Synfacts

Issue 11 · November 2022

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SYNFORM ISSUE 2022/11 FREE ACCESS

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Synthesis of Natural Products
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1167
Synthesis of (–)-10-Deoxydaphnipaxianine A, (+)-Daphlongamine E and (+)-Calyciphylline R

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1168
Total Synthesis of Indole Alkaloid (+)-Alstonlarsine A

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1169
Total Synthesis of the Grayanoid (+)-Mollanol A FREE ACCESS

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1170
Synthesis of (+)-Mutilin

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1171
Total Syntheses of (–)-Napelline

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1172
Total Synthesis of (+)-Aberrarone

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1173
Total Synthesis of (–)-Ircinol A, (+)-Ircinal A FREE ACCESS

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Synthesis of Heterocycles
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1175
Selective N2-Alkylation of 1H-Azaindazoles

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1176
Synthesis of 6-Phenanthridines by Photocatalytic Deoxygenation of Alcohols

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1177
Synthesis of Versatile Enantiopure Morpholine Fragments from Chiral-Pool Starting Materials FREE ACCESS

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1178
Multicomponent-Reaction-Triggered Cascade Approach to Functionalized Fused 2,6-Diketopiperazines

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1179
Design and Synthesis of Azaborine-Based Steroid Mimics

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1180
Silver-Catalyzed Synthesis of Densely Functionalized gem-Difluorinated Molecules

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1181
Mechanistic Insights into Light-Mediated C–H Functionalization of 2-Phenylpyridines

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1182
Furans by Rhodium-Catalyzed Tandem Cyclization of Acrylic Acids

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1183
Microwave-Assisted Synthesis of Tertiary Amines from Carbamates

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1184
Synthesis of Spiro[furan-2,1′-isoindolin]-3′-ones by Intramolecular Sequential Prins and Ritter Reactions

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1185
Nickel-Mediated C(sp²)–C(sp³) Cross-Couplings

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Synthesis of Materials and Unnatural Products
z1187
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1187
Transition-Metal Catalyzed Chain-Growth Conjugated Polymers

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1188
Bisurea-Functionalized Tetraazaperylene

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1189
Traceless Template for All-benzene Catenane FREE ACCESS

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1190
Expanded Radialenes and Their Aromatic Dianions

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1191
Silver and Gold Go Hand in Hand

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1192
Metathesis of Electron-Deficient Alkenes

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1193
Biomimetic Synthesis of Benzothiophene Sulfoxides

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1194
Acenes Fused with Azulene

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1195
Highly Strained Naphthalenonaphthalenophane

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1196
Ring-Fused Hexameric Perylene Diimide

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1197
Ester Exchange as Pivot to Block Polyolefins

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1198
A Triplet Ground State Kekulé Hydrocarbon

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Metals in Synthesis
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1199
Palladium-Catalyzed Butafulvene Synthesis FREE ACCESS

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1200
Iridium-Catalyzed Enantioselective and Diastereodivergent Propargylic C(sp³)–H Allylation

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1201
1,1-Difunctionalization of Terminal Alkenes to Chiral Allylboronates under Nickel Catalysis FREE ACCESS

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1202
Enantioselective Synthesis of gem-Diarylmethylsilanes via a Three-Component Coupling Reaction

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1203
Accessing Cyclopropenium Cations via a Rh-Catalyzed Oxidative [2+1] Reaction

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1204
Copper-Catalyzed Vinylogous and Bisvinylogous Asymmetric Propargylic Substitution

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1205
Stereodivergent Cross-Coupling of Aryl Halides with Redox-Active Imines

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1206
Enantioconvergent Benzylic C–H Azidation of Indolines Enabled by a Cationic Manganese Salen Catalyst

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1207
Palladium-Catalyzed Diolefination/Cyclization Reaction of o-Toluidine with Acrylates

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1208
Synthesis of Isocytosine Analogues via Palladium-Catalyzed Ring-Opening/Arylation/Cyclization Cascade

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1209
Copper(I)-Catalyzed Kinugasa/C–C Coupling Domino Reaction Towards Spirocyclic Oxindoles

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1210
Turning Aliphatic Carboxylic Acids into Fluorides under Iron Catalysis and Visible Light

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1211
Pd-Catalyzed Synthesis of Diaryl Difluoromethanes from Aryl Halides and Aryldifluoromethyl Trimethylsilanes

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1212
Palladium-Catalyzed Cross-Coupling of Silicon-Masked Diazenyl Anions and (Hetero)Aryl Halides

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1213
Cu-Catalyzed Borylallylation of in situ Generated Imines – Lewis Base Additive Prevents Direct C–N Coupling

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1214
Photoinduced Ring Opening of Cycloalkanols under Dual Organophotoredox and Copper Catalysis

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1215
Nickel-Catalyzed Dearomative Arylcyanation of Indoles

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1216
Palladium-Catalyzed, Directing Group-Enabled Perfluoroselenolation of Vinylic C–H Bonds

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1217
Let’s Do The Twist: Atroposelective Suzuki–Miyaura Cross-Coupling to Access Axially Chiral Biphenols

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1218
Nickel-Catalyzed Enantioselective Tandem Aza-Heck Cyclization and Cross-Coupling with Alkyl Iodides

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1219
Modular Palladium-Catalyzed Synthesis of Highly Conjugated Benzophosphole Derivatives

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1220
A Bench-Stable Bismuth(III) Precursor Promotes theα-Arylation of 1,3-Diketones with Arylboronic Acids

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1221
The Hirao Reaction: Palladium-Catalyzed Cross-Coupling of Dialkyl Phosphites with Aryl Halides FREE ACCESS

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1222
Copper-Catalyzed Conjugate Borylation of Enones FREE ACCESS

