DOI: 10.1055/s-00000131

Synfacts

Issue 06 · Volume 2011 · June 2011 DOI: 10.1055/s-002-22013

Synform

A46
Zanda, Matteo: SYNFORM ISSUE 2011/06

Synthesis of Natural Products and Potential Drugs

z577
All PDFs of this category
0577
Malmgren, H.; Cotton, H.; Frøstrup, B.; Jones, D. S.; Loke, M.-L.; Peters, D.; Schultz, S.; Sölver, E.; Thomsen, T.; Wennerberg, J.: Synthesis of NS9544 Acetate
0578
Campos, K. R.; Klapars, A.; Kohmura, Y.; Polard, D.; Ishibashi, H.; Kato, S.; Takezawa, A.; Waldman, J. H.; Wallace, D. J.; Chen, C.-y.; Yasuda, N.: Synthesis of an hNK-1 Receptor Antagonist
0579
Ouellet, S. G.; Roy, A.; Molinaro, C.; Angelaud, R.; Marcoux, J.-F.; O’Shea, P. D.; Davies, I. W.: Synthesis of the Biaryl Core of Anacetrapib
0580
Schubert, M.; Metz, P.: Synthesis of Kempene-2
0581
Takada, A.; Hashimoto, Y.; Takikawa, H.; Hikita, K.; Suzuki, K.: Synthesis of ent-Seragakinone A
0582
Wang, Y.; Zhu, L.; Zhang, Y.; Hong, R.: Synthesis of (±)-Stemoamide
0583
Chan, J.; Burke, B. J.; Baucom, K.; Hansen, K.; Bio, M. M.; DiVirgilio, E.; Faul, M.; Murry, J.: Synthesis of a CXCR3 Antagonist
0584
Albert, B. J.; Yamaoka, Y.; Yamamoto, H.: Synthesis of EBC-23
0585
Chinkov, N.; Warm, A.; Carreira, E. M.: Synthesis of Efavirenz
0586
Yazaki, R.; Kumagai, N.; Shibasaki, M.: Synthesis of AMG 837
0587
Hanessian, S.; Stoffman, E.; Mi, X.; Renton, P.: n-Nitric Oxide Synthase Inhibitor
0588
Kuttruff, C. A.; Zipse, H.; Trauner, D.: Synthesis of Variecolortides A and B
0589
Ishikawa, H.; Honma, M.; Hayashi, Y.: Synthesis of ABT-341
0590
Levin, S.; Nani, R. R.; Reisman, S. E.: Enantioselective Synthesis of (+)-Salvileucalin B
0591
Gampe, C. M.; Carreira, E. M.: Syntheses of Guanacastepenes N and O

Synthesis of Heterocycles

z593
All PDFs of this category
0593
Zhang, X.; Chen, D.; Zhao, M.; Zhao, J.; Jia, A.; Li, X.: Rhodium-Catalyzed Synthesis of Isoquinolines from Oximines and Alkynes
0594
Zhao, J.; Zhao, Y.; Fu, H.: Transition-Metal-Free SNAr-Type Synthesis of Chromones
0595
Weiß, K. M.; Wei, S.; Tsogoeva, S. B.: Synthesis of 1,3-Thiazoles from Nitrostyrenes and Aromatic Thioamides
0596
Kumar, R. K.; Ali, Md. A.; Punniyamurthy, T.: Palladium-Catalyzed C-H Activation/C-N Coupling Route to 1-Aryl-1H-benzotriazoles
0597
Hirano, K.; Inaba, Y.; Takahashi, N.; Shimano, M.; Oishi, S.; Fujii, N.; Ohno, H.: Gold-Catalyzed Hydroamination-Hydroarylation Route to Fused Indoles
0598
Lei, M.; Ma, L.; Hu, L.: Tetrahydropyranoquinolinone via a Knoevenagel Reaction
0599
Xu, W.; Jin, Y.; Liu, H.; Jiang, Y.; Fu, H.: Synthesis of Quinazolinones by Combined Ullmann Coupling-Oxidative C-H Amidation
0600
Kim, J. H.; Lee, S.-g.: One-Pot Synthesis of Indoles and N-Fused Indoles from Nitriles
0601
Nakao, Y.; Morita, E.; Idei, H.; Hiyama, T.: Nickel-Catalyzed Dehydrogenative [4+2]-Cycloaddition Route to Dihydropyridones
0602
Xu, J.; Wei, J.; Bian, L.; Zhang, J.; Chen, J.; Deng, H.; Wu, X.; Zhang, H.; Cao, W.: A Catalyst-Free MCR Approach to 1,5-Benzodiazepines
0603
Frutos, R. P.; Tampone, T.; Mulder, J. A.; Xu, Y.; Reeves, D.; Wang, X.-J.; Zhang, L.; Krishnamurthy, D.; Senanayake, C. H.: A Boronic Acid Catalyzed Route to Imidazoles. Synthesis of LFA-1 Antagonists
0604
Blanchot, M.; Candito, D. A.; Larnaud, F.; Lautens, M.: Phenanthridine Synthesis via a Pd-Catalyzed Direct Arylation/N-Arylation Sequence
0605
Attanasi, O. A.; Berretta, S.; De Crescentini, L.; Favi, G.; Giorgi, G.; Mantellini, F.; Nicolini, S.: Zinc(II)-Catalyzed Synthesis of Poly-functionalized Pyrroles
0606
Ng, E. P. J.; Wang, Y.-F.; Chiba, S.: Mn(III)-Catalyzed Synthesis of Pyrroles from Vinyl Azides and β-Keto Acids
0607
Kang, J. Y.; Connell, B. T.: Synthesis of Furans via Indium-Catalyzed Rearrangement of Acetylenic Epoxides

