DOI: 10.1055/s-00000131

Synfacts

Ausgabe 11 · Volume 10 · November 2014 DOI: 10.1055/s-004-27934

Synform

  • A143

    SYNFORM ISSUE 2014/11

    • Synthesis of Natural Products and Potential Drugs

  • z1117

    All PDFs of this category

  • 1117

    Syntheses of (+)-Flabellidine and (–)-Lycodine

  • 1118

    Synthesis of Fibrinolysis Inhibitor AZD6564

  • 1119

    Synthesis of a CETP Inhibitor

  • 1120

    Synthesis of (−)-Methyl Atisenoate and (−)-Isoatisine

  • 1121

    Formal Synthesis of Rosuvastatin and Pitavastatin

  • 1122

    Total Synthesis of Aspeverin

  • 1123

    Synthesis of (–)-Lepistine

  • 1124

    Synthesis of VX-787

  • 1125

    Synthesis of Δ12-Prostaglandin J3

  • 1126

    Total Synthesis of Gymnothelignan N

  • 1127

    Synthesis of (–)-Xanthatin

  • 1128

    Synthesis of SGLT-2 Inhibitor Empagliflozin

  • 1129

    Synthesis of Thrombin Inhibitor AZD8165

    • Synthesis of Heterocycles

  • z1131

    All PDFs of this category

  • 1131

    Spirocyclic and Ring-Expanded Fused Pyrazoles

  • 1132

    Synthesis of Aminotriazoloazepinone-Containing Di- and Tripeptides

  • 1133

    N-Aryl Heterocycles by Catalytic Photoredox Olefin Hydroamination

  • 1134

    Synthesis of the SF5 Analogue of Umemoto Salt

  • 1135

    An Organocatalytic Cascade Route to Functionalized Azepines

  • 1136

    Iron-Catalyzed Synthesis of Difluoromethylsulfonylated Oxindoles

  • 1137

    Quinoxaline N-Oxides by Dehydrogenative N-Incorporation of Imines

  • 1138

    Synthesis of Spiroaminals by Au/Sc Relay Catalysis

  • 1139

    NHC-Promoted Annulation Approach to Pyranyl Aldehydes

  • 1140

    C-8 Alkylation and Alkynylation of Quinoline N-Oxides by Rhodium Catalysis

  • 1141

    Copper-Catalyzed Synthesis of Dibenzodiazepinones

  • 1142

    Copper-Catalyzed Synthesis of Sulfonylated Oxindoles

  • 1143

    Synthesis of Benzotriazoles from 2-(Arylamino)aryliminophosphoranes

  • 1144

    Synthesis of Heterocycles by Palladium-Catalyzed Intramolecular C–H Amination

  • 1145

    Three-Component Reaction Approach to Aminopyrazoles and Iminopyrimidines

    • Synthesis of Materials and Unnatural Products

  • z1147

    All PDFs of this category

  • 1147

    A Starphene is Born: Largest and Most Soluble to Date

  • 1148

    Covalent Cage Construction via Alkyne Metathesis

  • 1149

    Every Cloud Has a Silver(I) or Tetramethylammonium Lining

  • 1150

    Iterative Benzannulation for Rapid Build-up of Congested Aromatic Systems

  • 1151

    Playing Dominoes with Palladium: Synthesis of Biaryl Tertiary Amines

  • 1152

    Rearrange Your Way to Tricyclic Heteroaromatics

  • 1153

    Taming the Wild Terminal Aryl Alkyne for High-Yield Cross-Metathesis

  • 1154

    Complex Polyphenylenes from Bromo-Oligophenylboronic Acids

  • 1155

    Platinum(II)-Catalyzed Synthesis of Substituted Azulenes

  • 1156

    The Road to Rotanes is Paved with Exocyclic Alkenes

  • 1157

    Synthetic Strategy Toward Enantiopure Helicene Quinones

  • 1158

    Nitrogen-Doped Zigzag-Edge Nanographenes

    • Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

  • z1159

    All PDFs of this category

  • 1159

    Mannich–Cyclization Cascade Reaction Catalyzed by Squaramide/AgOAc

  • 1160

    Asymmetric Hydrogenation of Sterically Hindered Enones

  • 1161

    Asymmetric Synthesis of Tetrahydrofurans Bearing Multiple Stereocenters

  • 1162

    Ruthenium-Catalyzed Synthesis of Enantioenriched γ-Substituted Lactones

  • 1163

    Iridium-Mediated Asymmetric Synthesis of Branched Allylic Sulfilimines

  • 1164

    Diastereoselective Cyanation and Trifluoromethylation of Ketimines

  • 1165

    Palladium-Catalyzed Asymmetric Allyl–Aryl Cross-Coupling Using Allylboronates

  • 1166

    Synthesis of (+)-Discodermolide via Borylation

  • 1167

    Asymmetric Hydrogenation of α,β-Unsaturated Nitriles

  • 1168

    Stereoselective Synthesis of cis-4-Aryl-cyclopent-2-en-1-ols

  • 1169

    Enantioselective C–H Addition of Pyridines to Alkenes

  • 1170

    Palladium-Catalyzed Stereoselective Cascade Reaction for a Planar Core Structure

  • 1171

    Rhodium/Phosphoric Acid Co-Catalyzed Asymmetric Csp2–H Functionalization

  • 1172

    Ruthenium-Catalyzed Cylization of Aromatic Nitriles with Alkenes

  • 1173

    Pd/Cu-Catalyzed Alkynylative Ring Opening of Oxabenzonorbornadienes

  • 1174

    Diastereoselective Amination of Alcohols Catalyzed by Ruthenium

