DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 13 · September 2017 DOI: 10.1055/s-007-34626

Synform

A140
Zanda, Matteo: SYNFORM ISSUE 2017/09

Synthesis of Natural Products and Potential Drugs

z0895
All PDFs of this category
0895
Synthesis of (±)-Waihoensene
0896
Synthesis of P4Q-391
0897
Synthesis of Vericiguat
0898
Syntheses of Ovafolinin A and B
0899
Synthesis of (–)-Tubingensin B
0900
Synthesis of a Serine Hydroxymethyltransferase Inhibitor
0901
Total Syntheses of Cheloviolenes A and B and Dendrillolide C
0902
Stille Cross-Coupling Route to HIV NNRTI Doravirine Analogues
0903
Syntheses of (–)-Alotaketal A and (–)-Phorbaketal
0904
Synthesis of (S)-Duloxetine
0905
Total Syntheses of Aspidosperma Alkaloids
0906
Biomimetic Syntheses of (±)-Homodimericin A

Synthesis of Heterocycles

z0907
All PDFs of this category
0907
Catalytic C(sp3)–CF3 Bond Formation
0908
Scalable Synthesis of Haloquinolin-2(1H)-ones and Quinolines
0909
Synthesis of 2-Spiropiperidines by the Aza-Maitland–Japp Reaction
0910
Conversion of Endoperoxides into Furans by the Appel Reaction
0911
Synthesis of Tetrahydropyridines by Enantioselective Cyclization of 1,6-Dienes
0912
Visible Light Assisted Synthesis of Imidazoles by Intramolecular C–H Imination
0913
Synthesis of Isoquinolinones by Amide Umpolung
0914
Copper-Catalyzed Annulation of Tetronic Acids with Azirines: Scope and Mechanism
0915
Chiral Binaphthylsulfonate Cluster Catalyst for Cycloaddition Reaction
0916
Diastereoselective Synthesis of Difluoromethylated Spirooxindoles
0917
Synthesis of Dihydrophenanthridines by Dehydrogenative Coupling
0918
Asymmetric Synthesis of Chiral 3,4-Dihydro-2H-pyrancarbonitriles
0919
One-Pot Synthesis of 1,2-Disubstituted Benzimidazoles
0920
Rhodium(III)-Catalyzed Synthesis of Pyrano[2,3,4-de]-quinolines

Synthesis of Materials and Unnatural Products

z0921
All PDFs of this category
0921
1,3- and 1,4-Benzdiyne Equivalents
0922
Ramping up to Thiophene: Sulfur-Containing Helicenes
0923
Utilizing Cyclopentadiene for the Design of New Polyenyne Motifs
0924
Facile Route to Fused Cyclobutanes
0925
Longer Arms Make It More Optically Active
0926
Catch and Release: Reversible Binding in a pH-Responsive Macrocycle
0927
Switching up the Synthesis of Molecular Switches
0928
Compounds with ABC’s (Electron-Acceptor, Boron, Chromophore)
0929
Bent Porphyrin Tapes Enabled by Seven-Membered Rings
0930
A New Addition to the BN-Phenanthrene Family
0931
π-Extended Antiaromatic Polycyclic Hydrocarbons
0932
Carbon Nanostructures for a 3D World

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0933
All PDFs of this category
0933
Silver-Catalyzed Intramolecular Aziridination
0934
Rhodium-Catalyzed Asymmetric Synthesis of γ-Keto Carboxylic Acids
0935
Enantioselective Palladium-Catalyzed Synthesis of Diarylsulfoxides
0936
Palladium-Catalyzed Reaction of α,α-Dithioacetonitriles with Imines
0937
Asymmetric Copper Hydride Catalyzed Coupling Reaction to Access Chiral Ketones
0938
Enantioselective Hydroamination of Olefins Forming Chiral Aziridines
0939
Iridium-Catalyzed Asymmetric Arylation of Allylic Alcohols with Anilines
0940
Spirocyclic Ketones through a Copper-Catalyzed Arylation-Semipinacol Rearrangement
0941
Asymmetric Dysprosium-Catalyzed [3+2] Cycloaddition Reaction
0942
Asymmetric Synthesis of γ-Alkenyl Butenolides
0943
Asymmetric Nickel-Catalyzed Desymmetrization Reaction
0944
Copper-Catalyzed [2+2] Cycloaddition of Quinones and Fulvenes
0945
Chiral-at-Metal Iridium(III) Nucleophilic Catalyst
0946
Construction of Oxindoles Catalyzed by a Chiral-at-Rhodium Complex
0947
Copper/Borinic Acid-Catalyzed Enantioselective Propargylation of Polyols
0948
Enantioselective Palladium-Catalyzed Diboration Reaction
0949
Cyclopropanation of β,γ-Unsaturated α-Keto Esters with Diazo Esters
0950
Enantioselective Rhodium-Catalyzed Markovnikov Hydroboration of Alkenes
0951
Asymmetric Carbomagnesiation of Cyclopropanes
0952
Palladium-Catalyzed Iminoarylation: Domino Narasaka–Heck/Arene C–H Alkylation
0953
Enantioselective Iridium-Catalyzed Hydro-hydroxymethylation of Trifluoromethyl Allenes
0954
Enantioselective Radical Addition of CX4 to Olefins
0955
Iridium-Catalyzed Enantio- and Diastereoselective Spiroketalization
0956
Asymmetric Protoboration to Form Chiral α-Amino Boronate Esters
0957
Synthesis of Dihydrophenazasilines via an Asymmetric 1,5-Palladium Migration
0958
Stereoselective Synthesis of Aryl Glycines by Ruthenium-Catalyzed Hydrogenation
0959
Copper-Catalyzed 1,2-Addition of gem-Diborylalkanes to Imines
0960
Iridium-Catalyzed Asymmetric Hydrogenation of Cyclic Enones
0961
Copper- and Lewis-Base-Catalyzed Asymmetric Synthesis of Quinolones
0962
Enantioselective Nickel-Catalyzed Mizoroki–Heck Reaction