Synthesis of Materials and Unnatural Products

z609
All PDFs of this category
0609
Oh, K.; Fuchibe, K.; Ichikawa, J.: Greener 1,1-Difluoroallenes
0610
Néabo, J. R.; Tohoundjona, K. I. S.; Morin, J.-F.: Bulky, Solid…but still Topochemical!
0611
Pacholska-Dudziak, E.; Szterenberg, L.; Latos-Grażyński, L.: Porphyrin-Annulene Hybrid
0612
Wang, Y.-H.; Liu, H.; Zhu, L.-L.; Li, X.-X.; Chen, Z.: Polyaromatic Furans from Diynyl-1,6-diols
0613
Kao, M.-T.; Chen, J.-H.; Chu, Y.-Y.; Tseng, K.-P.; Hsu, C.-H.; Wong, K.-T.; Chang, C.-W.; Hsu, C.-P.; Liu, Y.-H.: A Concise Route to Functionalized Truxenes
0614
Katsuta, S.; Miyagi, D.; Yamada, H.; Okujima, T.; Mori, S.; Nakayama, K.-i.; Uno, H.: Cyanated Pentacene and Naphthacene as Air-Stable Acene Derivatives
0615
Hübner, A.; Qu, Z.-W.; Englert, U.; Bolte, M.; Lerner, H.-W.; Holthausen, M. C.; Wagner, M.: 9-H-9-Borafluorene: Hydroboration and Oligomerization
0616
Liu, X.; Ma, Y.; Duan, W.; He, F.; Zhao, L.; Song, C.: A New Twist to [2.2]Paracyclophanes
0617
Abla, M.; Durand, G.; Pucci, B.: The Tale (Tail) of Hemifluorinated Surfactants
0618
Yamaguchi, I.; Jonai, S.; Matsuda, Y.: Through-Space in a Boat
0619
Akhigbe, J.; Zeller, M.; Brückner, C.: Red-Shifted Porphyrins
0620
Tverskoy, O.; Rominger, F.; Peters, A.; Himmel, H.-J.; Bunz, U. H. F.: A More Efficient Access to Tetraaza-pentacenes
0621
Zeng, Z.; Guan, Z.; Xu, Q.-H.; Wu, J.: Octupolar HBC Chromophores

