DOI: 10.1055/s-00000083

Synlett

Issue 14 · Volume 28 · September 2017 DOI: 10.1055/s-007-34652

Synform

A140
Zanda, Matteo: SYNFORM ISSUE 2017/09

synpacts

1663
Hu, Long; Zhao, Junfeng: Ynamide: A New Coupling Reagent for Amide and Peptide Synthesis
https://www.thieme-connect.de/media/synlett/201714/i_p0279_ga_10-1055_s-0036-1588860.gif
1671
Lu, Dapeng; Cui, Shengsheng; Du, Pingwu: Large π-Extension of Carbon Nanorings by Incorporating Hexa-peri-hexabenzocoronenes
https://www.thieme-connect.de/media/synlett/201714/i_p0201_ga_10-1055_s-0036-1588830.gif

cluster

1678
Reiser, Oliver: Heterocyclic Chemistry – Old Science or the Forefront of Chemistry?
https://www.thieme-connect.de/media/synlett/201714/i_b3000_ga_10-1055_s-0036-1589511.jpg

account

1680
Morimoto, Koji; Dohi, Toshifumi; Kita, Yasuyuki: Metal-free Oxidative Cross-Coupling Reaction of Aromatic Compounds Containing Heteroatoms
https://www.thieme-connect.de/media/synlett/201714/i_a0218_ga_10-1055_s-0036-1588455.gif
1695
Deng, Yongming; Cheng, Qing-Qing; Doyle, Michael P.: Asymmetric [3+3] Cycloaddition for Heterocycle Synthesis
https://www.thieme-connect.de/media/synlett/201714/i_a0230_ga_10-1055_s-0036-1588453.gif

cluster

1707
Hossain, Asik; Pagire, Santosh K.; Reiser, Oliver: Visible-Light-Mediated Synthesis of Pyrazines from Vinyl Azides Utilizing a Photocascade Process
https://www.thieme-connect.de/media/synlett/201714/i_b0533_ga_10-1055_s-0036-1590888.gif
Supporting Information
1715
Mei, Ruhuai; Zhang, Shou-Kun; Ackermann, Lutz: Concise Synthesis of Lamellarin Alkaloids by C–H/N–H Activation: Evaluation of Metal Catalysts in Oxidative Alkyne Annulation
https://www.thieme-connect.de/media/synlett/201714/i_b0539_ga_10-1055_s-0036-1591209.gif
Supporting Information
1719
Sato, Shogo; Kawada, Takuma; Takikawa, Hiroshi; Suzuki, Keisuke: Preparation of 2-Substituted 3-Methoxycarbonyl-4-methoxyfurans that Allow Access to Highly Functionalized Naphthalenes via Regioselective Cycloaddition with Alkoxybenzyne
https://www.thieme-connect.de/media/synlett/201714/i_b0332_ga_10-1055_s-0036-1590825.gif
Supporting Information
1724
Jarrige, Lucie; Merad, Jeremy; Zaied, Siwar; Blanchard, Florent; Masson, Géraldine: Easy Access to Quinolin-2(1H)-ones via a One-Pot Tandem Oxa-Michael–Aldol Sequence
https://www.thieme-connect.de/media/synlett/201714/i_b0305_ga_10-1055_s-0036-1588470.gif
Supporting Information
1729
Patil, Pravin C.; Luzzio, Frederick A.: Unnatural Amino Acid Derivatives through Click Chemistry: Synthesis of Triazolylalanine Analogues
https://www.thieme-connect.de/media/synlett/201714/i_b0340_ga_10-1055_s-0036-1588510.gif
Supporting Information
1733
Kippo, Takashi; Kimura, Yuki; Ueda, Mitsuhiro; Fukuyama, Takahide; Ryu, Ilhyong: Bromine-Radical-Mediated Synthesis of β-Functionalized β,γ- and δ,ε-Unsaturated Ketones via C–H Functionalization of Aldehydes
https://www.thieme-connect.de/media/synlett/201714/i_b0292_ga_10-1055_s-0036-1588494.gif
Supporting Information
1738
Aitken, R. Alan; Harper, Andrew D; Slawin, Alexandra M. Z.: Base-Induced Cyclisation of ortho-Substituted 2-Phenyloxazolines to Give 3-Aminobenzofurans and Related Heterocycles
https://www.thieme-connect.de/media/synlett/201714/i_b0311_ga_10-1055_s-0036-1588503.gif
Supporting Information
1743
Lessing, Timo; Müller, Thomas J. J.: One-Pot Coupling–Cyclization–Alkylation Synthesis of 1,2,5-Trisubstituted 7-Azaindoles in a Consecutive Three-component Fashion
https://www.thieme-connect.de/media/synlett/201714/i_b0330_ga_10-1055_s-0036-1590837.gif
Supporting Information
1748
Talero, Alexánder G.; Burtoloso, Antonio C. B.: Sharpless Asymmetric Dihydroxylation on α,β-Unsaturated Diazoketones: A New Entry for the Synthesis of Disubstituted Furanones
https://www.thieme-connect.de/media/synlett/201714/i_b0414_ga_10-1055_s-0036-1590977.gif
Supporting Information
1753
Parra, Claudio; Solís, Pablo; Bonjoch, Josep; Bradshaw, Ben: A One-Pot Methodology for the Synthesis of the Yohimban Skeleton
https://www.thieme-connect.de/media/synlett/201714/i_b0420_ga_10-1055_s-0036-1589092.gif
Supporting Information
1758
Mai, Duy N.; Uchenik, Dmitriy; Vanderwal, Christopher D.: Efforts Toward a Synthesis of Crotogoudin and Crotobarin
https://www.thieme-connect.de/media/synlett/201714/i_b0554_ga_10-1055_s-0036-1588560.gif
Supporting Information

