SynOpen

Kotha, Sambasivarao; Singh, Deepshikha: Tetraphenylmethane Derivatives Containing Nitrogen Heterocycles

Stampolaki, Marianna; Kolocouris, Antonios: Improved Synthesis of the Antitubercular Agent SQ109

Levchenko, Kostiantyn; Virstiuk, Ivan; Menshykova, Daria; Pokhodylo, Nazariy: A convenient synthesis of CHF₂O-containing pyrrolidines and related compounds — Perspective building blocks for drug discovery

Ramteke, Prachi; Gill, Manjinder Singh: Retraction Note: Novel and efficient process for the synthesis of 1,3,4 Oxadiazole containing MBX-4132

Xu, Zhongnan; Liang, Xin-Ting; Song, Jian-Guo; White, Lorenzo V.; Banwell, Martin G.; Tan, Shen: Total Synthesis of the Prenylated Indole Alkaloid (±)-Notoamide N via an Electrochemically Mediated Vilsmeier–Haack Formylation of a Chlorinated Indole

Shehta, Wael; Alsaiari, Norah A.; Farag, Basant; Abdel-Aziz, Marwa M.; Youssif, Shaker; Elfeky, Sherin M; El-Kalyoubi, Samar; Osman, Nermine A.: Synthesis, In Vitro and In Silico Molecular Docking Studies of Novel Phthalimide–Pyrimidine Hybrid Analogues to Thalidomide as Potent Antitubercular Agents

Nakao, Michiyasu; Okamoto, Marie; Isetani, Satoshi; Imai, Ayato; Kitaike, Syuji; Sano, Shigeki: Development of a Novel Horner–Wadsworth–Emmons Reagent for the Facile Preparation of Mixed Phosphonoacetates

Levchenko, Kostiantyn; Virstiuk, Ivan; Menshykova, Daria; Pokhodylo, Nazariy: A Convenient Synthesis of CHF₂O-Containing Pyrrolidines and Related Compounds — Prospective Building Blocks for Drug Discovery

Koidan, Georgyi; Tsyzoryk, Nazar; Rusanov, Eduard B.; Shishkina, Svitlana V.; Vovk, Mykhailo; Kostyuk, Aleksandr: Functionalization of Position 7 of Pyrazolo[1,5-a]pyrazines

Gaikwad, Shweta S.; Chaturbhuj, Ganesh U.: Thiourea/NCBSI/HCl System: Telescoping Alkyl Halide to Alkyl Sulfonyl Chloride by Recyclable N-Chloro-N-(phenylsulfonyl)benzene Sulfonamide (NCBSI)

Schade, Alexander: Synthesis of 5-(4-Formylphenyl)barbituric Acid to Access Enolizable Chromophoric Barbituric Acids

Lipson, Victoria V.; Yaremenko, Fedyr G.; Vakula, Volodymyr M.; Kovalenko, Svitlana V.; Kyrychenko, Alexander V.; Desenko, Sergiy M.; Borysko, Petro О.; Zozulya, Sergiy O.: Discovery of Novel N-Acylhydrazone Derivatives as Potent Inhibitors of Sirtuin-1

Subramanyam, Amudala; Sumit, Sumit; Aidhen, Indrapal S.: Synthesis of C-Glucoside Analogues of Naturally Occurring Phenyl­ethanoid O-Glucosides

Polanco, Jocelyn; Knoell, Theresa; Bakhoda, Abolghasem Gus: Cobalt–Magnesium and Cobalt–Calcium Heterotrimetallic Dinitrogen Complexes

Balázsi, Áron; Bognár, Balázs; Jekő, József; Kálai, Tamás: Synthesis of 3,4-Disubstituted Pyrroline Nitroxides Containing Diphenylphosphane or Diphenylphosphane Oxide Substituents

Pitchai, Manivel; Kaspady, Mahammed; Indasi, Gopikumar; Krishnan, Rajesh; Maheswarappa, Gururaju Sannakki; Vetrichelvan, Muthalagu; Mathur, Arvind; Gupta, Anuradha: Regioselective C3-Formylation of 2H-Indazoles Using Selectfluor under Microwave-Assisted Conditions

Li, Li; Dai, Guo-Liang; Zhu, Xue Hua; Yu, Lei; Li, Hai Yan: Synthesis and Characterization of an Eight-Membered Heterocyclic 1,3,5,7-Tetra(3-pyridyl)-1,3,5,7-tetrazacyclooctane

Vetrichelvan, Muthalagu; Lanke, Veeranjaneyulu; Chandu, Bellam; Mathur, Arvind; Gupta, Anuradha: Cost-Effective and Scalable Synthesis of 4-Bromo-1,2-dimethyl-1H-imidazole: A Key Building Block for Bioactive Molecules

