DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 9 · September 2013 DOI: 10.1055/s-003-25490

Synform

A107
Zanda, Matteo: SYNFORM ISSUE 2013/09

Synthesis of Natural Products and Potential Drugs

z915
All PDFs of this category
0915
Total Synthesis of (–)-Bolivianine
0916
Synthesis of (–)-Rhazinilam and (–)-Rhazinicine
0917
Synthesis of a Retinoic Acid Receptor Agonist
0918
Biomimetic Synthesis of the Major Colorants of Red Sandalwood
0919
Syntheses of (–)-Scabronines A and G, and (–)-Episcabronine A
0920
Total Synthesis of Daphenylline
0921
Synthesis of Almorexant
0922
Synthesis of Entecavir
0923
Synthesis of Vabicaserin
0924
Synthesis of a Mineralocorticoid Antagonist
0925
Synthesis of (1R,3S)-HPA-12
0926
Synthesis of (–)-Nakadomarin A
0927
Synthesis of (1R,3S)-HPA-12
0928
Synthesis of a Serotonin Norepinephrine Reuptake Inhibitor
0929
Total Synthesis of (±)-Rhazinal by a Catellani Ortho-Arylation

Synthesis of Heterocycles

z931
All PDFs of this category
0931
Palladium(II)-Catalyzed Dehydrogenative Heck Route to Pyrroles
0932
Synthesis of Homobenzotetramisole Organocatalysts by Heteroannulation
0933
Iron-Catalyzed Synthesis of Pyrrolidines via C–H Bond Amination
0934
A One-Pot Amine-Catalyzed de novo Synthesis of Highly Substituted Pyridines
0935
Synthesis of Perimidines and 1,5-Benzodiazepines
0936
Regioselective Functionalization of Pyrimidines and Pyrazines via Metalation
0937
One-Pot, Three-Component Sonogashira–Heterocyclization–Heck Reactions
0938
Benzimidazoisoquinoline Synthesis by Ru-Catalyzed Oxidative C–C and C–N Coupling
0939
Synthesis of Pyrazoloisoquinolines from Alkynes and Pyrazoles
0940
Benzyne-Mediated Heteroannulation Route to Indolines and Carbazoles
0941
Cu-Catalyzed C–N Cross-Coupling of Iodopyridines with Nitrogen Heterocycles
0942
Ag-Catalyzed Isocyanide-Alkyne Cycloaddition Route to Pyrroles
0943
Ru-Catalyzed Heteroannulation Route to Isoquinolines and Thienopyridines
0944
Pyrido[1,2-a]benzimidazoles via Iodine(III)-Mediated Demethylenation
0945
Gold-Catalyzed Synthesis of (Z)-1,2-Dihydro-1-tosylbenzo[b]azepin-3-ones

Synthesis of Materials and Unnatural Products

z947
All PDFs of this category
0947
One-Pot Synthesis of Poly(phenylenebutadiynylenes)
0948
Nitrile-Directed Palladium-Catalyzed Syntheses of Fluorenones
0949
Direct Conversion of Terminal Alkynes into Nitriles
0950
Triphenylenes and Azatriphenylenes by [2+2+2] Cycloadditions
0951
Ru-Based Metathesis Catalysts Yield Highly cis, Syndiotactic Polymers
0952
Low Temperature Synthesis of Aryl Sulfides
0953
A New Route to Zethrene
0954
Fullerene Functionalization under Kulinkovich Reaction Conditions
0955
Distorted Calix[4]arenes via Organomercurials
0956
Cross-Coupling at the 2-Positions of Indoles and Pyrroles by Chelation Assistance
0957
Tuning Photochromic Properties Through Molecular Conformation
0958
Mild and Metal-Free Synthesis of 2,4-Disubstituted Thiophenes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z959
All PDFs of this category
0959
Copper-Catalyzed Asymmetric Conjugate Addition of Organozinc Reagents
0960
Ruthenium-Catalyzed Dearomatization of Indoles
0961
Stereoselective [3+2] Cycloadditions Catalyzed by AgNTf2
0962
Gold-Catalyzed Synthesis of Medium-Sized Carbocycles
0963
Multicomponent Cyclobutane Synthesis in One Pot
0964
Ru-Catalyzed Asymmetric Hydrogenation of α-Arylcyclohexanones via DKR
0965
Asymmetric Hydrogenation of Cyclic Unsaturated Heterocyclic Acids
0966
Nickel-Catalyzed Asymmetric Michael Additions with 2-Acetylazaarenes
0967
Cooperative Lewis Acid Catalyzed Fluoride Ring Opening of Aziridines
0968
Asymmetric Allylic Alkylation of Cyclobutanones
0969
Enantioselective Aminoborylation of Aldehydes by a Chiral Pt Complex
0970
Mannich-Type Reaction of α-Sulfanyl Lactones by a Chiral Ag Complex
0971
Sc(III)-Catalyzed Enantioselective Conjugate Addition and α-Alkynylation of Oxindoles
0972
Zn-Mediated Asymmetric Allylation of N-tert-Butanesulfinyl Ketimines
0973
Indium-Catalyzed Hetero-Diels–Alder Cycloaddition
0974
Asymmetric Synthesis of Carbocycles by Pd/Chiral Amine Co-catalysis
0975
Cooperative Enamine–Copper–Brønsted Acid Catalyzed Cross-Aldol Reaction
0976
Enantioenriched CF3-Substituted Amino Acid Derivatives via Rh-Catalyzed Alkynylation
0977
Synthesis of Enantioenriched 1,2-Diamines L10013
0978
Synthesis of BIPI Ligands for the Asymmetric Hydrogenation
0979
Palladium-Catalyzed Enantioselective Allylation of Ketimines
0980
Pd-Catalyzed Asymmetric Allylic Alkylation of Pyrazol-5-ones
0981
Asymmetric Rh-Catalyzed Hydrogenation Using a Mixed Ligand Approach
0982
Enantioenriched Diarylcarbinols via Ru-Catalyzed Boronic Acid Addition of Aldehydes
0983
Cu–NHC-Catalyzed Asymmetric Conjugate Silylation
0984
Synthesis of Enantioenriched 3-Hydroxy-3,4-dihydroquinolin-2(1H)-ones
0985
Copper-Catalyzed Enantioselective 1,3-Dipolar Cycloaddition
0986
Dirhodium-Catalyzed Enantioselective Synthesis of Cyclopropanes
0987
Cu-Oxazoline-Imidazoline Catalyst for Asymmetric Friedel–Crafts Alkylation
0988
Palladium-Catalyzed Enantioselective Dehydrogenative Heck Reaction

