DOI: 10.1055/s-00000131

Synfacts

Issue 01 · Volume 14 · January 2018 DOI: 10.1055/s-007-35964

Synform

A1
Zanda, Matteo: SYNFORM ISSUE 2018/01

Synthesis of Natural Products and Potential Drugs

z0001
All PDFs of this category
0001
Pilot-Scale Synthesis of TV-45070
0002
Total Synthesis of (+)-Pancratistatins
0003
Synthesis of (–)-Longeracinphyllin A
0004
Cooperative Catalysis in the Synthesis of Chroman-2-ones: NNC 45-0781
0005
Syntheses of Foveoglin A and Perviridisin B
0006
Synthesis of Disorazole A1
0007
Total Synthesis of Resiniferatoxin
0008
Syntheses of (–)-Tetrapetalones A and C
0009
Synthesis of a trans-Cyclopropoxy Building Block for Grazoprevir
0010
Synthesis of GSK3036656

Synthesis of Heterocycles

z0011
All PDFs of this category
0011
Phosphinoboration of Pyridines and Related N-Heteroaromatic Systems
0012
Organocatalytic Synthesis of Cyclopenta[b]benzofurans
0013
Synthesis of Substituted Aziridines by Michael Addition Triggered Cyclization
0014
Synthesis of 2,3-Disubstituted Indoles by C–H Functionalization of Azobenzenes
0015
Synthesis of Fluorinated Oxazolines from Allylamides
0016
Iodine-Mediated Intramolecular C–H Ami-nation Route to 1H-Indazoles and 1H-Pyrazoles
0017
Phosphine-Catalyzed Synthesis of Chiral Spiro[cyclopentene-indole]ones
0018
Synthesis of Fluorocoumarins by a Photoredox Reaction
0019
Synthesis of Pyrrolidinoazepines and Pyrrolidinooxazoles by Cycloaddition
0020
Gold Catalysis in an Asymmetric Synthesis of Tetrahydrofurans
0021
Synthesis of Lactones and Lactams by Nickel-Catalyzed Transfer Hydrogenation
0022
Three Rings in One Shot: Diastereo- and Enantioselective Ring-System Synthesis
0023
Spirocyclic Pyrazoles by Ring Expansion of Cyclic Ketones
0024
Practical Synthesis of Azaheterocycles Con-taining a gem-Difluorocyclopropane Moiety

Synthesis of Materials and Unnatural Products

z0025
All PDFs of this category
0025
Tetraarylmethanes by Cross-Dehydrogenative Coupling
0026
Robust Ruthenium Catalysis to Poly(ortho ester)s
0027
Oxidation in the Direction of Increasing Aromaticity
0028
Efficient Nanographene BN-Doping
0029
Selenophene-Containing [7]Helicenes
0030
Lewis Acid Initiated Polymerization of Benzofurans
0031
[1+1+1+1] Cyclization to Obtain Four-Membered Rings
0032
Diels–Alder Reaction for New Fluorophores
0033
An Old Reaction for New Polymer Chemistry
0034
Easy Access to Zn2+-Responsive Fluorophores
0035
Fusing Furans with Thiophenes
0036
Caged Radicals

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0037
All PDFs of this category
0037
Gold(I)-Catalyzed Stereoselective Synthesis of Deoxyglycosides
0038
Asymmetric Palladium-Catalyzed Cascade Synthesis of Polycyclic Indoles
0039
Enantioselective Iridium-Catalyzed Cycloisomerization of N-Methylanilines
0040
Palladium/Amine-Cooperative Allylation
0041
Iridium-Catalyzed C–H Oxidative Reaction
0042
Palladium-Catalyzed Enantioselective Allylic Alkylation of Thiopyranones
0043
Enantioenriched Quaternary γ-Amino Acids through Copper-Catalyzed Amination
0044
Asymmetric Hydrogenation of Vinylsilanes by Iridium Catalysis
0045
Palladium(0)-Catalyzed Allylic Alkylation of Difficult Substrates
0046
Asymmetric Synthesis of Biaryldiols
0047
Copper-Catalyzed Borylallylation
0048
Synthesis of Cyclobutenes via a Palladium-Catalyzed Asymmetric Heck Reaction
0049
Palladium-Catalyzed Asymmetric Allylic Alkylations of N-Allyl Imines
0050
Copper-Catalyzed Cyclopropanation with Diazomalonates
0051
Iridium-Catalyzed Hydrogenation of α-Keto Amides
0052
Asymmetric Synthesis of Tetrahydroquinoline-Based Spirooxindoles
0053
Enantioselective Synthesis of γ-Lactams by [3+2] Cycloaddition
0054
Cobalt-Catalyzed Hydroboration/Hydrogenation Sequence
0055
Selective Synthesis of (Z)- and (E)-Mono-fluoroalkenes
0056
Anti-Markovnikov Hydroboration of Unactivated 1,1-Disubstituted Olefins
0057
Rhodium-Catalyzed Enantioselective Synthesis of Heterocycles
0058
Rhodium-Catalyzed Asymmetric Alkenylation of Aliphatic Imines
0059
Enantioselective Iridium-Catalyzed Allylic Dearomatization
0060
Rhodium-Catalyzed Asymmetric Allylation of Pyrimidines
0061
Synthesis of Crinine-Type Alkaloids by Asymmetric Hydrogenation
0062
Cobalt-Catalyzed Regioselective Hydroboration
0063
Manganese-Catalyzed Asymmetric Addition of β-Dicarbonyl Compounds
0064
Nickel-Catalyzed Enantioselective Synthesis of β-Amino Acids
0065
Cobalt-Catalyzed Interrupted Povarov Reaction
0066
Gold-Catalyzed Enantioselective [2+2] Cyclo-addition of Terminal Alkynes and Alkenes

