DOI: 10.1055/s-00000084

Synthesis

Issue 23 · Volume 44 · December 2012 DOI: 10.1055/s-002-24066

synform

  • A122
    Zanda, Matteo:

    SYNFORM ISSUE 2012/12

    • review

  • 3551
    Trstenjak, Uroš; Ilaš, Janez; Kikelj, Danijel:

    Advances in the Synthesis of Morpholin-3-ones and Morpholin-2-ones

    Image for article: Advances in the Synthesis of Morpholin-3-ones and Morpholin-2-ones

    • feature article

  • 3579
    Ghosh, Arun K.; Kass, Jorden; Nicponski, Daniel R.; Keyes, Chad:

    Diastereoselective Synthesis of Substituted Tetrahydropyrans by Copper(II)–Bisphosphine-Catalyzed Olefin Migration and Prins Cyclization

    Image for article: Diastereoselective Synthesis of Substituted Tetrahydropyrans by Copper(II)–Bisphosphine-Catalyzed Olefin Migration and Prins Cyclization

    • practical synthetic procedures

  • 3590
    Blay, Gonzalo; Fernández, Isabel; Pedro, José R.; Vila, Carlos:

    Enantioselective Synthesis of Substituted Indoles Through Zirconium(IV)-Catalyzed Friedel–Crafts Alkylation

    Image for article: Enantioselective Synthesis of Substituted Indoles Through Zirconium(IV)-Catalyzed Friedel–Crafts Alkylation

    • short paper

  • 3595
    Edelbach, Brian L.; Pharoah, Blaze M.; Bellows, Sarina M.; Thayer, Peter R.; Fennie, Charles N.; Cowley, Ryan E.; Holland, Patrick L.:

    An Expedient Synthesis of 2,4,6-Tris(trifluoromethyl)aniline

    Image for article: An Expedient Synthesis of 2,4,6-Tris(trifluoromethyl)aniline

    • paper

  • 3598
    Ni, Feng; Li, Jianqi:

    A New Route to Roflumilast via Copper-Catalyzed Hydroxylation

    Image for article: A New Route to Roflumilast via Copper-Catalyzed Hydroxylation
    Supporting Information (PDF)
  • 3603
    Koguchi, Shinichi; Izawa, Kazuki:

    A New Method for the Synthesis of 1,5-Disubstituted 1,2,3-Triazoles via Triazolium Salt Intermediates

    Image for article: A New Method for the Synthesis of 1,5-Disubstituted 1,2,3-Triazoles via Triazolium Salt Intermediates
  • 3609
    Bae, Hoon; Jeon, Hongjun; Baek, Dong Jae; Lee, Dongjoo; Kim, Sanghee:

    Stereochemically Reliable Syntheses of Pachastrissamine and Its 2-epi-Congener via Oxazolidinone Precursors from an Established Starting Material N-tert-Butoxycarbonyl-Protected Phytosphingosine

    Image for article: Stereochemically Reliable Syntheses of Pachastrissamine and Its 2-<i>epi</i>-Congener via Oxazolidinone Precursors from an Established Starting Material <i>N</i>-<i>tert</i>-Butoxycarbonyl-Protected Phytosphingosine
    Supporting Information (PDF)
  • 3613
    Ahn, Sang-Hyun; Kim, Young Keun; Hyun, Jina; Lee, Kee-Jung:

    A Synthetic Pathway to the 1,4-Dihydro-2H-3-benzoxocine System from Morita–Baylis–Hillman Cinnamyl Alcohols with 2,5-Dimethoxy-2,5-dihydrofuran via the Heck Reaction

    Image for article: A Synthetic Pathway to the 1,4-Dihydro-2<i>H</i>-3-benzoxocine System from Morita–Baylis–Hillman Cinnamyl Alcohols with 2,5-Dimethoxy-2,5-dihydrofuran via the Heck Reaction
  • 3623
    Kimura, Tsutomu; Kobayashi, Gen; Ishigaki, Masashi; Inumaru, Mio; Sakurada, Jo; Satoh, Tsuyoshi:

    Coupling Reaction of Magnesium Alkylidene Carbenoids with α-Sulfonyl­allyllithiums: An Efficient Route to Multi-Substituted Vinylallenes

    Image for article: Coupling Reaction of Magnesium Alkylidene Carbenoids with α-Sulfonyl­allyllithiums: An Efficient Route to Multi-Substituted Vinylallenes
    Supporting Information (PDF)
  • 3633
    Jiang, Hui; Na, Risong; Zhang, Lei; Liu, Honglei; Li, Zhen; Wang, Bo; Guo, Hongchao:

    Samarium Diiodide Mediated Highly Diastereoselective Conjugate Reduction of the α,β-Unsaturated Ester Moiety in Heterocyclic Compounds

    Image for article: Samarium Diiodide Mediated Highly Diastereoselective Conjugate Reduction of the α,β-Unsaturated Ester Moiety in Heterocyclic Compounds
    Supporting Information (PDF)
  • 3639
    McDonald, Frank E.; Pereira, Claney L.:

    Stereo- and Regioselective Synthesis of 2-Amino-3,5-diols via Stereospecific Crotyl Transfer and Regioselective Aminohydroxylation

    Image for article: Stereo- and Regioselective Synthesis of 2-Amino-3,5-diols via Stereospecific Crotyl Transfer and Regioselective Aminohydroxylation
  • 3649
    Mahdavi, Mohammad; Asadi, Mehdi; Saeedi, Mina; Ebrahimi, Mostafa; Rasouli, Mohammad A.; Ranjbar, Parviz R.; Foroumadi, Alireza; Shafiee, Abbas:

    One-Pot, Four-Component Synthesis of Novel Imidazo[2,1-b]thiazol-5-amine Derivatives

    Image for article: One-Pot, Four-Component Synthesis of Novel Imidazo[2,1-<i>b</i>]thiazol-5-amine Derivatives
  • 3655
    Kálai, Tamás; Bognár, Balázs; Zsolnai, Dániel; Berente, Zoltán; Hideg, Kálmán:

    Synthesis of Nitroxide-Annulated Carbocycles and Heterocycles

    Image for article: Synthesis of Nitroxide-Annulated Carbocycles and Heterocycles
    Supporting Information (PDF)
  • 3661
    Gratzer, Katharina; Waser, Mario:

    Investigations Concerning the Syntheses of TADDOL-Derived Secondary Amines and Their Use To Access Novel Chiral Organocatalysts

    Image for article: Investigations Concerning the Syntheses of TADDOL-Derived Secondary Amines and Their Use To Access Novel Chiral Organocatalysts
    Open Access
    Supporting Inform.ation (PDF)
  • 3671
    Ahmad, Anees; Silva, Luiz F.:

    Synthesis of Chromanes and 4H-Chromenes: Exploring the Oxidation of 2H-Chromenes and Dihydro-1-benzoxepines by Hypervalent Iodine(III)

    Image for article: Synthesis of Chromanes and 4<i>H</i>-Chromenes: Exploring the Oxidation of 2<i>H</i>-Chromenes and Dihydro-1-benzoxepines by Hypervalent Iodine(III)
    Supporting Information (PDF)
  • 3678
    Goud, D. Raghavender; Pathak, Uma:

    A Mild and Efficient Synthesis of 2-Oxazolines via Transamidation–Cyclodehydrosulfurisation­ of Thioamides with 2-Aminoethanol

    Image for article: A Mild and Efficient Synthesis of 2-Oxazolines via Transamidation–Cyclodehydrosulfurisation­ of Thioamides with 2-Aminoethanol
    Supporting Information (PDF)
  • 3683
    Skonieczny, Kamil; Charalambidis, Georgios; Tasior, Mariusz; Krzeszewski, Maciej; Kalkan-Burat, Ayfer; Coutsolelos, Athanassios G.; Gryko, Daniel T.:

    General and Efficient Protocol for Formylation of Aromatic and Heterocyclic Phenols

    Image for article: General and Efficient Protocol for Formylation of Aromatic and Heterocyclic Phenols
    Supporting Information (PDF)
  • 3688
    Scarpi, Dina; Avataneo, Ottavia; Prandi, Cristina; Venturello, Paolo; Occhiato, Ernesto G.:

    Synthesis of Both Enantiomers of the Streptomyces Alkaloid 4-epi-SS20846A

    Image for article: Synthesis of Both Enantiomers of the <i>Streptomyces</i> Alkaloid 4-<i>epi</i>-SS20846A
    Supporting Information (PDF)
  • 3693
    Cheng, Xue-Ming; Chen, Min; Huang, Zhi-Tang; Zheng, Qi-Yu:

    Stereocontrolled Photodimerization of (E)-3-Benzylidene-4-chromanones in the Crystalline State: The Effect of a Halogen Group on the Chromanone Moiety

    Image for article: Stereocontrolled Photodimerization of (<i>E</i>)-3-Benzylidene-4-chromanones in the Crystalline State: The Effect of a Halogen Group on the Chromanone Moiety
    Supporting Information (PDF)