DOI: 10.1055/s-00000131

Synfacts

Issue 11 · Volume 15 · November 2019 DOI: 10.1055/s-009-44705

Synform

  • A162

    SYNFORM ISSUE 2019/11

    • Synthesis of Natural Products and Potential Drugs

  • z1215

    All PDFs of this category

  • 1215

    Nanomolar Inhibitor of Trypanosoma brucei Trypanothione Reductase

  • 1216

    Total Synthesis of (±)-Atlanticone C

  • 1217

    Total Synthesis of Illisimonin A

  • 1218

    Artificial Intelligence Guides the Synthesis of SCH 47949

  • 1219

    Synthesis of the Immunosuppressant FR252921

  • 1220

    Synthesis of GSK2798745

  • 1221

    Synthesis of (±)-Rhabdastrellic Acid A

  • 1222

    Total Synthesis of (–)-Himeradine A

  • 1223

    Synthesis of (+)-Jungermatrobrunin A

  • 1224

    Synthesis of Antibacterial LpxC Inhibitors

  • 1225

    Synthesis of Esketamine

  • 1226

    Synthesis of (±)-Isocomene

  • 1227

    Synthesis of Omecamtiv Mecarbil

    • Synthesis of Heterocycles

  • z1229

    All PDFs of this category

  • 1229

    Copper-Catalyzed Synthesis of Di(het)arylamines

  • 1230

    Synthesis of Enaminones and Thiazoles Using Iodonium Ylides as Carbene Equivalents

  • 1231

    Cooperative Catalysis for the Asymmetric Synthesis of Piperidines

  • 1232

    Selective C-2 Directed-Carbonylation of Indoles and Pyrroles

  • 1233

    Synthesis of Substituted Morpholines by Fragmentation of Tetrazoles

  • 1234

    Rhodium-Catalyzed Synthesis of 2‑Arylindoles from N‑Aryl-2-aminopyridines

  • 1235

    Synthesis of Benzazepinones Involving an Unexpected Intramolecular Cyclization

  • 1236

    Electrocatalytic Synthesis of Imidazo[1,5-a]quinoline-3-carbonitriles

  • 1237

    Asymmetric Radical C–H Amination for the Synthesis of Azoles

  • 1238

    Three-Component Assembly of 3,4-Dihydroquinazolines

  • 1239

    Synthesis of Phosphinolines and Phosphepines

  • 1240

    Buchwald–Hartwig Coupling of Piperidines with Hetaryl Bromides

  • 1241

    Synthesis of 3-Phenylimidazo[1,2-a]pyridines by Annulation of Tetrazoles with Phenylacetylenes

  • 1242

    Copper-Catalyzed Cyclization of Enaminones to Polycyclic N-Fused Indoles

  • 1243

    An Illuminating Synthesis of Benzimidazoles

    • Synthesis of Materials and Unnatural Products

  • z1245

    All PDFs of this category

  • 1245

    Developing a Dye for Lysosome

  • 1246

    Synthesis of a π-Conjugated Macrocyclic Oligofuran: The First of Many to Come

  • 1247

    peri-Disubstituted Naphthalimides via Decarboxylative Arylation

  • 1248

    Finally, Furfural Flourishes

  • 1249

    Unmasked ‘Click Chemistry’

  • 1250

    Proton Hole-in-One With TriQuinoline

  • 1251

    Synthesis of Carbon-Skeleton-Like Molecules

  • 1252

    Going Full Circle: From Linear to Cyclic pH-Responsive Water-Soluble Cyclic Polymer

  • 1253

    Aryl Sulfones and Aryl Boronic Acids Make a Nice Couple

  • 1254

    Ring-Opening Doors to Controlled Polymerization with Hydrogen-Bond-Driven Organocatalysis

  • 1255

    Stepwise Synthesis of an Axially Chiral 1,1′-Biazulene and its π-Extended Derivative

