DOI: 10.1055/s-00000084

Synthesis

Issue 01 · Volume 44 · January 2012 DOI: 10.1055/s-002-22693

synform

  • A1
    Zanda, Matteo:

    SYNFORM ISSUE 2012/1

    • review

  • 1
    Zhang, Ming; Zhang, Aiqin:

    Non-Cyclizing Direct Transformation of Arene Carbon-Hydrogen Bonds into Carbon-Nitrogen Bonds

    Image for article: Non-Cyclizing Direct Transformation of Arene Carbon-Hydrogen Bonds into Carbon-Nitrogen Bonds
  • 15
    Kandepi, V. V. Krishna Mohan; Narender, Nama:

    Ecofriendly Oxidative Nuclear Halogenation of Aromatic Compounds Using Potassium and Ammonium Halides

    Image for article: Ecofriendly Oxidative Nuclear Halogenation of Aromatic Compounds Using Potassium and Ammonium Halides

    • feature article

  • 27
    Marti, Alex; Peruncheralathan, Saravanan; Schneider, Christoph:

    Cationic Late-Transition-Metal Complexes Catalyze the Ring Opening of Aziridines with Amines

    Image for article: Cationic Late-Transition-Metal Complexes Catalyze the Ring Opening of Aziridines with Amines

    • practical synthetic procedures

  • 37
    Rossy, Cybille; Fouquet, Eric; Felpin, François-Xavier:

    A Sustainable Procedure Combining the Advantages of Both Homogeneous and Heterogeneous Catalysis for the Heck-Matsuda Reaction

    Image for article: A Sustainable Procedure Combining the Advantages of Both Homogeneous and Heterogeneous Catalysis for the Heck-Matsuda Reaction

    • paper

  • 42
    Kim, Bo Ram; Lee, Hyung-Geun; Kang, Seung-Beom; Sung, Gi Hyeon; Kim, Jeum-Jong; Park, Jong Keun; Lee, Sang-Gyeong; Yoon, Yong-Jin:

    tert-Butoxide-Assisted Amidation of Esters under Green Conditions

    Image for article: <EM EMTYPE="ITALIC">tert</EM>-Butoxide-Assisted Amidation of Esters under Green Conditions
    Supporting Information (PDF)
  • 51
    Ye, Haiwei; Yu, Chuanming; Zhong, Weihui:

    New Procedure for the Preparation of (1R,2R)-2-[(R)-3-(Benzyloxy)pyr­rolidin-1-yl]cyclohexanol

    Image for article: New Procedure for the Preparation of (1<EM EMTYPE="ITALIC">R</EM>,2<EM EMTYPE="ITALIC">R</EM>)-2-[(<EM EMTYPE="ITALIC">R</EM>)-3-(Benzyloxy)pyr­rolidin-1-yl]cyclohexanol
    Supporting Information (PDF)
  • 57
    McElhinny Jr., Charles J.; Carroll, F. I.; Lewin, Anita H.:

    A Practical, Laboratory-Scale Synthesis of Perampanel

    Image for article: A Practical, Laboratory-Scale Synthesis of Perampanel
  • 63
    Maeng, Jun-Ho; Yang, Zhicai; Manning, David D.; Masih, Liaqat; Cao, Yeyu; Pattamana, Kevin G.; Bois, Frederic; Molino, Bruce F.:

    Organozirconium Chemistry on Cyclosporin: A Novel Process for the Highly Stereoselective Synthesis of (E)-ISA247 (Voclosporin) and Close Analogues

    Image for article: Organozirconium Chemistry on Cyclosporin: A Novel Process for the Highly Stereoselective Synthesis of (<EM EMTYPE="ITALIC">E</EM>)-ISA247 (Voclosporin) and Close Analogues
  • 69
    Antoine, Maud; Gerlach, Matthias; Günther, Eckhard; Schuster, Tilmann; Czech, Michael; Seipelt, Irene; Marchand, Pascal:

    A Convenient Synthesis of Novel 2,8-Disubstituted Pyrido[3,4-b]pyrazines Possessing Biological Activity

    Image for article: A Convenient Synthesis of Novel 2,8-Disubstituted Pyrido[3,4-<EM EMTYPE="ITALIC">b</EM>]pyrazines Possessing Biological Activity
  • 83
    Damodar, Kongara; Das, Biswanath:

    (N-tert-Butanesulfinyl)imines in Alkaloid Synthesis: Concise Formal Syntheses of the Dendrobate Alkaloid (+)-241D and Its C-4 Epimer

    Image for article: (<EM EMTYPE="ITALIC">N</EM>-<EM EMTYPE="ITALIC">tert</EM>-Butanesulfinyl)imines in Alkaloid Synthesis: Concise Formal Syntheses of the Dendrobate Alkaloid (+)-241D and Its C-4 Epimer
    Supporting Information (PDF)
  • 87
    Majumdar, K. C.; De, Nirupam; Ghosh, Debankan; Ponra, Sudipta; Roy, B.:

    Copper(II) Triflate Promoted One-Pot Synthesis of Coumarin-, Quinolone-, and Naphthalene-Annulated 2-Aminothiazoles under Ligand-Free Conditions

