Synthesis

Issue 04 · February 2014

Recommend Journal

review
403
Olszewski, Tomasz K.:
Environmentally Benign Syntheses of α-Substituted Phosphonates: Preparation of α-Amino- and α-Hydroxyphosphonates in Water, in Ionic Liquids, and under Solvent-Free Conditions

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short review
430
Sidduri, Achyutharao; Tilley, Jefferson W.; Fotouhi, Nader:
Functionalized Organozinc Reagents in Medicinal Chemistry: Discovery of Novel Drug Candidates

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practical synthetic procedures
445
Zajdlik, Adam; He, Zhi; St Denis, Jeffrey D.; Yudin, Andrei K.:
Efficient Preparation of α-Aminoboronic Acid Derivatives via Boroalkyl Group Migration

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paper
455
Kawase, Yasushi; Yamagishi, Takehiro; Kato, Jun-ya; Kutsuma, Teruo; Kataoka, Tadashi; Iwakuma, Takeo; Yokomatsu, Tsutomu:
Reductive Alkylation of Hydrazine Derivatives with α-Picoline-Borane and Its Applications to the Syntheses of Useful Compounds Related to Active Pharmaceutical Ingredients

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465
Vuppalapati, Srinivasu V. N.; Xia, Likai; Edayadulla, Naushad; Lee, Yong Rok:
Mild and Efficient One-Pot Synthesis of Diverse Flavanone Derivatives via an Organocatalyzed Mannich-Type Reaction

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475
Kretschmer, Florian; Wild, Andreas; Hager, Martin D.; Schubert, Ulrich S.:
Synthesis of a Rigid Tetrahedral Linker with Thioether End Groups

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479
Banoth, Linga; Chandarrao, Bhukya; Pujala, Brahmam; Chakraborti, Asit K.; Banerjee, U. C.:
Efficient Chemoenzymatic Synthesis of (RS)-, (R)-, and (S)-Bunitrolol

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489
Gao, Hong; Sun, Jing; Yan, Chao-Guo:
Povarov Reaction of β-Enamino Esters and Isatin-3-imines for Diastereoselective Synthesis of Spiro[indoline-3,2′-quinolines]

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496
Miura, Takuya; Fujioka, Saki; Takemura, Naoto; Iwasaki, Hiroki; Ozeki, Minoru; Kojima, Naoto; Yamashita, Masayuki:
Synthesis of 6-Substituted 3-(Alkoxycarbonyl)-5-aryl-α-pyrones

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503
Han, Liuquan; Zhang, Bijun; Xiang, Changbin; Yan, Jie:
One-Pot Synthesis of Isoxazolines from Aldehydes Catalyzed by Iodobenzene

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510
Hu, Manman; He, Xinwei; Niu, Zhiqiang; Yan, Zhenglei; Zhou, Fuyin; Shang, Yongjia:
Synthesis of 3,4,5-Trisubstituted Isoxazoles by the 1,3-Dipolar Cycloaddition Reaction of α-Azido Acrylates and Aromatic Oximes

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515
Smith, D. David; Gallagher, Audrey T.; Crowley, Vincent M.; Gergens, Wayne M.; Abel, Peter W.; Hulce, Martin:
An Efficient Synthesis of 4(5)-Benzyl-l-histidines Employing Catalytic Transfer Hydrogenolysis at Elevated Temperatures

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522
Nordmann, Jan; Müller, Thomas J. J.:
Anilines as Substrates in Consecutive Four-Component Synthesis of Novel 1-Aryl-5-benzoyl-6-phenyl-3,4-dihydropyridin-2(1H)-ones

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531
Gaitzsch, Jens; Rogachev, Victor; Zahel, Martin; Metz, Peter:
Synthesis of m-Terphenyl Derivatives via Domino Diels–Alder/Retro-Diels–Alder Reaction of 1,3-Dienic δ-Sultones with Alkynes

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