DOI: 10.1055/s-00000083

Synlett

eFirst

Publication Date: 03 November 2025

Synpacts

  • Hartley, Will; Kasten, Kevin; Smith, Andrew D.:

    Enantiocontrol in Radical Coupling Reactions: A Catalytic [1,2]-Rearrangement of Allylic Ammonium Ylides

    Image for article: Enantiocontrol in Radical Coupling Reactions: A Catalytic [1,2]-Rearrangement of Allylic Ammonium Ylides
    Open Access

    • Publication Date: 31 October 2025

    Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Jadhav, Pramod M.; Jamdade, Akash Bandu; Gnanaprakasam, Boopathy:

    Ru-Catalyzed Domino C-4 Alkylation and Hydroxylation of Pyrazolones Using Alcohols via Borrowing-Hydrogen Catalysis

    Image for article: Ru-Catalyzed Domino C-4 Alkylation and Hydroxylation of Pyrazolones Using Alcohols via Borrowing-Hydrogen Catalysis
    Supplementary Material (PDF)

    • Letter

  • Takahashi, Toshifumi; Tonbe, Rihoko; Hiramatsu, Daishi; Kurahashi, Takuya:

    Nickel-Catalyzed Enantioconvergent Cycloadditions of Aziridines and Imines

    Image for article: Nickel-Catalyzed Enantioconvergent Cycloadditions of Aziridines and Imines
    Supplementary Material (PDF)

    • Publication Date: 30 October 2025

    Account > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Dam, Binoyargha; Das, Bubul; Patel, Bhisma K.:

    Deciphering the Reactivity of Quinoxaline

    Image for article: Deciphering the Reactivity of Quinoxaline

    • Publication Date: 29 October 2025

    Letter

  • Bouda, Maria; Xhili, Dea; Hana, Grace E.; Sripada, Archita; Bertke, Jeffery A.; Wolf, Christian:

    Environmentally Benign Atroposelective Synthesis of Fluorinated Oxindole–Coumarin Hybrid Structures

    Image for article: Environmentally Benign Atroposelective Synthesis of Fluorinated Oxindole–Coumarin Hybrid Structures
    Supplementary Material (PDF)

    • Synpacts

  • Wang, Zi-Chao; Wang, Peng; Shi, Shi-Liang:

    Ni-Catalyzed Addition of Arylborons to Alkenes for the Synthesis of Quaternary Carbon Centers

    Image for article: Ni-Catalyzed Addition of Arylborons to Alkenes for the Synthesis of Quaternary Carbon Centers

    • Publication Date: 28 October 2025

    Account > Alkynes in Organic Synthesis

  • Acharya, Swadhin Swaraj; Rout, Padma Ranjan; Parida, Bibhuti Bhusan:

    The Application of Alkynes as 1,2-Dicarbonyl Substitutes in Organic Synthesis Through Iodination and Kornblum Oxidation

    Image for article: The Application of Alkynes as 1,2-Dicarbonyl Substitutes in Organic Synthesis Through Iodination and Kornblum Oxidation

    • Account > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Kotha, Sambasivarao; Solanke, Balaji U.:

    Diversity-Oriented Approach to Furan Building Blocks and Their Relevance in Organic Synthesis, Materials Science, and Medicinal Chemistry

    Image for article: Diversity-Oriented Approach to Furan Building Blocks and Their Relevance in Organic Synthesis, Materials Science, and Medicinal Chemistry

    • Synpacts

  • Wanderley, Taciano Antonio Santos; Crisenza, Giacomo Ercole Martino:

    The Electrosynthetic Toolkit for Stereoselective Alkene 1,2-Difunctionalization

    Image for article: The Electrosynthetic Toolkit for Stereoselective Alkene 1,2-Difunctionalization

    • Publication Date: 27 October 2025

    New Tools

  • Bansal, Diksha; Sivaganesan, Pooja; Sivaprasad, Ghanashyam; Ilango, Janani; Das, Mrinal K.; Chaudhuri, Saikat:

    Halogen Bond-Driven Oxa-Pictet–Spengler Cyclization Using CBr₄: A Metal-Free and Regioselective Approach for the Synthesis of Tetracyclic Dihydrochromenoindole Scaffolds

    Image for article: Halogen Bond-Driven Oxa-Pictet–Spengler Cyclization Using CBr₄: A Metal-Free and Regioselective Approach for the Synthesis of Tetracyclic Dihydrochromenoindole Scaffolds
    Supplementary Material (PDF)