    Image for article: Copper(II) Triflate Promoted One-Pot Synthesis of Coumarin-, Quinolone-, and Naphthalene-Annulated 2-Aminothiazoles under Ligand-Free Conditions
  • 93
    Lagadic, Elodie; Garcia, Yann; Marchand-Brynaert, Jacqueline:

    Selective Protection and Deprotection of ortho-Functionalized Arylphosphonates

    Image for article: Selective Protection and Deprotection of <EM EMTYPE="ITALIC">ortho</EM>-Functionalized Arylphosphonates
  • 99
    Pu, Ye; Gao, Liumian; Liu, Huijun; Yan, Jie:

    An Effective Catalytic α-Phosphoryloxylation of Ketones with Iodobenzene

    Image for article: An Effective Catalytic α-Phosphoryloxylation of Ketones with Iodobenzene
  • 104
    Ye, Jia-Hai; Wang, Guangpu; Huang, Chengmei; Hu, Zhengjuan; Zhang, Whenchao; Zhang, Yan:

    An Efficient and Convenient Bromination of BODIPY Derivatives with Copper(II) Bromide

    Image for article: An Efficient and Convenient Bromination of BODIPY Derivatives with Copper(II) Bromide
    Supporting Information (PDF)
  • 111
    Cui, Bing; Kong, Shasha; Wu, Guiping; Miao, Zhiwei; Chen, Ruyu:

    Lewis Acid Catalyzed Diastereoselective Vinylogous Mannich Reaction Induced by O-Pivaloylated d-Galactosylamine as the Chiral Auxiliary: Stereoselective Synthesis of 6-Arylpiperidin-2-ones

    Image for article: Lewis Acid Catalyzed Diastereoselective Vinylogous Mannich Reaction Induced by O-Pivaloylated <EM EMTYPE="CAPS">d</EM>-Galactosylamine as the Chiral Auxiliary: Stereoselective Synthesis of 6-Arylpiperidin-2-ones
    Supporting Information (PDF)
  • 120
    Farahat, Abdelbasset A.; Boykin, David W.:

    Unusual Regioselective Reactions of 2,4-Bis(methylsulfanyl)pyrimidine under Modified Suzuki and Stille Cross-Coupling Conditions

    Image for article: Unusual Regioselective Reactions of 2,4-Bis(methylsulfanyl)pyrimidine under Modified Suzuki and Stille Cross-Coupling Conditions
  • 125
    Martínez, Andrea R.; Vega, Daniel R.; Aguirre, José M.; Lantaño, Beatriz; Moltrasio, Graciela Y.:

    Synthesis of a Phenanthridine Analogue of Natural Isocarbostyril Alkaloids

    Image for article: Synthesis of a Phenanthridine Analogue of Natural Isocarbostyril Alkaloids
    Supporting Information (PDF)
  • 130
    Sokolova, Nadezhda V.; Vorobyeva, Daria V.; Osipov, Sergey N.; Vasilyeva, Tamara P.; Nenajdenko, Valentine G.:

    Synthesis of α-Trifluoromethyl-α-hydroxy Acid-Peptide Conjugates via Click Chemistry

    Image for article: Synthesis of α-Trifluoromethyl-α-hydroxy Acid-Peptide Conjugates via Click Chemistry
  • 137
    Billamboz, Muriel; Legeay, Jean Christophe; Hapiot, Frédéric; Monflier, Eric; Len, Christophe:

    Novel Strategy for the Bis-Butenolide Synthesis via Ring-Closing Metathesis

    Image for article: Novel Strategy for the Bis-Butenolide Synthesis via Ring-Closing Metathesis
  • 144
    Mirabal-Gallardo, Yaneris; Soriano, Maria D. P. C.; Caballero, Julio; Alzate-Morales, Jans; Simirgiotis, Mario J.; Santos, Leonardo S.:

    Synthesis of the Indolo[2,3-a]quinolizidine Ring through the Addition of 2-Siloxyfurans to Imines and Intrinsic Reaction Coordinate Calculations

    Image for article: Synthesis of the Indolo[2,3-<EM EMTYPE="ITALIC">a</EM>]quinolizidine Ring through the Addition of 2-Siloxyfurans to Imines and Intrinsic Reaction Coordinate Calculations
  • 151
    Potkin, Vladimir I.; Bumagin, Nikolay A.; Petkevich, Sergey K.; Lyakhov, Alexander S.; Rudakov, Dmitrii A.; Livantsov, Michail V.; Golantsov, Nikita E.:

    5-(p-Tolyl)isoxazol-3-amine-Palladium(II) Complex: Preparation, Structure, and Catalytic Application in the Suzuki-Miyaura Reaction in Water

    Image for article: 5-(<EM EMTYPE="ITALIC">p</EM>-Tolyl)isoxazol-3-amine-Palladium(II) Complex: Preparation, Structure, and Catalytic Application in the Suzuki-Miyaura Reaction in Water

    • addenda and errata

  • 0158

    Synthesis of 1-Chloroalkynes from Alkynylsilanes Using Trichloroisocyanuric Acid as Chlorinating Agent

  • e1

    tert-Butoxide-Assisted Amidation of Esters under Green Conditions