DOI: 10.1055/s-00000084

Synthesis

Issue 22 · Volume 48 · November 2016 DOI: 10.1055/s-006-32752

review

  • 3821
    Rossi, Renzo; Lessi, Marco; Manzini, Chiara; Marianetti, Giulia; Bellina, Fabio:

    Direct (Hetero)arylation Reactions of (Hetero)arenes as Tools for the Step- and Atom-Economical Synthesis of Biologically Active Unnatural Compounds Including Pharmaceutical Targets

    Image for article: Direct (Hetero)arylation Reactions of (Hetero)arenes as Tools for the Step- and Atom-Economical Synthesis of Biologically Active Unnatural Compounds Including Pharmaceutical Targets

    • short review

  • 3863
    Rintjema, Jeroen; Kleij, Arjan W.:

    Substrate-Assisted Carbon Dioxide Activation as a Versatile Approach for Heterocyclic Synthesis

    Image for article: Substrate-Assisted Carbon Dioxide Activation as a Versatile Approach for Heterocyclic Synthesis
  • 3879
    Besson, Thierry; Fruit, Corinne:

    Recent Developments in Microwave-Assisted Metal-Catalyzed C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications

    Image for article: Recent Developments in Microwave-Assisted Metal-Catalyzed C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications
  • 3890
    Vargas-Caporali, Jorge; Juaristi, Eusebio:

    The Diamino Analogues of Privileged Corey–Bakshi–Shibata and Jørgensen–Hayashi Catalysts: A Comparison of Their Performance

    Image for article: The Diamino Analogues of Privileged Corey–Bakshi–Shibata and Jørgensen–Hayashi Catalysts: A Comparison of Their Performance

    • paper

  • 3907
    Lesma, Giordano; Luraghi, Andrea; Rainoldi, Giulia; Mattiuzzo, Elena; Bortolozzi, Roberta; Viola, Giampietro; Silvani, Alessandra:

    Multicomponent Approach to Bioactive Peptide–Ecdysteroid Conjugates: Creating Diversity at C6 by Means of the Ugi Reaction

    Image for article: Multicomponent Approach to Bioactive Peptide–Ecdysteroid Conjugates: Creating Diversity at C6 by Means of the Ugi Reaction
    Supporting Information (PDF)
  • 3917
    Coman, Anca G.; Paraschivescu, Codruta C.; Hadade, Niculina D.; Juncu, Andrei; Vlaicu, Ovidiu; Popescu, Costin-Ioan; Matache, Mihaela:

    New Acyloxymethyl Ketones: Useful Probes for Cysteine Protease Profiling

    Image for article: New Acyloxymethyl Ketones: Useful Probes for Cysteine Protease Profiling
    Supporting Information (PDF)
  • 3924
    Zhang, Lutao; Tang, Dong; Gao, Jing; Wang, Jing; Wu, Ping; Meng, Xu; Chen, Baohua:

    Direct Access to 1,3,5-Trisubstituted 1H-1,2,4-Triazoles from N-Phenylbenzamidines via Copper-Catalyzed Diamination of Aryl Nitriles

    Image for article: Direct Access to 1,3,5-Trisubstituted 1<i>H</i>-1,2,4-Triazoles from <i>N</i>-Phenylbenzamidines via Copper-Catalyzed Diamination of Aryl Nitriles
    Supporting Information (PDF)
  • 3931
    Akimura, Nozomi; Fujii, Ayaka; Kamada, Fuma; Nogiwa, Ryoki; Yamamoto, Syota; Sato, Teppei; Ishikawa, Syuji; Okazaki, Tatsuya; Kaneda, Kyosuke:

    Synthesis of Tetracyclic Molecules Containing Medium-Sized Heterocycles: Scope Expansion of Cascade Nicholas and Pauson–Khand Methodology

    Image for article: Synthesis of Tetracyclic Molecules Containing Medium-Sized Heterocycles: Scope Expansion of Cascade Nicholas and Pauson–Khand Methodology
    Supporting Information (PDF)
  • 3941
    Yu, Yanhan; Yue, Yixia; Wang, Deqiang; Li, Xue; Chen, Chunxia; Peng, Jinsong:

    Modular Synthesis of Quinazolinone-Fused Phenanthridinones by a Palladium-Catalyzed Cascade C–H/N–H Arylation Process

