Synthesis 2021; 53(02): 383-390
DOI: 10.1055/s-0040-1707356
paper
© Georg Thieme Verlag Stuttgart · New York

Palladium-Catalyzed Cross-Coupling Reactions of 4-Tosyl­oxyquinazolines with Indoles: An Efficient Approach to 4-(1H-Indol-1-yl)quinazolines

Xinglin Ye
a   Department of Chemistry and Environmental Engineering, Jiujiang University, Jiujiang, Jiangxi 330025, P. R. of China
b   Key Laboratory of Small Functional Organic Molecule, Ministry of Education and Key Laboratory of Green Chemistry, Jiangxi Province, Jiangxi Normal University, Nanchang, Jiangxi 330022, P. R. of China   Email: yypeng@jxnu.edu.cn   Email: yiyuanpeng@yahoo.com
,
Jian Huang
b   Key Laboratory of Small Functional Organic Molecule, Ministry of Education and Key Laboratory of Green Chemistry, Jiangxi Province, Jiangxi Normal University, Nanchang, Jiangxi 330022, P. R. of China   Email: yypeng@jxnu.edu.cn   Email: yiyuanpeng@yahoo.com
,
Zhihong Deng
b   Key Laboratory of Small Functional Organic Molecule, Ministry of Education and Key Laboratory of Green Chemistry, Jiangxi Province, Jiangxi Normal University, Nanchang, Jiangxi 330022, P. R. of China   Email: yypeng@jxnu.edu.cn   Email: yiyuanpeng@yahoo.com
,
Jianjun Yuan
b   Key Laboratory of Small Functional Organic Molecule, Ministry of Education and Key Laboratory of Green Chemistry, Jiangxi Province, Jiangxi Normal University, Nanchang, Jiangxi 330022, P. R. of China   Email: yypeng@jxnu.edu.cn   Email: yiyuanpeng@yahoo.com
,
Yiyuan Peng
b   Key Laboratory of Small Functional Organic Molecule, Ministry of Education and Key Laboratory of Green Chemistry, Jiangxi Province, Jiangxi Normal University, Nanchang, Jiangxi 330022, P. R. of China   Email: yypeng@jxnu.edu.cn   Email: yiyuanpeng@yahoo.com
› Author Affiliations
Financial support from National Natural Science Foundation of China (no. 21362014 and 21762020), Jiangxi Provincial Department of Science and Technology (no. 20171BAB203006), and Key Laboratory of Functional Small Organic Molecule, Ministry of Education, Jiangxi Normal University (no. KLFS-KF-201408) is gratefully acknowledged.
Further Information

Publication History

Received: 14 June 2020

Accepted after revision: 27 July 2020

Publication Date:
25 August 2020 (online)


Abstract

In this paper, exploration of our continuous interests on late-stage derivation of quinozaline core is described. A wide array of 4-(1H-indol-1-yl)quinazolines were obtained in good to excellent yields through palladium-catalyzed cross-coupling of 4-tosyloxyquinazolines with indole derivatives under mild reaction conditions.

Supporting Information

 
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