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Synfacts 2005(1): 0155-0155  
DOI: 10.1055/s-2005-872130
Metal-Mediated Synthesis
© Georg Thieme Verlag Stuttgart · New York

Pd-Catalyzed Coupling of Arylboronic Esters with Carbamoyl Chlorides

Contributor(s): Paul Knochel, Andrei Gavryushin
M. Lysén, S. Kelleher, M. Begtrup, J. L. Kristensen*
Danish University of Pharma­-ceutical Sciences, Copenhagen, Denmark
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Publication History

Publication Date:
21 September 2005 (online)

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Significance

A wide range of boronic acids and esters are available. The acylation of these ‘bench-stable’ organoboron compounds would be of great interest and is reported in the article by using simple palladium catalysis. The resulting benzamides are important compounds having a number of applications.