DOI: 10.1055/s-00000084

Synthesis

Issue 04 · Volume 2010 · February 2010 DOI: 10.1055/s-002-20768

review

543
Czekelius, Constantin; Tzschucke, Carl Christoph: Synthesis of Halogenated Carboxylic Acids and Amino Acids
https://www.thieme-connect.de/media/synthesis/201004/e255_ga.jpg

paper

567
Enders, Dieter; Krüll, Ralf; Bettray, Wolfgang: Microwave-Assisted Organocatalytic Quadruple Domino Reactions of Acetaldehyde and Nitroalkenes
https://www.thieme-connect.de/media/synthesis/201004/z218_ga.jpg
573
Ravinder, Mettu; Sadhu, Partha Sarathi; Santhoshi, Amlipur; Narender, Puli; Swamy, Gundimella Y. S. K.; Ravikumar, Krishnan; Jayathirtha Rao, Vaidya: Synthesis of New Aminonicotinate Derivatives from Acetylated Baylis-Hillman Adducts and Enamino Esters via a Consecutive [3+3]-Annulation Protocol
https://www.thieme-connect.de/media/synthesis/201004/t163_ga.jpg
579
Naidu, Ajay B.; Sekar, Govindasamy: Synthesis of Benzoxazoles by an Efficient Ullmann-Type Intramolecular C(aryl)-O Bond-Forming Coupling Cyclization with a BINAM-Copper(II) Catalyst
https://www.thieme-connect.de/media/synthesis/201004/z206_ga.jpg
Supporting Information
587
Wu, Mengde; Wang, Shaozhong: An Alternative to Pictet-Gams Reaction Triggered by Hendrickson Reagent: Isoquinolines and β-Carbolines from Amides
https://www.thieme-connect.de/media/synthesis/201004/f187_ga.jpg
593
Saavedra, Luis Astudillo; Vallejos C., Gabriel; Kouznetsov, Vladimir V.; Gutierrez C., Margarita; Meléndez Gómez, Carlos Mario; Vargas Méndez, Leonor Y.; Bermúdez Jaimes, John Hervin: Synthesis of New Diversely Linked Biquinoline Derivatives by Multicomponent Imino-Diels-Alder Cycloaddition and Intramolecular Friedel-Crafts Cyclization
https://www.thieme-connect.de/media/synthesis/201004/m053_ga.jpg
601
La Ferla, Barbara; Orsato, Alexandre; Zona, Cristiano; Cervi, Giovanni; Papeo, Gianluca; Felder, Eduard R.; Nicotra, Francesco: Synthesis of a β-Carboline Scaffold Properly Functionalized for the Generation of Libraries of Bioactive Compounds
https://www.thieme-connect.de/media/synthesis/201004/t115_ga.jpg
605
Aurrecoechea, José M.; Gorgojo, José M.; Saornil, Carlos: A Two-Step Synthesis of 3,4-Disubstituted Piperidines from Acyclic Precursors through Tetrahydropyridine Intermediates
https://www.thieme-connect.de/media/synthesis/201004/t137_ga.jpg
613
Aladzheva, Inga M.; Bykhovskaya, Olga V.; Nelyubina, Yulya V.; Korlyukov, Alexander A.; Petrovskii, Pavel V.; Odinets, Irina L.: Facile One-Pot Synthesis and X-ray Characterization of N-(Thio)phosphoryl-2-oxo-1,2-azaphospholanes: First Example of Cyclic O,O- and O,S-Bidentate Ligands with the P-N-P Backbone
https://www.thieme-connect.de/media/synthesis/201004/t148_ga.jpg
619
Sliman, Faten; Desmaële, Didier: Synthesis of 5-Aryl- and 5-Heteroaryl-7-carboxyl-8-hydroxyquinaldines through Suzuki Cross-Coupling Reaction with Potassium Organotrifluoroborates
https://www.thieme-connect.de/media/synthesis/201004/t155_ga.jpg
631
