SynOpen

Issue 01 · March 2017

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0173
Musolino, M.; Dall’Angelo, S.; Zanda, M.:
Synthesis and Radiosynthesis of Prospective 2-Nitroimidazole Hypoxia PET Tracers via Thiazolidine Ligation with 5-Fluorodeoxyribose (FDR)
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0166
Maheshwar Reddy, A.; Sabitha, Gowravaram:
Synthesis of the C1–C9, C11–C19 Pyran Core and C19–C24 Fragments of Macrolactin 3
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0156
Barcia, Jose C.; Cruces, Jacobo; Salas, Cristian O.; Estévez, Juan C.; Cuellar, Mauricio A.; Tapia, Ricardo A.; Estévez, Ramón J.:
A New Approach to the Synthesis of Benzo[b]naphtho[2,3-b]furan-6,11-diones and 2-Benzyl-3-hydroxynaphthalene-1,4-diones
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0147
Yang, Yi-Qiu; Ke, Long-Zhi; Wang, Gui-Fei; Song, Shu-Yong; Qiu, Ming-Ning; Liu, Jian-Jun; Huang, Yun-Sheng:
Synthesis of N-Pyridin-2-ylmethyl and N-Quinolin-2-ylmethyl Substituted Ethane-1,2-diamines
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letter
0143
Ghanbari, N.; Ghafuri, H.; Zand, H. R. Esmaili; Eslami, M.:
Ball-Milling Promoted Monobromination Reactions: One-pot Regioselective Synthesis of Aryl Bromides and α-Bromoketones by NBS and Recyclable MCM-41-SO₃H at Room Temperature
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0138
Halimehjani, Azim Ziyaei; Nosood, Yazdanbakhsh Lotfi; Didaran, Shaghayegh; Aryanasab, Fezzeh:
Metal-Free Oxidative Dimerization of Dithiocarbamates: Direct Access to 3,5-Bis-mercapto-1,2,4-thiadiazoles
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paper
0129
Zhao, Lingyu; Shen, Guodong; Zhang, Tongxin; Wang, Zhen; Liang, Yuhua:
Pd/C-Catalyzed Intramolecular C–H Arylation for the Synthesis of Phenanthridinones and Dibenzo-α-pyrones
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0125
Majeed, Anju; Nagabhushanam, Kalyanam; Majeed, Muhammed; Thomas, Samuel Manoharan; Thajuddin, Nooruddin:
An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues
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letter
0121
Burmistrov, Vladimir; Pitushkin, Dmitry; Butov, Gennady:
New Facile Synthesis of Adamantyl Isothiocyanates
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0117
Bhaumik, Ishani; Misra, Anup Kumar:
Rapid Transformation of Alkyl Halides into Symmetrical Disulfides Using Sodium Sulfide and Carbon Disulfide
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paper
0103
Don Lawson, Chioma; Maza-Iglesias, Max; Sirhan, Muthana M.; Al Dulayymi, Jumaa R.; Baird, Mark S.:
The Synthesis of Single Enantiomers of α-Mycolic Acids of Mycobacterium tuberculosis and Related Organisms, with Alternative Cyclopropane Stereochemistries
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letter
0097
Boekell, Nicholas G.; Cerone, Dana J.; Boucher, Maria M.; Quach, Phong K.; Tentchou Nganyak, Wilfried B.; Reavis, Christine G.; Okoh, Ifeanyi I.; Reid, Jordan O. A.; Berg, Hayley E.; Chang, Briana A.; Brindle, Cheyenne S.:
Triarylmethyl Cation Catalysis: A Tunable Lewis Acid Organocatalyst for the Synthesis of Bisindolylmethanes
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paper
0091
Cívicos, José F.; Costa, Paulo R. R.; Domingos, Jorge L. O.:
Palladium-Catalyzed α-Arylation of Dimethyl Malonate and Ethyl Cyanoacetate with o-Alkoxybromobenzenes for the Synthesis of Phenylacetic Acid, Esters and Phenylacetonitriles
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0084
Nosik, Pavel S.; Artamonov, Oleksiy S.; Ryabukhin, Sergey V.; Grygorenko, Oleksandr O.:
An Approach to 1,1-Disubstituted Pyrazolylcyclopropane Building Blocks
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0076
Li, Jihui; Yu, Weiguang; Hou, Yifeng; Fu, Wenxing; Xu, Shuying; Zhang, Yucang:
An Efficient Protocol for the Synthesis of O-Fluoroalkylisoureas through Copper-Catalysed, Three-Component Reaction of Cyanamides, Fluoroalcohols and Diaryliodonium Triflates
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0068
Ge, Haihong; Liu, Shuang; Cai, Yan; Gao, Zenghui; Du, Siyi; Miao, Zhiwei; Xie, Guixian:
Diastereoselective [Cu(MeCN)₄BF₄/BF₃·Et₂O]-Catalyzed Cyclopropenation of Alkynes: Asymmetric Synthesis of β-Amino-α-cyclopropenyl Phosphonates
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letter
0063
Nallamala, Sirisha; Mannem, Srikumar; Raghavachary, Raghunathan:
Highly Efficient Construction of Sugar-Fused Spirochromanono Pyrrolidines/Pyrrolizidines/Thiolizidines via 1,3-Dipolar Cycloaddition of Azomethine Ylides
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0059
Otomo, Ikumi; Watanabe, Kanna; Kuroda, Chiaki; Kobayashi, Kenichi:
Chain Length of Amphipathic-Type Thioesters Dramatically Affects Reactivity in Aqueous Amidation Reactions with Cysteine Esters
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paper
0050
Panda, Siva S.; Asiri, Abdullah M.; Elagawany, Mohamed; Buchanan, Devan D.; Torkian, Behrad; Bathala, Keerthana; Thomas, Sean J.; Capito, Jason E.; Arshad, Muhammad N.; Al-Romaizan, Abeer N.:
Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates
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letter
0045
Kalita, Subarna Jyoti; Das, Bidyut; Deka, Dibakar Chandra:
l-Proline-Catalysed One-Pot Regio- and Diastereoselective Synthesis of Spiro[pyrido[2,3-d]pyrimidin-2-amine-6,5′-pyrimidines] in Water
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0041
Helgeland, Ida T. Urdal; Sydnes, Magne O.:
A Concise Synthesis of Isocryptolepine by C–C Cross-Coupling Followed by a Tandem C–H Activation and C–N Bond Formation
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paper
0029
Diez-Martinez, Alba; Krishnamurthy, Ramanarayanan:
Investigations towards the Synthesis of 5-Amino-l-lyxofuranosides and 4-Amino-lyxopyranosides and NMR Analysis
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letter
0024
Rodríguez-Aguilar, José; Ordóñez, Beatriz; Vidal, Matías; Rezende, Marcos Caroli; Domínguez, Moisés:
Microwave-Promoted Synthesis of 4-Arylpyrimidines by Pd-Catalysed Suzuki–Miyaura Coupling of 4-Pyrimidyl Tosylates in Water
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paper
0015
Ghosal, Nirnita Chakraborty; Mahato, Sachinta; Chatterjee, Rana; Santra, Sougata; Zyryanov, Grigory V.; Majee, Adinath:
A Mild and Efficient Method for the Syntheses and Regioselective Ring-Opening of Aziridines
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letter
0011
Arakawa, Yukihiro; Kohda, Takahiro; Minagawa, Keiji; Imada, Yasushi:
Brønsted Acid Catalysed Aerobic Reduction of Olefins by Diimide Generated In Situ from Hydrazine
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0008
Sharma, N.; Kumari, P.; Sharma, P.; Bhagat, N.; Bhagat, S.:
Ultrasound-Accelerated Amide Coupling Reactions Directed toward the Synthesis of 1-Acetyl-3-carboxamide-β-carboline Derivatives of Biological Importance
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0001
Zeng, Meng-Tian; Xu, Wan; Liu, Min; Liu, Xing; Chang, Cai-Zhu; Zhu, Hui; Dong, Zhi-Bing:
Iodobenzene-Promoted Pd-Catalysed ortho-Directed C–H Activation: The Synthesis of Benzothiazoles via Intramolecular Coupling
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Erratum
e1
Zeng, Meng-Tian; Xu, Wan; Liu, Min; Liu, Xing; Chang, Cai-Zhu; Zhu, Hui; Dong, Zhi-Bing:
Iodobenzene-Promoted Pd-Catalysed ortho-Directed C–H Activation: The Synthesis of Benzothiazoles via Intramolecular Coupling
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e2
Majeed, Anju; Nagabhushanam, Kalyanam; Majeed, Muhammed; Thomas, Samuel Manoharan; Thajuddin, Nooruddin:
An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues
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SynOpen