Yang, Qi-Liang; Lei, Ping-Ping; Hao, Er-Jun; Zhang, Bei-Ning; Zhou, Hong-Hao; Li, Wan-Wan; Guo, Hai-Ming: Oxidative C–H Sulfonylation of Hydrazones Enabled by Electrochemistry

Mudgal, Deeksha; Singh, Ravi Pratap; Yadav, Nisha; Bharti, Tapeesh; Mishra, Vivek: Exploring the Catalytic Efficiency of Copper-Doped Magnetic Carbon Aerogel for the Coupling Reaction of Isatin Oxime with Phenylboronic Acid Derivatives

Gavali, Kanchan D.; Chaturbhuj, Ganesh U.: Truly Catalytic Gewald Synthesis of 2-Aminothiophenes Using Piperidinium Borate (Pip Borate), a Conjugate Acid–Base Pair

Prakash, Supriya; Sreedhar, Bojja; Naidu, N. V. S.: Gum Acacia Stabilized Ag-TiO₂ and Ag-SiO₂: Sustainable Nanocatalysts for Direct and Convenient Synthesis of 5-Substituted 1H-tetrazoles

Lipson, Victoria; Zhikol, Oleg; Shishkina, Svetlana; Semenenko, Alexander; Kulyk, Karina; Mateychenko, Pavel; Musatov, Vladimir; Mazepa, Alexander; Vakula, Vladimir; Borisov, Alexander; Kyrychenko, Alexander: Low Molecular Weight Supramolecular Allobetuline-, Cyclohexanol-, or Undecanol-Appended 1,2,3-Triazole-Based Gelators: Synthesis and Molecular Dynamics Simulation Study

Prasanthi, A. V. G.; Babu, Bathini Nagendra: DMSO arbitrated Oxidative Annulation Followed by Homologated N-Alkylation: Microwave-Assisted Efficient and Greener Approach to Access 3-(3-Oxo-3-arylpropyl) Quinazolinones

Phull, Manjinder Singh; Jadav, Surender Singh; Bohara, Chander Singh; Gundla, Rambabu; Mainkar, Prathama S: Multi-step Flow Synthesis of the Anthelmintic Drug Praziquantel

Banwell, Martin G.; Marshall, Sarah; Ward, Jas S.; Schwartz, Brett D.: Synthesis of the Key Saccharide Fragments of the Glucuronic Acid-Containing Repeat Unit of Pentosan Polysulfate, a Heparin Sulfate Mimetic

Nakao, Michiyasu; Nakamura, Akihito; Takesue, Tomoyuki; Kitaike, Syuji; Ito, Hiro-O; Sano, Shigeki: Synthesis of Novel Phosphorus-Substituted Stable Isoindoles by a Three-Component Coupling Reaction of ortho-Phthalaldehyde, 9,10-Dihydro-9-oxa-10-phosphaphenanthrene 10-Oxide, and Primary Amines

Katla, Ramesh; Katla, Rakhi: Pyrrolidinium Acetate (PyrrIL) as a Green and Recyclable Catalyst: Synthesis of 2-Phenyl Benzimidazoles and 2-Phenyl Benzothiazoles under Solvent-Free Conditions at Room Temperature

Prachi, Ramteke; Gill, Manjinder Singh: A Practical and Efficient Method for the Synthesis of Sorafenib and Regorafenib

Kumar, Sunil; Yadav, Mangal S.; Singh, Sumit K.; Rajkhowa, Sanchayita; Tiwari, Vinod K.: Synthesis of Calix[4]arene Appended Lactosylated G₁ and Galacto­sylated G₂ Generation Glycodendrimers using a ‘CuAAC’ Click Approach

Sakhno, Yana; Radchenko, Oleksandr; Saraev, Vyacheslav; Shliapkina, Yuliia; Kaidash, Mariia; Shyshkina, Mariia; Shishkina, Svitlana; Musatov, Vladimir; Desenko, Sergey; Chebanov, Valentyn: Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction

Inyurt, Fevzi Can; Mammadova, Flora; Dengiz, Cagatay: Click-Type Synthesis of Homoconjugated Push–Pull Chromophores: Computational Investigation of Optical and Nonlinear Optical (NLO) Properties

Miyata, Ryo; Shigeta, Takashi; Kumazawa, Shigenori; Egi, Masahiro: Selective Syntheses of Coumarin and Benzofuran Derivatives Using Phenols and α-Methoxy-β-ketoesters

