DOI: 10.1055/s-00000084

Synthesis

Issue 02 · Volume 54 · January 2022 DOI: 10.1055/s-012-52652

table of contents

V
Linked PDF of Table of Contents

review

217
Larionova, Natalia A.; Shestopalov, Anatoliy M.; Rodinovskaya, Lyudmila A.; Zubarev, Andrey A.: Synthesis of Biologically Active Heterocycles via a Domino Sequence Involving an SN2/Thorpe–Ziegler Reaction Step
https://www.thieme-connect.de/media/synthesis/202202/i_z0084_ga_10-1055_a-1526-8160.gif

short review

246
Wei, Baosheng; Knochel, Paul: Recent Advances in Cross-Couplings of Functionalized Organozinc Reagents
https://www.thieme-connect.de/media/synthesis/202202/i_r0450_ga_10-1055_a-1589-0150.gif
255
Oroz, Paula; Avenoza, Alberto; Busto, Jesús H.; Corzana, Francisco; Zurbano, María M.; Peregrina, Jesús M.: Strategies for the Synthesis of Selenocysteine Derivatives
https://www.thieme-connect.de/media/synthesis/202202/i_r0354_ga_10-1055_a-1588-9763.gif
271
Glueck, David S.: Asymmetric Synthesis of P-Stereogenic Secondary Phosphine ­Oxides (SPOs)
https://www.thieme-connect.de/media/synthesis/202202/i_r0413_ga_10-1055_a-1582-0169.gif
281
Zhang, Yong; Sun, Wenxuan; Li, Chao: Nickel-Catalyzed Paired Electrochemical Cross-Coupling of Aryl Halides with Nucleophiles
https://www.thieme-connect.de/media/synthesis/202202/i_r0417_ga_10-1055_a-1581-0934.gif
295
Fokin, Igor; Kuessner, Kai-Thorben; Siewert, Inke: Transition Metal Complex Catalyzed Photo- and Electrochemical (De)hydrogenations Involving C=O and C=N Bonds
https://www.thieme-connect.de/media/synthesis/202202/i_r0488_ga_10-1055_a-1645-3254.jpg
Supporting Information
315
Feng, Yanping; Ye, Xiajuan; Huang, Dayun; Guo, Sheng-rong: α-Csp3–H Bond Functionalization of Simple Ethers in Radical Reactions
https://www.thieme-connect.de/media/synthesis/202202/i_r0422_ga_10-1055_a-1631-1606.gif

feature

334
Beckers, Igor; O’Rourke, Galahad; De Vos, Dirk: Late-Stage C–H Arylation of Azepinoindole via Pd/Cu Catalysis: A Step Efficient and Convergent Synthesis of Rucaparib
https://www.thieme-connect.de/media/synthesis/202202/i_z0392_ga_10-1055_s-0037-1610784.gif
341
Chand-Thakuri, Pratibha; Alahakoon, Indunil; Liu, Daniel; Kapoor, Mohit; Kennedy, John F.; Jenkins, Kenneth W.; Rabon, Allison M.; Young, Michael C.: Native Amine-Directed ortho-C–H Halogenation and Acetoxylation /Condensation of Benzylamines
https://www.thieme-connect.de/media/synthesis/202202/i_m0506_ga_10-1055_a-1625-9095.jpg
Supporting Information
355
El-Tunsi, Ashraf; Carter, Nicholas; Yeo, Song-Hee; Priest, Joshua D.; Choi, Anthony; Kobras, Carolin M.; Ndlovu, Soneni; Proietti Silvestri, Ilaria; Fenton, Andrew K.; Coldham, Iain: Kinetic Resolution by Lithiation: Highly Enantioselective Synthesis of Substituted Dihydrobenzoxazines and Tetrahydroquinoxalines
https://www.thieme-connect.de/media/synthesis/202202/i_z0502_ga_10-1055_a-1638-2478.gif
Supporting Information
369
Tatevosyan, Stepan S.; Kotovshchikov, Yury N.; Latyshev, Gennadij V.; Lukashev, Nikolay V.; Beletskaya, Irina P.: Facile Access to Triazole-Fused 3,1-Benzoxazines Enabled by Metal-Free Base-Promoted Intramolecular C–O Coupling
https://www.thieme-connect.de/media/synthesis/202202/i_z0398_ga_10-1055_a-1623-2333.gif
Supporting Information

psp

378
Janicki, Ignacy; Kiełbasiński, Piotr: A Straightforward, Purification-Free Procedure for the Synthesis of Ando and Still–Gennari Type Phosphonates
https://www.thieme-connect.de/media/synthesis/202202/i_t0381_ga_10-1055_a-1628-7586.gif
Supporting Information

