DOI: 10.1055/s-00000084

Synthesis

Issue 22 · Volume 52 · November 2020 DOI: 10.1055/s-010-49660

table of contents

V
Linked PDF of Table of Contents

review

3295
Grover, Nitika; Senge, Mathias O.: Synthetic Advances in the C–H Activation of Rigid Scaffold Molecules
https://www.thieme-connect.de/media/synthesis/202022/i_z0178_ga_10-1055_s-0040-1707884.gif

short review

3326
Yorimitsu, Hideki; Yoshimura, Aya; Misaki, Yohji: Catalytic C–H Arylation of Tetrathiafulvalenes for the Synthesis of Functional Materials
https://www.thieme-connect.de/media/synthesis/202022/i_z0334_ga_10-1055_s-0040-1707256.gif
3337
Li, Dan; Chen, Xiaochao; Gao, Wei: Asymmetric Synthesis of C1-Chiral THIQs with Imines in Isoquinoline Rings
https://www.thieme-connect.de/media/synthesis/202022/i_m0299_ga_10-1055_s-0040-1707206.gif

feature

3356
Ivanov, Konstantin L.; Tukhtaev, Hamidulla B.; Tukhtaeva, Feruza O.; Bezzubov, Stanislav I.; Melnikov, Mikhail Ya.; Budynina, Ekaterina M.: One-Pot Synthesis of γ-Azidobutyronitriles and Their Intramolecular Cycloadditions
https://www.thieme-connect.de/media/synthesis/202022/i_z0275_ga_10-1055_s-0040-1706402.jpg
Supporting Information CIF File

psp

3374
Delpe Acharige, Anjana; Neri, Raul; Hodgson, James; Bossmann, Stefan H.: A Catalyst-Free, Temperature-Driven One-Pot Synthesis of 1-Adamantylhydrazine Hydrochloride
https://www.thieme-connect.de/media/synthesis/202022/i_m0358_ga_10-1055_s-0040-1707353.gif
Supporting Information

special topic

Synthesis in Industry

3378
Maligres, Peter E.; Song, Zhiguo Jake; Strotman, Neil A.; Yin, Jinquin; Pei, Tao; Strotman, Hallena R.; Itoh, Tetsuji; Sherer, Edward C.; Humphrey, Guy R.: Synthesis of Fused Oxepane HIV Integrase Inhibitor MK-1376
https://www.thieme-connect.de/media/synthesis/202022/i_c0045_ga_10-1055_s-0040-1707994.gif
Supporting Information

3389
Toussaint, Frédéric C.; Defrance, Thierry; Decouvreur, Serge; Carly, Nicolas; Merschaert, Alain: Intensification of Free-Radical Racemization for a Non-activated Amine in a Continuous Flow Reactor
https://www.thieme-connect.de/media/synthesis/202022/i_c0232_ga_10-1055_s-0040-1707339.jpg
3397
Wächtler, Andreas; Bremer, Matthias; Maillard, David; Mohr, Thomas: Controlling the All-trans Stereochemistry in Liquid Crystalline 4,4′-Dialkyl-[1,1′-bicyclohexyl] Compounds
https://www.thieme-connect.de/media/synthesis/202022/i_c0256_ga_10-1055_s-0040-1707349.gif
3406
Stumpf, Andreas; St-Jean, Frédéric; Lao, David; Cheng, Zhigang Ken; Angelaud, Remy; Gosselin, Francis: Practical Early Development Synthesis of Nav1.7 Inhibitor GDC-0310
https://www.thieme-connect.de/media/synthesis/202022/i_c0207_ga_10-1055_s-0040-1707859.gif
Supporting Information
3415
Chen, Chengsheng; Wu, Ling; Wang, Yuwen; Wu, Linglin; Zhang, Yongda: Copper-Catalyzed Asymmetric Hydroamination of Styrenes with pivZPhos as Ligand
https://www.thieme-connect.de/media/synthesis/202022/i_c0264_ga_10-1055_s-0040-1707346.gif
Supporting Information