Goel, Kapil Kumar; Rajput, Satyendra Kumar; Kharb, Rajeev: Design, Synthesis and Biological Evaluation of Imidazole-Substituted/Fused Aryl Derivatives Targeting Tubulin Polymerization as Anticancer Agents

Mitra, Trisha; Joardar, Soumen; Chakravorty, Santanu; Majumdar, Manoj; Kundu, Mrinalkanti; Roy, Brindaban: Palladium-Mediated Reductive Heck Cyclization for the Synthesis of Fused Retinoid Derivatives

Burke, Adam; Spiccio, Silvia; Di Filippo, Mara; Baumann, Marcus: Photochemical Synthesis of Pyrazolines from Tetrazoles in Flow

Mali, Suraj N.; Pandey, Anima; Thorat, Bapu: A Chitosan Hydrochloride Mediated, Simple and Efficient Approach for the Synthesis of Hydrazones, their in vitro Antimycobacterial Evaluations, and Molecular Modeling Studies (Part III)

Srivastava, Avinash K.; Khandaka, Himanshu; Joshi, Raj Kumar: CN-Doped Cobalt Oxide Composite: An Economic and Reusable Catalyst with Multitasking Catalytic Capability for Alkyne and Nitrile Hydrations and Nitro Reductions

Mallesham, Poosa; Raghavulu, Karri; Miriyala, Venkatesh; Doddipalla, Raju; Yennam, Satyanarayana; Sanasi, Paul Douglas; Behera, Manoranjan: Synthesis of Acidiphilamide A–C: Secondary Metabolites from the Genus Streptacidiphilus

Ali, Mohammad Saif; Ramesh, P. I.; Ghosh, Subhash; Babu Tatina, Madhu: Zinc Acetate Catalyzed Stereoselective 1,2-trans-Glycosylation Using Glycosyl Chlorides

Yasam, Bharath Kumar; Pabbaraja, Srihari: Total Synthesis of Marine-Derived Azole Resistant Antifungal Agent (–)-Melearoride A and Antibiotic (–)-PF1163B

Noble, Jeffrey M.; Chang, Le; Chen, Dan; Wang, Binglin; Dominey, Raymond N.; Cook, Daniel W.; Burns, Justina M.; Stringham, Rodger W.; Cardoso, Flavio S. P.; Snead, David R.: A Practical and Economical Route to (S)-Glycidyl Pivalate

Biradar, D. O.; Mane, Y. D.; Sarnikar, Y. P.; Kulkarni, S. G.; Reddy, B. V. Subba; Narsaiah, A. Venkat: Zn/ZnBr₂ Catalysed Reaction of Aldehydes with Allylbromide: Synthesis of 2,6-Disubstituted 4-Bromotetrahydropyrans

Tan, Shen; Lan, Ping; Banwell, Martin G.; White, Lorenzo V.: Practical, Multigram Preparation of Synthetically Useful, Enantiomerically Pure Building-Blocks from Quinic Acid

Biradar, Dhanraj O.; Mane, Yogesh D.; Subba Reddy, Basi V.: Stereoselective Synthesis of Euscapholide and Tetraketide via Prins Cyclisation and Ring-Closing Metathesis

Jesin, C. P. Irfana; Kataria, Ramesh; Nandi, Ganesh Chandra: Synthesis of α-Sulfoximino Tetrazoles via Azido-Ugi Four-Component Reaction

Lin, Zhongren; Tong, Lingfeng; Qiu, Hong; Li, Zheyao; Shen, Lunhua; Chen, Niangen; Yu, Xinhong: The Synthesis of 5-Hydroxybenzofurans via Tandem In Situ Oxidative Coupling and Cyclization

Liu, Ying; Zhang, Yiping; Zhou, Yingkai; Zhang, Min; Deng, Hongmei; Song, Liping: Concise One-Pot Multicomponent Reaction Approach to Mono­fluo­rinated Spiro-pyrazole-pyridine Derivatives without Additional Catalyst

Devi, Lalita; Mishra, Poornima; Pokhriyal, Ayushi; Rastogi, Namrata: Organo-photocatalytic Synthesis of Functionalized Pyrroles from 2H-Azirines and α-Substituted Nitroalkenes

Mkhonazi, Blessing D.; Mabila, Euphrent M.; Moshapo, Paseka T.: Palladium-Catalysed Reductive Aminocarbonylation of Aryl Bromides and Iodides with Nitroarenes

Nie, Hui; Wang, Nian; Huang, Jinwen; Ni, Zhuang; Xue, Kangyan; Song, Lixing; Wang, Mingwei; Wu, Fanhong: Radiosynthesis and Tumor MicroPET/CT Imaging of ¹⁸F-Fluoro­ethoxylerianin, an ¹⁸F-Labeled Erianin Analogue

