Pd-Catalyzed Coupling of Arylboronic Esters with Carbamoyl Chlorides
M. Lysén, S. Kelleher, M. Begtrup, J. L. Kristensen*
Danish University of Pharma-ceutical Sciences, Copenhagen, Denmark
21. September 2005 (online)
A wide range of boronic acids and esters are available. The acylation of these ‘bench-stable’ organoboron compounds would be of great interest and is reported in the article by using simple palladium catalysis. The resulting benzamides are important compounds having a number of applications.