An Efficient and Safe Method for
the Multigram Synthesis of trans-2-(Trifluoromethyl)cyclopropylamine
Vladimir S. Yarmolchuka,b, Andrii V. Bezdudnya, Nataliya A. Tolmachevaa, Oleg Lukin*c, Alexander N. Boykoc, Alexey Chekotyloc, Andrei A. Tolmacheva,c, Pavel K. Mykhailiuk*a,b a Enamine Ltd., Alexander Matrosov
St. 23, Kiev 01103, Ukraine e-Mail: pavel.mykhailiuk@gmail.com; b Department of Chemistry, Kiev
National Taras Shevchenko University, Volodymyrska
St. 64, Kiev 01033, Ukraine c ChemBioCenter, Kiev
National Taras Shevchenko University, Volodymyrska
St. 62, Kiev 01033, Ukraine Fax: +38(44)2351273; e-Mail: oleg.lukin@univ.kiev.ua;