DOI: 10.1055/s-00000175

Arzneimittelforschung

Issue 02 · Volume 53 · February 2003 DOI: 10.1055/s-002-22658

CNS-active Drugs · Hypnotics · Psychotropics · Sedatives

  • 73
    Jindal, Dharam Paul; Piplani, Poonam; Fajrak, Hassan; Prior, Chris; Marshall, Ian G.:

    Synthesis and Biological Evaluation of 16β-Pyrrolidinosteroidal Derivatives

  • 80
    Washio, Takuo; Kohsaka, Kazuhiro; Arisawa, Hirohiko; Masunaga, Hiroaki; Nagatsuka, Shin-ichiro; Satoh, Yoshiaki:

    Pharmacokinetics and Metabolism of Radiolabelled SNI-2011, a Novel Muscarinic Receptor Agonist, in Healthy Volunteers

  • 87
    Kees, Frieder; Jehkul, Andreas; Bucher, Michael; Mair, Georg; Kiermaier, Josef; Grobecker, Horst:

    Bioavailability of Opipramol from a Film-coated Tablet, a Sugar-coated Tablet and an Aqueous Solution in Healthy Volunteers

    • Antiallergic Drugs · Antiasthmatics · Antitussives · Bronchodilators · Bronchosecretogogues · Mucolytics

  • 93
    Llupià, Josep; Gras, Jordi; Llenas, Jesús:

    Comparative Antiallergic Effects of Second-generation H1-Antihistamines Ebastine, Cetirizine and Loratadine in Preclinical Models

    • Antiemetics · Gastrointestinal Drugs · Urologic Drugs · Uricosuric Drugs

  • 98
    Yoshikawa, Takashi; Mine, Yukiko; Morikage, Kazuo; Yoshida, Naoyuki:

    Pharmacological Profile of AS-9705, a Novel Benzotriazolecarboxamide Derivative, as a Gastroprokinetic Agent with Potent Anti-emetic Activity

    • Antibiotics · Antiviral Drugs · Chemotherapeutics · Cytostatics

  • 107
    Baraldi, Pier Giovanni; Tabrizi, Mojgan Aghazadeh; Pavani, Maria Giovanna; Nuñez, Maria del Carmen; Makaeva, Rimma; Gambari, Roberto; Colla, Paolo La; Romagnoli, Romeo:

    Design, Synthesis and in vitro Cytotoxicity of a cis-Dichloroplatinum (II) Complex Linked to the Minor Groove Binder Stallimycin

  • 114
    Gökhan, Nesrin; Erdoğan, Hakkı; Durlu, N. Tugˇba; Demirdamar, Rümeysa; Özalp, Meral:

    Synthesis and Evaluation of Analgesic, Anti-inflammatory and Antimicrobial Activities of 6-Acyl-3-piperazinomethyl-2-benzoxazolinones

  • 121
    Guzmán, Antonio; García, Concepción; Marŕna, Ana-Paz; Willoughby, Chris; Demestre, Isabel:

    Developmental Toxicity Studies of the Quinolone Antibacterial Agent Irloxacin in Rats and Rabbits

  • 126
    Müller, Rainer; Böttger, Christina; Wichmann, Georg:

    Suitability of Cefotiam and Cefuroxime Axetil for the Perioperative Short-term Prophylaxis in Tonsillectomy Patients

    • Special Themes

  • 133
    Kandemirli, Fatma; Tokay, Nesrin; Shvets, Nataly M.; Dimoglo, Anatoly S.:

    Electronic-Topological Study of the Structure-Activity Relationships in a Series of Steroids with Mineralocorticoid Binding Affinity

    • Information on Patents

  • 139
    Habernickel, Valentin J.:

    The Pharma Market as Reflected by Patents

    • Book Reviews

  • 143

    Book Reviews