DOI: 10.1055/s-00000131

Synfacts

Issue 12 · Volume 11 · December 2015 DOI: 10.1055/s-005-30464

Synform

A167
Zanda, Matteo: SYNFORM ISSUE 2015/11

Synthesis of Natural Products and Potential Drugs

z1231
All PDFs of this category
1231
Synthesis of (–)-Incarviatone A
1232
Synthesis of NVP-CGM097
1233
Synthesis of LY2886721
1234
Synthesis of Erlotinib
1235
Synthesis of Olmesartan Medoxomil
1236
Total Synthesis of (±)-Goniomitine
1237
Total Synthesis of (+)-Batzelladine B
1238
Synthesis of (S)-Pregabalin
1239
Synthesis of (–)-Conolutinine
1240
Synthesis of Silodosin
1241
Synthesis of Leustroducsin B
1242
Total Synthesis of (–)-Pallavicinin and (+)-Neopallavicinin
1243
Synthesis of KAE609 via an Asymmetric aza-Diels–Alder Reaction
1244
Synthesis of Pevonedistat
1245
Total Syntheses of Rhodomyrtosones A and B

Synthesis of Heterocycles

z1247
All PDFs of this category
1247
Synthesis of Highly Functionalized Oxetanes
1248
Acid-Catalyzed Synthesis of Carbazoles from Indoles and 2-Amidodihydrofurans
1249
Synthesis of Six- and Seven-Membered Heterocycles
1250
Synthesis of 2-Aminoindoles and 5-Amino-indolo[1,2-a]quinazolines
1251
Nickel-Catalyzed Anti-Markovnikov Hydroheteroarylation of Nonactivated Alkenes
1252
Synthesis of Cyclic Ethers by Alkoxylation of Nonactivated sp3 C–H Bonds
1253
Manganese(I)-Catalyzed C–H Bond Amidation of Heteroarenes
1254
Silver-Catalyzed Synthesis of 2-Aryl-5-(trifluoromethyl)tetrazoles
1255
Imidazotetrazolodiazepinones by a Ugi–Azide Multicomponent Reaction
1256
Rhodium Carbenoid-Catalyzed Synthesis of 2,5-Epoxybenzo[f][1,4]oxazepines
1257
Potassium Persulfate Mediated Synthesis of Dihydrofurans
1258
Oxidative Radical Decarboxylation Route to 6-Alkyl- or 6-Arylphenanthridines
1259
Radical-Mediated Difluoromethylenephosphonation
1260
Highly Substituted Pyrimidines by Multicomponent Reactions
1261
Synthesis of Tetrasubstituted Furopyridazinones from Nitrile Imines

Synthesis of Materials and Unnatural Products

z1263
All PDFs of this category
1263
Two Steps to Porosity
1264
2- and 6-Thienylazulenes by Direct Arylation
1265
Aminocyclopropanation on Fullerene
1266
Facile Method for the Synthesis of Dibenzo[g,p]chrysenes
1267
[2+2+2] Cyclotrimerization in a Porous Coordination Framework
1268
C–H Functionalization Furnishes Thieno-Fused Cycles and Heterocycles
1269
Persistent COF: A Stable Platform for Asymmetric Organocatalysis
1270
A New Class of Classical and Nonclassical Aggregation-Induced Emitters
1271
Dimerized to Bend: Radilenes from Cumulenes
1272
Electrophilic Borylation Leads to Efficient OLED Materials
1273
High Mobility Conjugated Polymers through Direct Arylation
1274
One Stone Two Birds with a NHC Sponge

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1275
All PDFs of this category
1275
Ruthenium-Catalyzed Asymmetric Yne–Enone Cyclizations
1276
Asymmetric Oxygen Atom Transfer to Oxindoles by Copper Catalysis
1277
Asymmetric Gold(I)-Catalyzed [3+2] Cycloadditions
1278
Tetrahydrofurans by Enantioselective Gold(I)-Catalyzed Desymmetrization of 1,3-Diols
1279
Enantioselective Palladium-Catalyzed 1,1-Fluoroarylation
1280
Asymmetric Alkoxycarbonylative Amination of Allenes
1281
Scandium-Catalyzed Asymmetric Ring-Opening of Cyclopropanes
1282
Diastereodivergent Asymmetric [4+2] Cycloaddition
1283
Palladium-Catalyzed Enantioselective Synthesis of Chromans
1284
Copper-Catalyzed Asymmetric Synthesis of 3,4-Diaminopyrrolidines
1285
Enantioselective Synthesis of Pyrrolidine-thia(oxa)zolidinediones
1286
Rhodium-Catalyzed Asymmetric Ring Opening of Oxabicycles
1287
Enantioselective Palladium-Catalyzed Carboalkyoxylation Forming Tetrahydrofurans
1288
8-Oxa-6-Azabicyclo[3.2.1]octanes by Asymmetric Copper-Catalyzed Iodocyclization
1289
Asymmetric Copper-Catalyzed Propargylic Substitution
1290
Rhodium(I)-Catalyzed Asymmetric 1,4-Addition of Boronic Acids to Cumarins
1291
Transfer Hydrogenation with Chiral N-Heterocyclic Carbene/Iridium Complex
1292
Enantioselective Fluorination of Allylic Trichloroacetimidates
1293
Enantioselective Palladium-Catalyzed Ene Reaction and [2+2] Cyclization
1294
Asymmetric Zinc-Catalyzed Synthesis of Polycyclic Spirooxindoles
1295
Povarov Reaction Catalyzed by Anionic Chiral Cobalt(III) Complexes
1296
Synthesis of trans-1,2-Diamine through Asymmetric Ring-Opening Reaction
1297
Asymmetric Hydrophosphination of α,β,γ,δ-Unsaturated Ketones
1298
Asymmetric Addition of Heteroarylboronates to Arylimines
1299
Cobalt-Catalyzed Allylation and Asymmetric Ring-Opening of Heterobicyclic Alkenes
1300
Enantioselective Copper-Catalyzed Synthesis of Benzofuranones
1301
Enantioselective Intramolecular C–H Arylation of Cyclopropanes
1302
Functionalized Furans by Asymmetric Gold-Catalyzed Intermolecular Annulation

