DOI: 10.1055/s-00000083

Synlett

eFirst

Publication Date: 10 June 2025

letter > Hydrogen Atom Transfer Reactions

Mori, Soichiro; Entgelmeier, Lukas-Maximilian; Kansaku, Yaoki; Truong, Duc An; Mancheño, Olga García; Ohmatsu, Kohsuke; Ooi, Takashi: Zwitterionic Acridinium Amidate for Photocatalytic Acceptorless Dehydrogenation
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synpacts

Wheatley, Emilie; Silvi, Mattia: One Carbon at a Time: Unlocking Iterative Carboxylic Acid Homologation
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Publication Date: 05 June 2025

letter > Small Molecules in Medicinal Chemistry

Das, Debojyoti; Sadhukhan, Juheli; Mandal, Pabitra; Pramanik, Smritimoy; Kabir, Alomgir Shah; Adhikari, Susanta Sekhar: Synthesis of Novel Coumarin-Appended Dihydrothiopyrimidinones and Evaluation of Their Binding Interactions with Bovine Serum Albumin
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Supporting Information

Publication Date: 04 June 2025

letter

Sakamoto, Kaori; Oda, Wakana; Kobayashi, Yusuke; Matsuo, Jun-ichi; Furuta, Takumi; Hamada, Shohei: Accelerating Effect of the Addition of HFIP on the Oxidation of Alcohols Using TEMPO/PIDA
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perspectives > Small Molecules in Medicinal Chemistry

Sanjaykumar, Randhe Siddhant; Basavaraj, Chavan Sagar; Arshad, Anam Sania Md.; Singh, Rohit; Mahindroo, Neeraj: A Decade of FDA-Approved Pharmacophore-Based Small Molecules: Advances in Medicinal Chemistry from 2014 to 2024
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Publication Date: 03 June 2025

account > Emerging Trends in Organic Chemistry: A Focus on India

Handique, Prapti Priyam; Paul, Subham; Dutta, Papia; Gogoi, Pinky; Morang, Jita; Dutta, Minmoy; Borah, Ruli: Advances in Organic Synthesis on Ionic Liquid Platforms: An Account of Indian Research Contributions
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letter > Small Molecules in Medicinal Chemistry

Dastari, Sowmya; Panda, Biswajit; Rasane, Sai; Reddyrajula, Rajkumar; Godugu, Chandraiah; Shankaraiah, Nagula: Design, Synthesis, and In Vitro Cytotoxicity Studies of 1H-Benzimidazol-2-yl–Enaminone Hybrids as Tubulin Polymerization Inhibitors
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letter

Fang, Huasu; Yuwen, Liyan; Qi, Yayu; Wang, Jingwen; Zhang, Qing-Wei: Nickel-Catalyzed Nucleophilic Substitution of Cyclopropenes by Secondary Phosphines
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Publication Date: 02 June 2025

letter > Emerging Trends in Organic Chemistry: A Focus on India

Alam, Mohammad Sarwar; Kale, Balkrishna Ramchandra; Hamid, Hinna; Kale, Raju: Zinc Triflate Catalyzed Tandem One-Pot Regioselective Synthesis of Highly Functionalized Pyrrole Derivatives
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Publication Date: 28 May 2025

letter > Emerging Trends in Organic Chemistry: A Focus on India

Kurella, Sreenivasulu; Mamidipalli, Phani; Alla, Sampath; Kumari, Neha; Reddy V, Prabhakar; Sharon, Ashoke; Achanta, Srinivas; Bandichhor, Rakeshwar: Synthesis of Sacubitril Isomers Governed by Differential Facial Selectivity during the Hydrogenation of Conjugated System
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letter > First-Row Transition-Metal Catalysis for Organic Synthesis

Li, Guanbo; Liu, Weiping: Manganese-Catalyzed α-Trideuteromethylation of Sulfones
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letter

Samsonenko, Anna L.; Kostyuchenko, Anastasia S.; Zheleznova, Tatyana Y.; Uliankin, Evgenii B.; Chernenko, Sergei A.; Shuvalov, Vladislav Y.; Shatsauskas, Anton L.; Fisyuk, Alexander S.: Divergent Approach to the Synthesis of 2-Aryl-5-(thiophen-2-yl)-1,3,4-oxadiazoles and -1,3,4-thiadiazoles
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letter

Wen, Yuanjie; Wang, Yurou; Liang, Jianqing; Yan, Yaolong; Chen, Weifeng: Direct Alkynylation of Carbonyl Compounds Using an Efficient Catalytic System: Triisopropylsilanol/KOH
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synpacts

Gan, Yu; Li, Xuejiao; Zhou, Jun-Feng; Ye, Baihua: Selective Open-Shell Nickel Catalysis Driven by Redox-Transmetalation
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Publication Date: 27 May 2025

letter

Miyasaka, Tadachika; Kudo, Yuta; Mari, Yotsu-Yamashita; Adachi, Masaatsu; Nishikawa, Toshio: Synthetic Studies toward 4,9-Anhydro-10-hemiketal-5-deoxy-tetrodotoxin, a Proposed Biosynthetic Precursor of Tetrodotoxin
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letter

Shao, Hai-Yang; Sun, Meng; Yu, Yan-Cheng; Sun, Shan-Liang; Li, Nian-Guang; Cao, Peng: Semi-Synthesis of (+)-Digitoxigenin: Selective Bromination for Construction of the Key Intermediate
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Publication Date: 26 May 2025

letter > Small Molecules in Medicinal Chemistry

Chvatal, Jo; Nguyen, Dat T.; Xie, Alexondra S.; Parsons, William H.: Synthesis and Evaluation of N-Arylsulfonylated Succinimides as Activity-Based Probes
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Publication Date: 23 May 2025

letter > Small Molecules in Medicinal Chemistry

Alaeddini, AmirHossein; Karimian, Somaye; Noori, Milad; Dastyafteh, Navid; Mohammadi-Khanaposhtani, Maryam; Ghomi, Minoo Khalili; Bararjanian, Morteza; Iraji, Aida; Javanshir, Shahrzad; Larijani, Bagher; Ranjbar, Parviz Rashidi; Mahdavi, Mohammad: Design, Synthesis, Enzymatic Inhibition, and Antioxidant Activity of New 4-Phenylpiperazin-phenoxy-1,2,3-triazol-acetamide Derivatives as Tyrosinase Inhibitors
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letter > Small Molecules in Medicinal Chemistry

Peprah, Paul K.; Spitznagel, Brittany D.; Du, Yu; Nguyen, Dalena; Weaver, C. David; Emmitte, Kyle A.: Efficient Regioselective Synthesis of Benzimidazoles and Azabenz­imidazoles to Enable the Rapid Development of Structure–Activity Relationships for Activation of SLACK Potassium Channels
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Publication Date: 22 May 2025

letter > First-Row Transition-Metal Catalysis for Organic Synthesis

Ye, Fu; Liu, Peiwen; Yang, Yiqian; Gao, Wei; Yuan, Weiming: Nickel/Photoredox-Catalyzed Three-Component Dialkylation of Alkenes for the Synthesis of β-Amino Acid Derivatives
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