Synfacts

Issue 04 · April 2023

Recommend Journal

Issue
Synform
A59
SYNFORM ISSUE 2023/04 FREE ACCESS

Full Text

PDF (4070 kb)
Synthesis of Natural Products
z0323
All PDFs of this category

Full Text

PDF (331 kb)
0323
Synthesis of (+)-Chejuenolide A

Full Text

HTML

PDF (88 kb)
0324
Total Synthesis of (–)-Taxol

Full Text

HTML

PDF (78 kb)
0325
Total Synthesis of (+)-Bufogargarizin B FREE ACCESS

Full Text

HTML

PDF (136 kb)
0326
Total Synthesis of (–)-Prorocentin

Full Text

HTML

PDF (86 kb)
0327
Synthesis of (–)-Lissodendoric acid A

Full Text

HTML

PDF (74 kb)
0328
Synthesis of Atrachinenins A and B

Full Text

HTML

PDF (90 kb)
0329
Total Synthesis of (–)-Strychnine FREE ACCESS

Full Text

HTML

PDF (131 kb)
Synthesis of Heterocycles
z0331
All PDFs of this category

Full Text

PDF (364 kb)
0331
Modular Synthesis of Benzimidazoles from Nitroarenes

Full Text

HTML

PDF (83 kb)
0332
Oxidant-Free Synthesis of Fully Substituted Pyrroles through Multicomponent Cyclization

Full Text

HTML

PDF (94 kb)
0333
Circumventing the Aryldiazonium Salt Isolation in Intramolecular Heck–Matsuda Coupling

Full Text

HTML

PDF (98 kb)
0334
Direct and Practical Approach for the Synthesis of δ-Carbolines and Benzofuro[3,2-b]pyridines

Full Text

HTML

PDF (92 kb)
0335
Rational Design of a Palladium Catalyst System for C–N Bond Formation of Five-Membered Heteroaryl Halides

Full Text

HTML

PDF (85 kb)
0336
Robust Conditions for Nickel-Catalyzed Suzuki–Miyaura Cross-Couplings of Complex Molecules

Full Text

HTML

PDF (91 kb)
0337
Palladium-Catalyzed Synthesis of Benzazocines via [6+2] Double Allene Annulation

Full Text

HTML

PDF (87 kb)
0338
Catalyst-Free Synthesis of Oxacyclic Spirooxindoles through Oxonium Ylide Mediated Ring Expansion

Full Text

HTML

PDF (74 kb)
0339
Scalable Syntheses of Functionalized 2-Oxabicyclo[2.2.2]octanes

Full Text

HTML

PDF (81 kb)
0340
Construction of Functionalized Oxazole via Three-Component Cyclization Using a Lewis Acid

Full Text

HTML

PDF (79 kb)
0341
Bicyclic Silaazacycles Featuring Silicon at the Ring Junction: Synthesis and Further Transformations

Full Text

HTML

PDF (75 kb)
0342
Nickel-Catalyzed One-Pot Cascade Synthesis of N‑Substituted Indoles

Full Text

HTML

PDF (82 kb)
0343
Three-Step Modular Synthesis of N-Substituted Bicyclic Systems

Full Text

HTML

PDF (79 kb)
0344
Efficient Access to Pharmacologically Relevant 2-Arylpiperazines

Full Text

HTML

PDF (85 kb)
Synthesis of Materials and Unnatural Products
z0345
All PDFs of this category

Full Text

PDF (567 kb)
0345
9-Fluorenol-Assisted Tertiary Radical Generation and Functionalization

Full Text

HTML

PDF (75 kb)
0346
Build-Up BN-Rings Step by Step

Full Text

HTML

PDF (75 kb)
0347
Catenation of Chiral Cubes FREE ACCESS

Full Text

HTML

PDF (291 kb)
0348
Double Annulation with Three C–C Bond Formations

Full Text

HTML

PDF (84 kb)
0349
“Click” a Phenanthrene

Full Text

HTML

PDF (72 kb)
0350
Three-Component Synthesis of Bicyclic Diphosphacycles

Full Text

HTML

PDF (89 kb)
0351
B(III)Br-B(II)-Stabilized Neutral Boryl Radical

Full Text

HTML

PDF (69 kb)
0352
Carbene-Mediated Polyaminoborane Depolymerization

Full Text

HTML

PDF (147 kb)
0353
How Does 5+7 Compare to 6+6

Full Text

HTML

PDF (78 kb)
0354
Desymmetrized Chiral Calix[4]arenes

Full Text

HTML

PDF (87 kb)
0355
Aromatic Ring Expansions by Iminosilylene

Full Text

HTML

PDF (70 kb)
0356
o-Nitrobenzyl Ether-Enabled Polymer Photo-Degradation

Full Text

HTML

PDF (77 kb)
Metals in Synthesis
z0357
All PDFs of this category

Full Text

PDF (737 kb)
0357
ortho Difunctionalization of Arenes by Iron/Titanium Synergistic Interaction FREE ACCESS