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z623
All PDFs of this category
0623
Meek, S. J.; O’Brien, R. V.; Llaveria, J.; Schrock, R. R.; Hoveyda, A. H.: Catalytic Z-Selective Olefin Cross-Metathesis
0624
Wang, D.-S.; Tang, J.; Zhou, Y.-G.; Chen, M.-W.; Yu, C.-B.; Duan, Y.; Jiang, G.-F.: Synthesis of 2,3-Disubstituted Indolines by Asymmetric Hydrogenation
0625
Sonawane, R. P.; Jheengut, V.; Rabalakos, C.; Larouche-Gauthier, R.; Scott, H. K.; Aggarwal, V. K.: Construction of Quaternary Stereogenic Centers from Tertiary Boronic Esters
0626
Brozek, L. A.; Sieber, J. D.; Morken, J. P.: Catalytic Asymmetric Allylation of Unsaturated Methylidene Ketones
0627
Schotes, C.; Mezzetti, A.: Ruthenium-Catalyzed Asymmetric [2+2] Cycloaddition of Ynamides with Enones
0628
Gavrilov, K. N.; Zheglov, S. V.; Shiryaev, A. A.; Groshkin, N. N.; Rastorguev, E. A.; Benetskiy, E. B.; Davankov, V. A.: P*,P*-Bidentate Diamidophosphite Ligands in Palladium-Catalyzed Reactions
0629
Liu, T.-L.; He, Z.-L.; Tao, H.-Y.; Cai, Y.-P.; Wang, C.-J.: [3+2] Cycloaddition of Azomethine Ylides and Cyclopropylidene Acetates
0630
Ye, L.; He, W.; Zhang, L.: Gold-Catalyzed Stereoselective Synthesis of Azetidin-3-ones
0631
Camelio, A. M.; Barton, T.; Guo, F.; Shaw, T.; Siegel, D.: Palladium-Catalyzed Enyne Cyclization towards Complex Cyclopentanes
0632
Zheng, K.; Yin, C.; Liu, X.; Lin, L.; Feng, X.: Catalytic Asymmetric Addition of Alkyl Enol Ethers to 1,2-Dicarbonyls
0633
Urban, S.; Ortega, N.; Glorius, F.: Ligand-Controlled Highly Regioselective and Asymmetric Hydrogenation of Quinoxalines
0634
Zhao, Q.-Y.; Yuan, Z.-L.; Shi, M.: Vinylogous Mannich Reactions of Fluorinated Aldimines and Siloxyfurans
0635
Gonzáles, A. Z.; Benitez, D.; Tkatchouk, E.; Goddard III, W. A.; Toste, F. D.: Diastereo- and Enantioselective Synthesis of Pyrrolidines
0636
Yanagisawa, A.; Kushihara, N.; Yoshida, K.: Synthesis of Chiral γ-Butyrolactones by a Domino Aldol-Cyclization Reaction
0637
Ochi, Y.; Kurahashi, T.; Matsubara, S.: Nickel-Catalyzed Cycloaddition between Phthalic Anhydrides and Allenes
0638
Hansen, J. H.; Parr, B. T.; Pelphrey, P.; Jin, Q.; Autschbach, J.; Davies, H. M. L.: Rh(II)-Catalyzed Stereoselective Cross-Coupling of Diazo Compounds
0639
Mao, B.; Geurts, K.; Fañanás-Mastral, M.; van Zijl, A. W.; Fletcher, S. P.; Minnaard, A. J.; Feringa, B. L.: Asymmetric Synthesis of γ-Butenolides via Sequential Metal-Catalyzed Reactions
0640
Melhado, A. D.; Amarante, G. W.; Wang, Z. J.; Luparia, M.; Toste, F. D.: Au(I)-Catalyzed Asymmetric Cycloadditions and Mannich Reactions of Azlactones
0641
Nadeau, C.; Aly, S.; Belyk, K.: Asymmetric Addition of Boronic Acids to N-Benzylnicotinate Salts
0642
Teichert, J. F.; Feringa, B. L.: Copper-Catalyzed Asymmetric Conjugate Addition of Grignard Reagents
0643
Wolf, C.; Zhang, P.: Copper-Catalyzed Asymmetric Friedel-Crafts Reaction of Indoles
0644
Endo, K.; Tanaka, K.; Ogawa, M.; Shibata, T.: Ring Opening of Oxabicyclic Alkenes Catalyzed by Multinuclear Complexes
0645
Li, Q.; Dong, Z.; Yu, Z.-X.: Novel Chiral Diene Ligand for Rhodium-Catalyzed Asymmetric 1,4-Addition
0646
Wisniewska, H. M.; Jarvo, E. R.: Asymmetric Propargylation of Imines
0647
Aksin-Artok, Ö.; Krause, N.: Combined Rh/Au Catalysis to Form 2,5-Dihydrofurans
0648
Hong, A. Y.; Krout, M. R.; Jensen, T.; Bennett, N. B.; Harned, A. M.; Stoltz, B. M.: Synthesis of γ-Quaternary Acylcyclopentenes via a Ring-Contraction Strategy
0649
Iwata, M.; Yazaki, R.; Chen, I-H.; Sureshkumar, D.; Kumagai, N.; Shibasaki, M.: Enantio- and Diastereoselective Aldol Reaction of Thioamides
0650
Hoshi, T.; Sasaki, K.; Sato, S.; Ishii, Y.; Suzuki, T.; Hagiwara, H.: Asymmetric Palladium-Catalyzed Allylic Alkylation of Indoles
0651
Nguyen, T. D.; Webster, R.; Lautens, M.: Rapid Access to Stereochemically Defined Heterocyclic Scaffolds
0652
Steib, A. K.; Thaler, T.; Komeyama, K.; Mayer, P.; Knochel, P.: Highly Diastereoselective Iron-Mediated C(sp²)-C(sp³) Cross-Couplings

