Scaling Complexity: A Streamlined Route to the Northern Fragment of Enlicitide

Dirk H. Trauner; Christoph Etling

doi:10.1055/a-2601-4828

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Synfacts 2025; 21(07): 735
DOI: 10.1055/a-2601-4828

Innovative Drug Discovery and Development

Scaling Complexity: A Streamlined Route to the Northern Fragment of Enlicitide

Contributor(s):

Dirk H. Trauner

,

Christoph Etling

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Keywords

enlicitide decanoate - PCSK9 inhibitor - fragment synthesis - process development - one-pot reactions - macrocyclization - chemoselectivity - regioselectivity

Publication History

Article published online:
23 June 2025

Georg Thieme Verlag KG
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