DOI: 10.1055/s-00000131

Synfacts

Issue 04 · Volume 2010 · April 2010 DOI: 10.1055/s-002-20900

Synform

A33
Zanda, Matteo: SYNFORM ISSUE 2010/04

Synthesis of Natural Products and Potential Drugs

z375
All PDFs of this category
0375
Ishida, N.; Shimamoto, Y.; Murakami, M.: Synthesis of (E)- and (Z)-Tamoxifen
0376
Magauer, T.; Mulzer, J.; Tiefenbacher, K.: Syntheses of (+)-Echinopine A and B
0377
Chen, K.; Baran, P. S.: Synthesis of Eudesmane Terpenes by C-H Activation
0378
Walker, M. D.; Andrews, B. I.; Burton, A. J.; Humphreys, L. D.; Kelly, G.; Schilling, M. B.; Scott, P. W.: Synthesis of SB-406725A
0379
al., J. L. Vennerstrom et: Synthesis of Arterolane and Analogues
0380
Osato, H.; Jones, I. L.; Chen, A.; Chai, C. L. L.: Synthesis of Tamiflu
0381
Penner, M.; Rauniyar, V.; Kaspar, L. T.; Hall, D. G.: Asymmetric Synthesis of Palmerolide A
0382
Ni, Y.; Kassab, R. M.; Chevliakov, M. V.; Montgomery, J.: Syntheses of Isodomoic Acids G and H
0383
Karadeolian, A.; Kerr, M. A.: Synthesis of (+)-Isatisine A
0384
Webel, M.; Palmer, A. M.; Scheufler, C.; Haag, D.; Müller, B.: Synthesis of the Benzimidazole Fragment of BYK405879
0385
Fray, M. J.; Gillmore, A.T.; Glossop, M. S.; McManus, D. J.; Moses, I. B.; Praquin, C. F. B.; Reeves, K. A.; Thompson, L. R.: Synthesis of PF-1247324, a NaV1.8 Sodium Channel Modulator
0386
Wu, Y.-C.; Zhu, J.: Syntheses of (-)-Renieramycin M and G and (-)-Jorumycin
0387
Ohmiya, H.; Makida, Y.; Li, D.; Tanabe, M.; Sawamura, M.: Synthesis of (+)-Sertraline
0388
Kang, S.; Lee, H.-K.: Synthesis of (S)-(+)-Dapoxetine
0389
Gallagher, B. D.; Taft, B. R.; Lipshutz, B. H.: Synthesis of (R)-Tolterodine
0390
Cribiú, R.; Jäger, C.; Nevado, C.: Synthesis of Iriomoteolide 3a
0391
Denmark, S. E.; Liu, J. H.-C.; Muhuhi, J. M.: Syntheses of Isodomoic Acids G and H
0392
Tietze, L. F.; Tölle, N.; Kratzert, D.; Stalke, D.: Formal Synthesis of (+)-Erysotramidine
0393
Yu, S.; Haight, A.; Kotecki, B.; Wang, L.; Lukin, K.; Hill, D. R.: Synthesis of a TRPV1 Receptor Antagonist