Metal-Mediated Synthesis

z653
All PDFs of this category
0653
Auvinet, A.-L.; Harrity, J. P. A.: Ni-Catalyzed Alkyne Cycloaddition to Give Boronic Esters
0654
Aggarwal, V. K.; Binanzer, M.; de Ceglie, M. C.; Gallanti, M.; Glasspoole, B. W.; Kendrick, S. J. F.; Sonawane, R. P.; Vázquez-Romero, A.; Webster, M. P.: Synthesis of Tertiary and Quaternary Allyl- and Crotylsilanes
0655
Chen, Z.; Zheng, D.; Wu, J.: Synthesis of Polysubstituted Indoles via Three-Component Reaction
0656
Kaim, L. El; Grimaud, L.; Patil, P.: Three-Component Cascade Reaction towards Substituted Tetrazoles
0657
Molander, G. A.; Colombel, V.; Braz, V. A.: C-H Alkylation of Heteroarenes with Alkyl- and Alkoxymethyltrifluoroborates
0658
Zhang, L.; Ang, G. Y.; Chiba, S.: Cu-Catalyzed Benzylic C-H Oxidation Using Imines as Directing Groups
0659
Chai, G.; Wu, S.; Fu, C.; Ma, S.: Cyclobutenone Synthesis from 2,3-Allenoates and Organozincs
0660
Song, Z.; Kui, L.; Sun, X.; Li, L.: A Stereoselective Approach to Tetrasubstituted Silyl Enol Ethers
0661
Tissot, M.; Hernández, A. Pérez; Müller, D.; Mauduit, M.; Alexakis, A.: Cu-Catalyzed Highly Enantioselective 1,4-Addition of Grignard Reagents
0662
Joshi-Pangu, A.; Ganesh, M.; Biscoe, M. R.: Ni-Catalyzed Negishi Cross-Coupling of Secondary Alkylzinc Halides
0663
Truong, T.; Daugulis, O.: Base-Mediated Biaryl Formation via Benzyne Intermediates
0664
Ohashi, M.; Kambara, T.; Hatanaka, T.; Saijo, H.; Doi, R.; Ogoshi, S.: Pd-Catalyzed Coupling of Tetrafluoroethylene with Arylzinc Compounds
0665
Cohen, D. T.; Cardinal-David, B.; Roberts, J. M.; Sarjeant, A. A.; Scheidt, K. A.: Titanium-Mediated Diastereo- and Enantioselective Dimerization of Enals
0666
Molander, G. A.; Fleury-Brégeot, N.; Hiebel, M.-A.: Synthesis and Cross-Coupling of Sulfonamidomethyltrifluoroborates
0667
Maury, J.; Feray, L.; Bertrand, M. P.: anti-Carbozincation of Diethyl Acetylenedicarboxylate