Jagadeesha, Gullahalli S.; Mantelingu, Kempegowda; Thimmegowda, Naraganahalli R.; Rangappa, Kanchugarakoppal S.: Microwave-Assisted, Metal-Free, Chemoselective N-Formylation of Amines using 2-Formyl-1,3-dimethyl-1H-imidazol-3-ium Iodide and In Situ Synthesis of Benzimidazole and Isocyanides

Prabhakaran, Srinivasan; Velmathi, Sivan: Synthesis and Molecular Docking Studies of N,N-Dimethyl Arylpyranopyrimidinedione Derivatives

Tonekaboni, Maryam-Sadat; Tanbakouchian, Zahra; Majedi, Soma; Shiri, Morteza: Synthesis of [1,4]Oxathiepino[5,6-b]quinolines via Base-Mediated Intramolecular Hydroalkoxylation

Li, Zhongyuan; Huang, Jinwen; Ni, Zhuang; Sun, Ran; Nie, Hui; Tang, Hui; Song, Lixing; Wu, Fanhong: Indium-Mediated Reformatsky Reaction of Iododifluoro Ketones with Aldehydes: Preparation of α,α-Difluoro-β-hydroxyketone Derivatives in Water

Jagot, Fatema; Minnie, Izak; Rahman, Aliyaah; Ntsimango, Songeziwe; Ngwira, Kennedy J.; de Koning, Charles B.: Hydrogen-Bonded Xanthones as Potential UV Absorbers: The Synthesis of Xanthones from Bio-Renewable Cardanol Utilizing a Ceric Ammonium Sulfate (CAS)-Mediated Oxidation Reaction

Sosunovych, Bohdan; Brown, Alexander J.; Clarke, Paul A.: Amino Imidate Catalyzed Asymmetric Michael Reactions of Ketones and Nitroalkenes

Veverková, Eva; Molnosiová, Pavlína; Šebesta, Radovan: Asymmetric Sequential Michael Addition and Cyclization Reactions of 2-(2-Nitrovinyl)phenols Catalyzed by Bifunctional Amino-Squaramides

Kumar, Nemilikonda Sravan; Ramulu, B. Janaki; Ghosh, Subhash: Stereoselective Synthesis of the C19–C39 Fragment of Bastimolide A

Yadav, Mangal S.; Jaiswal, Manoj K.; Kumar, Sunil; Tiwari, Vinod K.: Trichloroacetimidate-Triggered Expeditious and Novel Synthesis of N-Acylbenzotriazoles

Duda, Addison M.; Giurini, Michael T.; Gillmore, Jason G.; Guarr, Thomas F.: Intramolecular Oxidative Diaryl Coupling of Tetrasubstituted Diphenylamines for the Preparation of Bis(trifluoromethyl) Dimethyl Carbazoles

Bardovskyi, Rostyslav; Fabre, Marie; Ronco, Cyril; Benhida, Rachid: Mild Biamidine-Transfer Conditions for the Synthesis of Aliphatic Biguanides

Liang, Zhi-Peng; Yu, Ying-Xin; Sun, Yuan-Yuan; Wang, Yang; Wu, Zheng-Guang: Oxidative Annulation of Diphenylpropanamides via In Situ Hypervalent Iodine-Promoted Intramolecular C–N/C–O Bond Formation

Zullo, Valerio; Petri, Antonella; Iuliano, Anna: An Efficient and Practical Chemoenzymatic Route to (3R,3aR,6R,6aR)-Hexahydrofuro[3,2-b]furan-6-amino-3-ol (6-Aminoisomannide) from Renewable Sources

Farhid, Hassan; Rostami, Mohammad Mahdi; Shaabani, Ahmad; Notash, Behrouz: Synthesis of Depsipeptides via Isocyanide-Based Consecutive Bargellini–Passerini Multicomponent Reactions

Saeedi, Marziyeh; Khoshdoun, Maryam; Taheri, Salman; Ziyaei Halimehjani, Azim; Mohammadi, Aliasghar; Halvagar, Mohammad Reza; Amani, Vahid: Synthesis of Functionalized Bicyclic Pyridones Containing the Dithiocarbamate Group Using Thioazlactones, Diamines, and Nitroketene Dithioacetal

Sathish, Kota; Nagaraju, Sakkani; Kashinath, Dhurke: Synthesis of Spiro Pyrazolone-Oxindole and Bicyclic Pyrazolone Derivatives via Solvent-Dependent Regioselective Aza-1,4/1,6-Michael and Intramolecular Cycloaddition under Catalyst-Free Conditions

