DOI: 10.1055/s-00000131

Synfacts

Issue 11 · Volume 2011 · November 2011 DOI: 10.1055/s-002-22386

Synform

A100
Zanda, Matteo: SYNFORM ISSUE 2011/11

Synthesis of Natural Products and Potential Drugs

z1149
All PDFs of this category
1149
Paleček, J.; Zweigerdt, R.; Olmer, R.; Martin, U.; Kirschning, A.; Dräger, G.: Synthesis of Rho-Kinase Inhibitor Y-27632
1150
Zhuo, X.; Xiang, K.; Zhang, F.-M.; Tu, Y.-Q.: Synthesis of (+)-Przewalskin B
1151
Stivala, C. E.; Zakarian, A.: Synthesis of a γ-Secretase Modulator
1152
Michalak, M.; Stodulski, M.; Stecko, S.; Mames, A.; Panfil, I.; Soluch, M.; Furman, B.; Chmielewski, M.: Formal Synthesis of Ezetimibe
1153
Benson, S.; Collin, M.-P.; Arlt, A.; Gabor, B.; Goddard, R.; Fürstner, A.: Synthesis of Spirastrellolide F Methyl Ester
1154
Wan, Z.-K.; Chenail, E.; Li, H.-Q.; Kendall, C.; Wang, Y.; Gingras, S.; Xiang, J.; Massefski, W. W.; Mansour, T. S.; Saiah, E.: Synthesis of HSD-016
1155
Herrmann, A. T.; Martinez, S. R.; Zakarian, A.: Synthesis of (+)-Brevisamide
1156
Chandra, A.; Johnston, J. N.: Synthesis of (±)-Hapalindoles K, A, and G
1157
Wohlfahrt, M.; Harms, K.; Koert, U.: Synthesis of (+)-Awajanomycin
1158
Yamamoto, T.; Muto, K.; Komiyama, M.; Canivet, J.; Yamaguchi, J.; Itami, K.: Synthesis of Febuxostat, Tafamadis, and Texaline
1159
Jiang, Y.; Chen, X.; Zheng, Y.; Xue, Z.; Shu, C.; Yuan, W.; Zhang, X.: Synthesis of Cholesterol Transporter NPC1L1 Inhibitor
1160
Kobayashi, S.; Kinoshita, T.; Kawamoto, T.; Wada, M.; Kuroda, H.; Masuyama, A.; Ryu, I.: Synthesis of (±)-Communiol E
1161
Fujii, S.; Chang, S. Y.; Burke, M. D.: Synthesis of Synechoxanthin

Synthesis of Heterocycles

z1163
All PDFs of this category
1163
Tsvelikhovsky, D.; Buchwald, S. L.: Concise Palladium-Catalyzed Synthesis of Dibenzodiazepines
1164
Zheng, D.; Wang, Z.; Wu, J.: Synthesis of 1-Aroxyisoquinolines from Phenols and 2-Alkynylbenzaldoximes
1165
Varela-Fernández, A.; Varela, J. A.; Saá, C.: Ru-Catalyzed Heteroannulation to Indoles, Dihydroisoquinolines, and Dihydroquinolines
1166
Zhao, J.; Wu, C.; Li, P.; Ai, W.; Chen, H.; Wang, C.; Larock, R. C.; Shi, F.: [3+2] Cycloaddition to Pyrido[1,2-b]indazoles
1167
Ackermann, L.; Pospech, J.: Ruthenium-Catalyzed Synthesis of Phthalides in Water via C-H Alkenylation
1168
Wu, Z.; Huang, Q.; Zhou, X.; Yu, L.; Li, Z.; Wu, D.: One-Pot Cu-Catalyzed C-N Coupling Approach to Pyrido[1,2-a]benzimidazoles
1169
Pews-Davtyan, A.; Beller, M.: Efficient Zinc-Mediated Heteroannulation Route to 3-Amidoindoles
1170
Candito, D. A.; Panteleev, J.; Lautens, M.: Base-Mediated Intramolecular Aryne-Ene Cyclization
1171
Ylijoki, K. E. O; Kündig, E. P.: Synthesis of Benzoxazinones via Palladium-Catalyzed Intramolecular C-O Coupling
1172
Hong, D.; Zhu, Y.; Li, Y.; Lin, X.; Lu, P.; Wang, Y.: Copper-Catalyzed Three-Component Synthesis of Polysubstituted Pyrroles
1173
Zhu, D.; Zhao, J.; Wei, Y.; Zhou, H.: Sonogashira-Hydroamination Route to 1,2,4-Trisubstituted Pyrroles
1174
Davies, P. W.; Cremonesi, A.; Dumitrescu, L.: Gold-Catalyzed [3+2]-Cycloaddition Approach to 2,4,5-Trisubstituted Oxazoles
1175
Radi, M.; Casaluce, G.; Botta, M.: Microwave-Facilitated Synthesis of Pyrimidinones
1176
Sperança, A.; Godoi, B.; Pinton, S.; Back, D. F.; Menezes, P. H.; Zeni, G.: Iron-Mediated Heteroannulation Route to Isochromenones
1177
Wang, Y.; Wang, H.; Peng, J.; Zhu, Q.: Pd-Catalyzed Heteroannulation Route to 4-Aminoquinazolines via C-H Amidination

