Fluorescent-Labeled Amino Acid–Antibiotic Conjugates

Anand D. Tiwari; Siva S. Panda; Abdullah M. Asiri; C. Dennis Hall; Alan R. Katritzky

doi:10.1055/s-0033-1340193

Synthesis, Inhaltsverzeichnis

Synthesis 2014; 46(18): 2430-2435
DOI: 10.1055/s-0033-1340193

paper

Fluorescent-Labeled Amino Acid–Antibiotic Conjugates

Anand D. Tiwari

^aCenter for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, FL 32611-7200, USA

,

Siva S. Panda*

^aCenter for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, FL 32611-7200, USA

,

Abdullah M. Asiri

^bChemistry Department, King Abdulaziz University, Jeddah, 21589, Saudi Arabia

^cCenter for Advanced Materials Research (CEAMR), King Abdulaziz University, Jeddah 21589, Saudi Arabia Fax: +1(352)3929199 eMail: sspanda12@gmail.com eMail: charlesdennishall@gmail.com

,

C. Dennis Hall*

^aCenter for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, FL 32611-7200, USA

,

Alan R. Katritzky †

^aCenter for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, FL 32611-7200, USA

^bChemistry Department, King Abdulaziz University, Jeddah, 21589, Saudi Arabia

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Abstract

Alle Artikel dieser Rubrik

Abstract

Benzotriazole-mediated synthesis provides novel fluorescent-labeled amino acid–quinolone antibiotic conjugates in good yields with retention of chirality. The photophysical properties of all the fluorescent-labeled antibiotic conjugates were determined.

Key words

antibiotics - amino acid - drug design - microwave assisted reaction - fluorescent labels

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Referenzen

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