Metal-Mediated Synthesis

z0963
All PDFs of this category
0963
Bi(OTf)3-Mediated Olefinic Cyclization
0964
Palladium-Catalyzed Desulfonative Coupling
0965
Nickel-Catalyzed Reductive Cross-Coupling
0966
Diastereoselective α-Arylation of Cyclic Nitriles
0967
Enantioselective Synthesis of Homopropargyl Alcohols
0968
Selective Addition of Allylboron Compounds to Fluoroalkyl Ketones
0969
Suzuki–Miyaura Cross-Coupling of N-Acylpyrroles and -Pyrazoles
0970
Allene Synthesis by Decomposition of Alkynyl N-Nosylhydrazones
0971
An 3-Aryl H8-BINOL Ligand for the Alkylation and Arylation of Aldehydes
0972
Borylative Cyclization of In Situ Generated o-Allenylaryl Nitriles
0973
Three-Component Coupling between Alkynes, Iodoarenes, and Bis(iodozincio)methane
0974
Gold-Catalyzed Alkylsulfonylation of Boronic Acids
0975
Utilizing Flow Conditions for the Production of Grignard Reagents
0976
ortho-Selective C–H Borylation of 2-Phenylpyridines
0977
Addition Reactions of Organomagnesium Halides

Organo- and Biocatalysis

z0979
All PDFs of this category
0979
Enzyme-Catalyzed Enantioselective Reductive Amination
0980
Enantioselective Aza-pinacol Rearrangement of Indoles
0981
Directed Evolution toward an Iron-Heme Enzyme for Asymmetric C–H Amination
0982
Enzymatic Friedel–Crafts Acylation and Fries Rearrangement
0983
Enantioselective Photocatalytic α-Alkylation of Aldehydes
0984
Asymmetric α-Fluorination of α-Branched Enals
0985
Catalyst-Controlled Diastereoselectivity Switch in Conjugate Additions
0986
Enantioselective Diels–Alder Cycloaddition to Construct Carbazolespirooxindoles
0987
Organo- and Biocatalytic Sequential Transformation of Alcohols into Amines
0988
Enantioselective Conjugate Additions of Indoles Catalyzed by Fiaud’s Acid

Polymer-Supported Synthesis

z0989
All PDFs of this category
0989
Parallel Carbonylation and Decarbonylative Heck Reaction on Palladium/Carbon
0990
Metal–Organic Frameworks as Multifunctional Heterogeneous Asymmetric Catalysts
0991
N-Arylation of Anilines and Imidazoles on Copper(II) Oxide Nanoparticles
0992
Palladium Nanocatalysts for Aryl Halogenation and Cross-Coupling Reactions
0993
Hydrogenation of Alkynes and Alkenes on Silica-Supported Palladium Nanoparticles
0994
Controlled Hydrogenation of Alkynes on Photogenerated Palladium Nanoparticles
0995
Hydrogenation with Ruthenium Nanoparticles in Ionic Liquids
0996
Dehydrogenative Imine Transformations on a Platinum/Titania Catalyst
0997
A Polymeric Pyridine–Zinc Catalyst for Synthesis of Cyclic Carbonates
0998
Synthesis of 2,2-Diphenylethanol Derivatives from Aromatic Aldehydes
0999
Enantioselective Tandem Hydrogenation/Coupling on a Palladium–Ruthenium Catalyst
1000
Continuous-Flow Palladium/Carbon-Catalyzed Fujiwara–Moritani Reaction
1001
Indium-Catalyzed Oxidative Amination of 2-Aminopyridines
1002
One-Pot Synthesis of Tetrahydropyridines on Graphene Oxide
1003
Photocatalytic Oxidation with Carbon-Nanodot-Doped Carbon Nitride
1004
Diazotation of o-Phenylenediamines on Montmorillonite K-10