Full Text

HTML

PDF (133 kb)
0358
Enantioselective Molybdenum-Catalyzed Cyclopropanation via Carbonyl Activation

Full Text

HTML

PDF (82 kb)
0359
Ni-Catalyzed Formation of Two Vicinal Enantioenriched C(sp³) Centers Stemming from Two Starting Materials FREE ACCESS

Full Text

HTML

PDF (126 kb)
0360
Enantioselective Rhodium-Catalyzed Synthesis of Cyclobutene Derivatives Using Boronic Acids

Full Text

HTML

PDF (76 kb)
0361
Enantioselective Copper-Catalyzed Inverse-Electron-Demand Diels–Alder Using Phenyl Vinyl Selenide

Full Text

HTML

PDF (78 kb)
0362
Catalytic Asymmetric Conjugate Addition of 1,4-Dienes to β-Substituted Alkenyl Azaarenes

Full Text

HTML

PDF (97 kb)
0363
Nickel-Catalyzed Acylzincation of Ynamides with Alkylzinc Reagents Under CO Atmosphere

Full Text

HTML

PDF (77 kb)
0364
Photoinduced Decarboxylative C–C and C–N Couplings of Carboxylic Acids under Dual Iron/Copper Catalysis

Full Text

HTML

PDF (78 kb)
0365
Synthesis of Oxaspirolactones via Palladium-Catalyzed Hydrocarbonylation of Alcohol-Tethered Styrenes

Full Text

HTML

PDF (75 kb)
0366
Enantioselective Cobalt-Catalyzed Double Hydrogenation for Chiral Z-Allylamide Syntheses

Full Text

HTML

PDF (89 kb)
0367
Iron-Catalyzed and Electrochemical Dehydrogenative Synthesis of Monofluorinated Oxindoles

Full Text

HTML

PDF (82 kb)
0368
Copper-Catalyzed Benzo[d][1,3,2]dithiazole-1-oxide Synthesis via Cross-Coupling with Elemental Sulfur

Full Text

HTML

PDF (89 kb)
0369
Copper-Catalyzed Addition of Terminal Alkynes across Dialkyl Azodicarboxylates

Full Text

HTML

PDF (70 kb)
0370
Syntheses of Difluorocarbonyl Oxindoles and Isoquinoline-1,3-diones via Radical Nickel Catalysis

Full Text

HTML

PDF (74 kb)
0371
Asymmetric α-Acylation of N-Heterocycles with Carboxylic Acids by Dual Nickel/Photoredox Catalysis

Full Text

HTML

PDF (91 kb)
0372
Nickel-Catalyzed Regiodivergent Cross-Electrophile Coupling of Alkyl Bromides Steered by the Ligand

Full Text

HTML

PDF (103 kb)
0373
Photocatalytic C(sp²)−H Fluoromethoxylation of Arenes

Full Text

HTML

PDF (81 kb)
0374
Silver-Catalyzed Synthesis of Spirocycles via an Enamine–Iminium Umpolung Step

Full Text

HTML

PDF (79 kb)
0375
Gold-Catalyzed Synthesis of Alkynylated Pyrrolidines from N,O-Acetals via Cyclic Iminium Ion Intermediates

Full Text

HTML

PDF (84 kb)
0376
Synthesis of Pyrrolines via Ni-Catalyzed Iminoarylation of Alkene-Tethered Oxime Esters

Full Text

HTML

PDF (72 kb)
0377
Enantioconvergent Cross-Electrophile Coupling of Two Alkyl Halides to Access Chiral α-Alkylboronic Esters

Full Text

HTML

PDF (97 kb)
0378
Stereoconvergent 1,3-Rearrangement of (Homo)Allylic Alcohols Using Crabtree’s Catalyst

