DOI: 10.1055/s-00000083

Synlett

Issue 12 · Volume 2003 · October 2003 DOI: 10.1055/s-002-2820

editorial

  • I

    Editorial

    • account

  • 1759
    Jun, Jong-Gab:

    Introduction of Bicyclic Ketal Chemistry: Synthesis and Transformation Reaction of 6,8-Dioxabicyclo[3.2.1]octane Skeletal System

    Image for article: Introduction of Bicyclic Ketal Chemistry: Synthesis and Transformation Reaction of 6,8-Dioxabicyclo[3.2.1]octane Skeletal System

    • letter

  • 1778
    Bernardi, Luca; Bonini, Bianca F.; Capitò, Elena; Dessole, Gabriella; Fochi, Mariafrancesca; Comes-Franchini, Mauro; Ricci, Alfredo:

    A New and Practical Procedure for the Bruylants Reaction. Zinc-Mediated Synthesis of Tertiary Homoallylamines and β-Aminoesters

    Image for article: A New and Practical Procedure for the Bruylants Reaction. Zinc-Mediated Synthesis of Tertiary Homoallylamines and β-Aminoesters
  • 1783
    Schumann, Herbert; Kaufmann, Jens; Schmalz, Hans-Günther; Böttcher, Andreas; Gotov, Battsengel:

    Pd-Catalyzed Cross-Coupling of Haloarenes and Chloroarene-Cr(CO)3 Complexes with Stabilized Vinyl- and Allylaluminium Reagents

    Image for article: Pd-Catalyzed Cross-Coupling of Haloarenes and Chloroarene-Cr(CO)<SUB>3</SUB> Complexes with Stabilized Vinyl- and Allylaluminium Reagents
  • 1789
    Wu, Yong-Jin; He, Huan:

    Copper-Catalyzed Cross-Coupling of Aryl Halides and Thiols Using Microwave Heating

    Image for article: Copper-Catalyzed Cross-Coupling of Aryl Halides and Thiols Using Microwave Heating
  • 1791
    Lingard, Iain; Bhalay, Gurdip; Bradley, Mark:

    Hexadienyloxycarbonyl (Hdoc) - A Mild Acid Labile Protecting Group for Amines

    Image for article: Hexadienyloxycarbonyl (Hdoc) - A Mild Acid Labile Protecting Group for Amines
  • 1793
    Palaniappan, Srinivasan; Narender, Puli; Saravanan, Chandrasekaran; Rao, Vaidya Jayathirtha:

    Polyaniline-Supported Sulfuric Acid Salt as a Powerful Catalyst for the Protection and Deprotection of Carbonyl Compounds

    Image for article: Polyaniline-Supported Sulfuric Acid Salt as a Powerful Catalyst for the Protection and Deprotection of Carbonyl Compounds
  • 1797
    Quayle, Peter; Fengas, David; Richards, Stuart:

    Atom Transfer Radical Cyclisations Mediated by the Grubbs Ruthenium Metathesis Catalyst

    Image for article: Atom Transfer Radical Cyclisations Mediated by the Grubbs Ruthenium Metathesis Catalyst
  • 1801
    Wolf, Christian; Tumambac, Gilbert E.; Villalobos, Cristina N.:

    Acid-Mediated Halogen Exchange in Heterocyclic Arenes: A Highly Effective Iodination Method

    Image for article: Acid-Mediated Halogen Exchange in Heterocyclic Arenes: A Highly Effective Iodination Method
  • 1805
    Chakraborti, Asit K.; Gulhane, Rajesh; Shivani:

    Bismuth Oxide Perchlorate as a Highly Efficient Catalyst for Heteroatom Acylation Under Solvent-Free Conditions

    Image for article: Bismuth Oxide Perchlorate as a Highly Efficient Catalyst for Heteroatom Acylation Under Solvent-Free Conditions
  • 1809
    Ito, Katsuji; Akashi, Suemi; Saito, Bunnai; Katsuki, Tsutomu:

    Asymmetric Intramolecular Allylic Amination: Straightforward Approach to Chiral C1-Substituted Tetrahydroisoquinolines