new tools

1763
Richert, Clemens; Krupp, Felix: Encapsulating Organic Crystals (EnOCs)
https://www.thieme-connect.de/media/synlett/201714/i_b0458_ga_10-1055_s-0036-1590971.gif

letter

1767
He, Jie; Kimani, Flora W.; Jewett, John C.: Rapid in Situ Generation of Benzene Diazonium Ions under Basic Aqueous Conditions from Bench-Stable Triazabutadienes
https://www.thieme-connect.de/media/synlett/201714/i_r0097_ga_10-1055_s-0036-1588797.gif
Supporting Information
1771
Zhang, Xiao-Ru; Zhou, Su-Lan; Yuan, Yi; Du, Wei; Chen, Ying-Chun: Chemo- and Regioselective Asymmetric Friedel–Crafts Reaction of Furans and Thiophenes with α,β-Unsaturated Aldehydes through Dual Activation
https://www.thieme-connect.de/media/synlett/201714/i_w0173_ga_10-1055_s-0036-1588831.gif
Supporting Information
1775
Inamori, Daiki; Miwa, Takuya; Fujihara, Tetsuaki; Tsuji, Yasushi; Terao, Jun: Thieme Chemistry Journals Awardees – Where Are They Now?
Synthesis of a Dinuclear Copper NHC Complex Bearing a Rigid π-Conjugated Cyclic Framework
https://www.thieme-connect.de/media/synlett/201714/i_u0199_ga_10-1055_s-0036-1588824.gif
Supporting Information
1780
Sun, Pengcheng; Tang, Wenli; Huang, Yu; Hu, Bi-Huang: Improved Fmoc Solid-Phase Peptide Synthesis of Oxytocin with High Bioactivity
https://www.thieme-connect.de/media/synlett/201714/i_w0240_ga_10-1055_s-0036-1589037.gif
Supporting Information
1785
Yavari, Issa; Khajeh-Khezri, Aliyeh; Bahemmat, Samira; Halvagar, Mohammad Reza: A Synthesis of Novel Dioxapropellanes from the Knoevenagel Adducts of Acenaphthoquinone and 3-Oxo-3-arylpropionitriles in Aqueous Methanol
https://www.thieme-connect.de/media/synlett/201714/i_d0023_ga_10-1055_s-0036-1588822.gif
Supporting Information
1789
Szantai-Kis, D. Miklos; Walters, Christopher R.; Barrett, Taylor M.; Hoang, Eileen M.; Petersson, E. James: Thieme Chemistry Journals Awardees – Where Are They Now?
Improved Fmoc Deprotection Methods for the Synthesis of Thioamide-Containing Peptides and Proteins
https://www.thieme-connect.de/media/synlett/201714/i_r0178_ga_10-1055_s-0036-1589027.gif
Supporting Information
1795
Chen, Zhengkai; Cao, Gangjian; Zhang, Fengjin; Li, Hongli; Xu, Jianfeng; Miao, Maozhong; Ren, Hongjun: Metal-Free Mediated C-3 Methylsulfanylation of Imidazo[1,2-a]-pyridines with Dimethyl Sulfoxide as a Methylsulfanylating Agent
https://www.thieme-connect.de/media/synlett/201714/i_w0152_ga_10-1055_s-0036-1588419.gif
Supporting Information
1801
Zhao, Mingzhu; Tian, Yawei; Zhao, Xiaoming: Thieme Chemistry Journals Awardees – Where Are They Now?
Chiral Sulfinamide Ligands and Pd-Catalyzed Asymmetric Allylic Alkylations of Ethyl 2-Fluoroacetoacetate
https://www.thieme-connect.de/media/synlett/201714/i_w0191_ga_10-1055_s-0036-1589033.gif
Supporting Information
1807
