DOI: 10.1055/s-00000083

Synlett

Issue 05 · Volume 33 · March 2022 DOI: 10.1055/s-012-53050

table of contents

synpacts

account

415
Bols, Mikael; Frihed, Tobias Gylling; Pedersen, Martin Jæger; Pedersen, Christian Marcus: Silylated Sugars – Synthesis and Properties
https://www.thieme-connect.de/media/synlett/202205/i_a0353_ga_10-1055_s-0040-1719854.gif

cluster

Design and Chemical Synthesis of Antivirals

458
Fischer, Christian; Vepřek, Nynke A.; Peitsinis, Zisis; Rühmann, Klaus-Peter; Yang, Chao; Spradlin, Jessica N.; Dovala, Dustin; Nomura, Daniel K.; Zhang, Yingkai; Trauner, Dirk: De novo Design of SARS-CoV-2 Main Protease Inhibitors
https://www.thieme-connect.de/media/synlett/202205/i_b0252_ga_10-1055_a-1582-0243.gif
464
Hung, Kevin; Liu, Yugang; Simon, Oliver; Zhang, Lei; Lu, Peichao; Yeung, Bryan K. S.; Sarko, Christopher; Yokokawa, Fumiaki: Synthesis of a Potent Pan-Serotype Dengue Virus Inhibitor Having a Tetrahydrothienopyridine Core
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letter

468
Hosseini, S. Sina; Abdi, Aida; Nikbakht, Ali; Bijanzadeh, Hamid Reza; Rominger, Frank; Werz, Daniel B.; Balalaie, Saeed: Hydrothiolation of Donor–Acceptor Cyclopropanes through Er(OTf)3-Promoted Three-Component Ring-Opening Reaction
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473
Abronina, Polina I.; Malysheva, Nelly N.; Zinin, Alexander I.; Karpenko, Maxim Y.; Kolotyrkina, Natalya G.; Kononov, Leonid O.: Trifluoroacetic Acid Promoted Ring Contraction in 2,3-Di-O-silylated O-Galactopyranosides and Hemiacetals
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478
Liu, Yang; Zhao, Ziyang; Hu, Chao; Zhao, Chuanfang; Liu, Jun; Du, Yuguo: Chiron Approach for the Total Synthesis of Brevipolide M
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495

addendum

502
Zhong, Zhuliang; Lyu, Mao-Yun; Ma, Hao-Ran; Wong, Henry N. C.; Peng, Xiao-Shui: Pivotal Reactions in the Creation of the Polycyclic Skeleton of Cryptotrione