DOI: 10.1055/s-00000083

Synlett

Issue 14 · Volume 28 · September 2017 DOI: 10.1055/s-007-34652

Synform

  • A140
    Zanda, Matteo:

    SYNFORM ISSUE 2017/09

    • synpacts

  • 1663
    Hu, Long; Zhao, Junfeng:

    Ynamide: A New Coupling Reagent for Amide and Peptide Synthesis

    Image for article: Ynamide: A New Coupling Reagent for Amide and Peptide Synthesis
  • 1671
    Lu, Dapeng; Cui, Shengsheng; Du, Pingwu:

    Large π-Extension of Carbon Nanorings by Incorporating Hexa-peri-hexabenzocoronenes

    Image for article: Large π-Extension of Carbon Nanorings by Incorporating Hexa-<i>peri</i>-hexabenzocoronenes

    • cluster

  • 1678
    Reiser, Oliver:

    Heterocyclic Chemistry – Old Science or the Forefront of Chemistry?

    Image for article: Heterocyclic Chemistry – Old Science or the Forefront of Chemistry?

    • account

  • 1680
    Morimoto, Koji; Dohi, Toshifumi; Kita, Yasuyuki:

    Metal-free Oxidative Cross-Coupling Reaction of Aromatic Compounds Containing Heteroatoms

    Image for article: Metal-free Oxidative Cross-Coupling Reaction of Aromatic Compounds Containing Heteroatoms
  • 1695
    Deng, Yongming; Cheng, Qing-Qing; Doyle, Michael P.:

    Asymmetric [3+3] Cycloaddition for Heterocycle Synthesis

    Image for article: Asymmetric [3+3] Cycloaddition for Heterocycle Synthesis

    • cluster

  • 1707
    Hossain, Asik; Pagire, Santosh K.; Reiser, Oliver:

    Visible-Light-Mediated Synthesis of Pyrazines from Vinyl Azides Utilizing a Photocascade Process

    Image for article: Visible-Light-Mediated Synthesis of Pyrazines from Vinyl Azides Utilizing a Photocascade Process
    Supporting Information (PDF)
  • 1715
    Mei, Ruhuai; Zhang, Shou-Kun; Ackermann, Lutz:

    Concise Synthesis of Lamellarin Alkaloids by C–H/N–H Activation: Evaluation of Metal Catalysts in Oxidative Alkyne Annulation

    Image for article: Concise Synthesis of Lamellarin Alkaloids by C–H/N–H Activation: Evaluation of Metal Catalysts in Oxidative Alkyne Annulation
    Supporting Information (PDF)
  • 1719
    Sato, Shogo; Kawada, Takuma; Takikawa, Hiroshi; Suzuki, Keisuke:

    Preparation of 2-Substituted 3-Methoxycarbonyl-4-methoxyfurans that Allow Access to Highly Functionalized Naphthalenes via Regioselective Cycloaddition with Alkoxybenzyne

    Image for article: Preparation of 2-Substituted 3-Methoxycarbonyl-4-methoxyfurans that Allow Access to Highly Functionalized Naphthalenes via Regioselective Cycloaddition with Alkoxybenzyne
    Supporting Information (PDF)
  • 1724
    Jarrige, Lucie; Merad, Jeremy; Zaied, Siwar; Blanchard, Florent; Masson, Géraldine:

    Easy Access to Quinolin-2(1H)-ones via a One-Pot Tandem Oxa-Michael–Aldol Sequence

    Image for article: Easy Access to Quinolin-2(1<i>H</i>)-ones via a One-Pot Tandem Oxa-Michael–Aldol Sequence
    Supporting Information (PDF)
  • 1729
    Patil, Pravin C.; Luzzio, Frederick A.:

    Unnatural Amino Acid Derivatives through Click Chemistry: Synthesis of Triazolylalanine Analogues

    Image for article: Unnatural Amino Acid Derivatives through Click Chemistry: Synthesis of Triazolylalanine Analogues
    Supporting Information (PDF)
  • 1733
    Kippo, Takashi; Kimura, Yuki; Ueda, Mitsuhiro; Fukuyama, Takahide; Ryu, Ilhyong:

    Bromine-Radical-Mediated Synthesis of β-Functionalized β,γ- and δ,ε-Unsaturated Ketones via C–H Functionalization of Aldehydes

    Image for article: Bromine-Radical-Mediated Synthesis of β-Functionalized β,γ- and δ,ε-Unsaturated Ketones via C–H Functionalization of Aldehydes
    Supporting Information (PDF)
  • 1738
    Aitken, R. Alan; Harper, Andrew D; Slawin, Alexandra M. Z.:

    Base-Induced Cyclisation of ortho-Substituted 2-Phenyloxazolines to Give 3-Aminobenzofurans and Related Heterocycles

    Image for article: Base-Induced Cyclisation of <i>ortho</i>-Substituted 2-Phenyloxazolines to Give 3-Aminobenzofurans and Related Heterocycles
    Supporting Information (PDF)
  • 1743
    Lessing, Timo; Müller, Thomas J. J.:

    One-Pot Coupling–Cyclization–Alkylation Synthesis of 1,2,5-Trisubstituted 7-Azaindoles in a Consecutive Three-component Fashion

    Image for article: One-Pot Coupling–Cyclization–Alkylation Synthesis of 1,2,5-Trisubstituted 7-Azaindoles in a Consecutive Three-component Fashion
    Supporting Information (PDF)
  • 1748
    Talero, Alexánder G.; Burtoloso, Antonio C. B.:

    Sharpless Asymmetric Dihydroxylation on α,β-Unsaturated Diazoketones: A New Entry for the Synthesis of Disubstituted Furanones

    Image for article: Sharpless Asymmetric Dihydroxylation on α,β-Unsaturated Diazoketones: A New Entry for the Synthesis of Disubstituted Furanones
    Supporting Information (PDF)
  • 1753
    Parra, Claudio; Solís, Pablo; Bonjoch, Josep; Bradshaw, Ben:

    A One-Pot Methodology for the Synthesis of the Yohimban Skeleton

    Image for article: A One-Pot Methodology for the Synthesis of the Yohimban Skeleton
    Supporting Information (PDF)
  • 1758
    Mai, Duy N.; Uchenik, Dmitriy; Vanderwal, Christopher D.:

    Efforts Toward a Synthesis of Crotogoudin and Crotobarin

    Image for article: Efforts Toward a Synthesis of Crotogoudin and Crotobarin
    Supporting Information (PDF)

    • new tools

  • 1763
    Richert, Clemens; Krupp, Felix:

    Encapsulating Organic Crystals (EnOCs)

    Image for article: Encapsulating Organic Crystals (EnOCs)
    Open Access

    • letter

  • 1767
    He, Jie; Kimani, Flora W.; Jewett, John C.:

    Rapid in Situ Generation of Benzene Diazonium Ions under Basic Aqueous Conditions from Bench-Stable Triazabutadienes

    Image for article: Rapid <i>in Situ</i> Generation of Benzene Diazonium Ions under Basic Aqueous Conditions from Bench-Stable Triazabutadienes
    Supporting Information (PDF)
  • 1771
    Zhang, Xiao-Ru; Zhou, Su-Lan; Yuan, Yi; Du, Wei; Chen, Ying-Chun:

    Chemo- and Regioselective Asymmetric Friedel–Crafts Reaction of Furans and Thiophenes with α,β-Unsaturated Aldehydes through Dual Activation

    Image for article: Chemo- and Regioselective Asymmetric Friedel–Crafts Reaction of Furans and Thiophenes with α,β-Unsaturated Aldehydes through Dual Activation
    Supporting Information (PDF)
  • 1775
    Inamori, Daiki; Miwa, Takuya; Fujihara, Tetsuaki; Tsuji, Yasushi; Terao, Jun:

    Thieme Chemistry Journals Awardees – Where Are They Now?
    Synthesis of a Dinuclear Copper NHC Complex Bearing a Rigid π-Conjugated Cyclic Framework