Metal-Mediated Synthesis

z989
All PDFs of this category
0989
Regioselective Co-Catalyzed Reactions of 1,3,5-Hexatrienes
0990
Al-Amides as Chemoselective Reagents in Additions to Carbonyl Groups
0991
Fe-, Co- and Cu-Catalyzed Coupling Reactions Using N2O
0992
Ru-Catalyzed Reduction of Alkynes, Ketones, and Nitro Compounds
0993
Synthesis of β-Alkynyl Ketones via Ti-Catalyzed Three-Component Couplings
0994
Aldol and Mannich Reactions with Supersilyl-Protected Carboxylic Acids
0995
Indole Synthesis via Intramolecular Carbocupration of N-Aryl-ynamides
0996
Highly Regioselective Synthesis of 3-Trifluoromethylpyrazoles
0997
An Aryl Sulfonamide Synthesis Using tert-Butyllithium
0998
Cu-Mediated Trifluoromethylation of Quinones
0999
Lithium-Base-Induced Aryne Formation Using Arylboronic Esters
1000
Stereoretentive Stille Coupling Using Secondary Alkyl Azastannatranes
1001
TmI2-Mediated C–N Bond Cleavage in Amides and Reduction of Esters
1002
Co-Catalyzed sp3–sp3 Cross-Coupling with Tertiary Alkyl Grignard Reagents
1003
Synthesis of Enantiopure Sulfinamides and Sulfinyl Ketimines

Organo- and Biocatalysis

z1005
All PDFs of this category
1005
Catalytic Asymmetric Oxidation of Imines to Oxaziridines
1006
Kinetic Resolution of Oxaziridines
1007
Amphiphilic Proline and CO2
1008
Enantioselective 6π-Electrocyclization to 1,4-Dihydropyridazines
1009
NHC-Catalyzed [4+3] Annulation of Enals and o-Quinone Methides
1010
Catalytic Asymmetric Fluoroamination
1011
Homo-Ene Cyclizations by SOMO Catalysis
1012
Hantzsch Esters Reacting Like Metal-Free Grignard Reagents
1013
Intramolecular Anti-Markovnikov Hydroamination of Alkenes
1014
Asymmetric Benzidine Rearrangement

Polymer-Supported Synthesis

z1015
All PDFs of this category
1015
Synthesis of 4H-Chromenes with ZnO Nanoparticles in Water
1016
The Suzuki–Miyaura Coupling with Pd NPs Supported on Nafion–Graphene
1017
Asymmetric Nitroaldol Reaction Using a Nd/Na Heterobimetallic Catalyst
1018
Synthesis of Tetrahydro-4H-chromenes Using Nano γ-Fe2O3 in H2O
1019
Alkylation of Indoles with Diazo Esters at the C3 Position Using CuO/SiO2
1020
C–H Arylation of Imidazo[1,2-a]pyridine with Pd-Fe3O4 NPs
1021
Flow Oxidation of Olefins with OsO4 Immobilized on Microreactor
1022
Solid-Phase Synthesis of Inverse Poly(amidoamine) Dendrons
1023
Supported Ionic Liquid-Rh Catalysts for Hydroaminomethylation
1024
N-Arylation of Indoles with Aryl Halides Using MCM-41-2N-CuI
1025
Amberlite IR-120H for Nucleophilic Substitution of Propargylic Alcohols
1026
Pyridines from β-Enaminones Using ZnO Nanoparticles
1027
Friedländer Reaction with a Supported Prolinamide Organocatalyst
1028
Aerobic Oxidation of Alcohols Using SBA-15-TEMPO/FeCl3

Erratum

1029
Fix, A. G.; Deal, P. E .; Vonnegut, C. L.; Rose, B. D.; Zakharov, L. N.; Haley, M. M.: A Novel Electron-Accepting Scaffold for Organic Electronics
1029
Dou, L.; Chen, C.-C.; Yoshimura, K.; Ohya, K.; Chang, W.-H.; Gao, J.; Liu, Y.; Richard, E.; Yang, Y.: A New, Strongly Electron-Donating Building Block for Low-Bandgap Polymers
1030
Dalton, D. M.; Rovis, T.: Rhodium-Catalyzed Enantioselective [2+2+2] Cycloaddition