    Image for article: Asymmetric Intramolecular Allylic Amination: Straightforward Approach to Chiral C1-Substituted Tetrahydroisoquinolines
  • 1813
    Berkenbusch, Thilo; Brückner, Reinhard:

    Concise Synthesis of Optically Pure syn-1,3-Diols by Stereoselective Desymmetrization of a Divinylcarbinol

    Image for article: Concise Synthesis of Optically Pure <EM EMTYPE="ITALIC">syn</EM>-1,3-Diols by Stereoselective Desymmetrization of a Divinylcarbinol
  • 1817
    Zhang, Dong-hui; Zhou, Wei-shan:

    Synthetic Studies Towards Phorboxazole B: Stereoselective Synthesis of the C3-C19 Bis-oxane Oxazole Fragment

    Image for article: Synthetic Studies Towards Phorboxazole B: Stereoselective Synthesis of the C3-C19 Bis-oxane Oxazole Fragment
  • 1822
    Maes, Bert U. W.; Loones, Kristof T. J.; Lemière, Guy L. F.; Dommisse, Roger A.:

    The First Rapid Palladium-Catalyzed Aminations of (Azahetero)aryl Chlorides under Temperature-Controlled Microwave Heating

    Image for article: The First Rapid Palladium-Catalyzed Aminations of (Azahetero)aryl Chlorides under Temperature-Controlled Microwave Heating
  • 1826
    Radics, Gábor; Koksch, Beate; El-Kousy, Salah M.; Spengler, Jan; Burger, Klaus:

    l-α-Methylhomoisoserine: A New Versatile Building Block for Peptide and Depsipeptide Modification

    Image for article: <EM EMTYPE="CAPS">l</EM>-α-Methylhomoisoserine: A New Versatile Building Block for Peptide and Depsipeptide Modification
  • 1830
    Müller, Paul; Ghanem, Ashraf:

    Asymmetric Cyclopropanation of Olefins with an in situ Generated Phenyliodonium Ylide

    Image for article: Asymmetric Cyclopropanation of Olefins with an in situ Generated Phenyliodonium Ylide
  • 1834
    Boucard, Valérie; Larrieu, Karen; Lubin-Germain, Nadège; Uziel, Jacques; Augé, Jacques:

    C-Glycosylated Phenylalanine Synthesis by Palladium-Catalyzed Cross-Coupling Reactions

    Image for article: <EM EMTYPE="BOLDITALIC">C</EM>-Glycosylated Phenylalanine Synthesis by Palladium-Catalyzed Cross-Coupling Reactions
  • 1838
    Kim, Su Jeong; Bang, Eun-Kyoung; Kim, Byeang Hyean:

    Synthesis of Novel Phosphoramidite Building Blocks from Pentaerythritol

    Image for article: Synthesis of Novel Phosphoramidite Building Blocks from Pentaerythritol
  • 1841
    Ballini, Roberto; Fiorini, Dennis; Palmieri, Alessandro:

    Highly Convenient, One-Pot Synthesis of Nitriles from Aldehydes Using the NH2OH·HCl/NaI/MeCN System

    Image for article: Highly Convenient, One-Pot Synthesis of Nitriles from Aldehydes Using the NH<SUB>2</SUB>OH·HCl/NaI/MeCN System
  • 1844
    El Kaïm, Laurent; Gautier, Laurent; Grimaud, Laurence; Michaut, Valerie:

    New Insight into the Azaenamine Behaviour of N-Arylhydrazones: First Aldol and Improved Mannich Reactions with Unactivated Aldehydes

    Image for article: New Insight into the Azaenamine Behaviour of <EM EMTYPE="ITALIC">N</EM>-Arylhydrazones: First Aldol and Improved Mannich Reactions with Unactivated Aldehydes
  • 1847
    Martínez-Palou, Rafael; de Paz, Gerardo; Marín-Cruz, Jesús; Zepeda, Luis Gerardo:

    Synthesis of Long Chain 2-Alkyl-1-(2-hydroxyethyl)-2-imidazolines under Microwave in Solvent-Free Conditions

    Image for article: Synthesis of Long Chain 2-Alkyl-1-(2-hydroxyethyl)-2-imidazolines under Microwave in Solvent-Free Conditions
  • 1850
    Koike, Tooru; Mori, Atsunori:

    Palladium-Catalyzed Cross-Coupling Reaction of Silicone with Aryl Chlorides

    Image for article: Palladium-Catalyzed Cross-Coupling Reaction of Silicone with Aryl Chlorides<SUP></SUP>
  • 1853
    Atkinson, Sov; Meredith, Paul:

    Synthesis of Acetoxy Stabilised Indolequinones as Precursors to Model Eumelanin Polymers

    Image for article: Synthesis of Acetoxy Stabilised Indolequinones as Precursors to Model Eumelanin Polymers
  • 1856
    Viseux, E. M. E.; Parsons, P. J.; Pavey, J. B. J.; Carter, C. M.; Pinto, I.:

    Model Studies Towards the Total Synthesis of the Anticancer Agent Roseophili­n

    Image for article: Model Studies Towards the Total Synthesis of the Anticancer Agent Roseophili­n
  • 1859
    van Otterlo, Willem A. L.; Pathak, Rakhi; de Koning, Charles B.:

    Ruthenium-Mediated Isomerization and Ring-Closing Metathesis: Versatile Syntheses of 6-, 7- and 8-Membered Benzo-Fused Heterocycles

    Image for article: Ruthenium-Mediated Isomerization and Ring-Closing Metathesis: Versatile Syntheses of 6-, 7- and 8-Membered Benzo-Fused Heterocycles
  • 1862
    Stanetty, Peter; Schnürch, Michael; Mihovilovic, Marko D.:

    Synthesis of Pyridinyl-Pyrimidines via Pd-Catalyzed Cross-Coupling Reactions: A Comparison of Classical Thermal and Microwave Assisted Reaction Conditions

    Image for article: Synthesis of Pyridinyl-Pyrimidines via Pd-Catalyzed Cross-Coupling Reactions: A Comparison of Classical Thermal and Microwave Assisted Reaction Conditions
  • 1865
    Tamai, Tetsuo; Asano, Shingo; Totani, Kiichiro; Takao, Ken-ichi; Tadano, Kin-ichi:

    Highly Stereoselective [3+2] Cycloadditions of Nitrile Oxides to Methyl 4-O-Acryloyl-6-deoxy-2,3-O-(t-butyldimethylsilyl)-α-d-glucopyranoside

    Image for article: Highly Stereoselective [3+2] Cycloadditions of Nitrile Oxides to Methyl 4-<EM EMTYPE="ITALIC">O</EM>-Acryloyl-6-deoxy-2,3-<EM EMTYPE="ITALIC">O</EM>-(<EM EMTYPE="ITALIC">t</EM>-butyldimethylsilyl)-α-<EM EMTYPE="CAPS">d</EM>-glucopyranoside
  • 1868
    Tashiro, Aya; Mitsuishi, Akimasa; Irie, Ryo; Katsuki, Tsutomu:

    (NO)Ru(salen)-Catalyzed Aerobic Oxidation of o-Hydroxybenzyl Alcohol Derivatives­

    Image for article: (NO)Ru(salen)-Catalyzed Aerobic Oxidation of <EM EMTYPE="ITALIC">o</EM>-Hydroxybenzyl Alcohol Derivatives­
  • 1871
    Cämmerer, Simon S.; Viciu, Mihai S.; Stevens, Edwin D.; Nolan, Steven P.:

    Use of (NHC)Pd(η3-allyl)Cl (NHC = N-Heterocyclic Carbene) in a Palladium-mediated Approach to Cryptocarya Alkaloids

    Image for article: Use of (NHC)Pd(η<SUP>3</SUP>-allyl)Cl (NHC = <EM EMTYPE="ITALIC">N</EM>-Heterocyclic Carbene) in a Palladium-mediated Approach to <EM EMTYPE="ITALIC">Cryptocarya</EM> Alkaloids
  • 1874
    Maerten, Eddy; Hassouna, Fatima; Couve-Bonnaire, Samuel; Mortreux, André; Carpentier, Jean-François; Castanet, Yves:

    Direct Synthesis of Benzoylpyridines from Chloropyridines via a Palladium-Carbene Catalyzed Carbonylative Suzuki Cross-Coupling Reaction