Synthesis of Materials and Unnatural Products

z1179
All PDFs of this category
1179
Sun, Z.; Huang, K.-W.; Wu, J.: A Stabilized Singlet Biradical Compound
1180
Maeda, C.; Yoneda, T.; Aratani, N.; Yoon, M.-C.; Lim, J. M.; Kim, D.; Yoshioka, N.; Osuka, A.: Alkynes en Route to Porphyrinoides
1181
Tejedor, D.; López-Tosco, S.; González-Platas, J.; García-Tellado, F.: Substitute This!
1182
Kuniobu, Y.; Tatsuzaki, T.; Matsuki, T.; Takai, K.: A Facile Route to Polycylic Aromatic Hydrocarbons
1183
Kang, E.-H.; Lee, I. S.; Choi, T.-L.: ‘Ticktock’ Cyclopolymerization
1184
Kurtz, J. P.; Grusenmeyer, T.; Tong, L.; Kosgei, G.; Schmehl, R. H.; Mague, J. T.; Pascal, Jr., R. A.: Polyaryl Mesobenzanthrones
1185
Okujima, T.; Jin, G.; Matsumoto, N.; Mack, J.; Mori, S.; Ohara, K.; Kuzuhara, D.; Ando, C.; Ono, N.; Yamada, H.; Uno, H.; Kobayashi, N.: Expanded Cyclo[8]pyrroles Made Easy
1186
Chen, J.-H.; Wang, S.-A.; Liu, Y.-H.; Wong, K.-T.: C3-Symmetric Chromophores with 6,5,5-Fused Ring Systems
1187
Mikie, T.; Asahara, H.; Nagao, K.; Ikuma, N.; Kokubo, K.; Oshima, T.: High-Yielding Thermal [2+2] Addition to Fullerene
1188
Bew, S. P.; Sharma, S. V.: Controlling Calixarene Size with Metal Salts: The First Brønsted-Free Synthesis
1189
Guo, X.; Watson, M. D.: Ultra-Low Bandgap Donor-Acceptor Polymers Based on Pyromellitic Diimide
1190
Liu, J.; Deng, C.; Tseng, N.-W.; Chan, C. Y. K.; Yue, Y.; Ng, J. C. Y.; Lam, J. W. Y.; Wang, J.; Hong, Y.; Sung, H. H. Y.; Williams, I. D.; Tang, B. Z.: Conjugated Polymers via Aroyl Chloride-Alkyne Polymerization
1191
Matano, Y.; Saito, A.; Fukushima, T.; Tokudome, Y.; Suzuki, F.; Sakamaki, D.; Kaji, H.; Ito, A.; Tanaka, K.; Imahori, H.: Acenaphthene-Fused Phospholes with Enhanced Electronic Properties

