DOI: 10.1055/s-00000084

Synthesis

Issue 05 · Volume 57 · March 2025 DOI: 10.1055/s-015-61105

table of contents

  • V

    Linked PDF of Table of Contents

    • review

  • 891
    Sajjad, Farrukh; Zhang, Shuyue; Xu, Ming-Hua:

    Advances in Transition-Metal Catalysis and Organocatalysis Approaches towards Asymmetric Synthesis of β-Amino Acid Derivatives

    Image for article: Advances in Transition-Metal Catalysis and Organocatalysis Approaches towards Asymmetric Synthesis of β-Amino Acid Derivatives

    • short review

  • 917
    Liu, Xigong; Liu, Lei:

    Catalytic Asymmetric Syntheses of 3-Monosubstituted Oxindoles

    Image for article: Catalytic Asymmetric Syntheses of 3-Monosubstituted Oxindoles
  • 925
    Horwitz, Matthew A.:

    Discovery Process Chemistry: An Innovation Hub at the Interface of Academia, the Pharmaceutical Industry, and Contract Research Organizations

    Image for article: Discovery Process Chemistry: An Innovation Hub at the Interface of Academia, the Pharmaceutical Industry, and Contract Research Organizations
  • 937
    Xie, Ke; Li, Ao; Kong, Bao-Rui; Chen, Zhi-Chao; Du, Wei; Chen, Ying-Chun:

    Recent Advances in Asymmetric Addition Reactions to Isatins

    Image for article: Recent Advances in Asymmetric Addition Reactions to Isatins

    • Dual Catalysis

  • 953
    Atriardi, Shafrizal R.; Anita, Yulia; Woo, Sang Kook:

    Harnessing Photoredox and Weak Brønsted Base Dual Catalysis for Selective C(sp3)–H Bond Activation

    Image for article: Harnessing Photoredox and Weak Brønsted Base Dual Catalysis for Selective C(sp<sup>3</sup>)–H Bond Activation

    • feature

  • 965
    Mizobuchi, Eduardo F.; Burtoloso, Antonio C. B.:

    The Acylation of α-Carbonyl Sulfoxonium Ylides with N-Hydroxyphthalimide Esters

    Image for article: The Acylation of α-Carbonyl Sulfoxonium Ylides with <i>N</i>-Hydroxyphthalimide Esters
    Supporting Information (PDF)

    • psp

  • 973
    Chaudhury, Subhabrata; Thennakoon, Dulanjali; Wetzel, Edward A.; Donaldson, William A.:

    A Scalable, Chromatography-Free Synthesis of the Potent and Highly Selective ERβ Agonist EGX358

    Image for article: A Scalable, Chromatography-Free Synthesis of the Potent and Highly Selective ERβ Agonist EGX358
    Supporting Information (PDF)

    • paper

  • 978
    Guo, Taijie; Wang, Wei; Xu, Long; Dong, Jiajia:

    RNHSO2F as Reliable Azasulfene Precursors for the Construction of Sulfamates

    Image for article: RNHSO<sub>2</sub>F as Reliable Azasulfene Precursors for the Construction of Sulfamates
    Supporting Information (PDF)

    • SuFEx Chemistry

  • 991
    Tao, Guang; Fayad, Eman; Abu Ali, Ola A.; Oyom, Bright; Qin, Hua-Li:

    A Convenient One-Pot Process for Converting Thiols into Sulfonyl Fluorides Using H2O2 as an Oxidant

    Image for article: A Convenient One-Pot Process for Converting Thiols into Sulfonyl Fluorides Using H<sub>2</sub>O<sub>2</sub> as an Oxidant
    Supporting Information (PDF)
  • 999
    Yang, Na; Pei, Guanhua; Li, Hao; Han, Junwei; Wang, Peng; Xie, Lili; Liao, Saihu:

    Synthesis of FSO2-Functionalized Oxindoles via a Radical Fluorosulfonylation/Intramolecular Arylation Cascade

    Image for article: Synthesis of FSO<sub>2</sub>-Functionalized Oxindoles via a Radical Fluorosulfonylation/Intramolecular Arylation Cascade
    Supporting Information (PDF)
  • 1007
    Dasmahapatra, Upala; Choudhury, Badruzzaman; Ahmad, Md Gulzar; Maiti, Barnali; Chanda, Kaushik:

    Direct Access to 5,6-Dihydropyrido[2′,1′:2,3]pyrido-Fused Imidazo [4,5-c]quinolines via Consecutive C–N and C–C Bond Formation in Deep Eutectic Solvent under Microwave Irradiation

    Image for article: Direct Access to 5,6-Dihydropyrido[2′,1′:2,3]pyrido-Fused Imidazo [4,5-<i>c</i>]quinolines via Consecutive C–N and C–C Bond Formation in Deep Eutectic Solvent under Microwave Irradiation
    Supporting Information (PDF)
  • 1015
    Olu-Igbiloba, Oluwaseun A.; Sitzmann, Helmut; Manolikakes, Georg:

    Cobalt-Catalyzed Three-Component Synthesis of α-Substituted N-Sulfonyl Amines via C(sp2)–H Bond Activation

    Image for article: Cobalt-Catalyzed Three-Component Synthesis of α-Substituted <i>N</i>-Sulfonyl Amines via C(sp<sup>2</sup>)–H Bond Activation
    Supporting Information (PDF)

    • Dual Catalysis

  • 1025
    Wang, Mingze; Zi, Weiwei:

    Synergistic Pd/Cu-Catalyzed Asymmetric Csp3–Csp3 Coupling of 1,3-Dienes with 2-Acylimidazoles

    Image for article: Synergistic Pd/Cu-Catalyzed Asymmetric Csp<sup>3</sup>–Csp<sup>3</sup> Coupling of 1,3-Dienes with 2-Acylimidazoles
    Supporting Information (PDF) CIF File (OTHER)

    • C–S Bond Forming and Cleaving Reactions

  • 1034
    Bugaenko, Dmitry I.; Karchava, Alexander V.:

    Synthesis of 2-Aminobenzo[b]thiophenes via an Intramolecular Dehydrogenative C–S Bond Formation Effected by Iodine(III) Reagents

    Image for article: Synthesis of 2-Aminobenzo[<i>b</i>]thiophenes via an Intramolecular Dehydrogenative C–S Bond Formation Effected by Iodine(III) Reagents
    Supporting Information (PDF)
  • 1043
    Endo, Koki; Shibahara, Fumitoshi:

    Imidazo[1,5-a]pyridin-3-ylidene-Catalyzed Oxidative Esterification of Aldehydes: Remarkable Electronic Effect Regarding π-Accepting Character of Ring-Fused N-Heterocyclic Carbene

    Image for article: Imidazo[1,5-<i>a</i>]pyridin-3-ylidene-Catalyzed Oxidative Esterification of Aldehydes: Remarkable Electronic Effect Regarding π-Accepting Character of Ring-Fused N-Heterocyclic Carbene
    Supporting Information (PDF)
  • 1050
    Singroha, Rekha; Onen, Patrick; Yadav, Usha; Kant, Ruchir; Mohanan, Kishor:

    Three-Component Synthesis of Cyanopyrazoles Employing Diazo­acetonitrile

    Image for article: Three-Component Synthesis of Cyanopyrazoles Employing Diazo­acetonitrile
    Supporting Information (PDF) CIF File (OTHER)
  • 1059
    Buravov, Oleksandr V.; Tomak, Victor O.; Shishkina, Svitlana V.; Chebanov, Valentyn A.:

    First Example of Aryl–Hetaryl Cross-Coupling via [5,5]-Sigmatropic Rearrangement

    Image for article: First Example of Aryl–Hetaryl Cross-Coupling via [5,5]-Sigmatropic Rearrangement
    Supporting Information (PDF)
  • 1072
    Michon, Synthia; Garcia, Maxime; Cavelier, Florine; Salom-Roig, Xavier J.:

    Divergent Synthetic Strategy To Access the Polyketide Subunits of Aurilides: Synthesis of the Southern Fragment of Lagunamides D and D′

    Image for article: Divergent Synthetic Strategy To Access the Polyketide Subunits of Aurilides: Synthesis of the Southern Fragment of Lagunamides D and D′
    Supporting Information (PDF)