    Image for article: Modular Synthesis of Quinazolinone-Fused Phenanthridinones by a Palladium-Catalyzed Cascade C–H/N–H Arylation Process
    Supporting Information (PDF)
  • 3951
    Yin, Hongli; Meng, Zhe; Liu, Bo:

    Construction of the Core Structure of Trichotomone

    Image for article: Construction of the Core Structure of Trichotomone
    Supporting Information (PDF)
  • 3957
    Kamiyama, Takuya; Sigrist, Lukas; Cvengroš, Ján:

    Synthesis of Tröger’s Base Analogues via a Phase-Transfer-Catalyzed Double Aza-Michael Reaction under Base-Free Conditions

    Image for article: Synthesis of Tröger’s Base Analogues via a Phase-Transfer-Catalyzed Double Aza-Michael Reaction under Base-Free Conditions
    Supporting Information (PDF)
  • 3965
    Lashmanova, Eugeniya A.; Rybakov, Victor B.; Shiryaev, Andrey K.:

    Synthesis of Adamantylated Pyrimidines Using the Biginelli Reaction

    Image for article: Synthesis of Adamantylated Pyrimidines Using the Biginelli Reaction
    Supporting Information (PDF)
  • 3971
    Omura, Ryuji; Fujiya, Akitoshi; Yamaguchi, Eiji; Tada, Norihiro; Miura, Tsuyoshi; Itoh, Akichika:

    One-Pot Aerobic Photooxidative Darzens Reaction from Styrene and Benzyl Alcohol via Phenacyl Iodide and Benzaldehyde by Using­ Iodine

    Image for article: One-Pot Aerobic Photooxidative Darzens Reaction from Styrene and Benzyl Alcohol via Phenacyl Iodide and Benzaldehyde by Using­ Iodine
    Supporting Information (PDF)
  • 3976
    Ye, Xinglin; Yuan, Jianjun; Zhou, Yirong; Deng, Zhihong; Mao, Xuechun; Peng, Yiyuan:

    Palladium-Catalyzed Cross-Coupling of 4-Tosyloxyquinazolines with Organoindium Reagents: An Efficient Route to 4-Substituted Quinazolines

    Image for article: Palladium-Catalyzed Cross-Coupling of 4-Tosyloxyquinazolines with Organoindium Reagents: An Efficient Route to 4-Substituted Quinazolines
    Supporting Information (PDF)
  • 3985
    Wang, Qi; Wang, Meirong; Li, Hui-Jing; Zhu, Shuai; Liu, Ying; Wu, Yan-Chao:

    Synthesis of Quinolines via Iron-Catalyzed Redox Condensation of Alcohols with 2-Nitrobenzyl Methyl Ether/2-Nitrobenzyl Alcohols

    Image for article: Synthesis of Quinolines via Iron-Catalyzed Redox Condensation of Alcohols with 2-Nitrobenzyl Methyl Ether/2-Nitrobenzyl Alcohols
    Supporting Information (PDF)
  • 3996
    Kadam, Kishorkumar S.; Gandhi, Thirumanavelan; Gupte, Amol; Gangopadhyay, A. K.; Sharma, Rajiv:

    Alkyl Nitrites: Novel Reagents for One-Pot Synthesis of 3,5-Disubstituted Isoxazoles from Aldoximes and Alkynes

    Image for article: Alkyl Nitrites: Novel Reagents for One-Pot Synthesis of 3,5-Disubstituted Isoxazoles from Aldoximes and Alkynes
    Supporting Information (PDF)
  • 4009
    Mondal, Susmita; Samanta, Sadhanendu; Singsardar, Mukta; Mishra, Subhajit; Mitra, Shubhanjan; Hajra, Alakananda:

    Zwitterionic-Type Molten Salt Catalyzed Iodination in Water: Synthesis of Iodoimidazoheterocycles

    Image for article: Zwitterionic-Type Molten Salt Catalyzed Iodination in Water: Synthesis of Iodoimidazoheterocycles
    Supporting Information (PDF)

    • book review

  • 4016
    Lutz, Ackermann:

    Science of Synthesis: Catalytic Transformations via C–H Activation, Workbench Edition, 2 Vol.