DOI: 10.1055/s-00000131

Synfacts

Issue 05 · Volume 16 · May 2020 DOI: 10.1055/s-010-47716

Synform

  • A66

    SYNFORM ISSUE 2020/05

    • Synthesis of Natural Products and Potential Drugs

  • z0493

    All PDFs of this category

  • 0493

    Synthesis of (–)-Canataxpropellane

  • 0494

    Total Synthesis of (–)-Stypodiol

  • 0495

    Synthesis of BACE1 Inhibitor LY3202626

  • 0496

    Synthesis of Balovaptan

  • 0497

    Synthesis of Glacaprevir by Ring-Closing Metathesis

  • 0498

    Synthesis of (–)-Farnesin

  • 0499

    Synthesis of (–)-Rhodomollanol A

  • 0500

    Synthesis of (–)-Cannabidiol

  • 0501

    Synthesis of Tryptophan Hydroxylase Inhibitor LX1031

  • 0502

    Synthesis of an Allosteric HIV-1 Integrase Inhibitor

  • 0503

    Total Synthesis of (–)-Rauwolscine Enabled Through NHC Catalysis

  • 0504

    Synthesis of Olutasidenib

  • 0505

    Synthesis of (–)-Batrachotoxinin A

  • 0506

    Total Synthesis of Isochrysohermidin

    • Synthesis of Heterocycles

  • z0507

    All PDFs of this category

  • 0507

    SNAr Reaction of Aminooxetanes with Quinazolines: Synthesis of Imidazo[1,2-c]quinazolines

  • 0508

    Synthesis of Five-Membered Heterocycles by H3PO2-Catalyzed Cyclization of Stereodefined Alcohols

  • 0509

    Pyrylium Reagent for the Radical C–N Borylation of Aromatic Amines

  • 0510

    Iridium-Catalyzed Synthesis of Fused Isoquinolines

  • 0511

    Photochemical Electrocyclization Synthesis of Azaanthraquinones

  • 0512

    AuCl3-Catalyzed Synthesis of Cyclopentenes, Polycycles, Benzocarbocycles, and N-Heterocycles

  • 0513

    Copper(I) Chloride-Catalyzed Synthesis of Benzo[4,5]thieno[2,3‑d]thiazoles

  • 0514

    Enantioselective Synthesis of Functionalized 1,3-Thiazin-4-ones

  • 0515

    Synthesis of 1,2,4-Thiadiazoles and Fused Analogues by Electrochemical S–N Bond Formation

  • 0516

    Synthesis of Ethyl 3-Fluoro-1-Pyrrole-2-Carboxylate

  • 0517

    Synthesis of Spiropyrazoline Oxindoles and Spiropyrazoline Indanones

  • 0518

    Phosphorus-free Reagent for the Chlorination of Aza-Arenes

  • 0519

    Dirhodium(II)-Catalyzed C(sp2)–H Azidation for the Synthesis of Azidobenzaldehydes

  • 0520

    Three-Component Synthesis of Morpholine Derivatives

  • 0521

    Copper-Mediated Synthesis of N-Arylpyrazoles from Cyclopropanols and Aryl Diazonium Salts

    • Synthesis of Materials and Unnatural Products

  • z0523

    All PDFs of this category

  • 0523

    Propeller-Like Fluorescent Dyes

  • 0524

    Efficient Route to Alkynylated PHAs and Derived Macrocycles

  • 0525

    Activated Amides Yield a Facile Synthesis of Chalcogenide Esters

  • 0526

    Clipping Fullerene

  • 0527

    Leggo My Lego-cycles

  • 0528

    Tightening the Belt[n]arenes

  • 0529

    Sulfoxide, Give You the Coupling

  • 0530

    Triptycene Chirality as Easy as 2+2+2

  • 0531

    Ynamide Umpolung Palooza

  • 0532

    A Mild Way to Synthesize Triarylmethanes

  • 0533

    It Takes Three Electrons to Tango

  • 0534

    Fluoride-Ion-Catalyzed Synthesis of Ladder-Type Benzobisbenzofurans

    • Metals in Synthesis

  • z0535

    All PDFs of this category

  • 0535

    Ruthenium-Catalyzed Lemieux–Johnson-Type Oxidation of Olefins

  • 0536

    Nickel-Catalyzed Bis-Alkyl Electrophile Cross-Coupling for the Synthesis of Alkylcyclopropanes