De Marchi, Elisa; Arnodo, Davide; Maffeis, Elia; Scarpi, Dina; Prandi, Cristina; Occhiato, Ernesto G.: Enantiodivergent Synthesis of Halofuginone by Candida antarctica Lipase B (CAL-B)-Catalyzed Kinetic Resolution in Cyclopentyl Methyl Ether (CPME)

Katta, Narenderreddy; Murugan, Arumugavel; Sharma, Sonika; Sharada, Duddu S.: Visible-Light-Mediated Photocatalytic Oxidative C–C Bond Cleavage of Geminal Diazides: An Approach to Oxamates

Kutyashev, Igor B.; Sannikov, Maxim S.; Kochnev, Ivan A.; Barkov, Alexey Y.; Zimnitskiy, Nikolay S.; Korotaev, Vladislav Y.; Sosnovskikh, Vyacheslav Y.: Diversity-Oriented Synthesis of Novel Trihalomethyl-Containing Spirochromeno[3,4-a](thia)pyrrolizidines and Spirochromeno-[3,4-a]indolizidines by One-Pot, Three-Component [3+2]-Cyclo­addition Reaction

Bracken, Cormac; Batsanov, Andrei S.; Baumann, Marcus: Development of a Continuous Photochemical Benzyne-Forming Process

Guirado, Antonio; Vera, María; Martiz, Bruno; Ródenas, Francisco; Sandoval, José A.; Alarcón, Enrique; Bautista, Delia: Synthesis and Crystal Structures of 4,5-Dihydroimidazo[1,5-b]pyrazol-6-ones

Avula, Satya Kumar; Das, Biswanath; Csuk, Rene; Al-Rawahi, Ahmed; Al-Harrasi, Ahmed: Total Synthesis of Surinamensinols A and B

Nariki, Haruna; Miyamura, Takuya; Matsui, Daiki; Sonoda, Motohiro; Tanimori, Shinji: Iodine-Mediated Facile One-Pot Access to N-Aryl-2-benzoxazolamines

Faverio, Chiara; Boselli, Monica Fiorenza; Raimondi, Laura; Benaglia, Maurizio: Ammonia–Borane-Mediated Reduction of Nitroalkenes

Rickertsen, Dillon R. L.; Ma, Longle; Paul, Anirudra; Abboud, Khalil A.; Seidel, Daniel: Traceless Redox-Annulations of Alicyclic Amines

Raghunadh, Akula; Tadiparthi, Krishnaji; Meruva, Suresh Babu; Murthy, V. Narayana; Rao, L. Vaikunta; Kumar, U. K. Syam: Synthesis of Quinoxalin-2(1H)-ones and Hexahydroquinoxalin-2(1H)-ones via Oxidative Amidation–Heterocycloannulation

Raji Reddy, Chada; Sinare, Sudam N.: Expedient Approach to the Synthesis of Betrixaban

Qin, Ling; Wu, Hui-bin; Weng, Lidong; Shen, Qun; Chen, Huoji: Aerobic Iron(III)-Catalyzed Direct Thiolation of Imidazo[1,2-a]pyridine with Thiols

Sharma, Pooja; Singh, Gurdial; Bhongade, Bhoomendra A.; Noolvi, Malleshappa N.; Gadad, Andanappa K.: Synthesis of 5-Fluoroaminobenzothiazoles

Singh, Pargat; Nath, Mahendra: A Modified Vilsmeier–Haack Strategy to Construct β-Pyridine-Fused 5,10,15,20-Tetraarylporphyrins

Jain, Vipin Kumar; Kumar, Mrityunjay: Synthesis of (–)-Bulgecinine and 5-epi-Bulgecinine through Proline-Catalysed Asymmetric α-Hydroxylation of an Aldehyde Derived from l-Glutamic Acid

Dacho, Vladimír; Nitrayová, Dária; Šoral, Michal; Machyňáková, Andrea; Moncoľ, Ján; Szolcsányi, Peter: Access to N-Alkylpyrazin-2-ones via C–O to C–N Rearrangement of Pyrazinyl Ethers

Jain, Vipin Kumar: Diastereoselective Synthesis of (–)-Bestatin, Epibestatin, Phebestin and (3S,4R)-4-Amino-3-hydroxy-5-phenylpentanoic Acid from an Aldehyde Derived from d-Phenylalanine

Sonawane, Rahul B.; Sonawane, Swapnali R.; Rasal, Nishant K.; Jagtap, Sangeeta V.: Room-Temperature, Base-Mediated Selective Synthesis of 2-(Arylamino)ethanols and 2-Aryloxyethanols