Full Text

HTML

PDF (96 kb)
0379
Nickel-Catalyzed Enantioselective C(sp)–P Cross-Coupling of Secondary Phosphines with Bromoalkynes

Full Text

HTML

PDF (71 kb)
0380
Highly Linear- or Branched-Selective Ni-Catalyzed Mizoroki–Heck Reaction of 1,3-Dienes

Full Text

HTML

PDF (73 kb)
0381
Intercepted Kinugasa Reaction with Ir Catalysis: Asymmetric Synthesis of Allylated β-Lactams

Full Text

HTML

PDF (94 kb)
0382
Desymmetrization of 1,3-Diols by Copper(I)-Catalyzed S–O Cross-Coupling with Aryl Sulfonyl Chlorides

Full Text

HTML

PDF (71 kb)
Polymer-Supported Synthesis
z0383
All PDFs of this category

Full Text

PDF (1600 kb)
0383
Semi-Hydrogenation of Alkynes and Suzuki Coupling with a Polyurethane Foam-Supported Pd Catalyst FREE ACCESS

Full Text

HTML

PDF (719 kb)
0384
C3-Formylation of Indoles with Methanol by g-C₃N₄/rGO/BiVO₄ Heterojunction Photocatalyst

Full Text

HTML

PDF (75 kb)
0385
MOF-Supported Chiral Frustrated Lewis Pair for Asymmetric Hydrogenation

Full Text

HTML

PDF (731 kb)
0386
Photocatalytic Dehydrative Etherification of Alcohols by an Unsupported Nanoporous Gold Catalyst

Full Text

HTML

PDF (75 kb)
0387
Aerobic Oxidative Annulation of N-Arylpyrrolidines Catalyzed by Pt/C

Full Text

HTML

PDF (91 kb)
0388
Synthesis of Amino Phenazines through the Oxidative Cyclization of Anilines with o-Phenylenediamines

Full Text

HTML

PDF (80 kb)
0389
1,4-Arylation of α,β-Unsaturated Ketones with Arylboronic Acids Using NHC–Coordinated Rh on Ceria

Full Text

HTML

PDF (96 kb)
0390
Heterogeneous Photocatalytic Multicomponent Reaction for the Synthesis of Imidazolidines

Full Text

HTML

PDF (91 kb)
0391
Hydrogenation of Nitroarenes Catalyzed by a COF-Based Photocatalyst

Full Text

HTML

PDF (85 kb)
0392
Oxidative Coupling of Carbon Monoxide with Amines by Gold Nanoparticles Supported on ZnO

Full Text

HTML

PDF (71 kb)
0393
Synthesis of α‑Haloketones from Vinylarenes Catalyzed by Cu-Modified Graphitic Carbon Nitride

Full Text

HTML

PDF (80 kb)
0394
Asymmetric Allylic Amination Using PS-Supported Phosphoramidite Ligands–Ir Complex

Full Text

HTML

PDF (79 kb)
Organo- and Biocatalysis
z0395
All PDFs of this category

Full Text

PDF (428 kb)
0395
Formal Electronically Mismatched Radical Additions

Full Text

HTML

PDF (81 kb)
0396
Carbene Transferases as Catalysts for Chemodivergent Activation of C(sp²)–H and C(sp³)–H Bonds

Full Text

HTML

PDF (94 kb)
0397
Enantioselective Synthesis of Tertiary Nitroalkanes Enabled by Enzyme Catalysis FREE ACCESS

Full Text

HTML

PDF (165 kb)
0398
Aminocatalytic Enantio-, Diastereo- and Periselective [4+4] Cycloaddition

Full Text

HTML

PDF (86 kb)
0399
Hydrogen-Bond-Donor Catalyst Permits Asymmetric Transformation of Sulfonyl Cyanides toward Sulfinates

Full Text

HTML

PDF (76 kb)
0400
Photocatalytic Cyclopropanation of Unactivated Olefins with α-Bromomalonates and α-Bromo-β-Keto Esters

Full Text

HTML

PDF (87 kb)
0401
Borenium-Catalyzed Hydrogenative Cleavage of Unactivated C(Aryl)–C(Alkyl) Bonds

Full Text

HTML

PDF (75 kb)
0402
Conformation-Switching DNA Photocatalyst for Radical Polymerization

Full Text

HTML

PDF (121 kb)
0403
Asymmetric Enolexo-Aldol Condensations of Siladials via Enamine Catalysis