Metal-Mediated Synthesis

z1303
All PDFs of this category
1303
Asymmetric Bromine–Lithium Exchange
1304
Diastereoselective Addition of Organozinc Reagents to 1,2-Anhydro Sugars
1305
Enantioselective Bromocyclopropanation of Allylic Alcohols
1306
Negishi Cross-Coupling of Aminotriazoles
1307
Palladium-Catalyzed Carbofluoroalkylation
1308
Zinc-Catalyzed Borylation
1309
Enantioselective Homocrotylation of Aldehydes
1310
Palladium-Catalyzed Alkylsulfonylation of Boronic Acids
1311
Ruthenium-Catalyzed Cross-Coupling of Naphthamides
1312
Nickel-Catalyzed Direct Borylation of Unactivated Fluoroarenes
1313
Copper-Catalyzed Carboxylation of Alkenylzirconocenes
1314
Silver-Catalyzed Diastereoselective Coupling
1315
Trifluoromethylation of Carbonyl Compounds
1316
Addition of Boronic Acids to Cyclic Sulfonylketimines
1317
3-Substituted 2-Aminochromones by Tin(IV)-Promoted Annulation

Organo- and Biocatalysis

z1319
All PDFs of this category
1319
Organocatalytic Photoredox C–H Amination of Arenes
1320
1,6-Conjugate Addition of Pyrroles to para-Quinone Methides
1321
Biocatalytic Hydrogen-Borrowing Amination of Ketones
1322
Organocatalytic Carbonyl–Ene Cyclization
1323
C–H Alkylation of Alcohols
1324
The Mitsunobu Reaction Catalytic in Phosphine and Azodicarboxylate

Polymer-Supported Synthesis

z1325
All PDFs of this category
1325
Silver-Foil-Catalyzed Cyclopropanation of Alkenes Under Mechanochemical Conditions
1326
Bisoxazoline/Palladium Complex Microsphere Catalyzed Heck Reactions
1327
Ullmann-Type Coupling of Phenols with Aryl Halides on Cuprian Zeolite USY
1328
Cobalt Ferrite Nanoparticle Catalyzed Petasis–Borono–Mannich Reaction
1329
Enantiospecific C–H Activation with Ruthenium Nanocatalysts
1330
Microwave-Assisted Click Reaction Using Copper(I) Iodide on Alumina
1331
C–C Bond Formation with Heterogeneous Lewis Acids in Aqueous Media
1332
Oxidation of Alcohols by Using a Supported Manganese(lll) Salophen Complex
1333
Solid-Phase Total Synthesis of Spiruchostatin A
1334
Synthesis of Benzothiazoles by Using Piperazinylpyrimidine-Modified MCM-41
1335
Zirconia–β-Cyclodextrin Catalyst for Synthesis of Substituted Imidazoles
1336
Palladium/Carbon-Catalyzed Aminocarbonylation of Aryl Iodides
1337
Copper/Manganese(II) Oxide Catalyzed ortho-Halogenation of 2-Arylpyridines
1338
Multicomponent Synthesis of Dibenzo-diazepines with Iron(III) Tosylate/Silica
1339
Sulfonated Carbon Nanotubes: A Supported Acid Catalyst for Pyrrole Synthesis
1340
Synthesis of β-Enaminones by Using a Ag/γ-Fe3O4@meso-TiO2 Nanocatalyst

Erratum

1341
Prakash, G. K. S.; Rapp, A.; Munoz, S. B.; May, N.; Jones, J.-P.; Haiges, R.; Esteves, P. M.; Mathew, T.: Lewis Acid Catalyzed Synthesis of Di/Trifluoromethyl- 1,2,3,4-Tetrahydroquinazolines
1341
Prakash, S.; Muralirajan, K; Cheng, C.-H.: Rhodium-Catalyzed Vinylation
1342
Lao, J. R.; Fernández-Pérez, H.; Vidal-Ferran, A.: Kinetic Resolution of Vinyl Sulfoxides by Rhodium Catalysis