  • 1256

    Synthesis of Sumanene

    • Metals in Synthesis

  • z1257

    All PDFs of this category

  • 1257

    Palladium-Catalyzed Synthesis of Carboxylic Acids

  • 1258

    Copper-Mediated Trifluoromethylation of Aryl Sulfonium Salts

  • 1259

    Asymmetric C–H Alkylation of Fluoroarenes with Alkenes via Nickel/NHC Catalysis

  • 1260

    C–H Acetoxylation of Carboxylic Acids

  • 1261

    Reductive Dicarbofunctionalization of Alkenes

  • 1262

    Zinc-Catalyzed Tandem Asymmetric Friedel–Crafts Alkylation/Michael Addition

  • 1263

    Hydroalkylation of Terminal Alkynes with Primary or Secondary Alkyl Iodides

  • 1264

    Synthesis of 2-Arylquinazolines via Visible-Light-Induced Benzylic C–H Functionalization

  • 1265

    Enantioselective Allylic Substitution with Nucleophiles in Aqueous Solution under Iridium Catalysis

  • 1266

    Catalytic Interrupted Click/Acylation Reactions

  • 1267

    Enantioselective Preparation of Chiral Diamines

  • 1268

    Base-Catalyzed Synthesis of Fully Substituted Silyl Enol Ethers

  • 1269

    Photoredox/Nickel-Catalyzed C(sp3)–C(sp3) Cross-Coupling

  • 1270

    Anti-Markovnikov Hydroamination and Hydroamidation of Allylic Alcohols through Iron Catalysis

  • 1271

    Rhodium(III)-Catalyzed C–H Activation/Carbene Insertion/Lossen Rearrangement Sequence

  • 1272

    Nickel-Catalyzed Asymmetric Reductive Heck Cyclization

  • 1273

    Heteroaryl Thioether Directing Group in Oxidative Heck and C–H Functionalization Reactions

  • 1274

    Enantioselective Benzylic Arylations

  • 1275

    Photoreduction of Arenes and Heteroarenes

  • 1276

    Decarbonylative Suzuki–Couplings of Amides

  • 1277

    Ruthenium-Catalyzed Cross-Coupling of Anilines

  • 1278

    Enantioselective Access to Tetrahydroquinoxalines through Relay Epoxide Opening/Amination of Alcohols

  • 1279

    Photocatalysis: Asymmetric Intramolecular HAT in Photoexcited Catalyst–Substrate Complex

  • 1280

    β-C(sp3)-Methylation of Alcohols

  • 1281

    Preparation of β-Aminoboronates

  • 1282

    Copper-Catalyzed Asymmetric Annulation of Carbenes to Access Enantioenriched 2,3-Dihydrobenzofurans

  • 1283

    Palladium-Catalyzed C(sp3)–H Bond Activation of Phenylacetaldehydes

  • 1284

    Palladium-Catalyzed Aerobic Oxidative C-H Arylation

  • 1285

    The Hiyama–Denmark Cross-Coupling

    • Polymer-Supported Synthesis

  • z1287

    All PDFs of this category

  • 1287

    Zeolitic Imidazole Framework Encapsulated Copper Nanoparticles for Hydrogenation of Aldehydes

  • 1288

    Transfer Hydrogenation of Unsaturated Compounds by Co NPs Encapsulated in N-doped Graphene

  • 1289

    Copper-Catalyzed Oxidative Cyclization of Benzylamines with 1,3-Dicarbonyl Compounds

  • 1290

    Controlled Reduction of Nitroarenes to Azo Compounds with Iron–Nitrogen Co-Doped Mesoporous Carbon

  • 1291

    Rh-Catalyzed Asymmetric Arylation of α,β-Unsaturated Carbonyl Compounds, Nitroalkenes, or Imines

  • 1292

    Hybrid Palladium Catalyst for Suzuki–Miyaura and Heck Reactions

  • 1293

    Selective Deprotection of Benzyl Carbamates on Micellar Nickel–Palladium Nanoparticles in Water

  • 1294

    Ruthenium-Photocatalyzed Aerobic Oxidation of Benzylic Halides and Cyclization of Tertiary Anilines

  • 1295

    One-Pot Synthesis of 5-Substituted 1H-Tetrazoles on a Silica-Coated Fe3O4-Supported Copper(II) Complex

  • 1296

    Oxidative Synthesis of Nitriles from Primary Alcohols and Ammonia Catalyzed by Cobalt Nanoparticles

  • 1297

    Synthesis of Xanthene Derivatives by Using a Lewis Acidic Ionic Liquid Immobilized on Perlite NPs

