DOI:
10.1055/s-00000084
Synthesis
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References
For an example of palladium-catalysed
direct 3-arylation of a pyrazole, see: Brnardic EJ, Garbaccio RM, Fraley ME, Tasber ES, Steen JT, Arrington KL, Dudkin VY, Hartman GD, Stirdivant SM, Drakas BA, Rickert K, Walsh ES, Hamilton K, Buser CA, Hardwick J, Tao W, Beck SC, Mao X, Lobell RB, Sepp-Lorenzino L, Yan Y, Ikuta M, Munshi SK, Kuo LC, Kreatsoulas C,
Bioorg.
Med. Chem. Lett.. 2007; 17 5989
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