DOI: 10.1055/s-00000131

Synfacts

Issue 10 · Volume 15 · October 2019 DOI: 10.1055/s-009-44215

Synform

  • A148

    SYNFORM ISSUE 2019/10

    • Synthesis of Natural Products and Potential Drugs

  • z1089

    All PDFs of this category

  • 1089

    Total Synthesis of Gymnocin B

  • 1090

    Synthesis of (±)-Hirsutene

  • 1091

    Synthesis of AZD6738

  • 1092

    Synthesis of GDC-0077

  • 1093

    Synthesis of (–)-Salinosporamide A

  • 1094

    Synthesis of Aspidosperma Alkaloids by a Radical Cyclization Strategy

  • 1095

    Total Synthesis of (−)-Nemorosone and (−)-6-epi-Garcimultiflorone A

  • 1096

    Synthesis of GSK2981278A

  • 1097

    Synthesis of SIPI 6398

  • 1098

    Synthesis of M-89

  • 1099

    Synthesis of (+)-Dapholdhamine B

  • 1100

    Synthesis of Ziresovir

  • 1101

    Stereochemical Revision and Total Synthesis of Mytilipin B

  • 1102

    Synthesis of Dapagliflozin

  • 1103

    Synthesis of a CCR4 Antagonist

  • 1104

    Synthesis of ABBC-2222

    • Synthesis of Heterocycles

  • z1105

    All PDFs of this category

  • 1105

    Enantioselective Synthesis of Cyclic Dipeptides by Iridium-Catalyzed Hydrogenation

  • 1106

    Rhodium-Catalyzed Synthesis of Chiral Sulfoximines and 1,2-Benzothiazines

  • 1107

    Pyridine Synthesis by 6π-3-Azatriene Electrocyclization

  • 1108

    Copper-Catalyzed Iodine-Mediated Synthesis of Indolizines

  • 1109

    Palladium–NHC Catalyzed Coupling of Organolithium Reagents at Low Temperatures

  • 1110

    N-Acetyl-Directed Cyclopropanation of Indoles

  • 1111

    Synthesis of Spirocyclic Thiadiazino Quinazolinones

  • 1112

    3-Aroylquinolines by a Three-Component Reaction of Anilines, Enaminones, and DMSO

  • 1113

    Palladium(II)-Catalyzed Synthesis of Pyrroles from Alkynylimines and Isocyanides

  • 1114

    Brønsted Acid Catalyzed Synthesis of α-(3-Indolyl) Ketones

  • 1115

    Enantioselective Cyclization of Alkenyl Amides to Polycyclic Dihydroindoles

  • 1116

    Photoredox Approach to Fluorinated Pyrrolo[1,2-a][1,5]benzodiazepines

  • 1117

    Photoredox-Mediated Pyridonation of (Het)Arenes

  • 1118

    Decarboxylative Cross-Coupling of α-Amino Acids and α-Oxy Acids with Aryl Nitriles

  • 1119

    Cobalt-Catalyzed Synthesis of Benzoindol-2-ones from Naphthylamides

    • Synthesis of Materials and Unnatural Products

  • z1121

    All PDFs of this category

  • 1121

    Synthesis of Conjugated Nanohoops Containing Antiaromatic Units

  • 1122

    Ladies & Gentlemen: The Nanocone

  • 1123

    Get Your Chloride Here

  • 1124

    Synthesis of Cryptophane-Type Xenon Hosts with Biosensing Application

  • 1125

    Emerging from the Flatlands Using Diels–Alder Cycloaddition

  • 1126

    3D Aromaticity: Two Wrongs Do Make a Right in Antiaromatic Cyclophanes

  • 1127

    Tying the Molecular Knot

  • 1128

    Non-Aromatic Superbenzoquinones

  • 1129

    Stabilizing Imine-Based COFs by Oxidative Cyclization

  • 1130

    New Molecular Machines? Phosphonium Donor-π-Acceptor Dyes with Tunable Dual Emission

  • 1131

    When Aufbau Needs to Bow Down: Highly Photostable and Luminescent Donor–Acceptor Organic Radicals

  • 1132

    Rebuilding from the Dust: Suzuki–Miyaura Cross-Coupling Using Mechanical Grinding

    • Metals in Synthesis

  • z1133

    All PDFs of this category

  • 1133

    Regio- and Enantioselective Cobalt-Catalyzed Allylic Amination

  • 1134

    Decarboxylative Difluoromethylation via Copper Catalysis

  • 1135

    Gold-Catalyzed Enantioselective Cyclizations of Enynes through Remote Enantioinduction

  • 1136

    NiH-Catalyzed Remote Hydroarylation of Alkenes

  • 1137

    α-Arylation of Carboxylic Acids and Secondary Amides

  • 1138

    Nickel-Catalyzed Decarboxylative Allylation with C-Centered Nucleophiles

  • 1139

    Formation of Tertiary C–F Bonds through Enantioselective Palladium-Catalyzed Cross-Coupling

  • 1140

    Palladium-Catalyzed Synthesis of Alkenylated α,β-Unsaturated Lactams

  • 1141

    Copper-Catalyzed Enantioselective Alkylation of N-Heterocyclic Michael Acceptors

  • 1142

    Synthesis of β-Branched Arylethylamines

  • 1143

    The Kulinkovich Reaction

  • 1144

    Synthesis of Chiral α‑CF3 Thioethers

  • 1145

    Direct Photoredox-Mediated Giese Reactions

  • 1146

    Enantioselective Intramolecular Hydroarylation of Enones

  • 1147

    Palladium-Catalyzed Synthesis of Enantioenriched Tertiary Nitroalkanes

  • 1148

    Aminotrifluoromethylation of Alkenes via Copper Catalysis

  • 1149

    Iridium-Catalyzed Regiodivergent Oxyamination of Unactivated Alkenes

  • 1150

    Enantioselective Thiocarbonylation of Styrenes

  • 1151

    Gold(I)-Catalyzed Stereoselective Cyclization Reactions

  • 1152

    Enantioselective Ring-Opening of Cyclic Diaryliodonium Salts

  • 1153

    Cobalt-Catalyzed Acylation Using Thiopyridyl Ester Derivatives

  • 1154

    Nickel-Catalyzed Decarboxylative Coupling of Carboxylic Acid Esters

  • 1155

    Copper-Catalyzed 1,4-Reduction of Vinyl Epoxides and Epoxyenynes

  • 1156

    Palladium Catalyzed Atroposelective C–H Functionalization

  • 1157

    Enantioselective Copper-Catalyzed SN2′ Substitution on Allylic Phosphates using Allenyl Boronates

  • 1158

    Copper-Catalyzed Synthesis of Enantioenriched β-Hydroxy Allenes

  • 1159

    CO2-Based Carboxylation of C–F Bonds under Copper Catalysis

  • 1160

    A New Reductive Arylation of Redox-Active Sulfones

    • Polymer-Supported Synthesis

  • z1161

    All PDFs of this category

  • 1161

    Enantioselective Michael Addition Using Quinine Adsorbed in Alginate Gel

  • 1162

    Intramolecular Cyclization of 2-Allylanilines and 2-Allylphenols on Pd/C

  • 1163

    Stille Coupling Catalyzed by Gold Nanoparticles Formed In Situ on Active Carbon

  • 1164

    Heterogeneous Tungsten-Catalyzed Synthesis of 2-Azapyrrolizidines

  • 1165

    Ferrier Rearrangements Catalyzed by a Magnetic Iron(III) Nanocatalyst

  • 1166

    Asymmetric Epoxidation of Allylic Alcohols on Polystyrene-Supported Vanadium

  • 1167

    Palladium Nanoparticle Catalyzed Sonogashira Coupling in Water

  • 1168

    Hydrogenation of Carbonyl Compounds by Platinum on Ceria–Zirconia

  • 1169

    Reduction of Nitroarenes on Goethite-Supported Rhodium Nanoparticles

  • 1170

    Deacylation Coupling and Cyclization Catalyzed by a Magnetic Metal–Organic Framework