Metal-Mediated Synthesis

z0067
All PDFs of this category
0067
Chromium-Promoted Synthesis of Borylcyclopropanes
0068
Cobalt-Catalyzed Cross-Coupling of α-Bromo Amides
0069
Palladium-Catalyzed Cross-Coupling of (Hetero)Arenes with Low E-Factor
0070
Palladium-Catalyzed Diastereoselective Synthesis of Homoallylic Alcohols
0071
Trifluoromethylfluorosulfonylation of Unactivated Alkenes
0072
Diastereoselective [3+2] Annulation
0073
Rhodium-Catalyzed Asymmetric 1,4-Additions
0074
Cobalt-Catalyzed Addition of Allylarenes to Ketones
0075
Selective Carbonylation of β-Methylene C–H Bonds
0076
Copper-Mediated Formation of Allyl- and Homoallylboranes
0077
Photoredox Activation of Boronic Acids and Esters
0078
Synthesis of Biphenylenes
0079
Nickel/Photoredox-Catalyzed Amidation
0080
Synthesis of a Hemithioindigo-Motor
0081
Iridium-Catalyzed ortho-Selective Borylation

Organo- and Biocatalysis

z0083
All PDFs of this category
0083
Enzymatic Anti-Markovnikov Oxidations of Styrenes
0084
Kinetic Resolution of anti-1,3-Diols by Horeau Amplification
0085
Organic Photoredox-Catalytic Arene C–H Amination with Primary Amines
0086
Photoredox-Catalytic Nucleophilic Aromatic Substitution of Alkoxyarenes
0087
Corrigendum: Cyclobutadienes via an Organocascade
0088
Organocatalytic Asymmetric Reduction of N-Alkyl Aryl Imino Esters
0089
Phosphine-Catalyzed [4+4] Annulation to Construct Eight-Membered Rings
0090
Tetraarylphosphonium Salt-Catalyzed Synthesis of Oxazolidinones
0091
Enzymatic Olefin Cyclopropanation under Aerobic Conditions
0092
Lactate-Based Ionic Liquid Catalyzed Reductive Amination–Cyclization
0093
Oxidative Asymmetric [2+3] Annulation of Aldehydes with Azomethine Imines
0094
Catalytic Asymmetric Synthesis of Isoindolinones

Polymer-Supported Synthesis

z0095
All PDFs of this category
0095
Pd-Catalyzed Cross-Coupling Mediated by Polymer-Supported Siloxanes
0096
Deoxygenative Amination of Phenols on Palladium/Carbon
0097
Phosphorylated Polyacrylonitrile Fiber Catalyzed Acetalization of Aldehydes
0098
Reusable Magnetic Palladium Catalyst for the Suzuki–Miyaura Reaction
0099
Ruthenium-Catalyzed Carbon–Carbon Cleavage of Carbonyl Compounds
0100
Synthesis of N-Alkyl-2-Pyrrolidones by Using a Palladium Catalyst
0101
Platinum-Catalyzed Diels–Alder Photocycloaddition of Indoles
0102
Transfer Hydrogenolysis of β-O-4 Linkages in Lignin on Pd–Ni Nanoparticles
0103
Heterogeneous Nickel Catalysts for Reductive Amination of Levulinic Acid
0104
Synthesis of (Non)symmetrical Ureas Catalyzed by Sulfated Polyborate
0105
Controlled Hydrogenation of Alkynes on a TiO2/Pt/TiO2 Sandwich Catalyst
0106
Hydrogenation of Carboxylic Acid Derivatives and N-Alkylation of Amines
0107
Titanium-Catalyzed Hydroboration of Aldehydes and Ketones
0108
Oxidative Coupling of 2-Naphthols on Graphene Oxide
0109
Heterogeneous Gold(I) Catalysts for the Functionalization of Alkynes
0110
Palladium Nanoparticles Catalyzed Aerobic Oxidation of Benzylic Alcohols