    Image for article: Direct Synthesis of Benzoylpyridines from Chloropyridines via a Palladium-Carbene Catalyzed Carbonylative Suzuki Cross-Coupling Reaction
  • 1877
    Zolfigol, Mohammad Ali; Mohammadpoor-Baltork, Iraj; Mirjalili, Bi Bi Fatemeh; Bamoniri, Abdolhamid:

    Silica Sulfuric Acid: An Efficient Catalyst for the Direct Conversion of Primary and Secondary Trimethylsilyl Ethers to their Corresponding Ethers under Mild and Heterogeneous Conditions

    Image for article: Silica Sulfuric Acid: An Efficient Catalyst for the Direct Conversion of Primary and Secondary Trimethylsilyl Ethers to their Corresponding Ethers under Mild and Heterogeneous Conditions
  • 1880
    Zeni, Gilson; Stracke, Marcelo Paulo; Lissner, Elizeo; Braga, Antonio Luiz:

    A Convenient Preparation of Chalcogenoenynes from β-Bromovinyl Ketene Chalcogenoacetals

    Image for article: A Convenient Preparation of Chalcogenoenynes from β-Bromovinyl Ketene Chalcogenoacetals
  • 1883
    Motoyama, Yukihiro; Nishiyama, Hisao:

    Bis(oxazolinyl)phenylrhodium(III) Aqua Complex: Efficiency in Enantioselective Addition of Methallyltributyltin to Aldehydes under Aerobic Conditions

    Image for article: Bis(oxazolinyl)phenylrhodium(III) Aqua Complex: Efficiency in Enantioselective Addition of Methallyltributyltin to Aldehydes under Aerobic Conditions
  • 1886
    Kalogerakis, Aris; Groth, Ulrich:

    Total Synthesis of the Angucylinone Antibiotic (+)-Rubiginone B2

    Image for article: Total Synthesis of the Angucylinone Antibiotic (+)-Rubiginone B<SUB>2</SUB>
  • 1889
    Pisaneschi, Federica; Cordero, Franca M.; Brandi, Alberto:

    Resin Linked Dipolarophiles to Mask Nitrones

    Image for article: Resin Linked Dipolarophiles to Mask Nitrones
  • 1892
    Korn, Tobias J.; Cahiez, Gérard; Knochel, Paul:

    New Cobalt-Catalyzed Cross-Coupling Reactions of Heterocyclic Chlorides with Aryl and Heteroaryl Magnesium Halides

    Image for article: New Cobalt-Catalyzed Cross-Coupling Reactions of Heterocyclic Chlorides with Aryl and Heteroaryl Magnesium Halides
  • 1895
    Alexander, Varughese M.; Khandekar, Amit C.; Samant, Shriniwas D.:

    Solvent-Free Iodination of Arenes at Room Temperature

    Image for article: Solvent-Free Iodination of Arenes at Room Temperature
  • 1898
    Maguire, Naomi E.; McLaren, Andrew B.; Sweeney, J. B.:

    Asymmetric Synthesis of Arylalanines via Asymmetric aza-Darzens (ADZ) Reaction

    Image for article: Asymmetric Synthesis of Arylalanines via Asymmetric aza-Darzens (ADZ) Reaction

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  • 1901
    Martin, Harry J.; List, Benjamin:

    Mining Sequence Space for Asymmetric Aminocatalysis: N-Terminal Prolyl-Peptides Efficiently Catalyze Enantioselective Aldol and Michael Reactions

    Image for article: Mining Sequence Space for Asymmetric Aminocatalysis: <EM EMTYPE="ITALIC">N-</EM>Terminal Prolyl-Peptides Efficiently Catalyze Enantioselective Aldol and Michael Reactions
  • 1903
    Pojarliev, Peter; Biller, William T.; Martin, Harry J.; List, Benjamin:

    Highly Enantioselective Synthesis of 1,2-Amino Alcohol Derivatives via Proline-Catalyzed Mannich Reaction

    Image for article: Highly Enantioselective Synthesis of 1,2-Amino Alcohol Derivatives via Proline-Catalyzed Mannich Reaction
  • 1906
    Chowdari, Naidu S.; Ramachary, D. B.; Barbas III, Carlos F.:

    Organocatalysis in Ionic Liquids: Highly Efficient l-Proline-Catalyzed Direct Asymmetric Mannich Reactions Involving Ketone and Aldehyde Nucleophiles

    Image for article: Organocatalysis in Ionic Liquids: Highly Efficient <EM EMTYPE="CAPS">l</EM>-Proline-Catalyzed Direct Asymmetric Mannich Reactions Involving Ketone and Aldehyde Nucleophiles
  • 1910
    Ramachary, D. B.; Chowdari, Naidu S.; Barbas III, Carlos F.:

    The First Organocatalytic Hetero-Domino Knoevenagel-Diels-Alder-Epimerization Reactions: Diastereoselective Synthesis of Highly Substituted Spiro[cyclohexane-1,2′-indan]-1′,3′,4-triones

    Image for article: The First Organocatalytic Hetero-Domino Knoevenagel-Diels-Alder-Epimerization Reactions: Diastereoselective Synthesis of Highly Substituted Spiro[cyclohexane-1,2′-indan]-1′,3′,4-triones
  • 1915
    Bøgevig, Anders; Poulsen, Thomas B.; Zhuang, Wei; Jørgensen, Karl Anker:

    Formation of Optically Active Functionalized β-Hydroxy Nitrones Using a Proline Catalyzed Aldol Reaction of Aldehydes with Carbonyl Compounds and Hydroxylamines

    Image for article: Formation of Optically Active Functionalized β-Hydroxy Nitrones Using a Proline Catalyzed Aldol Reaction of Aldehydes with Carbonyl Compounds and Hydroxylamines
  • 1919
    Wenzel, Anna G.; Lalonde, Mathieu P.; Jacobsen, Eric N.:

    Divergent Stereoinduction Mechanisms in Urea-Catalyzed Additions to Imines

    Image for article: Divergent Stereoinduction Mechanisms in Urea-Catalyzed Additions to Imines
  • 1923
    Griswold, Keith S.; Horstmann, Thomas E.; Miller, Scott J.:

    Acyl Sulfonamide Catalysts for Glycosylation Reactions with Trichloroacetimidate Donors

    Image for article: Acyl Sulfonamide Catalysts for Glycosylation Reactions with Trichloroacetimidate Donors
  • 1927
    Hang, Jianfeng; Deng, Li:

    Dynamic Kinetic Resolution for Asymmetric Synthesis of α-Alkyl Amino Acids via Dual-Function Catalysis of Modified Cinchona Alkaloids

    Image for article: Dynamic Kinetic Resolution for Asymmetric Synthesis of α-Alkyl Amino Acids via Dual-Function Catalysis of Modified Cinchona Alkaloids
  • 1931
    Ooi, Takashi; Kubota, Yasushi; Maruoka, Keiji:

    A New N-Spiro C2-Symmetric Chiral Quaternary Ammonium Bromide Consisting of 4,6-Disubstituted Biphenyl Subunit as an Efficient Chiral Phase-Transfer Catalyst

    Image for article: A New <EM EMTYPE="ITALIC">N</EM>-Spiro C<SUB>2</SUB>-Symmetric Chiral Quaternary Ammonium Bromide Consisting of 4,6-Disubstituted Biphenyl Subunit as an Efficient Chiral Phase-Transfer Catalyst
  • 1934
    Kerr, Mark S.; Rovis, Tomislav:

    Effect of the Michael Acceptor in the Asymmetric Intramolecular Stetter Reaction

    Image for article: Effect of the Michael Acceptor in the Asymmetric Intramolecular Stetter Reaction
  • 1937
    Shah, Meha H.; France, Stefan; Lectka, Thomas:

    Bicarbonate Salts as Cost-Effective Bases for the Synthesis of Ketenes and Their Synthetic Equivalents Applied to the Asymmetric Synthesis of β-Lactams

    Image for article: Bicarbonate Salts as Cost-Effective Bases for the Synthesis of Ketenes and Their Synthetic Equivalents Applied to the Asymmetric Synthesis of β-Lactams

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  • 1940
    Goundry, William R. F.:

    Trimethylsilyl Trifluoromethanesulfonate (TMSOTf)

  • 1942
    Pasupathy, K.:

    Magnesium/Methanol