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1193
All PDFs of this category
1193
Chen, G.; Gui, J.; Li, L.; Liao, J.: Novel Ligand for Rh-Catalyzed Asymmetric Conjugate Addition
1194
Jenkins, A. D.; Herath, A.; Song, M.; Montgomery, J.: Ni-Catalyzed Reductive Cycloaddition
1195
Cheon, C. H.; Kanno, O.; Toste, F. D.: Gold-Catalyzed Enantioselective Protonation
1196
Cao, Z.; Liu, Z.; Lin, Y.; Du, H.: Pd-Catalyzed Enantioselective Allylic Etherizations of Oximes
1197
Soheili, A.; Tambar, U. K.: Tandem Catalytic Allylic Amination and [2,3]-Stevens Rearrangement of Tertiary Amines
1198
Nugent, T. C.; Negru, D. E.; El-Shazly, M.; Hu, D.; Sadiq, A.; Bibi, A.; Umar, M. N.: A One-Pot Synthesis of Challenging Chiral Primary Amines
1199
Liu, T.-L.; Hea, Z.-L.; Wang, C.-J.: Copper-Catalyzed Asymmetric 1,3-Dipolar Cycloadditions
1200
Kunisu, T.; Oguma, T.; Katsuki, T.: Iron-Catalyzed Oxidative Kinetic Resolution of Secondary Alcohols
1201
Ovalles, S. R.; Hansen, J. H.; Davies, H. M. L.: Thermally-Induced Cycloadditions of Diazo Compounds and Alkenes
1202
Lian, Y.; Davies, H. M. L.: Combined C-H Functionalization/Cope Rearrangement with Vinyl Ethers
1203
Okamoto, R.; Okazaki, E.; Nogushi, K.; Tanaka, K.: Enantioselective Alder-Ene Reactions towards Dihydrobenzofurans
1204
Chen, J.-P.; Peng, Q.; Lei, B.-L.; Hou, X.-L.; Wu, Y.-D.: Pd-Catalyzed Chemo- and Regioselective Allylic Alkylation
1205
Liu, T.-L.; He, Z.-L.; Li, Q.-H.; Tao, H.-Y.; Wang, C.-J.: Silver-Catalyzed Enantioselective 1,3-Dipolar Cycloaddition
1206
Hassan, A.; Townsend, I. A.; Krische, M. J.: Iridium-Catalyzed Asymmetric Allylations
1207
Gormisky, P. E.; White, M. C.: Palladium-Catalyzed Allylic C-H Oxidation
1208
Wu, Z.; Ayad, T.; Ratovelomanana-Vidal, V.: 3-Aminochroman Derivatives via Ruthenium-Catalyzed Asymmetric Hydrogenation
1209
Huang, X.-R.; Pan, X.-H.; Lee, G.-H.; Chen, C.: New Ligands for Catalytic Asymmetric NHK Allylation of Aldehydes
1210
Kuang, Y.; Liu, X.; Chang, L.; Wang, M.; Lin, L.; Feng, X.: Yb-Catalyzed Asymmetric Conjugate Allylation of Coumarins
1211
Chen, W.; Cai, Y.; Fu, X.; Liu, X.; Lin, L.; Feng, X.: Domino Knovenagel/Pinner/Friedel-Crafts Synthesis of Chiral Chromenes
1212
Lin, L.; Kuang, Y.; Liu, X.; Feng, X.: Hetero-Diels-Alder Reaction of Brassard’s Diene and Aliphatic Aldehydes
1213
Liu, Z.; Cao, Z.; Du, H.: Novel Phosphorus Amidite-Olefin Ligands for Allylic Alkylation of Indoles
1214
Nishimura, T.; Sawano, T.; Ou, K.; Hayashi, T.: Co-Catalyzed Conjugate Addition of Alkynes to α,β-Unsaturated Ketones
1215
Zibinsky, M.; Fokin, V.: Use of 1,2,4-Triazolyl-1,2,3-Triazoles as Carbene Precursors
1216
Wang, Y.; Feng, X.; Du, H.: Kinetic Resolution of Morita-Baylis-Hillman Adducts by 1,4-Addition
1217
Blay, G.; Fernández, I.; Muñoz, M. C.; Pedro, J. R.; Recuenco, A.; Vila, C.: Zirconium-Catalyzed Enantioselective Friedel-Crafts Alkylation of Pyrroles
1218
Wu, J.; Li, X.; Wu, F.; Wan, B.: Tetradentate Amine Ligands for Asymmetric Friedel-Crafts Alkylations
1219
Yin, L.; Kanai, M.; Shibasaki, M.: Pd-Catalyzed Asymmetric Intramolecular Arylation of α-Keto Amides
1220
Ghorai, M. K.; Nanaji, Y.; Yadav, A. K.: One-Pot Domino Ring Opening/C-N Bond Formations
1221
Berhal, F.; Wu, Z.; Genêt, J.-P.; Ayad, T.; Ratovelomanana-Vidal, V.: Rhodium-Catalyzed Asymmetric 1,4-Addition of Arylboronic Acids
1222
Matsuzawa, A.; Mashiko, T.; Kumagai, N.; Shibasaki, M.: Asymmetric Ene Reaction by La/Ag Heterobimetallic Cooperative Catalysis

