Palladium-Catalyzed Amination of Unprotected Halo-7-azaindoles

J. L. Henderson; S. M. McDermott; S. L. Buchwald

doi:10.1055/s-0030-1259416

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Synfacts 2011(3): 0317-0317
DOI: 10.1055/s-0030-1259416

Metal-Mediated Synthesis

Palladium-Catalyzed Amination of Unprotected Halo-7-azaindoles

Contributor(s): Paul Knochel, Andreas J. Wagner
J. L. Henderson, S. M. McDermott, S. L. Buchwald*
Massachusetts Institute of Technology, Cambridge, USA

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Publication History

Publication Date:
16 February 2011 (online)

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Significance

Efficient procedures for the palladium-catalyzed cross-coupling of primary and secondary amines with halo-7-azaindoles are presented. A wide range of aromatic and aliphatic amines can be used in this reaction.