Organo- and Biocatalysis

z669
All PDFs of this category
0669
Jia, Z.-J.; Jiang, H.; Li, J.-L.; Gschwend, B.; Li, Q.-Z.; Yin, X.; Grouleff, J.; Chen, Y.-C.; Jørgensen, K. A.: Trienamines in Organocatalysis
0670
Shibuya, M.; Osada, Y.; Sasano, Y.; Tomizawa, M.; Iwabuchi, Y.: Metal-Free Aerobic Oxidation of Alcohols
0671
Zilly, F. E.; Acevedo, J. P.; Augustyniak, W.; Deege, A.; Häusig, U. W.; Reetz, M. T.: How to Oxidize Methane with a P450 Enzyme
0672
Wu, R.; Chang, X.; Lu, A.; Wang, Y.; Wu, G.; Song, H.; Zhou, Z.; Tang, C.: Highly Efficient Hydrogen-Bond Catalysis with (Thio)Phosphorodiamides
0673
Chen, Q.-A.; Wang, D.-S.; Zhou, Y.-G.; Duan, Y.; Fan, H.-J.; Yang, Y.; Zhang, Z.: Reduction of Quinoxalines: A Convergent Disproportionation Reaction
0674
Ren, H.; Wulff, W. D.: Catalytic Asymmetric Aminoallylation of Aldehydes
0675
Klauber, E. G.; Mittal, N.; Shah, T. K.; Seidel, D.: Kinetic Resolution of Allylic Amines via a Dual-Catalysis Approach
0676
Bernardi, L.; Indrigo, E.; Pollicino, S.; Ricci, A.: Coupled Lewis Base and Phase-Transfer Catalysis for Imine Trifluoromethylation
0677
Misaki, T.; Kawano, K.; Sugimura, T.: Z-Selective 1,4-Addition of 5H-Oxazol-4-ones with Alkynyl Carbonyl Compounds
0678
Mori, K.; Ehara, K.; Kurihara, K.; Akiyama, T.: Activation of C(sp³)-H Bond via 1,5-Hydride Transfer-Cyclization
0679
Hamed, R. B.; Gomez-Castellanos, J. R.; Thalhammer, A.; Harding, D.; Ducho, C.; Claridge, T. D. W.; Schofield, C. J.: Biocatalytic, Decarboxylative Addition of Malonates to Imines, a ”Rodionovase"
0680
Terada, M.; Ando, K.: Asymmetric Vinylogous Michael Addition of Furanones to Nitroolefines
0681
Jaganathan, A.; Garzan, A.; Whitehead, D. C.; Staples, R. J.; Borhan, B.: Catalytic Asymmetric Chlorocyclization of Unsaturated Amides to Heterocycles

Polymer-Supported Synthesis

z683
All PDFs of this category
0683
Stein, M.; Wieland, J.; Steurer, P.; Tölle, F.; Mülhaupt, R.; Breit, B.: Hydrogenation with Iron Nanoparticles Supported on CDG
0684
Yu, Y.; Hu, T.; Chen, X.; Xu, K.; Zhang, J.; Huang, J.: Suzuki-Miyaura Coupling with Pd(OAc)2 Supported on an Ionic Copolymer
0685
Carter, C. F.; Lange, H.; Sakai, D.; Baxendale, I. R.; Ley, S. V.: Crotylation and Homopropargylation by Flow Technology
0686
Panda, N.; Jena, A. K.; Mohapatra, S.; Rout, S. R.: CuFe2O4 Nanoparticles for N-Arylation of Heterocycles
0687
D’Elia, V.; Liu, Y.; Zipse, H.: Immobilized DMAP Derivatives Rivaling Homogeneous DMAP
0688
Chen, J.-M.; Zeng, X.-M.; Middleton, K.; Zhdankin, V. V.: Recyclable Polystyrene-Supported (Dichloroiodo)benzene
0689
Yoshimura, K.; Oishi, T.; Yamaguchi, K.; Mizuno, N.: Synthesis of N,N-Bicyclic Pyrazolidinones Using Cu(OH)x/Al2O3
0690
Jang, Y.; Kim, S.; Jun, S. W.; Kim, B. H.; Hwang, S.; Song, I. K.; Kim, B. M.; Hyeon, T.: Reduction of Nitroarenes and Alkenes with Rh-Fe3O4 Nanocrystals
0691
Hoshiya, N.; Shuto, S.; Arisawa, M.: Suzuki-Miyaura Coupling with Sulfur-Modified Gold-Supported Palladium
0692
Schaffert, D.; Badgujar, N.; Wagner, E.: Solid-Phase Synthesis of Polyamidoamines
0693
Khan, S. N.; Kim, A.; Grubbs, R. H.; Kwon, Y.-U.: Ring-Closing Metathesis for the Preparation of Cyclic Peptoids
0694
Noujima, A.; Mitsudome, T.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Deoxygenation of Epoxides to Alkenes with H2 Using Au/HT