Metal-Mediated Synthesis

z1223
All PDFs of this category
1223
Ano, Y.; Tobisu, M.; Chatani, N.: Pd-Catalyzed Direct Alkynylation of Aliphatic C-H Bonds
1224
Bigovic, M.; Maslak, V.; Tokic-Vujosevic, Z.; Divjakovic, V.; Saicic, R. N.: In-Promoted Approach to Synthetic Equivalents of Hydroxyacetone Enolates
1225
Leermann, T.; Leroux, F. R.; Colobert, F.: One-Pot Synthesis of Functionalized Arylboronic Acids
1226
Molander, G. A.; McKee, S. A.: CuCl-Catalyzed β-Boration of α,β-Unsaturated Carbonyl Compounds
1227
Truong, T.; Daugulis, O.: Base-Mediated Transition-Metal-Free Alkynylation of Aryl Chlorides
1228
Shintani, R.; Takatsu, K.; Takeda, M.; Hayashi, T.: Asymmetric Allylic Substitution
1229
Li, J.; Burke, M. D.: Chiral C(sp³) Boronate Building Blocks
1230
Denmark, S. E.; Werner, N. S.: γ-Selective Cross-Coupling of Allylic Silanolate Salts
1231
Nishihara, Y.; Okada, Y.; Jiao, J.; Suetsugu, M.; Lan, M.-T.; Kinoshita, M.; Iwasaki, M.; Takagi, K.: Synthesis of Multialkylated Olefins through Carbozirconation and Coupling
1232
Barker, T. J.; Jarvo, E. R.: Ti-Mediated Coupling of Amines with Grignard Reagents
1233
Baidya, M.; Yamamoto, H.: Oxidation of Silyl Enol Ethers with Metal Nitrites
1234
Fei, N.; Yin, H.; Wang, S.; Wang, H.; Yao, Z.-J.: CuCl2-Mediated Chlorocyclization and Oxidative Aromatization Cascade
1235
Vrancken, E.; Gérard, H.; Linder, D.; Ouizem, S.; Alouane, N.; Roubineau, E.; Bentayeb, K.; Marrot, J.; Mangeney, P.: Lithium Cuprate Ion Pairs as a Key to Control Diastereoselectivity
1236
Tomashenko, O. A.; Escudero-Adán, E. C.; Belmonte, M. Martínez; Grushin, V. V.: CuCF3 Aromatic Trifluoromethylating Agents
1237
Huang, C.; Liang, T.; Harada, S.; Lee, E.; Ritter, T.: Ag-Mediated Caryl-OCF3 Bond Formation
1238
Kawai, H.; Tachi, K.; Tokunaga, E.; Shiro, M.; Shibata, N.: Trifluoromethylation of Aromatic Isoxazoles