Synthesis of Heterocycles

z395
All PDFs of this category
0395
Zhang, G.; Cui, L.; Wang, Y.; Zhang, L.: Gold-Catalyzed Synthesis of THFs and Pyrrolidines by Oxidative Coupling
0396
Huang, X.; Zhang, T.: Synthesis of C9-Functionalized Xanthenes and Acridines
0397
Liu, W.; Jiang, H.; Zhang, M.; Qi, C.: Synthesis of Highly Substituted Furans from Alkynoates and 1,3-Dicarbonyls
0398
Zhang, X.; Yao, T.; Campo, M. A.; Larock, R. C.: Halo-Induced Heteroannulation Route to Quinolines
0399
Han, J.; Xu, B.; Hammond, G. B.: Copper-Catalyzed Synthesis of Pyrrolidines and Piperidines
0400
Vovk, M. V.; Golovach, N. M.; Sukach, V. A.: Synthesis of 4-Aryl-4-trifluoromethyl-4H-1,3-oxa(thia)zines
0401
Zeng, X.; Kinjo, R.; Donnadieu, B.; Bertrand, G.: Gold(I)-Catalyzed Hydroammoniumation and Methylamination of Alkynes to Indoles
0402
Matsnev, A.; Noritake, S.; Nomura, Y.; Tokunaga, E.; Nakamura, S.; Shibata, N.: Synthesis of Thiophenium Salts: A Trifluoromethylation Reagent
0403
Peng, C.; Wang, Y.; Liu, L.; Wang, H.; Zhao, J.; Zhu, Q.: Synthesis of Substituted Quinolines from 2-Alkynylanilines
0404
He, Z.-Q.; Han, B.; Li, R.; Wu, L.; Chen, Y.-C.: Enantioselective Synthesis of Lactone-[2,3-b]piperidines
0405
Fontana, F.; Tron, G. C.; Barbero, N.; Ferrini, S.; Thomas, S. P.; Aggarwal, V. K.: Palladium-Catalyzed Synthesis of β-Lactams by Carbonylation of Vinyl Aziridines
0406
Liu, W.; Jiang, H.; Huang, L.: Synthesis of Polysubstituted Pyrroles by Condensation of Acetylenes and Amines
0407
Okitsu, T.; Nakazawa, D.; Kobayashi, A.; Mizohata, M.; In, Y.; Ishida, T.; Wada, A.: Iodocyclization-Based Synthesis of Spiro Heterocycles
0408
Zhao, T.; Xu, B.: Palladium-Catalyzed C-N Coupling-Hydroamination Route to 4-Quinolones