    • Publication Date: 24 October 2025

    Account

  • Kumari, Pallvi; Kumari, Anshu; Kumar, Ankush; Bhatia, Rohit:

    Five-Membered Heterocyclic Hybrids as Promising Anticancer Agents: SAR and Biological Activities (2020–2025)

    Image for article: Five-Membered Heterocyclic Hybrids as Promising Anticancer Agents: SAR and Biological Activities (2020–2025)

    • Account > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Mehta, Ronak; Chande, Vatsal Dhiraj; Appayee, Chandrakumar:

    Recent Applications of Aminocatalysis in Reactions of α,β-Unsaturated Aldehydes

    Image for article: Recent Applications of Aminocatalysis in Reactions of α<i>,</i>β-Unsaturated Aldehydes

    • Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Muthuvel, Karthick; Sivaraj, Chandrasekaran; Gandhi, Thirumanavelan:

    Heterobenzylic C(sp3)─H Acylation of Isoindolinones via Photoinduced Intermolecular Hydrogen Atom Transfer Strategy

    Image for article: Heterobenzylic C(sp<sup>3</sup>)─H Acylation of Isoindolinones via Photoinduced Intermolecular Hydrogen Atom Transfer Strategy
    Supplementary Material (PDF)

    • Letter

  • Xu, Ke; Zhou, Min-Jie; Liu, Xinrui; Chen, Guofei; Xie, Yinjun:

    Additive- and Catalyst-free Deoxygenative Reduction of Amides and Imides to Amines with Ammonia Borane

    Image for article: Additive- and Catalyst-free Deoxygenative Reduction of Amides and Imides to Amines with Ammonia Borane
    Supplementary Material (PDF)

    • Letter

  • Yuan, Xinxin; Zeng, Qian-Ding; Yao, Hongmiao; Jin, Wenjun; Ren, Jiangmeng; Zeng, Bu-Bing:

    Rapid Deprotection of O-Allyoxycarbonyl(alloc) Alcohols by NiCl2•6H2O and NaBH4

    Image for article: Rapid Deprotection of <i>O</i>-Allyoxycarbonyl(alloc) Alcohols by NiCl<sub>2</sub>•6H<sub>2</sub>O and NaBH<sub>4</sub>
    Supplementary Material (PDF)

    • Synpacts

  • Liu, Chang; Zhang, Mingyu; Dai, Mingji:

    Total Synthesis of (±)-Phaeocaulisin A Enabled Chemistry Innovation and Biological Discovery

    Image for article: Total Synthesis of (±)-Phaeocaulisin A Enabled Chemistry Innovation and Biological Discovery

    • Publication Date: 22 October 2025

    Letter

  • Chatragadda, Kranthi; Nagarajan, Rajagopal:

    Facile Synthesis of 11H-Indolo[3,2-c]quinolines Through Pictet–Spengler Cyclization and Aromatization by Oxygen

    Image for article: Facile Synthesis of 11<i>H</i>-Indolo[3,2-<i>c</i>]quinolines Through Pictet–Spengler Cyclization and Aromatization by Oxygen
    Supplementary Material (PDF)

    • Publication Date: 21 October 2025

    Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Afreen, Saista; Ghosh, Abhipsa; Kumar Banjare, Shyam; Ravikumar, Ponneri C.:

    Cobalt-Catalyzed C-2 Functionalization of N-Methylindole-1-carboxamide via Regioselective Hydroindolation of 1,6-Diyne

    Image for article: Cobalt-Catalyzed C-2 Functionalization of <i>N-Methylindole-1-carboxamide</i> via Regioselective Hydroindolation of 1,6-Diyne
    Supplementary Material (PDF)

    • Publication Date: 08 October 2025

    Letter > Published as part of the Special Issue dedicated to Prof. S. Chandrasekaran on his 80th birthday

  • Ramisetty, Mohana Krishna; Yadav, Vikas; Venkitasamy, Kesavan; Baskaran, Sundarababu:

    Exploration of Oxetanes and Azetidines in Structure-Based Drug Design

    Image for article: Exploration of Oxetanes and Azetidines in Structure-Based Drug Design
    Supplementary Material (PDF)

    • Publication Date: 07 October 2025

    Letter

  • Drury, Paige A.; Sullivan, Ciara L.; Pottle, Haley L.; Quinn, Kevin J.:

    Total Synthesis of Obolactone via Regioselective Carbonyl Desaturation

    Image for article: Total Synthesis of Obolactone via Regioselective Carbonyl Desaturation
    Supplementary Material (PDF)
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