Information (PDF)

    • letter

  • 79
    Patel, Bhaven; Hilton, Stephen T.:

    A Radical-Mediated Approach to the Total Synthesis of Fluorinated Marinoquinoline A and Related Tricyclic and Tetracyclic Congeners

    Image for article: A Radical-Mediated Approach to the Total Synthesis of Fluorinated Marinoquinoline A and Related Tricyclic and Tetracyclic Congeners
    Supporting Information (PDF)
  • 84
    Antoniak, Damian; Sakowicz, Arkadiusz; Loska, Rafał; Mąkosza, Mieczysław:

    Direct Conversion of Aromatic Aldehydes into Benzamides via Oxidation with Potassium Permanganate in Liquid Ammonia

    Image for article: Direct Conversion of Aromatic Aldehydes into Benzamides via Oxidation with Potassium Permanganate in Liquid Ammonia
    Supporting Information (PDF)
  • 87
    Sarbu, Laura G.; Hopf, Henning; Grunenberg, Jörg; Birsa, Lucian M.:

    Reduction of Pseudo-geminal Bis(ethynyl)-Substituted [2.2]Paracyclophanes

    Image for article: Reduction of Pseudo-geminal Bis(ethynyl)-Substituted [2.2]Paracyclophanes
  • 91
    Sarmah, Manas M.; Prajapati, Dipak:

    Ultrasound-Mediated One-Pot Synthesis of 7-Methyl-Substituted Pyrido[4,3-d]pyrimidine Scaffolds by a Catalyst-Free Protocol

    Image for article: Ultrasound-Mediated One-Pot Synthesis of 7-Methyl-Substituted Pyrido[4,3-<i>d</i>]pyrimidine Scaffolds by a Catalyst-Free Protocol
    Supporting Information (PDF)
  • 95
    Trillo, Paz; Gómez-Martínez, Melania; Alonso, Diego A.; Baeza, Alejandro:

    2-Aminobenzimidazole Organocatalyzed Asymmetric Amination of Cyclic 1,3-Dicarbonyl Compounds

    Image for article: 2-Aminobenzimidazole Organocatalyzed Asymmetric Amination of Cyclic 1,3-Dicarbonyl Compounds
    Supporting Information (PDF)
  • 101
    Teimouri, Mohammad Bagher; Asnaashari, Bita; Moayedi, Maryam; Naderi, Soheila:

    Diastereoselective One-Pot Synthesis of Succinimides Bearing a Chromone Unit

    Image for article: Diastereoselective One-Pot Synthesis of Succinimides Bearing a Chromone Unit
    Supporting Information (PDF)
  • 108
    Hajibabaei, Khadijeh; Zali-Boeini, Hassan:

    One-Pot Multicomponent Domino Synthesis of 4-Aminothiazole-2(3H)-thiones

    Image for article: One-Pot Multicomponent Domino Synthesis of 4-Aminothiazole-2(3<i>H</i>)-thiones
  • 111
    Stockton, Kieran P.; Glover, Stephen A.; Greatrex, Ben W.:

    Nucleophilic Trapping of Alkoxy-Stabilized Oxyallyl Systems Generated from Inosose 2-O-Mesylates

    Image for article: Nucleophilic Trapping of Alkoxy-Stabilized Oxyallyl Systems Generated from Inosose 2-<i>O-</i>Mesylates
    Supporting Information (PDF)
  • 116
    Li, Yanru; Zhang, Luyan; Yuan, Haiyan; Liang, Fushun; Zhang, Jingping:

    Rapid α-Amination of N-Substituted Indoles by Using DBU-Activated N-Haloimides as Nitrogen Sources

    Image for article: Rapid α-Amination of N-Substituted Indoles by Using DBU-Activated <i>N</i>-Haloimides as Nitrogen Sources
    Supporting Information (PDF)
  • 123
    Capitta, Francesca; Frongia, Angelo; Ollivier, Jean; Aitken, David J.; Secci, Francesco; Piras, Pier Paolo; Guillot, Régis:

    Enantioselective Organocatalyzed Desymmetrization of 3-Substituted Cyclobutanones through Michael Addition to Nitroalkenes

    Image for article: Enantioselective Organocatalyzed Desymmetrization of 3-Substituted Cyclobutanones through Michael Addition to Nitroalkenes
    Supporting Information (PDF)
  • 127
    Qian, Jinlong; Yi, Wenbin; Lv, Meifang; Cai, Chun:

    A Facile and Mild Approach for Stereoselective Synthesis of α-Fluoro-α,β-unsaturated Esters from α-Fluoro-β-keto Esters via Deacylation

    Image for article: A Facile and Mild Approach for Stereoselective Synthesis of α-Fluoro-α,β-unsaturated Esters from α-Fluoro-β-keto Esters via Deacylation
    Supporting Information (PDF)

    • spotlight

  • 133
    Gao, Kai:

    Hypophosphorous Acid

  • 135
    Mears, Paul R.:

    3,3,3-Bromodifluoro-1-propene: The Mild Introduction of CF2