Szabó, Tímea; Kormány, Róbert; Dancsó, András; Volk, Balázs; Milen, Mátyás: Total Synthesis of Bacterial 5-(3-Indolyl)oxazole Alkaloids: Pimprinols A–C

Talakokkula, Anil; Baikadi, Karunakar; Narsaiah, A. Venkat: First Total Synthesis of Artekeiskeanol A, C and Altissimacoumarin D

Sharada, Ambati; Kundeti, Lakshmi Srinivasa Rao; Ramakrishna, Kallaganti V. S.; Nagaiah, Kommu: First Stereoselective Total Synthesis of Ciryneol C

Kawtharani, Ranin.; Elmasri, Mirvat; Cherry, Khalil; Jacquemin, Johan; Abarbri, Mohamed: Highly Regio- and Stereoselective Hydrogermylation of Fluorinated Alkyl Propiolate

Debnath, Sudarshan; Mondal, Shovan: Palladium-Catalysed Intramolecular C–N versus C–C Coupling: The Effect of 1,8-peri-Interaction in the Naphthalene System

Kitagawa, Saori; Mori, Hiromitsu; Odagiri, Tatsuya; Suzuki, Katsuya; Kikkawa, You; Osugi, Rie; Takizawa, Shinobu; Kimura, Yoshikazu; Kirihara, Masayuki: A Concise, Catalyst-Free Synthesis of Davis’ Oxaziridines using Sodium Hypochlorite

Baikadi, Karunakar; Talakokkula, Anil; Narsaiah, A. Venkat: Stereoselective Total Synthesis of Macrolide Sch-725674 and C-7-epi-Sch-725674

Sarkar, Sujit; Devi, Namita; Porashar, Bikoshita; Ruidas, Santu; Saikia, Anil K: Stereoselective Synthesis of 4-O-Tosyltetrahydropyrans via Prins Cyclization Reaction of Enol Ethers

Kumar, Devarapalli Ravi; Kishore, Dakoju Ravi; Satyanarayana, Gedu: Palladium-Catalysed Coupling and Acid-Mediated Cyclisation: Synthesis of Fluorenones and Fluorenes

Panwar, Rahul; Shally; Shaw, Ranjay; Elagamy, Amr; Shah, Chandan; Pratap, Ramendra: Substituent-Dependent Chemoselective Synthesis of Highly Functionalized­ Benzo[h]quinolines and 4-Benzylpyrans from 2-Methyl-5-nitro-benzonitrile

Bandatmakuru, Sreenivasulareddy; Arava, Veerareddy: Novel Synthesis of 1,2-Substituted 4-Quinolones

Mayooufi, A.; Romdhani-Younes, M.; Thibonnet, J.: Efficient One-Pot Synthesis of Triazole-Linked Morpholinone Scaffolds by CuAAC in the Presence of 18-Crown-6

Delaye, Pierre-Olivier; Pénichon, Mélanie; Boudesocque-Delaye, Leslie; Enguehard-Gueiffier, Cécile; Gueiffier, Alain: Natural Deep Eutectic Solvents as Sustainable Solvents for Suzuki­–Miyaura Cross-Coupling Reactions Applied to Imidazo-Fused Heterocycles

Nagalatha, G.; Narala, Siva Ganesh; Narsaiah, A. Venkat: First Stereoselective Total Synthesis of Tumonoic Acid A and its Derivatives

Balalas, T. D.; Stratidis, G.; Papatheodorou, D.; Vlachou, E.-E.; Gabriel, C.; Hadjipavlou-Litina, D. J.; Litinas, K. E.: One-pot Synthesis of 2-Substituted 4H-Chromeno[3,4-d]oxazol-4-ones from 4-Hydroxy-3-nitrocoumarin and Acids in the Presence of Triphenylphosphine and Phosphorus Pentoxide under Microwave Irradiation

Ahsan, Mohamed J.; Kumawat, Bhawani S.; Kumawat, Sonu; Sharma, Piush; Bakht, Mohammad A.; Hassan, Mohd Z.; Hussain, Afzal; Saraswat, Pankaj; Khalilullah, Habibullah: Synthesis and Cytotoxic Evaluation of 3-(4-Fluorophenyl)-4,5-dihydro-5-(3,4,5-trimethoxy/4-nitrophenyl)-N-(substituted-phenyl)pyrazole-1-carboxamide Analogues