  • 1171

    Cyanation of Terminal Alkynes with Switchable Copper Metal–Organic Frameworks

  • 1172

    Suzuki–Miyaura Coupling Catalyzed by Ligand-Stabilized Palladium Nanoparticles

  • 1173

    Primary Aniline Synthesis by Dehydrogenative Aromatization on Pd Nanoparticles

  • 1174

    Palladium-Free Sonogashira Coupling with Supported Copper Nanoparticles

    • Organo- and Biocatalysis

  • z1175

    All PDFs of this category

  • 1175

    Sulfenylation/Semipinacol Reaction of Di- and Trisubstituted Allylic Alcohols

  • 1176

    Dehydrative Annulation of Amines with Carboxylic Acids via PIII/PV Catalysis

  • 1177

    Stereoselective Radical Cyclization by Photoexcited Flavoenzymes

  • 1178

    Organocatalytic Aldehyde Olefination: Synthesis of α,β-Disubstituted Acrylates

  • 1179

    Benzylic Photocarboxylation through C–H Bond Photoactivation

  • 1180

    Radical Chain Reaction Catalyzed by Organic Super Electron Donors

  • 1181

    Electrophotoredox Coupling Between Arenes and Nitrogen Heteroaromatics

  • 1182

    Coordinatively Saturated Phosphorus(V) Species Initiates Silylium Catalysis

  • 1183

    Asymmetric Lewis Base-Catalyzed Sulfenoacetalization of Alkenals

  • 1184

    Organocatalytic Synthesis of γ-Butyrolactones

  • 1185

    The Steglich Esterification

    • Chemistry in Medicine and Biology

  • z1187

    All PDFs of this category

  • 1187

    Binding-Site Hotspot Mapping using Photochemical Proteomics

  • 1188

    Structure-Guided Discovery of Selective Mcl-1 Inhibitors

  • 1189

    Ethynylphosphonamidates in the Synthesis of Antibody–Drug Conjugates

  • 1190

    A Reagent for Doubly Bioorthogonal Cysteine Labeling

  • 1191

    Staudinger Ligation in Living Animals

  • 1192

    Photocatalytic Defluoroalkylation of Unactivated Trifluoromethylarenes

  • 1193

    Targeted Degradation of Extracellular Proteins with ENDTACs

  • 1194

    Profiling of Inhibitor-Bound Kinase Complexes

  • 1195

    Selenophosph(V)azanes as Transporters and Sensors

  • 1196

    Defying the Odds – Drugging KRAS

  • 1197

    In vivo Visualization of Copper(II) in the Brain

    • Peptide Chemistry

  • z1199

    All PDFs of this category

  • 1199

    Modified KAHA Ligation for Protein Synthesis

  • 1200

    Selenium-Auxiliary-Mediated Chemical Ligation

  • 1201

    Sulfide-Mediated Peptide Ligation in Water

  • 1202

    Palladium-Catalyzed Hydrogenation of β-Fluoroalkyl β-Amino Acrylic Acids

  • 1203

    Stereoselective Synthesis of α-Allyl Amino Esters by Organocatalysis

  • 1204

    Formamide-Catalyzed Efficient Amidation and Esterification

  • 1205

    Atroposelective Couplings of Indoles with Amino Acid Derivatives

  • 1206

    Synthesis of Selenocysteine-Based Peptides

  • 1207

    Staudinger Ligation for the Synthesis of Peptides

  • 1208

    Cooperative Catalysis for Asymmetric Multicomponent Reactions

  • 1209

    Removal of Aminoquinoline Auxiliary from Protected α-Amino Acids

    • Flow Chemistry

  • z1211

    All PDFs of this category

  • 1211

    Ibuprofen in Continuous Flow without Headache

  • 1212

    Synthesis of α-CF2H-Substituted Ketones from Styrenes via Photoredox Catalysis in Flow

  • 1213

    Three-Step Streamlined Flow Synthesis of Imatinib and Analogues

  • 1214

    Continuous-Flow Photochemical Iodoperfluoroalkylation of Alkenes