DOI:
10.1055/s-00000083
Synlett
Issue Small-Molecule MedChem ·
Volume ·
2025
DOI: 10.1055/s-015-61587
Emerging Trends in Organic Chemistry: A Focus on India
Small Molecules in Medicinal Chemistry
Candito, David A.;
Simov, Vladimir;
Liu, Ping;
Ardolino, Michael J.;
Martinot, Theodore;
Lyons, Thomas;
Qi, Ji;
Yin, Jingjun;
Hao, Jinglai;
Hu, Bin;
Chen, Meng;
Zhang, Jun;
Lam, Yu-hong;
Fuller, Peter H.;
Ellis, J. Michael;
Maddess, Matthew:
A Concise Synthesis of a Key Azabicyclo[2.1.1]hexane Building Block for N-Heteroaryl Indazole LRRK2 Kinase Inhibitors
Alaeddini, AmirHossein;
Karimian, Somaye;
Noori, Milad;
Dastyafteh, Navid;
Mohammadi-Khanaposhtani, Maryam;
Ghomi, Minoo Khalili;
Bararjanian, Morteza;
Iraji, Aida;
Javanshir, Shahrzad;
Larijani, Bagher;
Ranjbar, Parviz Rashidi;
Mahdavi, Mohammad:
Design, Synthesis, Enzymatic Inhibition, and Antioxidant Activity of New 4-Phenylpiperazin-phenoxy-1,2,3-triazol-acetamide Derivatives as Tyrosinase Inhibitors
Goel, Kapil Kumar;
Singhal, Peeush;
Marianesan, Arockia Babu;
Pandey, Sarvesh Kumar;
Kumar, Roshan;
Singh, Thakur Gurjeet;
Tyagi, Yogita;
Gaidhane, Shilpa;
Singh, Mahendra Pratap;
Dwivedi, Ashish Ranjan:
A Decade of Piperazine-Based Small Molecules Approved by U.S. FDA: Exploring the Medicinal Chemistry Impact of this Versatile Pharmacophore
Shaw, Suman K.;
Dey, Rajdeep;
Yadav, Ruchi;
Baldiwala, Aliasgar;
Patel, Manan;
Patel, Bhumika D.;
Bhatt, Hardik G.;
Natesan, Gopal;
Jha, Abhishek;
Chaube, Udit:
Exploring Tetrahydroquinoline Derivatives: A New Frontier in Cancer Treatment
Khanka, Sonu;
Rawat, Kundan S.;
Pandey, Priyanka;
Pal, Shyamal;
Vats, Ravi P.;
Rathur, Rajat;
Sharma, Kriti;
Dipali, Divya;
Singh, Divya;
Goel, Atul:
An Efficient Synthesis of 3-Aryl-2H-chromene Derivatives as Potential Bone Anabolic Agents
Sakamoto, Masaharu;
Kai, Seriha;
Tateishi, Hiroshi;
Biswas, Tanima;
Sakamoto, Takashi;
Teshima, Misaki;
Iwanaga, Misaki;
Nishikawa, Akiko;
Sakamoto, Arisa;
Shimozono, Rie;
Kameyama, Hiroki;
Nambu, Masami;
Masunaga, Takuya;
Anraku, Kensaku;
Fujita, Mikako;
Otsuka, Masami:
Oxaprozin and SB-431542 Hybrid Molecule Inhibits Fibrosis and Cancer Cell Migration
Toledano-Pinedo, Mireia;
Diez-Iriepa, Daniel;
Porro-Pérez, Alicia;
Schäker-Hübner, Linda;
Hanl, Maria;
Samadi, Abdelouahid;
Almendros, Pedro;
Iriepa, Isabel;
Rodríguez-Fernández, M. Mercedes;
Griñán-Ferré, Christian;
Siwek, Agata;
Wolak, Małgorzata;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Doroż-Płonka, Agata;
Handzlik, Jadwiga;
Godyń, Justyna;
Knez, Damijan;
Gobec, Stanislav;
Więckowska, Anna;
Hansen, Finn K.;
Marco-Contelles, José:
Contilistat, a New Multitarget Small Polyfunctionalized Indole Derivative
Ateşoğlu, Şeyma;
Çakır, Furkan;
Şenol, Ayşe Merve;
Tokalı, Pelin;
Şenol, Halil;
Tokalı, Feyzi Sinan;
Akbaş, Fahri;
Kalay, Erbay:
Synthesis, Characterization and In Vitro and In Silico Biological Evaluation of New Mannich-Based Rhodanine and Thiazolidine-2,4-dione Derivatives as Potential Anti-Lung-Cancer Agents
Hamdy, Ahmed K.;
Araki, Hiroshi;
Tateishi, Hiroshi;
Toma, Tsugumasa;
Radwan, Mohamed O.;
Biswas, Shashwata;
Kuwata, Takeo;
Matsushita, Shuzo;
Fujita, Mikako;
Niwa, Shin-ichiro;
Otsuka, Masami:
Synthesis of a 5,6-Dihydropyran-2-one Derivative with Dual Anti-Cell-Migration and Anticancer Activity