DOI: 10.1055/s-00000131

Synfacts

References

Garcia-Losada P. * Frederick M. * et al. Centro de Investigación Lilly S.A., Alcobendas-Madrid, Spain and Lilly Research Laboratories, Windlesham, UK
Synthesis, Optimization, and Large-Scale Preparation of Low-Dose CNS-Penetrant BACE Inhibitor LY3202626 via a [3 + 2] Nitrone Cycloaddition.

Org. Process Res. Dev. 2020;
23: 306-314

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