A Mild and Efficient Method for the Syntheses and Regioselective Ring-Opening of Aziridines
Received: 02 March 2017
Accepted after revision: 09 April 2017
25 April 2017 (online)
We have developed a new synthetic method for the synthesis of aziridines using Chloramine-T as an effective reagent in the presence of NH2OH·HCl and NaIO4. We found that the same combination of NH2OH·HCl and NaIO4 is also very effective for nucleophilic ring opening of aziridines.