Bonazzi, Simone; Binaghi, Massimo; Fellay, Cindy; Wach, Jean-Yves; Gademann, Karl: Synthetic Studies on the Sporolides: Exploration of the Enediyne Route
https://www.thieme-connect.de/media/synthesis/201004/t178_ga.jpg
643
Bose, D. Subhas; Chary, M. Venu: First Total Synthesis of (-)-Circumdatin H, a Novel Mitochondrial NADH Oxidase Inhibitor
https://www.thieme-connect.de/media/synthesis/201004/z209_ga.jpg
651
Olimpieri, Francesca; Fustero, Santos; Volonterio, Alessandro; Zanda, Matteo: A Mild, Efficient Synthesis of gem-Difluorodihydrouracils
https://www.thieme-connect.de/media/synthesis/201004/z217_ga.jpg
661
Park, Jinhyung; Kwon, Young Bum; Yang, Kyungmo; Rhee, Hakjune; Yoon, Cheol Min: Efficient Palladium-Catalyzed Coupling of Baylis-Hillman Acetates with an Allylstannane
https://www.thieme-connect.de/media/synthesis/201004/f093_ga.jpg
666
Kobayashi, Kazuhiro; Shirai, Yuu; Fukamachi, Shuhei; Konishi, Hisatoshi: Synthesis of 2,3-Bis(arylamino)benzofurans and 2,3-Bis(arylimino)-2,3-dihydrobenzofurans by a Lewis Acid Catalyzed Reaction of 2-Aryliminophenols with Aryl Isocyanides
https://www.thieme-connect.de/media/synthesis/201004/f197_ga.jpg
671
Kotljarov, Anton; Sevenard, Dmitri V.; Iaroshenko, Viktor O.; Irgashev, Roman A.; Volochnyuk, Dmitriy M.; Langer, Peter; Tolmachev, Andrei A.; Sosnovskikh, Vyacheslav Ya.: Regioselective Synthesis of Novel Perfluoroalkylated Fused Pyridines and 3-(Aminomethylene)thiochroman-4-ones from 3-(Perfluoroalkanoyl)thio­chromenones and Amines
https://www.thieme-connect.de/media/synthesis/201004/p122_ga.jpg
678
Diez-Martinez, Alba; Gultekin, Zeynep; Delso, Ignacio; Tejero, Tomas; Merino, Pedro: Synthesis of N-(Benzyloxyethyl)- and N-(Alkoxycarbonylmethyl)nitrones
https://www.thieme-connect.de/media/synthesis/201004/p136_ga.jpg
689
Hansen, Finn K.; Geffken, Detlef: Synthesis of Novel N,3-Substituted 3H-[1,2,3]Triazolo[4,5-d]pyrimidin-5-amines
https://www.thieme-connect.de/media/synthesis/201004/t170_ga.jpg
694
Pattarozzi, Mariella; Roncaglia, Fabrizio; Giangiordano, Valerio; Davoli, Paolo; Prati, Fabio; Ghelfi, Franco: ‘Ligand-Free-Like’ CuCl-Catalyzed Atom Transfer Radical Cyclization of N-Substituted N-Allyl Polychloroamides to γ-Lactams
https://www.thieme-connect.de/media/synthesis/201004/z220_ga.jpg

feature article

701
Uria, Uxue; Vicario, Jose L.; Badía, Dolores; Carrillo, Luisa; Reyes, Efraim; Pesquera, Amaia: ‘On Water’ Iminium/Enamine Catalysis: Organocatalytic Enantioselective Cyclopropanation of α,β-Unsaturated Aldehydes
https://www.thieme-connect.de/media/synthesis/201004/e259_ga.jpg

practical synthetic procedures

714
Phillips, James G.; Jaworska, Maria; Lew, Willard: A Practical Synthesis of 1-N-SEM-Protected 3-Iodo-7-methyl-2-piperidin-3-ylindole
https://www.thieme-connect.de/media/synthesis/201004/m051_ga.jpg

book review

718
Schmidt, Bernd: The Mizoroki-Heck Reaction

addenda and errata

e2
‘Ligand-Free-Like’ CuCl-Catalyzed Atom Transfer Radical Cyclization of N-Substituted N-Allyl Polychloroamides to γ-Lactams