Synthesis of Materials and Unnatural Products

z409
All PDFs of this category
0409
Gsänger, M.; Oh, J. H.; Könemann, M.; Höffken, H. W.; Krause, A.-M.; Bao, Z.; Würthner, F.: A Twisted Perylene Semiconductor
0410
Wezenberg, S. J.; Kleij, A. W.: Co(III) Operation Makes it Happen
0411
Wang, Z.; Shi, J.; Wang, J.; Li, C.; Tian, X.; Cheng, Y.; Wang, H.: Helicene and Double Helicene
0412
Jiang, W.; Li, Y.; Yue, W.; Zhen, Y.; Qu, J.; Wang, Z.: Pyridyl Annelated Perylene Bisimides
0413
Kaur, I.; Jazdzyk, M.; Stein, N. N.; Prusevich, P.; Miller, G. P.: Nine in a Row
0414
Chen, T.-A.; Lee, T.-J.; Lin, M.-Y.; Sohel, S. M. A.; Diau, E. W.-G.; Lush, S.-F.; Liu, R.-S.: Polyaromatic Oligomers
0415
Choi, H.; Raabe, I.; Kim, D.; Teocoli, F.; Kim, C.; Song, K.; Yum, J.-H.; Ko, J.; Nazeeruddin, Md. K.; Grätzel, M.: Thienothiophene-Based Organic Sensitizers
0416
Bhalla, V.; Singh, H.; Kumar, M.: Fluoride-Induced Formation of Triphenylene Chemodosimeter
0417
Shirtcliff, L. D.; Xu, H.; Diederich, F.: Fluorophore-Appended Resorcin[4]arene Cavitands
0418
Ohmae, T.; Nishinaga, T.; Wu, M.; Iyoda, M.: Planarized Cyclooctatetraenes
0419
Mike, J. F.; Inteman, J. J.; Ellern, A.; Jeffries-EL, M.: Versatile Monomers for Conjugated Polymer Synthesis
0420
Qu, H.; Luo, J.; Zhang, X.; Chi, C.: A Novel n-Type PPV
0421
Yamago, S.; Watanabe, Y.; Iwamoto, T.: Concise Cycloparaphenylene Synthesis
0422
Morishita, T.; Yoshida, H.; Ohshita, J.: Copper-Catalyzed Domino Formation of (Alkynyl)bromoarenes
0423
Saino, N.; Kawaji, T.; Ito, T.; Matsushita, Y.; Okamoto, S.: Polyacenes from the Cyclotrimerization of Alkynes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z425
All PDFs of this category
0425
Lou, S.; Fu, G. C.: Asymmetric Kumada Couplings of α-Bromo Ketones
0426
Yamauchi, M.; Morimoto, M.; Miura, T.; Murakami, M.: Nickel-Catalyzed Denitrogenative Annulation
0427
Feske, M. I.; Santanilla, A. B.; Leighton, J. L.: Allylation of N-Heteroaryl Hydrazones
0428
Thaler, T.; Haag, B.; Gavryushin, A.; Schober, K.; Hartmann, E.; Gschwind, R. M.; Zipse, H.; Mayer, P.; Knochel, P.: Diastereoselective Negishi Coupling of Cycloalkylzinc Reagents
0429
Bai, W.-J.; Xie, J.-H.; Li, Y.-L.; Liu, S.; Zhou, Q.-L.: Asymmetric Synthesis of β-Aryloxy Alcohols via Dynamic Kinetic Resolution
0430
Rodrigues, A.; Lee, E. E.; Batey, R. A.: Synthesis of Chiral Pyridones by Palladium-Catalyzed Rearrangement
0431
Shen, X.; Buchwald, S. L.: Rhodium-Catalyzed Enantioselective Hydroamination of Alkenes
0432
Igawa, K.; Kokan, N.; Tomooka, K.: Synthesis of Chiral Silacarboxylic Acids and Esters
0433
Flynn, C. J.; Elcoate, C. J.; Lawrence, S. E.; Maguire, A. R.: Copper-Catalyzed Asymmetric C-H Insertion of α-Diazosulfones
0434
Larionov, O. V.; Corey, E. J.: Asymmetric Conjugate Addition of Acetylene Nucleophiles
0435
González, A. Z.; Toste, F. D.: Catalytic Asymmetric Cycloaddition of Allene-Dienes
0436
Simaan, S.; Goldberg, A. F. G.; Rosset, S.; Marek, I.: Metal-Catalyzed Ring-Opening Hydro-metalation of Alkylidenecyclopropanes
0437
Liu, Y.; Shang, D.; Zhou, X.; Zhu, Y.; Lin, L.; Liu, X.; Feng, X.: Metal-Controlled Reversal of Enantio-selectivity in the Alkylation of Indoles
0438
Ogata, K.; Sugasawa, J.; Atsuumi, Y.; Fukuzawa, S.-i.: Nickel-Catalyzed Reaction of Norbornene with Two Alkynes
0439
Sasaki, Y.; Zhong, C.; Sawamura, M.; Ito, H.: Copper-Catalyzed Asymmetric Mono-borylation of 1,3-Dienes
0440
LaLonde, R. L.; Wang, Z. J.; Mba, M.; Lackner, A. D.; Toste, F. D.: Gold-Catalyzed Intramolecular Hydroamination and Hydroalkoxylation
0441
Singh, P. K.; Singh, V. K.: Zn(II) Complexes Catalyzed Asymmetric Friedel-Crafts Alkylation of Pyrroles
0442
Olson, A. C.; Overman, L. E.; Sneddon, H. F.; Ziller, J. W.: Enantioselective Allylic Etherification Using a Novel COP Catalyst
0443
Brown, M. K.; Corey, E. J.: Preparation of Chiral-Bridged Dienes - Ligands for Enantioselective Catalysis
0444
Ito, H.; Okura, T.; Matsuura, K.; Sawamura, M.: Copper(I)-Catalyzed Desymmetrization of meso-2-Alkene-1,4-diol Derivatives
0445
Hatano, M.; Horibe, T.; Ishihara, K.: Asymmetric Direct Mannich-Type Reaction Catalyzed by Chiral Lithium Complexes
0446
He, H.; Liu, W.-B.; Dai, L.-X.; You, S.-L.: Synthesis of Chiral Benzoazepines through Allylic Substitution
0447
Tanaka, R.; Noguchi, K.; Tanaka, K.: Rhodium-Catalyzed Asymmetric Reductive Cyclization of Alkynals
0448
Suyama, K.; Sakai, Y.; Matsumoto, K.; Saito, B.; Katsuki, T.: Asymmetric Hydrophosphonylation of Aldehydes
0449
Hanhan, N. V.; Sahin, A. H.; Chang, T. W.; Fettinger, J. C.; Franz, A. K.: Asymmetric Addition of Aromatic Nucleophiles to Isatins
0450
Liao, S.; List, B.: Chiral Phosphate Counteranion Directed Enantioselective Expoxidation
0451
Robles-Machín, R.; González-Esguevillas, M.; Adrio, J.; Carretero, J. C.: Pyrrolidine Synthesis from Copper-Catalyzed 1,3-Dipolar Cycloadditions
0452
Kanbayashi, N.; Onitsuka, K.: Ruthenium-Catalyzed Asymmetric Allylic Substitution with Metal Carboxylates
0453
Overman, L. E.; Tanis, P. S.: Stereochemistry of the Prins-Pinacol Rearrangement
0454
Ueda, M.; Hartwig, J. F.: Iridium-Catalyzed Allylic Substitution with Aromatic and Aliphatic Sulfinates