  • 0537

    Nickel-Catalyzed anti-Markovnikov Hydroarylation of Unactivated Alkenes

  • 0538

    1,2-Difunctionalization of Unsaturated Amides Using Manganese Catalysis to Form C–C Bonds

  • 0539

    Remote Nickel/Photocatalyzed Arylation via a C–C Bond Cleavage of Cyclic Alcohols

  • 0540

    Palladium-Catalyzed C–H Alkenylation of Aryl Ethers

  • 0541

    Reductive Difunctionalization of Aryl Alkenes

  • 0542

    Rhodium-Catalyzed [2+2+2] Cycloaddition Forming Substituted Fluorenones

  • 0543

    Synthesis of Biaryl Ketones via Oxidative Coupling of Unactivated Arenes and Carbon Monoxide

  • 0544

    Preparation of Alkynylated and Alkylated Alkenes

  • 0545

    α-Oxidation of Carboxylic Acids

  • 0546

    Zinc-Catalyzed Enantio- and Diastereoselective Double Mannich Reaction

  • 0547

    Enantioselective Conjunctive Cross-Coupling Strategy for the Formation of anti-1,2-Dimetalloid Compounds

  • 0548

    Enantioselective α-Aminoketone Synthesis by Rhodium Indium Dual Catalysis

  • 0549

    Nickel-Catalyzed Ester Transfer to Aromatic Halides Using Phenyl Nicotinate

  • 0550

    Ruthenium(II)-Catalyzed Amination of Aryl Fluorides via η6-Coordination

  • 0551

    Regio- and Stereoselective Copper-Catalyzed Addition of γ,γ-Disubstituted Allyldiborons to Ketones

  • 0552

    Catalytic Acceptorless Dehydrogenation of Aliphatic Alcohols

  • 0553

    Bismacycles for the Selective C–H Arylation of Phenols and Naphthols

  • 0554

    Stereoselective Copper-Catalyzed Michael Reaction of 2,3-Dioxopyrrolidines with Nitroalkanes

  • 0555

    Reductive Amination of Ketones and Aldehydes Catalyzed by Cobalt Nanoparticles

  • 0556

    Iron-Catalyzed Difunctionalization of Vinyl Cyclopropanes

  • 0557

    Nickel-Catalyzed Hydrodefluorination of CF3-Substituted Alkenes

  • 0558

    Iridium-Based Visible-Light Photoredox Catalyst for Radical Alkylation

  • 0559

    Palladium-Catalyzed meta-Selective C–H Functionalization of Aryl Boronate Esters

  • 0560

    Preparation of anti-α-Amino Acids

  • 0561

    Reductive Vinylation of Tertiary Alkyl Oxalates

  • 0562

    Copper(I)-Catalyzed Oxidation of Aryl Olefins

  • 0563

    Grubbs Catalyst 2nd Generation: Synthesis and Activity of Ruthenium-Based Olefin Metathesis Catalysts

    • Polymer-Supported Synthesis

  • z0565

    All PDFs of this category

  • 0565

    Ring-Opening Hydroboration of Epoxides Catalyzed by a Silica-Supported Organolanthanum Complex

  • 0566

    Synthesis of 3-Ketopyridines on Titania-Immobilized Gold Nanoparticles

  • 0567

    Synthesis of 2-Arylbenzoxazinones on a Mesoporous Silica-Supported Palladium Catalyst

  • 0568

    Synthesis of ortho-Substituted Phenols from Cyclohexanones and Primary Alcohols

  • 0569

    Microwave-Assisted Synthesis of Xanthones Catalyzed by Palladium NPs Supported on Biochar

  • 0570

    Cross-Dehydrogenative Coupling of Alkyne and Thiols Catalyzed by Ni2P NPs on N,P-Codoped Carbon

  • 0571

    Visible-Light-Induced Hydroxyarylation of Alkenes with Aryl Diazonium Salts Using mpg-C3N4

  • 0572

    Pd NPs Immobilized on Silica-Coated Fe3O4 for C–C/C–O Coupling Reactions in Water

  • 0573

    Suzuki–Miyaura Reaction in Water Catalyzed by Covalent Organic Framework-Supported Pd NPs

  • 0574

    Domino Intramolecular Heck/Intermolecular Sonogashira Reactions Catalyzed by Palladium NPs