Full Text

HTML

PDF (68 kb)
0404
Identification of a Pericyclase that Catalyzes the Formation of cis-Decalins

Full Text

HTML

PDF (98 kb)
Innovative Drug Discovery and Development
z0405
All PDFs of this category

Full Text

PDF (459 kb)
0405
Bioorthogonal “Click-and-Release” of Iminosydnones to Give Water-Stable Isocyanates FREE ACCESS

Full Text

HTML

PDF (127 kb)
0406
Total Synthesis of Iridoid Oligomers Enlightens Efficacy of Folk Medicine

Full Text

HTML

PDF (90 kb)
0407
Process Understanding Enables Control of Hydrogen Fluoride Formation in a Nitroarene Reduction FREE ACCESS

Full Text

HTML

PDF (134 kb)
0408
Hydrolysis-Resistant Ester for Probe Development

Full Text

HTML

PDF (77 kb)
0409
Design and Synthesis of BCL6 BTB Inhibitor OICR12694

Full Text

HTML

PDF (77 kb)
0410
MK-8189: A Potent and Selective PDE10A Inhibitor for the Treatment of Schizophrenia

Full Text

HTML

PDF (78 kb)
0411
Photo-Decarboxylative Coupling of α-Amino Acids and Enones Enables Efficient Synthesis of a Drug Scaffold

Full Text

HTML

PDF (97 kb)
0412
A Scalable Asymmetric Total Synthesis of (–)-Emetine

Full Text

HTML

PDF (73 kb)
0413
Efficient Synthesis of DNA Interstrand Cross-Links

Full Text

HTML

PDF (72 kb)
0414
Stepwise, Controllable Electrochemical Reduction of Trifluoromethylarenes

Full Text

HTML

PDF (72 kb)
0415
Macrocyclization and Scaffold Hopping Improves Selectivity and ADME Properties of HPK1 Inhibitors

Full Text

HTML

PDF (68 kb)
0416
Synthesis of Anesthetic Ketamine FREE ACCESS

Full Text

HTML

PDF (129 kb)
Peptide Chemistry
z0417
All PDFs of this category

Full Text

PDF (339 kb)
0417
Rh(III)-Catalyzed Synthesis of Unnatural Peptides FREE ACCESS

Full Text

HTML

PDF (113 kb)
0418
Coupling of Amino Acid Terminal Alkyne with in situ Iminium Ion to Access N^ε‑Substituted Lysine Mimetics

Full Text

HTML

PDF (83 kb)
0419
Visible-Light-Mediated Continuous-Flow Technology for the Synthesis of α-(N-Hydroxy)amino Amides

Full Text

HTML

PDF (109 kb)
0420
Modification of Diamino Acid-Containing Hydrospirophosphoranes

Full Text

HTML

PDF (70 kb)
0421
Acetoxylation of Tyrosine-Containing Peptides Using a Palladium Catalyst

Full Text

HTML

PDF (77 kb)
0422
Palladium-Catalyzed C–H Alkenylation to Form Maleimide-Braced Peptides

Full Text

HTML

PDF (70 kb)
0423
Organocatalyzed Enantioselective N–H Insertion

Full Text

HTML

PDF (78 kb)
0424
Synthesis of N-Formyl Amino Acid Esters FREE ACCESS

Full Text

HTML

PDF (124 kb)
Flow Chemistry
z0425
All PDFs of this category

Full Text

PDF (71 kb)
0425
Segmented Continuous Flow Allows for Convenient Synthesis of Phenyl Glucosazone

Full Text

HTML

PDF (71 kb)
Erratum
0426
Erratum: 2-Amino-3,3-difluoro-2,3-dihydrofurans from Difluorocarbenes and Enaminones

Full Text

HTML

PDF (62 kb)
Most Read
Archive
Articles by Category
Free Sample Issue

Journal

More About This Journal
Synfacts Videos
Editorial Board
Editorial Office
Brochure

Authors

Instructions for Authors

Subscription

Subscription Information & Contacts
Institutional Licensing

Nobel Prize 2016

Instructions for Authors

Journals
Book Series
Login
Help
Portal
Return to Classic Website

German English

Thieme E-Books & E-Journals is a service of Georg Thieme Verlag and Thieme Medical Publishers, Inc.
© Georg Thieme Verlag KG

Imprint | Privacy policy statement

Your Current IP Address: 18.191.5.237