Metal-Mediated Synthesis

z455
All PDFs of this category
0455
Guan, B.-T.; Lu, X.-Y.; Zheng, Y.; Yu, D.-G.; Wu, T.; Li, K.-L.; Li, B.-J.; Shi, Z.-J.: Diaryl Sulfates as Electrophiles in Kumada Cross-Coupling Reactions
0456
Demir, A. S.; Findik, H.; Saygili, N.; Subasi, N. T.: Manganese(III)-Mediated Biaryl Synthesis
0457
Everson, D. A.; Shrestha, R.; Weix, D. J.: Nickel-Catalyzed Reductive Cross-Coupling of Aryl Halides with Alkyl Halides
0458
Zhang, Z.; Liu, Y.; Gong, M.; Zhao, X.; Zhang, Y.; Wang, J.: Palladium-Catalyzed Carbonylation/Acyl Migratory Insertion Sequence
0459
Gooßen, L. J.; Rodríguez, N.; Lange, P. P.; Linder, C.: Decarboxylative Coupling of Aryl Tosylates with Aromatic Carboxylate Salts
0460
Sada, M.; Matsubara, S.: 1,3-Diketone Synthesis via a Novel Tandem Reaction
0461
Fields, W. H.; Chruma, J. J.: Decarboxylative Benzylation of Diphenyl-glycinate Imines
0462
Luo, F.; Pan, C.; Wang, W.; Ye, Z.; Cheng, J.: Stereoselective Reduction of Alkynes to cis- and trans-Alkenes Using Pd/HSiEt3
0463
Mo, J.; Kim, S. H.; Lee, P. H.: Tandem One-Pot Diels-Alder/Cross-Coupling Reactions of Organoindium Reagents
0464
Kuninobu, Y.; Nishi, M.; Kawata, A.; Takata, H.; Hanatani, Y.; S., S. Yudha; Iwai, A.; Takai, K.: Re- and Mn-Catalyzed Formal Cycloaddition of 1,3-Dicarbonyl Compounds and Alkynes
0465
Bernoud, E.; Duc, G. Le; Bantreil, X.; Prestat, G.; Madec, D.; Poli, G.: Domino Palladium-Catalyzed Generation and Arylation of Sulfenate Anions
0466
Yamashita, M.; Hirano, K.; Satoh, T.; Miura, M.: Decarboxylative Coupling of Cinnamic Acids with Vinyl Bromides
0467
Han, J. H.; Kwon, Y. E.; Sohn, J.-H.; Ryu, D. H.: Simple and Selective Deprotection of MOM Ethers
0468
Mitsudome, T.; Mizumoto, K.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Palladium-Catalyzed Copper-Free Wacker Oxidation of Internal Olefins
0469
Kabir, M. S.; Lorenz, M.; Namjoshi, O. A.; Cook, J. M.: A New Ligand for Copper-Catalyzed Cross-Coupling of Heterocycles and Phenols