  • 0575

    C–H Sulfonylation of Enamides with Sodium Sulfinates Catalyzed by a Ruthenium Photocatalyst

  • 0576

    Aerobic Oxidation of Alcohols on a Gold Catalyst Supported on Ionic Liquid-Bridged Mesoporous Silica

  • 0577

    Reduction of Nitroarenes and Oxidation of Ethylbenzene on an N,S-Co-Doped Carbon Catalyst

    • Organo- and Biocatalysis

  • z0579

    All PDFs of this category

  • 0579

    Protonation by a Selenourea–Thiourea Catalyst Permits Highly Enantioselective Aza-Michael Additions

  • 0580

    Ureates as Chiral Strong Brønsted Base Catalysts

  • 0581

    Atroposelective Enzymatic Synthesis of Cyclophanes

  • 0582

    Organocatalytic Aziridination of Isolated Double Bonds

  • 0583

    Anionic Nucleophilic Dithiocarbamate Catalyst Permits α-Alkylation of Carbonyl Compounds

  • 0584

    Photoenolization/Diels–Alder Reaction of Aroyl Fluorides Catalyzed by N-Heterocyclic Carbenes

  • 0585

    Photoredox-Catalyzed Arene C–H Alkylation: No Need for Superstoichiometric Amounts of Substrate

  • 0586

    Enantioselective Redox-Divergent Diels–Alder Reaction of Quinones with Diene Carbamates

  • 0587

    Bisthiourea Organocatalysts Permit Stereospecific O-Furanosylations

    • Chemistry in Medicine and Biology

  • z0589

    All PDFs of this category

  • 0589

    Reversible Spatiotemporal Control of Induced Protein Degradation by Bistable PhotoPROTACs

  • 0590

    Salinipostin A Probe Identifies Potential Antimalarial Protein Targets

  • 0591

    PHOTACs Enable Optical Control of Protein Degradation

  • 0592

    Water-Soluble Benzene Mimetics

  • 0593

    Engelhardt’s Deoxofluorination 60 Years Later

  • 0594

    Introducing Phosphatase-Recruiting Chimeras

  • 0595

    Poppin’ Open Propellanes

  • 0596

    Late-Stage Epoxidation of Geldanamycin with Peptide-Based Organocatalysts

  • 0597

    Natural-Product-Inspired Covalent Telomerase Inhibitors

  • 0598

    Catching Cathepsin X in the Act

  • 0599

    How to Repurpose Sanger’s Reagent as a Photocage

  • 0600

    Sulfo-Click Conjugation

  • 0601

    Synthesis of Photo-Caged ATP

  • 0602

    cGAS/STING Antagonist Discovered in Butenolide Dimer Library

    • Peptide Chemistry

  • z0603

    All PDFs of this category

  • 0603

    Cooperative Catalysis in Amination of β-Hydroxy Carboxylic Acid Esters

  • 0604

    Stereoselective Synthesis of N-Allyl Amino Acids by Using Palladium Catalysts

  • 0605

    Zinc-Catalyzed Peptide Synthesis by Using a Nicotinate-Directed Protocol

  • 0606

    Site-Selective Modification of Selenocystine Peptides

  • 0607

    Lewis Acid Catalyzed Synthesis of α-Amino Acid Derivatives

  • 0608

    Nickel-Catalyzed Asymmetric Hydrogenation To Afford α-Amino Acid Derivatives

  • 0609

    Copper-Catalyzed Functionalization of Tryptophan-Containing Peptides

  • 0610

    Synthesis of 3,4-Dihydro-2H-naphtho-1,4-oxazin-2-ones from Amino Acids

  • 0611

    Rhodium(III)-Catalyzed C-2 Alkenylation of Tryptophan and Tryptophan-Containing Peptides

  • 0612

    Nickel-Catalyzed Synthesis of γ-Amino Acid Derivatives

  • 0613

    Organophotocatalytic Synthesis of α-Deuterated α-Amino Acids

  • 0614

    Acridine–Peptide Conjugates by Solid-Phase Synthesis

    • Flow Chemistry

  • z0615

    All PDFs of this category

  • 0615

    Metallaphotoredox Cross-Coupling of Drug-Like Aryl Halides with Bicyclo[1.1.1]pentane Trifluoroborate Salts