  • 1175

    Enantioselective Allyl–Allylsilane Cross-Coupling Catalyzed by Iridium

  • 1176

    Intramolecular Ruthenium-Mediated trans-Selective Silylvinylation of Alkynes

  • 1177

    Rhodium-Catalyzed Cyclopropanation of N-Enoxyphthalimides

  • 1178

    Synergistic Catalysis for Asymmetric Cascade Transformations

  • 1179

    Functionalized Azulenes via Rhodium-Mediated N-Sulfonylaminoalkenylation

  • 1180

    Rhodium-Catalyzed Asymmetric Synthesis of Tetrahydroquinolines

  • 1181

    Chiral Bicyclo[3,2,1]octanes via Domino Reaction

  • 1182

    Asymmetric aza-Henry Reaction Catalyzed by Copper

  • 1183

    Copper-Catalyzed Asymmetric Boron Conjugate Addition in Water

  • 1184

    Palladium-Catalyzed Stereospecific C-3 Arylation of Proline Derivatives

  • 1185

    Rhodium-Catalyzed Enantioselective Carbonyl–Ene Reaction

  • 1186

    Asymmetric Nickel-Catalyzed Synthesis of Spiro[isoxazolin-3,3′-oxindoles]

  • 1187

    Heterobimetallic Rare-Earth–Lithium Complexes for Asymmetric Epoxidations

    • Metal-Mediated Synthesis

  • z1189

    All PDFs of this category

  • 1189

    Synthesis of 2,3-Disubstituted Indoles from Isatins

  • 1190

    γ-Selective Arylation of Zincated Boc-Allylamines

  • 1191

    Ketones from Carbon Dioxide and Organolithium or Grignard Reagents

  • 1192

    Carbolithiation of Chloro-Substituted Alkynes

  • 1193

    Zinc-Catalyzed Synthesis of Aryl Boronates

  • 1194

    Synthesis of Polysubstituted Phenanthridines

  • 1195

    Trifluoromethylthiolation of Alcohols

  • 1196

    Alkoxide-Promoted Deborylative Alkylation of Bis(boronates)

  • 1197

    Indium-Mediated Intramolecular Allenylation of N-tert-Butanesulfinyl Imines

  • 1198

    Copper-Mediated ortho-Nitration of Aromatic Amides

  • 1199

    Cross-Coupling of N-Tosylaziridines with Organozinc Reagents

  • 1200

    Nickel-Catalyzed Difluoroalkylation of Organoboronic Acids

  • 1201

    Cross-Coupling Reactions of Diazo Compounds and Vinylboronic Acids

  • 1202

    Copper(II)-Mediated Ortho C–H Alkynylation

  • 1203

    Asymmetric Arylation of Cyclic N-Sulfonyl Ketimines

    • Organo- and Biocatalysis

  • z1205

    All PDFs of this category

  • 1205

    Organocatalytic Asymmetric Mannich Synthesis of α-Amino Esters

  • 1206

    ω-Transaminase-Catalyzed Reductive Amination of Ketones

  • 1207

    N-Heterocyclic Carbene Catalyzed Formal [3+2] Annulation of Enals

  • 1208

    Kinetic Resolution of Axially Chiral Diols and Amino Alcohols

  • 1209

    Kinetic Resolution of BINOL Derivative Catalyzed by Chiral DMAPs

  • 1210

    Enantioselective Formation of All-Carbon Quaternary Stereocenters

  • 1211

    Biocatalytic Oxidative Desymmetrization of Piperidine Carboxylates

  • 1212

    Disulfonimide-Catalyzed Enantioselective Torgov Cyclization

  • 1213

    Catalytic Asymmetric Synthesis of 4-Nitropyrazolidines

  • 1214

    Asymmetric Synthesis of Pyrrolines Using Bicyclic Phosphine Catalysts

  • 1215

    Enantioselective Route to Piperidines via Covalent Phosphoric Acid Catalysis

  • 1216

    Desymmetrization of 1,3-Diols via Oxidative Cleavage of Benzylidene Acetals

    • Polymer-Supported Synthesis

  • z1217

    All PDFs of this category

  • 1217

    1,3-Addition of Silyl Enol Ethers to Nitrones Using Al-MCM-41

  • 1218

    Allylation of Imines and Aldehydes Using Pd-POMs

  • 1219

    An Organo Porous Polymer Catalyst for Asymmetric Alkylation with Et2Zn

  • 1220

    Selenophenes and Selanyl Selenophenes Using CuO Nanoparticles

  • 1221

    C–C Cross-Couplings Using Triazole Dendrimer Stabilized Pd Nanoparticles

  • 1222

    Co–Pd Magnetic Nanoparticle Catalyst for the Aerobic Oxidation of Alcohols

  • 1223

    Oxidation of Alcohols Using CoFe2O4@APTES@Ni(OH)2

  • 1224

    Direct Glycosylation with Sc(OTf)2-NSMP Catalyst in Water

  • 1225

    Polymer-Incarcerated Gold Nanocluster Catalysts for Oxidation

  • 1226

    Chemoselective Hydrogenation of Chloronitrobenzenes Using Pt/C

  • 1227

    Deoxygenation of Sulfoxides Using Ruthenium Nanoparticles Supported on TiO2

  • 1228

    O-Arylation of Phenols with Aryl Halides Using Cu/Nf–Graphene Nanoribbons

  • 1229

    The Michael Addition of Aldehydes to Nitroalkenes with Carrageenan/MNPs

  • 1230

    Solid-Phase Synthesis of 1,2,3-Triazoles Using 4,4′-Bismethoxybenzhydryl Azide

  • 1231

    C(sp)–C(sp) and C(sp)–C(sp2) Cross-Coupling with CuFe2O4 Nanoparticles