Synthesis 2019; 51(12): 2564-2571
DOI: 10.1055/s-0037-1612421
DOI: 10.1055/s-0037-1612421
paper
Exploratory Process Development of Pexidartinib through the Tandem Tsuji–Trost Reaction and Heck Coupling
Dongsheng Chen
a
Novel Technology Center of Pharmaceutical Chemistry, Shanghai Institute of Pharmaceutical
Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China
b
Shanghai Engineering Research Center of Pharmaceutical Process, Shanghai Institute
of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China Email: lijianqb@126.com Email: liuyu_tianjin@126.com
,
Yi Zhang
a
Novel Technology Center of Pharmaceutical Chemistry, Shanghai Institute of Pharmaceutical
Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China
b
Shanghai Engineering Research Center of Pharmaceutical Process, Shanghai Institute
of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China Email: lijianqb@126.com Email: liuyu_tianjin@126.com
,
Jianqi Li*
a
Novel Technology Center of Pharmaceutical Chemistry, Shanghai Institute of Pharmaceutical
Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China
b
Shanghai Engineering Research Center of Pharmaceutical Process, Shanghai Institute
of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China Email: lijianqb@126.com Email: liuyu_tianjin@126.com
,
Yu Liu
*
a
Novel Technology Center of Pharmaceutical Chemistry, Shanghai Institute of Pharmaceutical
Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China
b
Shanghai Engineering Research Center of Pharmaceutical Process, Shanghai Institute
of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry, 285 Gebaini Road, Shanghai 201203, P. R. China Email: lijianqb@126.com Email: liuyu_tianjin@126.com
› Author Affiliations