    Image for article: Thieme Chemistry Journals Awardees – Where Are They Now?<break/>Synthesis of a Dinuclear Copper NHC Complex Bearing a Rigid π-Conjugated Cyclic Framework
    Supporting Information (PDF)
  • 1780
    Sun, Pengcheng; Tang, Wenli; Huang, Yu; Hu, Bi-Huang:

    Improved Fmoc Solid-Phase Peptide Synthesis of Oxytocin with High Bioactivity

    Image for article: Improved Fmoc Solid-Phase Peptide Synthesis of Oxytocin with High Bioactivity
    Supporting Information (PDF)
  • 1785
    Yavari, Issa; Khajeh-Khezri, Aliyeh; Bahemmat, Samira; Halvagar, Mohammad Reza:

    A Synthesis of Novel Dioxapropellanes from the Knoevenagel Adducts of Acenaphthoquinone and 3-Oxo-3-arylpropionitriles in Aqueous Methanol

    Image for article: A Synthesis of Novel Dioxapropellanes from the Knoevenagel Adducts of Acenaphthoquinone and 3-Oxo-3-arylpropionitriles in Aqueous Methanol
    Supporting Information (PDF)
  • 1789
    Szantai-Kis, D. Miklos; Walters, Christopher R.; Barrett, Taylor M.; Hoang, Eileen M.; Petersson, E. James:

    Thieme Chemistry Journals Awardees – Where Are They Now?
    Improved Fmoc Deprotection Methods for the Synthesis of Thioamide-Containing Peptides and Proteins

    Image for article: Thieme Chemistry Journals Awardees – Where Are They Now?<break/>Improved Fmoc Deprotection Methods for the Synthesis of Thioamide-Containing Peptides and Proteins
    Supporting Information (PDF)
  • 1795
    Chen, Zhengkai; Cao, Gangjian; Zhang, Fengjin; Li, Hongli; Xu, Jianfeng; Miao, Maozhong; Ren, Hongjun:

    Metal-Free Mediated C-3 Methylsulfanylation of Imidazo[1,2-a]-pyridines with Dimethyl Sulfoxide as a Methylsulfanylating Agent

    Image for article: Metal-Free Mediated C-3 Methylsulfanylation of Imidazo[1,2-<i>a</i>]-pyridines with Dimethyl Sulfoxide as a Methylsulfanylating Agent
    Supporting Information (PDF)
  • 1801
    Zhao, Mingzhu; Tian, Yawei; Zhao, Xiaoming:

    Thieme Chemistry Journals Awardees – Where Are They Now?
    Chiral Sulfinamide Ligands and Pd-Catalyzed Asymmetric Allylic Alkylations of Ethyl 2-Fluoroacetoacetate

    Image for article: Thieme Chemistry Journals Awardees – Where Are They Now?<break/>Chiral Sulfinamide Ligands and Pd-Catalyzed Asymmetric Allylic Alkylations of Ethyl 2-Fluoroacetoacetate
    Supporting Information (PDF)
  • 1807
    Tang, Ruotian; Jiang, Chunfeng; Li, Hongliang; Li, Wei; Xu, Youjun:

    Facile Synthesis of N-Substituted 4-Amino-6-methyl Resorcinols from Polysubstituted Cyclohexanone

    Image for article: Facile Synthesis of N-Substituted 4-Amino-6-methyl Resorcinols from Polysubstituted Cyclohexanone
    Supporting Information (PDF)
  • 1811
    Ho, Son Long; Dao, Pham Duy Quang; Cho, Chan Sik:

    Microwave-Assisted Synthesis of Benzo[4,5]imidazo[1,2-a]pyrimidines from β-Bromo-α,β-unsaturated Aldehydes and 2-Aminobenzimidazoles

    Image for article: Microwave-Assisted Synthesis of Benzo[4,5]imidazo[1,2-<i>a</i>]pyrimidines from β-Bromo-α,β-unsaturated Aldehydes and 2-Aminobenzimidazoles
  • 1816
    Yoshimura, Fumihiko; Saito, Hiroki; Abe, Taiki; Tanino, Keiji:

    Nucleophilic Addition of Alkanenitriles to Aldehydes via N-Silyl Ketene Imines Generated In Situ

    Image for article: Nucleophilic Addition of Alkanenitriles to Aldehydes via <i>N</i>-Silyl Ketene Imines Generated In Situ
    Supporting Information (PDF)
  • 1821
    Zhu, Yi-Fan; Geng, Xin-Le; Guan, Yong-Hong; Teng, Wei; Fan, Xiaohui:

    Poly(phosphoric acid) (PPA)-Promoted 5-exo-Cyclization of Iminium Ions Generated In Situ: A Facile Access to Functionalized Indene Derivatives

    Image for article: Poly(phosphoric acid) (PPA)-Promoted 5-<i>exo</i>-Cyclization of Iminium Ions Generated In Situ: A Facile Access to Functionalized Indene Derivatives
    Supporting Information (PDF)
  • 1828
    Yu, Haifeng; Zhao, Lijuan; Diao, Quanping; Li, Tiechun; Liao, Peiqiu; Hou, Dongyan; Xin, Guang:

    FeCl3·6H2O-Catalyzed Tandem Alkylation–Hydrolysis Reaction of Chain α-Oxo Ketene Dithioacetals with Alcohols: Efficient ­Synthesis of α-Alkylated β-Oxo Thioesters

    Image for article: FeCl<sub>3</sub>·6H<sub>2</sub>O-Catalyzed Tandem Alkylation–Hydrolysis Reaction of Chain α-Oxo Ketene Dithioacetals with Alcohols: Efficient ­Synthesis of α-Alkylated β-Oxo Thioesters
    Supporting Information (PDF)
  • 1835
    Peng, Zhihua; Yu, Zhi; Chen, Dong-Huang; Liang, Shuyuan; Zhang, Liwei; Zhao, Dezhi; Song, Linhua; Jiang, Cuiyu:

    Efficient C(sp3)–H Bond Arylation of Tetrahydroisoquinolines with Knochel-Type Arylzinc Reagents under Oxidative Conditions

    Image for article: Efficient C(sp<sup>3</sup>)–H Bond Arylation of Tetrahydroisoquinolines with Knochel-Type Arylzinc Reagents under Oxidative Conditions
    Supporting Information (PDF)
  • 1840
    Chen, Xiang-Xiang; Wang, Jia-Xin; Ren, Jiang-Tao; Xie, Hu; Zhao, Yanxia; Li, Ya-Min; Sun, Meng:

    A Convenient Strategy for Remote C–H Bond Halogenation of 8-Aminoquinolines in the C5 Position

    Image for article: A Convenient Strategy for Remote C–H Bond Halogenation of 8-Aminoquinolines in the C5 Position
    Supporting Information (PDF) Primary Data (ZIP)
  • 1845
    Guo, Tao; Wang, Hongyan:

    Copper-Mediated Direct Sulfenylation of 4-Hydroxyquinolinones and 4-Hydroxypyridones with Aryl Thiols via a C−H Functionalization Process

    Image for article: Copper-Mediated Direct Sulfenylation of 4-Hydroxyquinolinones and 4-Hydroxypyridones with Aryl Thiols via a C−H Functionalization Process
    Supporting Information (PDF)
  • 1852
    Gao, Hongjie; Xu, Xiangsheng; Xu, Jianfeng:

    Sc(OTf)3-Catalyzed Aza-Friedel–Crafts Reaction of Electron-Rich Arenes with Isatin-Derived Ketimines: Access to 3-Amino-3-Aryl-2-Oxindoles

    Image for article: Sc(OTf)<sub>3</sub>-Catalyzed Aza-Friedel–Crafts Reaction of Electron-Rich Arenes with Isatin-Derived Ketimines: Access to 3-Amino-3-Aryl-2-Oxindoles
    Supporting Information (PDF)