paper

383
Islam, Md. Rafikul; Nishinaga, Tohru; Hirabayashi, Kazunori; Shimizu, Toshio; Sugiura, Ken-ichi: Oxidative Intramolecular C–C Bond Formation Reactions of 1,2-Diarylbenzenes: Syntheses of Highly Conjugated Double-Bridged Polycyclic Aromatic Hydrocarbons
https://www.thieme-connect.de/media/synthesis/202202/i_f0378_ga_10-1055_a-1560-4791.gif
Supporting Information
393
Ghora, Santanu; Sreenivasulu, Chinnabattigalla; Satyanarayana, Gedu: A Domino Heck Coupling–Cyclization–Dehydrogenative Strategy for the One-Pot Synthesis of Quinolines
https://www.thieme-connect.de/media/synthesis/202202/i_f0412_ga_10-1055_a-1589-7548.gif
Supporting Information
403
Wu, Weilong; Jing, Yongkang; Zhang, Deyi; Yan, Xianghe; Liang, Rong; Lu, Zhiqiang; Ji, Baoming: Palladium-Catalyzed Butoxycarbonylation of Polybromo(hetero)arenes: A Practical Method for the Preparation of (Hetero)arenepolycarboxylates and -carboxylic Acids
https://www.thieme-connect.de/media/synthesis/202202/i_g0397_ga_10-1055_a-1587-8859.gif
Supporting Information
411
Zhang, Dongke; Zhang, Jingran; Li, Xiaoxian; Yu, Zhenyang; Li, Yadong; Sun, Fengxia; Du, Yunfei: Intramolecular Chalcogenylation of Isooxazolines Mediated by PhICl2 and Diorganyl Disulfides or Diselenides
https://www.thieme-connect.de/media/synthesis/202202/i_g0429_ga_10-1055_s-0040-1719833.gif
Supporting Information
421
Zhou, Likai; Jia, Kuiyong; Liu, Xigong; Liu, Lei: Enantioselective Transfer Hydrogenation of Oxocarbenium Ions Enables Asymmetric Access to α-Substituted 1,3-Dihydroisobenzofurans
https://www.thieme-connect.de/media/synthesis/202202/i_g0433_ga_10-1055_a-1643-8526.gif
Supporting Information
429
Zhou, Wei; Yao, Lan; Liu, Yongxiurong; Shen, Lichun; Chen, Jie; Deng, Hongmei; Shao, Min; Zhang, Hui; Tang, Xiaojun; Cao, Weiguo: A Catalyst-Free Synthesis of Fused Perfluoroalkylated 2,3-Dihydroisoxazoles via Oxa-Michael-Aldol Annulation
https://www.thieme-connect.de/media/synthesis/202202/i_g0457_ga_10-1055_a-1625-9538.gif
Supporting Information
439
Mittersteiner, Mateus; Aquino, Estefania C.; Budragchaa, Tuvshinjargal; Wessjohann, Ludger A.; Bonacorso, Helio G.; Martins, Marcos A. P.; Zanatta, Nilo: Synthesis of Methylene-Bridged Trifluoromethyl Azoles Using 5-(1,2,3-Triazol-1-yl)enones
https://www.thieme-connect.de/media/synthesis/202202/i_m0469_ga_10-1055_s-0040-1719837.gif
Supporting Information
451
Brahmachari, Goutam; Mandal, Mullicka; Karmakar, Indrajit: Facile and Straightforward Synthesis of Racemic Version of Substituted 3-[3-(2-Hydroxyphenyl)-3-oxo-1-arylpropyl]-4-hydroxycoumarins: Easy Access to a Series of Biorelevant Warfarin Analogues
https://www.thieme-connect.de/media/synthesis/202202/i_n0207_ga_10-1055_a-1624-2176.gif
Supporting Information
465
Heinemann, Maximilian J. B.; Voigt, Thomas; Menche, Dirk: Dihydroxylation Studies of Isoquinolinones: Synthesis of the EF-Ring of Lysolipin I
https://www.thieme-connect.de/media/synthesis/202202/i_t0405_ga_10-1055_a-1628-7972.gif
Supporting Information
475
Xia, Xu-Ling; Zhu, Qi-Long; Chen, Jin-Quan; Shi, Zhen; Dong, Zhi-Bing: Synthesis of Aryl Dithiocarbamates from Tetramethylthiuram Monosulfide (TMTM) and Aryl Boronic Acids: Copper-Catalyzed Construction of C(sp2)–S Bonds
https://www.thieme-connect.de/media/synthesis/202202/i_z0481_ga_10-1055_a-1645-6040.gif
Supporting Information
483
Fuchiya, Asuka; Miyamura, Takuya; Nariki, Haruna; Noda, Shizuki; Makiyama, Kouhei; Sonoda, Motohiro; Tanimori, Shinji: A Facile Synthesis of 2-Aminobenzoxazines Based on Iodine­Catalyzed Desulfurative Cyclization
https://www.thieme-connect.de/media/synthesis/202202/i_f0315_ga_10-1055_s-0040-1719832.gif
Supporting Information
490
He, Jing; Wei, Yueting; Li, Xuezhen; Dai, Bin; Liu, Ping: Tetrabutylammonium Iodide Mediated Sulfenylation of Poly­substituted 1H-Pyrazol-5-amines with Arylsulfonyl Hydrazides
https://www.thieme-connect.de/media/synthesis/202202/i_f0425_ga_10-1055_a-1592-6394.gif
Supporting Information
499
Ma, Yan-Hua; Meng, Fan-Xiao; Wang, Ruo-Nan; Fan, Ya-Xin; Su, Qing-Qiang; Du, Ji-Yuan: Diastereoselective Palladium-Catalyzed [4+1] Cycloadditions of 4-Vinyl-1,4-dihydro-2H-3,1-benzoxazin-2-ones with In Situ Formed Carbenes
https://www.thieme-connect.de/media/synthesis/202202/i_g0352_ga_10-1055_a-1561-5557.gif
Supporting Information
506
Krylov, Igor B.; Paveliev, Stanislav A.; Budnikov, Alexander S.; Segida, Oleg O.; Merkulova, Valentina M.; Vil’, Vera A.; Nikishin, Gennady I.; Terent’ev, Alexander O.: Hidden Reactivity of Barbituric and Meldrum’s Acids: Atom-Efficient Free-Radical C–O Coupling with N-Hydroxy Compounds
https://www.thieme-connect.de/media/synthesis/202202/i_m0443_ga_10-1055_a-1643-7642.gif
Supporting Information