  • 1298

    Cerium(IV) Oxide-Catalyzed Direct Phenolysis of Amides

    • Organo- and Biocatalysis

  • z1299

    All PDFs of this category

  • 1299

    A Newly Designed Catalyst for Additive-Free Mitsunobu Reactions

  • 1300

    Brønsted Acid Catalyzed Asymmetric House–Meinwald Rearrangement of p-Hydroxyphenyl Epoxides

  • 1301

    Asymmetric Functionalization of C(sp3)–H Bonds in 2-Alkylindoles

  • 1302

    NHC-Catalyzed Carboacylation of Alkenes

  • 1303

    Lewis Base Catalyzed Enantioselective Sulfenoamination of Olefins

  • 1304

    Asymmetric NHC-Catalyzed Rauhut–Currier Reaction of Weakly Electrophilic Bisenoates

  • 1305

    Phosphenium Ion Catalyzed Enantioselective Reduction of Cyclic Imines

  • 1306

    Asymmetric Phosphoric Acid Catalyzed Multi-Component Synthesis of Axially Chiral N-Arylindoles

  • 1307

    N-Heterocyclic Carbene Catalyzed Stetter Reaction of Cyclic Enones

  • 1308

    Organometallic Organocatalysts

    • Chemistry in Medicine and Biology

  • z1309

    All PDFs of this category

  • 1309

    Water-Soluble BODIPY Dyes for Voltage Imaging

  • 1310

    Pre-Exposure Prophylaxis (PrEP)

  • 1311

    Sign-Inversion in Photopharmacology

  • 1312

    HPLC-Free Synthesis of Nucleoside Triphosphates

  • 1313

    Targetable, Bright Small-Molecule Ca2+ Indicators

  • 1314

    Macrocycle Library Synthesis through Thiol-to-Amine Cyclization

  • 1315

    Membrane Probes for Super-Resolution Imaging of Plasma Membranes

  • 1316

    Activatable Photosensitizers for Photodynamic Therapy

  • 1317

    C–N Coupling of Aryl Thianthrenium Salts

  • 1318

    An Aromatic Brønsted Acid Catalyst for the Direct Glycosylation of Amides

  • 1319

    pH-Sensitive μ Opioid Receptor Agonists

  • 1320

    Conformational Restricted Cyclopropanated Nucleoside Derivatives

  • 1321

    SPiDER-Killer-βGal: A Photosensitizer for Targeted Cell Ablation with Single-Cell Resolution

    • Peptide Chemistry

  • z1323

    All PDFs of this category

  • 1323

    Synthesis of Cyclic and Bicyclic Peptides

  • 1324

    Palladium-Catalyzed Conversion of Phenyl Aspartates into Ketones

  • 1325

    Ruthenium-Catalyzed C–H Alkylation of Resin-Attached Tryptophan

  • 1326

    Asymmetric Hydrogenation of β-Aminoacrylates to β-Amino Acid Derivatives

  • 1327

    Palladium-Catalyzed Acylation of Phenylalanine-Containing Peptides

  • 1328

    Palladium-Catalyzed Arylation of Sulfonamide-Containing Peptides

  • 1329

    Synthesis of Diazirines from Amino Acids by Using Phenyliodonium Diacetate

  • 1330

    Synthesis of Dehydroamino Acid Containing Peptides

  • 1331

    Synthesis of Benzotriazole-Derived α-Amino Acids

  • 1332

    Synthesis of Activated Amides and Directed C(sp3)–H Arylation

  • 1333

    Peptide Nanoassemblies Promote Enantioselective Hydrogenation

    • Flow Chemistry

  • z1335

    All PDFs of this category

  • 1335

    Continuous Flow Electrochemical Oxidation of Alcohols

  • 1336

    Functionalized Alkyllithium Reagents Towards Heterotelechelic Polymers

  • 1337

    Radical-Based Late-Stage C−H 18F-Difluoromethylation of N-Heteroaromatics

  • 1338

    Organocatalyzed Photooxygenation of β-Dicarbonyl Compounds in Flow Photomicroreactors

  • 1339

    One-Step Synthesis of 2-Fluoroadenine in a Continuous Flow Operation