Organo- and Biocatalysis

z1239
All PDFs of this category
1239
Lykke, L.; Rodríguez-Escrich, C.; Jørgensen, K. A.: Catalytic Enantioselective Oxaziridination
1240
Cao, Y.; Jiang, X.; Liu, L.; Shen, F.; Zhang, F.; Wang, R.: Asymmetric Synthesis of Spirooxindoles
1241
Burns, N. Z.; Witten, M. R.; Jacobsen, E. N.: Thiourea-Catalyzed Intramolecular [5+2] Cycloadditions
1242
Gu, Q.; You, S.-L.: Desymmetrization of Cyclohexadienones via Cinchonine-Derived Thiourea
1243
Fujiwara, Y.; Sun, J.; Fu, G. C.: Synthesis of Aryl Alkyl Sulfides by γ-Addition of Aryl Thiols to Allenoates
1244
Zhang, B.; Xiang, S.-K.; Zhang, L.-H.; Cui, Y.; Jiao, N.: α-Alkylation of Aldehydes by Oxidative Coupling with Molecular Oxygen
1245
Ding, M.; Zhou, F.; Liu, Y.-L.; Wang, C.-H.; Zhao, X.-L.; Zhou, J.: Phosphoramide-Catalyzed Michael Addition of Oxindoles to Nitroolefins
1246
Lakhdar, S.; Ammer, J.; Mayr, H.: Electrophilic Reactivities of Photo-Generated α,β-Unsaturated Iminium Ions
1247
De, C. K.; Seidel, D.: Catalytic Enantioselective Desymmetrization of meso-Diamines

Polymer-Supported Synthesis

z1249
All PDFs of this category
1249
John, J.; Gravel, E.; Hagège, A.; Li, H.; Gacoin, T.; Doris, E.: Silane Oxidation Catalyzed by Carbon Nanotube-Gold Nanohybrids
1250
Verma, S.; Nandi, M.; Modak, A.; Jain, S. L.; Bhaumik, A.: Oxidation of Alcohols with PMO-Supported Oxo-Vanadium Schiff Base
1251
Gruttadauria, M.; Liotta, L. F.; Salvo, A. M. P.; Giacalone, F.; LaParola, V.; Aprile, [nl]C.; Noto, R.: Silica-Supported Polyimidazolium Pd Catalysts for Suzuki-Miyaura Coupling
1252
Vanderheiden, S.; Bulat, B.; Zevaco, T.; Jung, N.; Bräse, S.: Denitrogenative Deuteration of Solid-Supported Triazenes
1253
Putta, C. B.; Ghosh, S.: Suzuki-Miyaura Coupling in Water with Pd@CSP
1254
Akkilagunta, V. K.; Kakulapati, R. R.: Synthesis of Unsymmetrical Sulfides with CuO Nanoparticles
1255
Hobbs, C.; Yang, Y.-C.; Ling, J.; Nicola, S.; Su, H.-L.; Bazzi, H. S.; Bergbreiter, D. E.: Polyethylene Oligomer Supported Olefin Metathesis Catalysts
1256
Kim, S.; Kim, E.; Kim, B. M.: Reduction of Nitro Compounds with N2H4˙H2O Using Fe3O4 Nanoparticles
1257
Cao, W.; Yu, B.: A Recyclable Polystyrene-Supported Gold(I) Catalyst
1258
Niknam, K.; Deris, A.; Naeimi, F.; Majleci, F.: Synthesis of 1,2,4,5-Tetrasubstituted Imidazoles with Silica-Bonded PPSA
1259
Alonso, F.; Moglie, Y.; Radivoy, G.; Yus, M.: Copper Nanoparticles on Activated Carbon for Click Chemistry
1260
Ohta, H.; Yuyama, Y.; Uozumi, Y.; Yamada, Y. M. A.: A Polymeric Bimetallic Catalyst for
N-Alkylation of Amines with Alcohols
1261
Bogár, K.; Krumlinde, P.; Bacsik, Z.; Hedin, N.; Bäckvall, J.-E.: Transfer Hydrogenation with Immobilized Wilkinson’s Catalyst
1262
Kawamorita, S.; Ohmiya, H.; Iwai, T.; Sawamura, M.: Borylation of Aryl Halides with Silica-SMAP/Pd

Addenda and Errata

1263
Fe-Catalyzed Phenanthrene Synthesis via [4+2] Benzannulation
1263
Palladium-Catalyzed C-H Activation Induced Enantioselective Route to Fused Indolines
1264
Dysprosium(III) Triflate Catalyzed Aza-Piancatelli Rearrangement
1264
Organocatalytic Enantioselective Fluorocyclizations