Kour, M.; Gupta, R.; Saini, R.; Bansal, R. K.: Diastereoselectivity in the Aza-Michael Reaction of Chiral α-Methylbenzylamines with α,β-Unsaturated Carbonyl Compounds

Mourya, Mohini; Sharma, Himanshu; Joshi, Yogesh C.; Basak, Ashok K.: [4+3]-Annulation of 3-Cyano-4-aryl-2-iminochromenes with 1,2-Diaminobenzene: An Access to Novel Chromenobenzodiazepines

Tiwari, Raju; Nath, Mahendra: A Divergent Approach to β-Pyrazine-Fused meso-Tetraphenyl­diporphyrins

Gujjarappa, Raghuram; Vodnala, Nagaraju; Kabi, Arup K.; Kaldhi, Dhananjaya; Kumar, Mohan; Beifuss, Uwe; Malakar, Chandi C.: Efficient Syntheses of Diverse N-Heterocycles: The Molybdenum(VI)-Catalyzed Reductive Cyclization of Nitroarenes using Pinacol as a Deoxygenating­ Agent

Nagaraju, Kare; Rajesh, Nomula; Krishna, Palakodety Radha: Synthesis of Phthalimides: A New Entry via TBAI-Catalyzed Intramolecular Cyclization of 2-(Hydroxymethyl)benzamides

Pathan, Mosim Amin; Khan, Faiz Ahmed: Synthesis of Substituted Pyrido-oxazine through Tandem S_N2 and S_NAr Reaction

Matziari, Magdalini; Xie, Yixin: One-Pot Synthesis of α-Substituted Acrylates

Shields, Samuel W. J.; Buist, Peter H.; Manthorpe, Jeffrey M.: Asymmetric and Regiospecific Synthesis of Isotopically Labelled Cyclopropane Fatty Acid (9R,10S)-Dihydrosterculic Acid: Overcoming Spontaneous Protonation During Lithium-Sulfoxide Exchange­

Rana, Anil; Kumar, Varun; Tiwari, Lata; Thakur, Anamika; Meena, Chhuttan Lal; Mahajan, Dinesh: Triflic Anhydride Promoted Synthesis of Primary Amides and their Conversion into Nitriles

Grollmisch, A.; Kragl, U.; Großeheilmann, J.: Enzyme Immobilization in Polymerized Ionic Liquids-based Hydrogels for Active and Reusable Biocatalysts

Rahman, Masood ur; Ayoob, Iram; Rehman, Shakeel u; Bhat, Khursheed A.; Ara, Tabassum: Microwave-Assisted Synthesis of Andrographolide Analogues as Potent β-Glycosidase Inhibitors

Choudhary, Rakhee; Bai, Rekha; Singh, Pratibha; Sharma, Mahesh C.; Badsara, Satpal Singh: Room Temperature, Open-Flask C–P Bond-Formation on Water under Catalyst-Free Conditions

Songsichan, T.; Katrun, P.; Khaikate, O.; Soorukram, D.; Pohmakotr, M.; Reutrakul, V.; Kuhakarn, C.: Thiocyanation of Pyrazoles Using KSCN/K₂S₂O₈ Combination

Kummari, Bhaskar; Ramesh, Perla; Polkam, Naveen; Malthum, Shankaraiah; Vishnuvardhan, M. V. P. S.; Anireddy, Jaya Shree: Design, Synthesis, and Cytotoxic Evaluation of Etodolac-1,3,4-oxadiazole-1,2,3-triazole Molecules

Uma, Pathki; Rajanna, Kamatala Chinna; Sriram, Yelike Hemanth; Premalatha, Akarapu; Saipraksh, Pondichery Kuppuswamy: Synthesis of 3-(4-(Benzo[d]thiazol-2-yl)phenyl)-5-aryl-1,3,5-oxadiazinane-4-thiones and 1-(4-(Benzo[d]thiazol-2-yl)phenyl)-5-methyl-3-aryl-1,3,5-triazinane-2-thiones

Caillé, Julien; Setzer, Paul; Boeda, Fabien; Pearson-Long, Morwenna S. M.; Bertus, Philippe: Asymmetric Titanium-Catalyzed Cyclopropanation of Nitriles with Grignard Reagents

Nakao, Michiyasu; Nishikiori, Nanako; Nakamura, Akihito; Miyagi, Murasaki; Shibata, Nao; Kitaike, Syuji; Fukui, Makoto; Ito, Hiro-O; Sano, Shigeki: Synthesis of Sterically Protected Isoindoles from ortho-Phthalaldehyde

Reddy, A. Maheswara; Sabitha, Gowravaram: First Total Synthesis of Cryptopyranmoscatone A3 and Crypto­pyranmoscatone B4