Synthesis in Industry

3420
Crawford, James J.; Liao, Daohong; Kolesnikov, Aleksandr; Lee, Wendy; Landry, Matthew L.: Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation
https://www.thieme-connect.de/media/synthesis/202022/i_c0401_ga_10-1055_s-0040-1707279.gif
Supporting Information

paper

3427
Kolupaeva, Ekaterina V.; Ozeryanskii, Valery A.; Pozharskii, Alexander F.: N-Methylated 1,8-Diaminonaphthalenes as Bifunctional Nucleo­philes in Reactions with α,ω-Dihalogenoalkanes: A Facile Route to Heterocyclic and Double Proton Sponges
https://www.thieme-connect.de/media/synthesis/202022/i_z0206_ga_10-1055_s-0040-1707079.gif
Supporting Information
3439
Luo, Nianhua; Zhong, Yuhong; Liu, Ji-Tian; Ouyang, Lu; Luo, Renshi: An Efficient Hydration and Tandem Transfer Hydrogenation of Alkynes for the Synthesis of Alcohol in Water
https://www.thieme-connect.de/media/synthesis/202022/i_g0279_ga_10-1055_s-0040-1707233.gif
Supporting Information
3446
Xie, Dengbing; Wang, Yiqiong; Yang, Bo; Zhang, Songlin: Neodymium-Promoted Highly Selective Carbon–Carbon Double Bond Formation of Ketones with Allyl Halides in the Presence of Diethyl Phosphite
https://www.thieme-connect.de/media/synthesis/202022/i_g0223_ga_10-1055_s-0040-1707219.gif
Supporting Information
3452
Liza, Umme Aiman; Sugiura, Ken-ichi: Functionalization of Bipyrenol: Potential Precursors for Advanced Chiral Molecules
https://www.thieme-connect.de/media/synthesis/202022/i_f0258_ga_10-1055_s-0040-1707341.gif
Supporting Information
3461
Nakamura, Itaru; Shiga, Keigo; Suzuki, Mao; Terada, Masahiro: Efficient Synthesis of O-tert-Propargylic Oximes via Nicholas Reaction
https://www.thieme-connect.de/media/synthesis/202022/i_f0290_ga_10-1055_s-0040-1707191.gif
Supporting Information
3466
Li, Qiao; Jin, Hongwei; Liu, Yunkui; Zhou, Bingwei: Nickel-Catalyzed Multicomponent Coupling Reaction of Alkyl Halides, Isocyanides and H2O: An Expedient Way to Access Alkyl Amides
https://www.thieme-connect.de/media/synthesis/202022/i_f0341_ga_10-1055_s-0040-1707229.gif
Supporting Information
3473
Bonilla-Reyes, Edgar; Sánchez-Carrillo, Adrian; Vázquez, Alfredo: Synthesis of l-Kynurenine and Homo-l-Kynurenine via an Aza-Fries Rearrangement
https://www.thieme-connect.de/media/synthesis/202022/i_m0220_ga_10-1055_s-0040-1707223.gif
Supporting Information
3480
Chavan, Subhash P.; Pawar, Ambaji A.; Patil, Niteen B.; Kadam, Appasaheb L.; Shinde, Shrikrishna S.: Scalable Synthesis of 3-Ethyl-4-methyl-1,5-dihydro-2H-pyrrol-2-one: An Important Building Block of the Antidiabetic Drug Glimepiride
https://www.thieme-connect.de/media/synthesis/202022/i_n0639_ga_10-1055_s-0040-1707344.gif
Supporting Information
3485
Arabadzhi, Svetlana S.; Zharkov, Mikhail N.; Kuchurov, Ilya V.; Zlotin, Sergei G.: Synthesis of Chiral N-Nitro-oxazolidin-2-ones and O-(β-Nitraminoalkyl) Carbamates in Liquefied 1,1,1,2-Tetrafluoroethane Medium
https://www.thieme-connect.de/media/synthesis/202022/i_t0303_ga_10-1055_s-0040-1706762.gif
Supporting Information

book review

3492
Lakhdar, Sami: Science of Synthesis: Photocatalysis in Organic Synthesis