Organo- and Biocatalysis

z471
All PDFs of this category
0471
Durchschein, K.; Silva, B. Ferreira-da; Wallner, S.; Macheroux, P.; Kroutil, W.; Glueck, S. M.; Faber, K.: A Biocatalytic Equivalent to the Nef Reaction
0472
Murai, K.; Fukushima, S.; Hayashi, S.; Takahara, Y.; Fujioka, H.: Trisimidazolines in Asymmetric Conjugate Additions
0473
Rueping, M.; Tato, F.; Schoepke, F. R.: Enantioselective Transfer Hydrogenation of Quinoxalines and Quinoxalinones
0474
Zhang, X.; Zhang, S.; Wang, W.: Iminium-Allenamine Cascade
0475
Ube, H.; Shimada, N.; Terada, M.: Vinylogous Aldol Reaction of Furanones
0476
Sriramurthy, V.; Kwon, O.: Benzoheterocycle Synthesis via Diphosphine Catalysis
0477
Cai, Y.; Wang, W.; Shen, K.; Wang, J.; Hu, X.; Lin, L.; Liu, X.; Feng, X.: α-Chlorination of β-Keto Esters Catalyzed by a Bifunctional N-Oxide/Amide Catalyst
0478
Jiang, H.; Paixão, M. W.; Monge, D.; Jørgensen, K. A.: Asymmetric Additions to α,β-Unsaturated Acyl Phosphonates
0479
Kano, T.; Sakamoto, R.; Mii, H.; Wang, Y. G.; Maruoka, K.: Catalytic Enantioselective Synthesis of Cyclic α-Amino Acids
0480
Hu, J.; Wu, L.-Y.; Wang, X.-C.; Hu, Y.-Y.; Niu, Y.-N.; Liu, X.-Y.; Yang, S.; Liang, Y.-M.: Phase-Transfer-Catalyzed Intramolecular Cyclization of Phenyl Ether Derivatives
0481
Wu, Y.; Yao, W.; Pan, L.; Zhang, Y.; Ma, C.: 3-Halopropenals as β-Acylvinyl Anion Equivalents
0482
Ma, H.; Liu, K.; Zhang, F.-G.; Zhu, C.-L.; Nie, J.; Ma, J.-A.: Michael Addition Catalyzed by Chiral Bifunctional Thioureas Based on Saccharides
0483
Lao, J.-h.; Zhang, X.-j.; Wang, J.-j.; Li, X.-m.; Yan, M.; Luo, H.-b.: Hydrogen-Bonding Catalysts are Hard to Predict
0484
Sugiura, M.; Sato, N.; Sonoda, Y.; Kotani, S.; Nakajima, M.: Chiral Base-Catalyzed Reductive Aldol Reaction with Trichlorosilane
0485
Wei, Q.; Gong, L.-Z.: Formal [4+2] Cycloadditions Promoted by a Chiral Amine Urea Catalyst

Polymer-Supported Synthesis

z487
All PDFs of this category
0487
Lim, J.; Lee, S. S.; Ying, J. Y.: A Mesoporous Silica-Supported Ruthenium Catalyst for Metathesis
0488
Namitharan, K.; Pitchumani, K.: Synthesis of Propargyl Amines with Ni-Y Zeolite
0489
Tailhades, J.; Gidel, M.-A.; Grossi, B.; Lécaillon, J.; Brunel, L.; Subra, G.; Martinez, J.; Amblard, M.: Solid-Phase Synthesis of Peptide Alcohols
0490
Guérin, B.; Ait-Mohand, S.; Tremblay, M.-C.; Dumulon-Perreault, V.; Fournier, P.; Bénard, F.: Solid-Phase Synthesis of NOTA-Functionalized Peptides
0491
Liu, Y.; Tsunoyama, H.; Akita, T.; Tsukuda, T.: Epoxidation of Styrene with Au25 Clusters Grafted on Hydroxyapatite
0492
Quinn, J. F.; Bryant, C. E.; Golden, K. C.; Gregg, B. T.: Reduction of Nitroarenes with Hydrogen Transfer Catalysis
0493
Jammi, S.; Krishnamoorthy, S.; Saha, P.; Kundu, D. S.; Sakthivel, S.; Ali, Md. A.; Paul, R.; Punniyamurthy, T.: N-Arylation of Amides with Cu2O Nano-particles
0494
Zhou, W.-J.; Wang, K.-H.; Wang, J.-X.; Huang, D.-F.: Cross-Coupling of Aryl Halides and Triarylbismuths with PS-Supported Palladium
0495
Fujita, K.-i.; Ainoya, T.; Tsuchimoto, T.; Yasuda, H.: Dihydroxylation of Olefins with a Dendrimer-Supported Osmium Catalyst
0496
Kitahara, H.; Sakurai, H.: Gold Nanoclusters as a Catalyst for Intramolecular Hydroamination
0497
Cho, C.-H.; Kim, C.-B.; Park, K.: Polymer-Supported Synthesis of Stilbenes
0498
Suzuka, T.; Okada, Y.; Ooshiro, K.; Uozumi, Y.: Copper-Free Sonogashira Coupling in Water with a PS-PEG Palladium Complex
0499
Lang, L.; Li, B.; Liu, W.; Jiang, L.; Xu, Z.; Yin, G.: Synthesis of Tetrazoles with Mesoporous ZnS Nanospheres

Addenda and Errata

0500
Synthesis of Englerin A