Menczinger, B.; Nemes, A.; Csámpai, A.; Rábai, J.: Synthesis of 3-(Arylthio)propionic Acids from Nonactivated Aryl Iodides and their Use as Odorless Aryl Mercaptan Surrogates

Zeng, Meng-Tian; Xu, Wan; Liu, Min; Liu, Xing; Chang, Cai-Zhu; Zhu, Hui; Dong, Zhi-Bing: Iodobenzene-Promoted Pd-Catalysed ortho-Directed C–H Activation: The Synthesis of Benzothiazoles via Intramolecular Coupling

Ghosal, Nirnita Chakraborty; Mahato, Sachinta; Chatterjee, Rana; Santra, Sougata; Zyryanov, Grigory V.; Majee, Adinath: A Mild and Efficient Method for the Syntheses and Regioselective Ring-Opening of Aziridines

Diez-Martinez, Alba; Krishnamurthy, Ramanarayanan: Investigations towards the Synthesis of 5-Amino-l-lyxofuranosides and 4-Amino-lyxopyranosides and NMR Analysis

Panda, Siva S.; Asiri, Abdullah M.; Elagawany, Mohamed; Buchanan, Devan D.; Torkian, Behrad; Bathala, Keerthana; Thomas, Sean J.; Capito, Jason E.; Arshad, Muhammad N.; Al-Romaizan, Abeer N.: Efficient Synthesis of Pyrazinoic Acid Hybrid Conjugates

Ge, Haihong; Liu, Shuang; Cai, Yan; Gao, Zenghui; Du, Siyi; Miao, Zhiwei; Xie, Guixian: Diastereoselective [Cu(MeCN)₄BF₄/BF₃·Et₂O]-Catalyzed Cyclopropenation of Alkynes: Asymmetric Synthesis of β-Amino-α-cyclopropenyl Phosphonates

Li, Jihui; Yu, Weiguang; Hou, Yifeng; Fu, Wenxing; Xu, Shuying; Zhang, Yucang: An Efficient Protocol for the Synthesis of O-Fluoroalkylisoureas through Copper-Catalysed, Three-Component Reaction of Cyan­amides, Fluoroalcohols and Diaryliodonium Triflates

Nosik, Pavel S.; Artamonov, Oleksiy S.; Ryabukhin, Sergey V.; Grygorenko, Oleksandr O.: An Approach to 1,1-Disubstituted Pyrazolylcyclopropane Building Blocks

Cívicos, José F.; Costa, Paulo R. R.; Domingos, Jorge L. O.: Palladium-Catalyzed α-Arylation of Dimethyl Malonate and Ethyl Cyanoacetate with o-Alkoxybromobenzenes for the Synthesis of Phenylacetic Acid, Esters and Phenylacetonitriles

Don Lawson, Chioma; Maza-Iglesias, Max; Sirhan, Muthana M.; Al Dulayymi, Jumaa R.; Baird, Mark S.: The Synthesis of Single Enantiomers of α-Mycolic Acids of Mycobacterium­ tuberculosis and Related Organisms, with Alternative­ Cyclopropane Stereochemistries

Majeed, Anju; Nagabhushanam, Kalyanam; Majeed, Muhammed; Thomas, Samuel Manoharan; Thajuddin, Nooruddin: An Expeditious, Green and Protecting-Group-Free Synthesis of a Potent Secondary Metabolite Calebin-A and Its Analogues

Zhao, Lingyu; Shen, Guodong; Zhang, Tongxin; Wang, Zhen; Liang, Yuhua: Pd/C-Catalyzed Intramolecular C–H Arylation for the Synthesis of Phenanthridinones and Dibenzo-α-pyrones

Yang, Yi-Qiu; Ke, Long-Zhi; Wang, Gui-Fei; Song, Shu-Yong; Qiu, Ming-Ning; Liu, Jian-Jun; Huang, Yun-Sheng: Synthesis of N-Pyridin-2-ylmethyl and N-Quinolin-2-ylmethyl ­Substituted Ethane-1,2-diamines

Barcia, Jose C.; Cruces, Jacobo; Salas, Cristian O.; Estévez, Juan C.; Cuellar, Mauricio A.; Tapia, Ricardo A.; Estévez, Ramón J.: A New Approach to the Synthesis of Benzo[b]naphtho[2,3-b]furan-6,11-diones and 2-Benzyl-3-hydroxynaphthalene-1,4-diones

Maheshwar Reddy, A.; Sabitha, Gowravaram: Synthesis of the C1–C9, C11–C19 Pyran Core and C19–C24 Fragments­ of Macrolactin 3