Synthesis and Radiosynthesis of Prospective 2-Nitroimidazole Hypoxia PET Tracers via Thiazolidine Ligation with 5-Fluorodeoxyribose (FDR)

Synthesis of the C1–C9, C11–C19 Pyran Core and C19–C24 Fragments of Macrolactin 3

A New Approach to the Synthesis of Benzo[b]naphtho[2,3-b]furan-6,11-diones and 2-Benzyl-3-hydroxynaphthalene-1,4-diones

Synthesis of N-Pyridin-2-ylmethyl and N-Quinolin-2-ylmethyl Substituted Ethane-1,2-diamines

Ball-Milling Promoted Monobromination Reactions: One-pot Regioselective Synthesis of Aryl Bromides and α-Bromoketones by NBS and Recyclable MCM-41-SO₃H at Room Temperature

Metal-Free Oxidative Dimerization of Dithiocarbamates: Direct Access to 3,5-Bis-mercapto-1,2,4-thiadiazoles

Pd/C-Catalyzed Intramolecular C–H Arylation for the Synthesis of Phenanthridinones and Dibenzo-α-pyrones

An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues

New Facile Synthesis of Adamantyl Isothiocyanates

Rapid Transformation of Alkyl Halides into Symmetrical Disulfides Using Sodium Sulfide and Carbon Disulfide

The Synthesis of Single Enantiomers of α-Mycolic Acids of Mycobacterium tuberculosis and Related Organisms, with Alternative Cyclopropane Stereochemistries

Triarylmethyl Cation Catalysis: A Tunable Lewis Acid Organocatalyst for the Synthesis of Bisindolylmethanes

Palladium-Catalyzed α-Arylation of Dimethyl Malonate and Ethyl Cyanoacetate with o-Alkoxybromobenzenes for the Synthesis of Phenylacetic Acid, Esters and Phenylacetonitriles

An Approach to 1,1-Disubstituted Pyrazolylcyclopropane Building Blocks

An Efficient Protocol for the Synthesis of O-Fluoroalkylisoureas through Copper-Catalysed, Three-Component Reaction of Cyanamides, Fluoroalcohols and Diaryliodonium Triflates

Diastereoselective [Cu(MeCN)₄BF₄/BF₃·Et₂O]-Catalyzed Cyclopropenation of Alkynes: Asymmetric Synthesis of β-Amino-α-cyclopropenyl Phosphonates

Highly Efficient Construction of Sugar-Fused Spirochromanono Pyrrolidines/Pyrrolizidines/Thiolizidines via 1,3-Dipolar Cycloaddition of Azomethine Ylides

Chain Length of Amphipathic-Type Thioesters Dramatically Affects Reactivity in Aqueous Amidation Reactions with Cysteine Esters

Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates

l-Proline-Catalysed One-Pot Regio- and Diastereoselective Synthesis of Spiro[pyrido[2,3-d]pyrimidin-2-amine-6,5′-pyrimidines] in Water

A Concise Synthesis of Isocryptolepine by C–C Cross-Coupling Followed by a Tandem C–H Activation and C–N Bond Formation

Investigations towards the Synthesis of 5-Amino-l-lyxofuranosides and 4-Amino-lyxopyranosides and NMR Analysis

Microwave-Promoted Synthesis of 4-Arylpyrimidines by Pd-Catalysed Suzuki–Miyaura Coupling of 4-Pyrimidyl Tosylates in Water

A Mild and Efficient Method for the Syntheses and Regioselective Ring-Opening of Aziridines

Brønsted Acid Catalysed Aerobic Reduction of Olefins by Diimide Generated In Situ from Hydrazine

Ultrasound-Accelerated Amide Coupling Reactions Directed toward the Synthesis of 1-Acetyl-3-carboxamide-β-carboline Derivatives of Biological Importance

Iodobenzene-Promoted Pd-Catalysed ortho-Directed C–H Activation: The Synthesis of Benzothiazoles via Intramolecular Coupling

Iodobenzene-Promoted Pd-Catalysed ortho-Directed C–H Activation: The Synthesis of Benzothiazoles via Intramolecular Coupling

An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues