DOI: 10.1055/s-00000083

Synlett

eFirst

Publication Date: 11 December 2025

Letter > Published as part of the Special Topic Alkynes in Organic Synthesis

  • Prabhakaran, Mohan; Parthasarathy, Kanniyappan:

    Palladium-Catalyzed C−H/N−H Annulations of (E,Z)-3-Arylidene Indolin-2-ones with Alkynes: A Synthesis of Benzazepine Derivatives

    Image for article: Palladium-Catalyzed C−H/N−H Annulations of (<i>E,Z</i>)-3-Arylidene Indolin-2-ones with Alkynes: A Synthesis of Benzazepine Derivatives
    Supplementary Material (PDF)

    • Publication Date: 10 December 2025

    Letter

  • Jiang, Chunfeng; Wang, Xianrui; An, Changwei; Jiang, Jiaqi; Su, Tongjia; Liu, Meiwei; Xu, Xiaobo; Zeng, Qinglin:

    Synthesis and Activity Evaluation of Gemcitabine Prodrugs with 4-(Boronic acid) benzoylamide Structure

    Image for article: Synthesis and Activity Evaluation of Gemcitabine Prodrugs with 4-(Boronic acid) benzoylamide Structure
    Supplementary Material (PDF)

    • Publication Date: 09 December 2025

    Letter

  • Schroder, Chelsea M.; Kulawik, Isabella M.; Leadbeater, Nicholas:

    Aminoxyl-mediated Electrocatalytic C–N Coupling of Azoles with Cycloheptatriene

    Image for article: Aminoxyl-mediated Electrocatalytic C–N Coupling of Azoles with Cycloheptatriene
    Supplementary Material (PDF)

    • Letter

  • Sharma, Supriya; Chauhan, Amar Nath Singh; Gajare, Swaranjali D.; Kumar, Akhilesh; Erande, Rohan D.:

    Chemoselective Reduction of Conjugated Indole-maleimides and Oxindole-esters via Zn/TiCl₄-Assisted Unified Approach

    Image for article: Chemoselective Reduction of Conjugated Indole-maleimides and Oxindole-esters via Zn/TiCl₄-Assisted Unified Approach
    Supplementary Material (PDF)

    • Publication Date: 08 December 2025

    Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Harikrishna, A. S.; Kesavan, Venkitasamy:

    Identification of Natural Product Inhibitors against Human Nicotinamide N-Methyltransferase (hNNMT): An In Silico and invitro Approach

    Image for article: Identification of Natural Product Inhibitors against Human Nicotinamide <i>N</i>-Methyltransferase (hNNMT): An <i>In Silico</i> and <i>in</i><i>vitro</i> Approach
    Supplementary Material (PDF) Supplementary Material (PDF)

    • Publication Date: 05 December 2025

    Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Gharpure, Santosh J.; Bhujbal, Sandesh Balu; Somani, Shipra:

    HFIP-Promoted Intramolecular Oximation of O-Propargyl Hydroxylamines for the Synthesis of 2-Isoxazolines

    Image for article: HFIP-Promoted Intramolecular Oximation of <i>O</i>-Propargyl Hydroxylamines for the Synthesis of 2-Isoxazolines
    Supplementary Material (PDF)

    • Publication Date: 04 December 2025

    Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Kumar, Vipin; Yadav, Anup Kumar; Singh, Saurabh; Singh, Maya Shankar:

    Transition-Metal Free Chemoselective C(sp3)–S Cross-Coupling/Cyclization Cascade: Reagent-Controlled Divergent Synthesis of Methylene-functionalized Thiazolidines and 1,3-Thiazinanes

    Image for article: Transition-Metal Free Chemoselective C(sp<sup>3</sup>)–S Cross-Coupling/Cyclization Cascade: Reagent-Controlled Divergent Synthesis of Methylene-functionalized Thiazolidines and 1,3-Thiazinanes
    Supplementary Material (PDF)

    • Publication Date: 02 December 2025

    Correction

  • Xie, Ying; Li, Haiping; Hu, Xin; Lai, Yinlong:

    Correction: N-Heterocyclic Carbene-Catalyzed Acylalkylation of Indole via C–C Bond Cleavage/Dearomatization to Access the Multisubstituted Benzopyrrolizidinones

    • Letter

  • Wang, Qingxu; Zhao, Jianyou; Fang, Pengkai; Shen, Xiaoqian; Meng, Jingyu; Zhang, Lanlan; Han, Hongliang; Huang, Xianting; Zhang, Jiatai; Liu, Zhehuai; Wang, Fan; Liu, Zhong-Quan:

    Comparing the Effects of Solvents on Organic Thermochemical Reactions

    Image for article: Comparing the Effects of Solvents on Organic Thermochemical Reactions

    • Publication Date: 01 December 2025

    Account > Alkynes in Organic Synthesis

  • Choudhary, Shivani; Ghosh, Nayan:

    Ynamides as Linear Building Blocks for Aromatic N-Heterocycles in Metal-Catalyzed Transformations

    Image for article: Ynamides as Linear Building Blocks for Aromatic <i>N</i>-Heterocycles in Metal-Catalyzed Transformations

