Synthesis 2017; 49(12): 2743-2748
DOI: 10.1055/s-0036-1588159
paper
© Georg Thieme Verlag Stuttgart · New York

Coumaryl Triflate, a Versatile Building Block for the Modification of Coumarins and for Fluorescence Labeling

Uli Kazmaier*
a   Universität des Saarlandes, Organische Chemie, 66123 Saarbrücken, Germany   Email: u.kazmaier@mx.uni-saarland.de
,
Tamara Doroshenko
a   Universität des Saarlandes, Organische Chemie, 66123 Saarbrücken, Germany   Email: u.kazmaier@mx.uni-saarland.de
,
Kevin Bauer
a   Universität des Saarlandes, Organische Chemie, 66123 Saarbrücken, Germany   Email: u.kazmaier@mx.uni-saarland.de
,
Isabel Filbrich
a   Universität des Saarlandes, Organische Chemie, 66123 Saarbrücken, Germany   Email: u.kazmaier@mx.uni-saarland.de
,
Andreas Grueter
b   Universität des Saarlandes, Biophysikalische Chemie, 66123 Saarbrücken, Germany
,
Gregor Jung
b   Universität des Saarlandes, Biophysikalische Chemie, 66123 Saarbrücken, Germany
,
Angelika Ullrich
a   Universität des Saarlandes, Organische Chemie, 66123 Saarbrücken, Germany   Email: u.kazmaier@mx.uni-saarland.de
› Author Affiliations
Further Information

Publication History

Received: 11 January 2017

Accepted after revision: 06 March 2017

Publication Date:
23 March 2017 (online)


Abstract

Coumaryl triflate can be used for a wide range of substitution reactions, either under Pd-catalyzed conditions or via direct nucleophilic substitutions, and is therefore an ideal substrate for the fluorescence labeling of functionalized compounds, such as amino acids.

Supporting Information

 
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