DOI: 10.1055/s-00000084

Synthesis

eFirst

Publication Date: 05 February 2025

paper

Dupeux, Aurélien; Durant, Andrew G.; Rabeda, Karolina; Mirabi, Bijan; Marchese, Austin D.; Algera, Russell F.; Monfette, Sebastien; Roosen, Philipp C.; Lautens, Mark: CsCF3B(OMe)3: A Versatile Nucleophilic Source of the Trifluoromethyl Anion
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0450_ga_10-1055_s-0043-1775439.gif

paper

Ďurina, Lukáš; Kerti, Lukáš; Litecká, Miroslava; Moncol, Ján; Žídeková, Ivana; Fischer, Róbert: Zinc-Mediated Diastereoselective Acyloxyallylation of Isoxazolidine-4,5-diols
https://www.thieme-connect.de/media/synthesis/EFirst/i_t0401_ga_10-1055_a-2503-2981.gif

Publication Date: 04 February 2025

Publication Date: 03 February 2025

review

Lukin, Oleg; Shivanyuk, Alexander; Dolgonos, Grygoriy; Gerasov, Andrii; Mandzhulo, Aleksandr; Fetyukhin, Volodymyr: Spirocyclizations of Nortropanes
https://www.thieme-connect.de/media/synthesis/EFirst/i_r0399_ga_10-1055_a-2503-2459.gif

Publication Date: 29 January 2025

Publication Date: 27 January 2025

paper

Gao, Jun-Nan; Tan, Wen-Xin; Yang, Shuang; Wang, Ning-Yi; Han, Jiebin; Wang, Da-Hua; Zhang, Yu-Chen; Shi, Feng: Lewis Acid Catalyzed Regioselective Substitution of 2-Indolylmethanols with Pyrroles
https://www.thieme-connect.de/media/synthesis/EFirst/i_f0437_ga_10-1055_a-2503-3181.gif

Publication Date: 23 January 2025

Publication Date: 22 January 2025

paper

Niu, Yu-Dan; Lv, Pei; Hu, Hao-Lan; Shi, Jianghuan; Chen, Peng; Jiang, Yi-Jun: Scandium(III)-Catalyzed N-Alkylation of Carbazoles with Alcohols
https://www.thieme-connect.de/media/synthesis/EFirst/i_g0415_ga_10-1055_a-2502-7704.gif

psp

Chaudhury, Subhabrata; Thennakoon, Dulanjali; Wetzel, Edward A.; Donaldson, William A.: A Scalable, Chromatography-Free Synthesis of the Potent and Highly Selective ERβ Agonist EGX358
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0445_ga_10-1055_s-0043-1775433.gif

Publication Date: 21 January 2025

feature

paper

Manna, Priyadarshi; Chatterjee, Arunima; Kundu, Mrinalkanti; Rao, G. Prabhakar; Mukherjee, Rusmita; Podder, Swarnali; Datta, Bandita; Adhikari, Susanta: 3-Amino-1-methyl-1H-pyridin-2-one as Inbuilt Directing Group for Additive-Free Late-Stage ortho-Amination under Copper Catalysis towards Biologically Relevant Molecules
https://www.thieme-connect.de/media/synthesis/EFirst/i_m0441_ga_10-1055_s-0040-1720160.gif

Publication Date: 20 January 2025

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