    • Letter > Alkynes In Organic Synthesis

  • Hazarika, Nitumoni; Gogoi, Nitish Nayan; Gogoi, Manashjyoti; Ghosh, Nayan; Das, Animesh:

    One-Pot Synthesis of 1-Alkoxyisoquinoline Derivatives via Ru(II)-Catalyzed Aryl C−H Activation and Alkyne Annulation

    Image for article: One-Pot Synthesis of 1-Alkoxyisoquinoline Derivatives via Ru(II)-Catalyzed Aryl C−H Activation and Alkyne Annulation
    Supplementary Material (PDF)

    • Publication Date: 28 November 2025

    Letter

  • Yavari, Issa; Akbarzadeh, Somayeh; Ghorbanzadeh, Meysam:

    A Synthesis of Functionalized Benzimidazoles via the Three-Component Reaction of Terminal Alkynes, Phenylsulfonyl Azide, and Phenylenediamine-1,3-dicarbonyl Adducts

    Image for article: A Synthesis of Functionalized Benzimidazoles via the Three-Component Reaction of Terminal Alkynes, Phenylsulfonyl Azide, and Phenylenediamine-1,3-dicarbonyl Adducts
    Supplementary Material (PDF) Supplementary Material (PDF)

    • Publication Date: 27 November 2025

    Account > Published as part of the Special Topic Alkynes in Organic Synthesis

  • Maddaluno, Jacques; Fressigné, Catherine; Durandetti, Muriel:

    Intramolecular Carbolithiation of Alkynes: Observation, Mechanism, Applications

    Image for article: Intramolecular Carbolithiation of Alkynes: Observation, Mechanism, Applications

    • Letter > Published as part of the Special Topic Alkynes in Organic Synthesis

  • Bozzi, Ícaro A. O.; Borges, Dandara S.; Dival, Bruno; Oliveira, Willian X. C.; Machado, Luana A.; Almeida, Renata G.; Araujo, Maria H.; Gravel, Edmond; da Silva Júnior, Eufrânio N.; Jardim, Guilherme A. M.:

    Light-Induced, Iron-Promoted Formation of Benzotetraphenones via Paternò–Büchi Photorearrangement/Electrocyclization: A Route to Polyaromatic Scaffolds

    Image for article: Light-Induced, Iron-Promoted Formation of Benzotetraphenones <i>via</i> Paternò–Büchi Photorearrangement/Electrocyclization: A Route to Polyaromatic Scaffolds
    Supplementary Material (PDF)

    • Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Dhanalakshmi, Murugan; Anbarasan, Pazhamalai:

    Catalytic Cyanation of Aryl Halides with Electrophilic N–CN Reagent

    Image for article: Catalytic Cyanation of Aryl Halides with Electrophilic N–CN Reagent
    Supplementary Material (PDF)

    • Letter > Published as part of the Special Issue Dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Khobragade, Virendra R.; AR, Archana; Ramana, Chepuri Venkata:

    Asymmetric Total Synthesis of Streptoglycerides A and B

    Image for article: Asymmetric Total Synthesis of Streptoglycerides A and B
    Supplementary Material (PDF)

    • Letter

  • Kishore Kumar Reddy, Ramireddy; Raju, Mogalagani; Penke, Vijaya Babu; Kotanka, Ramakrishna Reddy; Gandolla, Chinna Reddy:

    Amberlyst-Promoted Eco-Friendly Route to 4-Arylpyrrolo [1,2-a]Quinoxalines

    Image for article: Amberlyst-Promoted Eco-Friendly Route to 4-Arylpyrrolo [1,2-a]Quinoxalines
    Supplementary Material (PDF)

    • Letter

  • Lu, Wenjie; Murai, Takuya; Kyan, Ryuji; Kobayashi, Yusuke; Kawabata, Takeo; Furuta, Takumi:

    Asymmetric intramolecular C–H insertion of N-tosyl diazoimine intermediate from triazole derivative by axially chiral dirhodium(II) carboxylate complex

    Image for article: Asymmetric intramolecular C–H insertion of <i>N</i>-tosyl diazoimine intermediate from triazole derivative by axially chiral dirhodium(II) carboxylate complex
    Supplementary Material (PDF)

    • Letter

  • Pandavadara, Atul R.; Khanvilkar, Aditya N.; Bedekar, Ashutosh V.; Butcher, Raymond; Abraham, Alex:

    Applications of Optically Pure Biphenyloxycyclohexanols in Deracemization of α-Substituted Aryloxypropanoic Acids by Dynamic Kinetic Resolution

    Image for article: Applications of Optically Pure Biphenyloxycyclohexanols in Deracemization of α-Substituted Aryloxypropanoic Acids by Dynamic Kinetic Resolution

    • Publication Date: 26 November 2025

    Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Koner, Mainak; Khan, Shabbir Ahmed; Baidya, Mahiuddin:

    Weak Coordination-Assisted Cobalt(III)-Catalyzed Regioselective Alkenylation of Indolines with Allenes

    Image for article: Weak Coordination-Assisted Cobalt(III)-Catalyzed Regioselective Alkenylation of Indolines with Allenes
    Supplementary Material (PDF)
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