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Polymer-Supported Synthesis
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1223
Aerobic Oxidation of Alcohols and Sulfides on Todorokite-Type Manganese Oxide Nanoparticles

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1224
Michael Addition of Aldehydes to Nitrostyrenes on a Tetrahydropyran-Based Dipeptide Catalyst

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1225
Amination and Trifluoroethylation of Fullerenes Promoted by Subphthalocyanine Capsules FREE ACCESS

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1226
Diastereoselective Hydrogenation of Arenes and Pyridines Promoted by a Ru-Phenanthroline Catalyst

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1227
Oxidation of Benzylic C–H Bonds with a Single-Atom-Like Zinc Catalyst

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1228
Preparation of α-Hydroxy Carboxylic Acids by Carboxylation of Aldehydes on a Nickel(II) Catalyst

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1229
Synthesis of 3,4-Dihydro-2H-Pyrroles by a Nickel-Catalyzed Hydrogenative Cyclization

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1230
Heterogeneous Photocatalytic Synthesis of Functionalized Dihydropyrazoles from Hydrazones

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1231
Photocatalytic Hydrogenation of Olefins and Nitro-benzenes with Al–H₂O on Pd-Doped Carbon Nitride

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1232
Asymmetric Alkylation of α,β-Unsaturated Ketones or Imines on a Polymeric Copper Catalyst

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1233
Nanohybrid Photocatalyst for the Synthesis of Aryl Carbonyl Compounds and Benzimidazoles

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Organo- and Biocatalysis
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1235
Thioxanthone-Catalyzed Single-Step Synthesis of β- and γ-Amino Acid Derivatives FREE ACCESS

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1236
Supramolecular Capsule Emulates Enzymatic Proton-Wire Mechanism in β-Selective O-Glycosylations

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1237
Biocatalytic Double- and Triple-Cascades Permit Highly Stereoselective Syntheses of Cyclohexene Derivatives

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1238
Photocatalytic Functionalization of Nonactivated C(sp³)–H Bonds

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1239
Photoredox-Catalyzed Imino Alkylation of Electronically Diverse Alkenes with Bifunctional Oxime Esters

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1240
N-Arylphenothiazine-Catalyzed Cross-Coupling of Allyl Bromides with Arylboronic Acids

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1241
Organocatalytic Construction of Heterobiaryl Atropisomers via Vinylidene–Quinone Methides

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1242
Disulfide Reagent for Catalytic Asymmetric α-Alkylsulfenylation of Carbonyl Compounds

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1243
Organocatalytic On-Water System for the Synthesis of α-Tertiary Amines

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1244
Intermolecular Organosulfide-Catalyzed Difunctionalization of Allylic Sulfonamides

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1245
Enzymatic Site-Selective and Atroposelective Bromination of 3-Aryl-4(3H)-Quinazolinones

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1246
Organocatalytic Cationic Polymerization toward High-Molecular-Weight Poly(2,3-Dihydrofuran)

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Innovative Drug Discovery and Development
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1247
Kinetic Target-Guided Synthesis of ERAP2 Inhibitors FREE ACCESS

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1248
α-Synuclein Proaggregators via C–H Arylation

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1249
A Non-Peptidic Protease Inhibitor for HIV Treatment

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1250
Lomaiviticin A Monomer – Not as Cytotoxic as the Dimer

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1251
Synthesis and Reevaluation of (+)- and (−)-Collybolide as kappa-Opioid Receptor Agonists

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1252
Dual-Controlled Tumor Imaging using an Enzyme-Responsive and Photoactivated Probe

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1253
Shortest Synthesis of Lysergol and its Binding to 5-HT_1/2Receptors

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1254
Dynamic Kinetic Resolution of Axially Chiral MRTX1719

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1255
A Medicinal Chemist's Guide to Decarboxylative Cross-Couplings

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1256
Atroposelective Annulations Afford Darobactin A

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1257
Targeting KRAS G12R with α,β-Diketoamides

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1258
Selective CYP11B1 Inhibitor Development via an Enantiomer Discrimination

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1259
Application of Continuous Processing for a Scalable High-Temperature Racemization

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1260
Design of a GPCR Antagonist from Agonist Scaffold

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1261
A Candidate for Potential Treatment of Heart Failure with Preserved Ejection Fraction

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1262
An Ene-reaction Ene-ables an α-Kainic Acid Synthesis FREE ACCESS

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Peptide Chemistry
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1263
Palladium-Catalyzed C(sp³)–H Arylation of Cyclic Peptides FREE ACCESS

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1264
C–H Alkylation for the Synthesis of Tetrasubstituted Amino Acid Derivatives

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1265
Primary Amine–Thiourea-Catalyzed Enantioselective Alkylation of Cyclic Ketones

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1266
Functionalization of Aspartic or Glutamic Acids through Photoinduced Decarboxylation

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1267
Iridium-Catalyzed Photochemical [2+2]-Cycloaddition of Dehydroamino Acids with Styrenes

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1268
Synthesis of α-Amino Acids by Enantioselective Carbene Insertion

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1269
Potassium Fluoride-Mediated Deprotection of Fmoc-Amino Acid Esters: One-Pot Peptide Synthesis FREE ACCESS

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1270
Chiral Calcium Phosphate-Catalyzed Amination of β-Keto Esters

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Flow Chemistry
z1271
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1272
Synthesis of α-Aminoamides by a Photocatalytic Continuous-Flow Reaction

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1273
Scalable Photoalkylation of Carbohydrates in Flow with a Sustainable Organocatalyst

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1274
Hydrogen-Transfer Reaction Using Packed-Column Catalysts in Flow

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1275
Photochemical Approach for the Synthesis of Tetrahydroimidazo[1,2-a]pyridine 1-Oxides

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