Tang, Ruotian; Jiang, Chunfeng; Li, Hongliang; Li, Wei; Xu, Youjun: Facile Synthesis of N-Substituted 4-Amino-6-methyl Resorcinols from Polysubstituted Cyclohexanone
https://www.thieme-connect.de/media/synlett/201714/i_w0263_ga_10-1055_s-0036-1590817.gif
Supporting Information
1811
Ho, Son Long; Dao, Pham Duy Quang; Cho, Chan Sik: Microwave-Assisted Synthesis of Benzo[4,5]imidazo[1,2-a]pyrimidines from β-Bromo-α,β-unsaturated Aldehydes and 2-Aminobenzimidazoles
https://www.thieme-connect.de/media/synlett/201714/i_u0161_ga_10-1055_s-0036-1588834.gif
1816
Yoshimura, Fumihiko; Saito, Hiroki; Abe, Taiki; Tanino, Keiji: Nucleophilic Addition of Alkanenitriles to Aldehydes via N-Silyl Ketene Imines Generated In Situ
https://www.thieme-connect.de/media/synlett/201714/i_u0185_ga_10-1055_s-0036-1588424.gif
Supporting Information
1821
Zhu, Yi-Fan; Geng, Xin-Le; Guan, Yong-Hong; Teng, Wei; Fan, Xiaohui: Poly(phosphoric acid) (PPA)-Promoted 5-exo-Cyclization of Iminium Ions Generated In Situ: A Facile Access to Functionalized Indene Derivatives
https://www.thieme-connect.de/media/synlett/201714/i_w0060_ga_10-1055_s-0036-1589009.gif
Supporting Information
1828
Yu, Haifeng; Zhao, Lijuan; Diao, Quanping; Li, Tiechun; Liao, Peiqiu; Hou, Dongyan; Xin, Guang: FeCl3·6H2O-Catalyzed Tandem Alkylation–Hydrolysis Reaction of Chain α-Oxo Ketene Dithioacetals with Alcohols: Efficient ­Synthesis of α-Alkylated β-Oxo Thioesters
https://www.thieme-connect.de/media/synlett/201714/i_w0079_ga_10-1055_s0036-1588982.gif
Supporting Information
1835
Peng, Zhihua; Yu, Zhi; Chen, Dong-Huang; Liang, Shuyuan; Zhang, Liwei; Zhao, Dezhi; Song, Linhua; Jiang, Cuiyu: Efficient C(sp3)–H Bond Arylation of Tetrahydroisoquinolines with Knochel-Type Arylzinc Reagents under Oxidative Conditions
https://www.thieme-connect.de/media/synlett/201714/i_w0113_ga_10-1055_s-0036-1589029.gif
Supporting Information
1840
Chen, Xiang-Xiang; Wang, Jia-Xin; Ren, Jiang-Tao; Xie, Hu; Zhao, Yanxia; Li, Ya-Min; Sun, Meng: A Convenient Strategy for Remote C–H Bond Halogenation of 8-Aminoquinolines in the C5 Position
https://www.thieme-connect.de/media/synlett/201714/i_w0174_ga_10-1055_s-0036-1588420.gif
Supporting Information Primary Data
1845
Guo, Tao; Wang, Hongyan: Copper-Mediated Direct Sulfenylation of 4-Hydroxyquinolinones and 4-Hydroxypyridones with Aryl Thiols via a C−H Functionalization Process
https://www.thieme-connect.de/media/synlett/201714/i_w0177_ga_10-1055_s-0036-1588829.gif
Supporting Information
1852
Gao, Hongjie; Xu, Xiangsheng; Xu, Jianfeng: Sc(OTf)3-Catalyzed Aza-Friedel–Crafts Reaction of Electron-Rich Arenes with Isatin-Derived Ketimines: Access to 3-Amino-3-Aryl-2-Oxindoles
https://www.thieme-connect.de/media/synlett/201714/i_w0202_ga_10-1055_s-0036-1588432.gif
Supporting Information